PEAQX tetrasodium salt |
| Catalog No.GC50089 |
Potent and GluN2A-selective NMDA antagonist
Products are for research use only. Not for human use. We do not sell to patients.
Sample solution is provided at 25 µL, 10mM.
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Potent NMDA receptor antagonist (IC50 = 8 nM). Exhibits >100-fold selectivity for hGluN2A (formally hNR2A) containing receptors over hGluN2B (hNR2B). Anticonvulsant in vivo. Please refer to IUPHAR Guide to Pharmacology for the most recent naming conventions.
Auberson et al (2002) 5-Phosphonomethylquinoxalinediones as competitive NMDA receptor antagonists with a preference for the human 1A/2A, rather than 1A/2B receptor composition. Bioorg.Med.Chem.Lett. 12 1099 PMID:11909726
Average Rating: 5 (Based on Reviews and 5 reference(s) in Google Scholar.)
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