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AChR

AChR, also known as acetylcholine receptor, is an integral membrane protein that responds to the binding of acetylcholine.

Products for  AChR

  1. Cat.No. Product Name Information
  2. GC26093 α-Conotoxin GI α-Conotoxin GI, a 13-residue peptide originally isolated from the venom of the fish-hunting cone snail Conus geographus, acts as a competitive antagonist for the muscle-type nicotinic acetylcholine receptor (nAChR) with excellent selectivity for α/δ receptor subunit binding over α/γ. α-Conotoxin GI  Chemical Structure
  3. GC11128 (±)-Vesamicol hydrochloride acetylcholine transport inhibitor (±)-Vesamicol hydrochloride  Chemical Structure
  4. GC11219 (R)-(+)-Tolterodine (R)-(+)-Tolterodine(PNU-200583) is a potent muscarinic receptor antagonists that show selectivity for the urinary bladder over salivary glands in vivo. (R)-(+)-Tolterodine  Chemical Structure
  5. GC15014 A-867744 A positive allosteric modulator of α7 nAChRs A-867744  Chemical Structure
  6. GC14142 Acetylcholine Chloride Major transmitter at many nervous sites Acetylcholine Chloride  Chemical Structure
  7. GC11786 Acetylcysteine Acetylcysteine is the N-acetyl derivative of CYSTEINE. Acetylcysteine  Chemical Structure
  8. GC13240 Arecoline Muscarinic acetylcholine receptors agonist Arecoline  Chemical Structure
  9. GC16526 Atropine MAChRs antagonist Atropine  Chemical Structure
  10. GC14419 Bethanechol chloride Muscarinic receptor agonist Bethanechol chloride  Chemical Structure
  11. GC16255 Decamethonium Bromide Nicotinic AChR partial agonist Decamethonium Bromide  Chemical Structure
  12. GC16635 Diphemanil Methylsulfate Diphemanil methylsulfate is a quaternary ammonium anticholinergic. Diphemanil Methylsulfate  Chemical Structure
  13. GC25387 Ethyl (triphenylphosphoranylidene) acetate Ethyl (triphenylphosphoranylidene) acetate (Triphenylcarbethoxymethylenephosphorane, (Carbethoxymethylene)triphenylphosphorane) may act as an inhibitor of cholinesterase that inhibits AChE and BChE. Ethyl (triphenylphosphoranylidene) acetate  Chemical Structure
  14. GC13361 Flavoxate hydrochloride muscarinic AChR antagonist Flavoxate hydrochloride  Chemical Structure
  15. GC16573 Galanthamine An alkaloid with AChE inhibitory and nAChR potentiating activities Galanthamine  Chemical Structure
  16. GC14624 Galanthamine HBr Acetylcholinesterase inhibitor Galanthamine HBr  Chemical Structure
  17. GC10972 Gallamine Triethiodide Cholinergic receptor blocker Gallamine Triethiodide  Chemical Structure
  18. GC15029 Glycopyrrolate Muscarinic competitive antagonist Glycopyrrolate  Chemical Structure
  19. GC15178 Hexamethonium Bromide Selective antagonist of neuronal-type nicotinic AChR Hexamethonium Bromide  Chemical Structure
  20. GC13897 Homatropine Bromide Muscarinic AChR antagonist Homatropine Bromide  Chemical Structure
  21. GC17908 Homatropine Methylbromide Muscarinic AChR antagonist Homatropine Methylbromide  Chemical Structure
  22. GC11035 Hyoscyamine Hyoscyamine (Daturine), a natural plant tropane alkaloid, is a potent and competitive muscarinic receptor (MR) antagonist. Hyoscyamine  Chemical Structure
  23. GC12717 Ipratropium Bromide AChR antagonist Ipratropium Bromide  Chemical Structure
  24. GC13314 L-Acetylcarnitine (hydrochloride) Acetyl-L-carnitine (O-Acetyl-L-carnitine) hydrochloride is a blood-brain permeable acetyl ester of the amino acid L-carnitine found in the body. L-Acetylcarnitine (hydrochloride)  Chemical Structure
  25. GC25583 Lobelin sulphate Lobelin sulphate (Lobeline sulfate, Bantron) is an alkaloid that has actions similar to nicotine on nicotinic cholinergic receptors but is less potent. It has a variety of therapeutic uses including in respiratory disorders, peripheral vascular disorders, insomnia, and smoking cessation. Lobelin sulphate  Chemical Structure
  26. GC13445 LY2119620 positive allosteric modulator of M2/M4 receptor LY2119620  Chemical Structure
  27. GC17825 Methscopolamine Muscarinic acetylcholine receptor blocker Methscopolamine  Chemical Structure
  28. GC12507 ML352 Non-competitive inhibitor of the presynaptic choline transporter ML352  Chemical Structure
  29. GC16056 Neostigmine Bromide Cholinesterase inhibitor Neostigmine Bromide  Chemical Structure
  30. GC17627 Nitenpyram nicotinic acetylcholine receptor (AchR) agonist Nitenpyram  Chemical Structure
  31. GC13779 Orphenadrine Citrate Antiparkinsonian and analgesic drug Orphenadrine Citrate  Chemical Structure
  32. GC10863 Otilonium Bromide AChR inhibitor Otilonium Bromide  Chemical Structure
  33. GC14113 Oxybutynin AChR antagonist Oxybutynin  Chemical Structure
  34. GC14703 Oxybutynin chloride Anticholinergic medication Oxybutynin chloride  Chemical Structure
  35. GC11773 Pancuronium dibromide AChR antagonist Pancuronium dibromide  Chemical Structure
  36. GC17229 Paroxetine HCl Paroxetine HCl is a potent selective serotonin-reuptake inhibitor, commonly prescribed as an and has GRK2 inhibitory ability with IC50 of 14μM. Paroxetine HCl  Chemical Structure
  37. GC11643 PNU-120596 α7 nAChR modulator,positive allosteric PNU-120596  Chemical Structure
  38. GC12920 Pregnenolone steroid hormone Pregnenolone  Chemical Structure
  39. GC10267 Rivastigmine A cholinesterase inhibitor Rivastigmine  Chemical Structure
  40. GC12994 Rivastigmine Tartrate AChR inhibitor Rivastigmine Tartrate  Chemical Structure
  41. GC13449 Rocuronium Bromide TGF-βR I kinase inhibitor Rocuronium Bromide  Chemical Structure
  42. GC10508 Solifenacin hydrochloride muscarinic receptor antagonist Solifenacin hydrochloride  Chemical Structure
  43. GC12453 Succinylcholine Chloride Dihydrate Nicotinic AChR agonist Succinylcholine Chloride Dihydrate  Chemical Structure
  44. GC13618 Tarafenacin M3 muscarinic receptor antagonist Tarafenacin  Chemical Structure
  45. GC16059 Tarafenacin D-tartrate Highly selective M3 muscarinic receptor antagonist Tarafenacin D-tartrate  Chemical Structure
  46. GC25994 Thonzylamine Thonzylamine (Neohetramine) is an antihistamine and anticholinergic drug. Thonzylamine  Chemical Structure
  47. GC12554 Tiotropium Bromide A muscarinic receptor antagonist Tiotropium Bromide  Chemical Structure
  48. GC13134 Tiotropium Bromide hydrate Muscarinic antagonist Tiotropium Bromide hydrate  Chemical Structure
  49. GC15150 Tropicamide Antimuscarinic drug Tropicamide  Chemical Structure
  50. GC17483 Trospium chloride Antimuscarinic agent Trospium chloride  Chemical Structure
  51. GC26032 Varenicline (CP 526555) dihydrochloride Varenicline (CP 526555, Chantix, Champix,CP 526555 dihydrochloride) dihydrochloride is a potent, partial agonist of α4β2 nicotinic acetylcholine receptor (nAChR) and α3β4 nAChR with EC50 of 2.3 μM and 55 μM, respectively. Varenicline dihydrochloride is a potent, full agonist of α7 nAChRs with EC50 of 18 μM. Varenicline is a prescription medication used for smoking cessation. Varenicline (CP 526555) dihydrochloride  Chemical Structure
  52. GC10948 Varenicline Tartrate Subtype-selective agonist of α4β2 nicotinic receptors,orally active Varenicline Tartrate  Chemical Structure
  53. GC11210 Vecuronium Bromide Nonpolarizing neuromuscular relaxant Vecuronium Bromide  Chemical Structure
  54. GC16819 VU0152100 M4 receptor allosteric modulators VU0152100  Chemical Structure
  55. GC17885 VU0364572 (trifluoroacetate salt) M1 agonist VU0364572 (trifluoroacetate salt)  Chemical Structure

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