AChR
AChR, also known as acetylcholine receptor, is an integral membrane protein that responds to the binding of acetylcholine.
Products for AChR
- Cat.No. Product Name Information
- GC26093 α-Conotoxin GI α-Conotoxin GI, a 13-residue peptide originally isolated from the venom of the fish-hunting cone snail Conus geographus, acts as a competitive antagonist for the muscle-type nicotinic acetylcholine receptor (nAChR) with excellent selectivity for α/δ receptor subunit binding over α/γ.
- GC11128 (±)-Vesamicol hydrochloride acetylcholine transport inhibitor
- GC11219 (R)-(+)-Tolterodine (R)-(+)-Tolterodine(PNU-200583) is a potent muscarinic receptor antagonists that show selectivity for the urinary bladder over salivary glands in vivo.
- GC15014 A-867744 A positive allosteric modulator of α7 nAChRs
- GC14142 Acetylcholine Chloride Major transmitter at many nervous sites
- GC11786 Acetylcysteine Acetylcysteine is the N-acetyl derivative of CYSTEINE.
- GC13240 Arecoline Muscarinic acetylcholine receptors agonist
- GC16526 Atropine MAChRs antagonist
- GC14419 Bethanechol chloride Muscarinic receptor agonist
- GC16255 Decamethonium Bromide Nicotinic AChR partial agonist
- GC16635 Diphemanil Methylsulfate Diphemanil methylsulfate is a quaternary ammonium anticholinergic.
- GC25387 Ethyl (triphenylphosphoranylidene) acetate Ethyl (triphenylphosphoranylidene) acetate (Triphenylcarbethoxymethylenephosphorane, (Carbethoxymethylene)triphenylphosphorane) may act as an inhibitor of cholinesterase that inhibits AChE and BChE.
- GC13361 Flavoxate hydrochloride muscarinic AChR antagonist
- GC16573 Galanthamine An alkaloid with AChE inhibitory and nAChR potentiating activities
- GC14624 Galanthamine HBr Acetylcholinesterase inhibitor
- GC10972 Gallamine Triethiodide Cholinergic receptor blocker
- GC15029 Glycopyrrolate Muscarinic competitive antagonist
- GC15178 Hexamethonium Bromide Selective antagonist of neuronal-type nicotinic AChR
- GC13897 Homatropine Bromide Muscarinic AChR antagonist
- GC17908 Homatropine Methylbromide Muscarinic AChR antagonist
- GC11035 Hyoscyamine Hyoscyamine (Daturine), a natural plant tropane alkaloid, is a potent and competitive muscarinic receptor (MR) antagonist.
- GC12717 Ipratropium Bromide AChR antagonist
- GC13314 L-Acetylcarnitine (hydrochloride) Acetyl-L-carnitine (O-Acetyl-L-carnitine) hydrochloride is a blood-brain permeable acetyl ester of the amino acid L-carnitine found in the body.
- GC25583 Lobelin sulphate Lobelin sulphate (Lobeline sulfate, Bantron) is an alkaloid that has actions similar to nicotine on nicotinic cholinergic receptors but is less potent. It has a variety of therapeutic uses including in respiratory disorders, peripheral vascular disorders, insomnia, and smoking cessation.
- GC13445 LY2119620 positive allosteric modulator of M2/M4 receptor
- GC17825 Methscopolamine Muscarinic acetylcholine receptor blocker
- GC12507 ML352 Non-competitive inhibitor of the presynaptic choline transporter
- GC16056 Neostigmine Bromide Cholinesterase inhibitor
- GC17627 Nitenpyram nicotinic acetylcholine receptor (AchR) agonist
- GC13779 Orphenadrine Citrate Antiparkinsonian and analgesic drug
- GC10863 Otilonium Bromide AChR inhibitor
- GC14113 Oxybutynin AChR antagonist
- GC14703 Oxybutynin chloride Anticholinergic medication
- GC11773 Pancuronium dibromide AChR antagonist
- GC17229 Paroxetine HCl Paroxetine HCl is a potent selective serotonin-reuptake inhibitor, commonly prescribed as an and has GRK2 inhibitory ability with IC50 of 14μM.
- GC11643 PNU-120596 α7 nAChR modulator,positive allosteric
- GC12920 Pregnenolone steroid hormone
- GC10267 Rivastigmine A cholinesterase inhibitor
- GC12994 Rivastigmine Tartrate AChR inhibitor
- GC13449 Rocuronium Bromide TGF-βR I kinase inhibitor
- GC10508 Solifenacin hydrochloride muscarinic receptor antagonist
- GC12453 Succinylcholine Chloride Dihydrate Nicotinic AChR agonist
- GC13618 Tarafenacin M3 muscarinic receptor antagonist
- GC16059 Tarafenacin D-tartrate Highly selective M3 muscarinic receptor antagonist
- GC25994 Thonzylamine Thonzylamine (Neohetramine) is an antihistamine and anticholinergic drug.
- GC12554 Tiotropium Bromide A muscarinic receptor antagonist
- GC13134 Tiotropium Bromide hydrate Muscarinic antagonist
- GC15150 Tropicamide Antimuscarinic drug
- GC17483 Trospium chloride Antimuscarinic agent
- GC26032 Varenicline (CP 526555) dihydrochloride Varenicline (CP 526555, Chantix, Champix,CP 526555 dihydrochloride) dihydrochloride is a potent, partial agonist of α4β2 nicotinic acetylcholine receptor (nAChR) and α3β4 nAChR with EC50 of 2.3 μM and 55 μM, respectively. Varenicline dihydrochloride is a potent, full agonist of α7 nAChRs with EC50 of 18 μM. Varenicline is a prescription medication used for smoking cessation.
- GC10948 Varenicline Tartrate Subtype-selective agonist of α4β2 nicotinic receptors,orally active
- GC11210 Vecuronium Bromide Nonpolarizing neuromuscular relaxant
- GC16819 VU0152100 M4 receptor allosteric modulators
- GC17885 VU0364572 (trifluoroacetate salt) M1 agonist