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Home >> Signaling Pathways >> Neuroscience >> Histamine Receptor

Histamine Receptor

Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.

Products for  Histamine Receptor

  1. Cat.No. Product Name Information
  2. GC33544 (±)-Methotrimeprazine (D6) (dl-Methotrimeprazine D6) (±)-Levomepromazine D6 ((±)-Methotrimeprazine D6) is the deuterium labeled Methotrimeprazine, which is a D3 dopamine and Histamine H1 receptor antagonist. (±)-Methotrimeprazine (D6) (dl-Methotrimeprazine D6) Chemical Structure
  3. GC31026 (±)-Tazifylline (±)-Tazifylline is a potent, selective and long-acting histamine H1 receptor antagonist. (±)-Tazifylline Chemical Structure
  4. GC69834 (R)-(+)-Dimethindene maleate

    (R)-(+)-Dimethindene maleate is an orally active H1-receptor blocker with anti-histamine properties in pigs.

     (R)-(+)-Dimethindene maleate Chemical Structure
  5. GC11809 (R)-(-)-α-Methylhistamine dihydrobromide (R)-(-)-α-Methylhistamine dihydrobromide is a potent, selective and brain-penetrant agonist of H3 histamine receptor, with a Kd of 50.3 nM. (R)-(-)-α-Methylhistamine dihydrobromide Chemical Structure
  6. GC41715 (R)-Cetirizine (hydrochloride) A selective histamine H1 receptor antagonist (R)-Cetirizine (hydrochloride) Chemical Structure
  7. GC10704 (S)-(+)-α-Methylhistamine dihydrobromide H3 histamine receptor agonist (S)-(+)-α-Methylhistamine dihydrobromide Chemical Structure
  8. GC11001 2-Pyridylethylamine dihydrochloride

    Histamine H1 receptor agonist

     2-Pyridylethylamine dihydrochloride Chemical Structure
  9. GC12737 4-Methylhistamine dihydrochloride H4 receptor agonist 4-Methylhistamine dihydrochloride Chemical Structure
  10. GC13537 A 331440 dihydrochloride H3 receptor antagonist,non-imidazole,high affinity A 331440 dihydrochloride Chemical Structure
  11. GC11121 A 943931 dihydrochloride Antagonist of histamine H4 receptor,potent and selective A 943931 dihydrochloride Chemical Structure
  12. GC17743 A 987306 H4 receptor antagonist,potent and selective A 987306 Chemical Structure
  13. GC35222 ABT-239 ABT-239 is a novel, highly efficacious, non-imidazole?class of H3R antagonist and a transient receptor potential vanilloid type 1 (TRPV1) antagonist. ABT-239 Chemical Structure
  14. GC31695 Acrivastine (BW825C) Acrivastine (BW825C) (BW825C) is a short acting histamine 1 receptor antagonist for the treatment of allergic rhinitis. Acrivastine (BW825C) Chemical Structure
  15. GC60563 Acrivastine D7 Acrivastine D7 (BW825C D7) is a deuterium labeled Acrivastine. Acrivastine D7 Chemical Structure
  16. GC17517 Alcaftadine H1 histamine receptor antagonist Alcaftadine Chemical Structure
  17. GC35284 Alimemazine D6 Alimemazine D6 is deuterium labeled Alimemazine, which is an antihistamine. Alimemazine D6 Chemical Structure
  18. GC16052 Aminopotentidine H2 antagonist Aminopotentidine Chemical Structure
  19. GC25060 Amitriptyline Amitriptyline (MK-230, N-750, Ro41575) is a tricyclic antidepressant (TCA) with analgesic properties, widely used to treat depression and neuropathic pain. Amitriptyline is an inhibitor of both serotonin transporter (SERT) and norepinephrine transporter (NET) with Ki of 3.45 nM and 13.3 nM, respectively. Amitriptyline also inhibits histamine receptor H1, histamine receptor H4, 5-HT2 and sigma 1 receptor with Ki of 0.5 nM, 7.31 nM, 235 nM and 287 nM, respectively. This product is a waxy solid. Amitriptyline Chemical Structure
  20. GC12472 Amthamine dihydrobromide H2 agonist Amthamine dihydrobromide Chemical Structure
  21. GC13899 Antazoline HCl Antazoline HCl is a 1st generation antihistamine with also anticholinergic properties used to relieve nasal congestion and in eye drops. Antazoline HCl Chemical Structure
  22. GC31141 Antihistamine-1 Antihistamine-1 is a H1-antihistamine (Ki=6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively. Antihistamine-1 Chemical Structure
  23. GC16945 Astemizole anti-histamine compound, potent Astemizole Chemical Structure
  24. GC14070 Azatadine Histamine and cholinergic inhibitor Azatadine Chemical Structure
  25. GC15776 Azatadine dimaleate Histamine and cholinergic inhibitor Azatadine dimaleate Chemical Structure
  26. GC33879 Azelastine Azelastine, an antihistamine, is a potent and selective histamine 1 (H1) antagonist. Azelastine Chemical Structure
  27. GC17297 Azelastine HCl Azelastine HClm, an antihistamine, is a potent and selective histamine 1 (H1) antagonist. Azelastine HCl Chemical Structure
  28. GC31840 Bamirastine (TAK-427) Bamirastine (TAK-427) inhibits ligand binding to recombinant human histamine H1 receptors (rhH1R) with an IC50 value of 17.3 nM. Bamirastine (TAK-427) Chemical Structure
  29. GC35471 Bavisant Bavisant (JNJ-31001074) is an orally active, potent, brain-penetrating and highly selective antagonist of the histamine H3 receptor. Bavisant Chemical Structure
  30. GC35472 Bavisant dihydrochloride Bavisant (JNJ-31001074) dihydrochloride is an orally active, potent, brain-penetrating and highly selective antagonist of the histamine H3 receptor. Bavisant dihydrochloride Chemical Structure
  31. GC35473 Bavisant dihydrochloride hydrate Bavisant dihydrochloride hydrate (JNJ31001074AAC) is an orally active, potent, brain-penetrating and highly selective antagonist of the histamine H3 receptor. Bavisant dihydrochloride hydrate Chemical Structure
  32. GC16791 Benztropine mesylate Dopamine transporter (DAT) inhibitor Benztropine mesylate Chemical Structure
  33. GC39479 Bepotastine Bepotastine is a selective and orally active second-generation histamine H1 receptor antagonist, can suppress the expression of nerve growth factor (NGF). Bepotastine Chemical Structure
  34. GC14250 Bepotastine Besilate Non-sedating, selective antagonist of histamine 1 (H1) receptor Bepotastine Besilate Chemical Structure
  35. GC60072 Betahistine Betahistine is an orally active histamine H1 receptor agonist and a H3 receptor antagonist. Betahistine Chemical Structure
  36. GC10127 Betahistine 2HCl Betahistine 2HCl is an orally active histamine H1 receptor agonist and a H3 receptor antagonist. Betahistine 2HCl Chemical Structure
  37. GC60641 Betahistine mesylate Betahistine mesylate is an orally active histamine H1 receptor agonist and a H3 receptor antagonist. Betahistine mesylate Chemical Structure
  38. GC63923 Betahistine-d3 dihydrochloride Betahistine-d3 dihydrochloride Chemical Structure
  39. GC61539 Betazole Betazole (Ametazole), a pyrazole analogue of histamine, is an orally active histamine H2 receptor agonist. Betazole Chemical Structure
  40. GC25136 Betazole Dihydrochloride Betazole Dihydrochloride (Ametazole, 2-(3-Pyrazolyl)ethanamine) is a histamine H2 agonist used clinically to test gastric secretory function. Betazole Dihydrochloride Chemical Structure
  41. GC17643 Bilastine H1 histamine receptor antagonist Bilastine Chemical Structure
  42. GC63318 Bilastine-d6 Bilastine-d6 Chemical Structure
  43. GC31877 BMY-25271 BMY-25271 is a histamine H2 receptor antagonist. BMY-25271 Chemical Structure
  44. GC13341 Brompheniramine hydrogen maleate Brompheniramine ((±)-Brompheniramine) maleate is a potent and orally active antihistamine of the alkylamine class. Brompheniramine hydrogen maleate Chemical Structure
  45. GC15068 Buclizine HCl Buclizine HCl is an orally active antihistamine antiallergic compound. Buclizine HCl Chemical Structure
  46. GC13757 CarbinoxaMine Maleate CarbinoxaMine Maleate is a histamine H1 receptor antagonist. CarbinoxaMine Maleate Chemical Structure
  47. GC13995 Carcinine ditrifluoroacetate H3 receptor antagonist Carcinine ditrifluoroacetate Chemical Structure
  48. GC18198 Carebastine Carebastine is an active metabolite of ebastine . Carebastine Chemical Structure
  49. GC10185 Cetirizine Cetirizine Chemical Structure
  50. GC67944 Cetirizine D4 Cetirizine D4 Chemical Structure
  51. GC35655 Cetirizine D4 dihydrochloride Cetirizine D4 dihydrochloride is a deuterium labeled Cetirizine. Cetirizine D4 dihydrochloride Chemical Structure
  52. GC68409 Cetirizine D8 Cetirizine D8 Chemical Structure
  53. GC35656 Cetirizine D8 dihydrochloride Cetirizine D8 dihydrochloride is a deuterium labeled Cetirizine. Cetirizine D8 dihydrochloride Chemical Structure
  54. GC11009 Cetirizine DiHCl Cetirizine DiHCl, a second-generation antihistamine and the carboxylated metabolite of hydroxyzine, is a specific, orally active and long-acting histamine H1-receptor antagonist. Cetirizine DiHCl Chemical Structure
  55. GC60691 Cetirizine Impurity C Cetirizine Impurity C is an impurity of Cetirizine. Cetirizine Impurity C Chemical Structure
  56. GC64577 Cetirizine Impurity C dihydrochloride Cetirizine Impurity C dihydrochloride is an impurity of Cetirizine. Cetirizine Impurity C dihydrochloride Chemical Structure
  57. GC63666 Chlorcyclizine Chlorcyclizine Chemical Structure
  58. GC13465 Chlorcyclizine (hydrochloride) histamine H1 receptor antagonist and inhibits HCV Chlorcyclizine (hydrochloride) Chemical Structure
  59. GC32979 Chloropyramine hydrochloride Chloropyramine hydrochloride is a histamine receptor H1 antagonist which can also inhibit the biochemical function of VEGFR-3 and FAK. Chloropyramine hydrochloride Chemical Structure
  60. GC16047 Chlorpheniramine Maleate Histamine H1 receptor antagonist Chlorpheniramine Maleate Chemical Structure
  61. GC30948 Chlorphenoxamine Chlorphenoxamine is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent. Chlorphenoxamine Chemical Structure
  62. GC31994 CI-949 CI-949 is an allergic mediator release inhibitor, which inhibits histamine, leukotriene C4/D4 (LTC4/LTD4), and thromboxane B2 (TXB2) release with IC50s of 11.4 μM, 0.5 μM and 0.1 μM, respectively. CI-949 Chemical Structure
  63. GC13486 Cimetidine H2 receptor antagonist Cimetidine Chemical Structure
  64. GC62267 Cimetidine sulfoxide Cimetidine sulfoxide (Cimetidine sulphoxide) is a sulfoxide metabolite of Cimetidine. Cimetidine sulfoxide Chemical Structure
  65. GC11695 Cinnarizine antihistamine and calcium channel blocker Cinnarizine Chemical Structure
  66. GC60709 Cinnarizine D8 An internal standard for the quantification of cinnarizine Cinnarizine D8 Chemical Structure
  67. GC31269 Cipralisant (GT-2331) Cipralisant (GT-2331) (GT-2331) is an orally active, low-toxicity, potent, selective, high affinity histamine H3 receptor full antagonist in vivo, and an agonist in vitro, with a pKi of 9.9 for histamine H3 receptor and a Ki of 0.47 nM for rat histamine H3 receptor. Cipralisant (GT-2331) Chemical Structure
  68. GC12924 Ciproxifan Histamine H3-receptor antagonist Ciproxifan Chemical Structure
  69. GC15847 Ciproxifan maleate Potent histamine H3 receptor antagonist Ciproxifan maleate Chemical Structure
  70. GC14892 Clemastine Fumarate Selective histamine H1 receptor antagonist Clemastine Fumarate Chemical Structure
  71. GC12444 Clemizole An antihistamine and TRPC5 channel blocker Clemizole Chemical Structure
  72. GC17701 Clemizole hydrochloride An antihistamine and TRPC5 channel blocker Clemizole hydrochloride Chemical Structure
  73. GC10490 Clobenpropit dihydrobromide

    histamine H3 antagonist/inverse agonist

     Clobenpropit dihydrobromide Chemical Structure
  74. GC12749 Conessine A histamine H3 receptor antagonist Conessine Chemical Structure
  75. GC30423 CP-66948 CP-66948 is a histamine H2-receptor antagonist with gastric antisecretory activity and mucosal protective properties. CP-66948 Chemical Structure
  76. GC64088 Cyclizine Cyclizine Chemical Structure
  77. GC12039 Cyclizine 2HCl Histamine H1 receptor antagonist Cyclizine 2HCl Chemical Structure
  78. GC43353 Cyproheptadine (hydrochloride hydrate) Cyproheptadine (hydrochloride hydrate) is an antihistamine and is an antagonist of serotonin and histamine2. Cyproheptadine (hydrochloride hydrate) Chemical Structure
  79. GC10698 Cyproheptadine hydrochloride serotonin and histamine antagonist as well as antimuscarinic reagent Cyproheptadine hydrochloride Chemical Structure
  80. GC10321 Decloxizine histamine 1 receptor antagonist Decloxizine Chemical Structure
  81. GC35826 Decloxizine dihydrochloride Decloxizine dihydrochloride(UCB-1402; NSC289116) is a histamine 1 receptor antagonist. Decloxizine dihydrochloride Chemical Structure
  82. GC16416 Desloratadine High affinity histamine H1 receptor antagonist Desloratadine Chemical Structure
  83. GC43427 Dexchlorpheniramine (maleate)

    Dexchlorpheniramine is a histamine H1 receptor antagonist with a pA2 value of 9.36 in guinea pig ileal tissue in vitro.

     Dexchlorpheniramine (maleate) Chemical Structure
  84. GC11883 Dimaprit dihydrochloride H2 agonist Dimaprit dihydrochloride Chemical Structure
  85. GC15723 Dimebolin antihistamine, orally-available Dimebolin Chemical Structure
  86. GC30902 Dimenhydrinate Dimenhydrinate is an anti-emetic and anti-histamine commonly available over-the-counter as a motion sickness remedy. Dimenhydrinate Chemical Structure
  87. GC66445 Dimethindene maleate Dimethindene maleate is a selective histamine H1 antagonist with antihistamine effects. Dimethindene maleate can be used for the research of hypersensitivity reactions. Dimethindene maleate Chemical Structure
  88. GC10445 Diphenhydramine HCl Diphenhydramine HCl is a first-generation histamine H1-receptor antagonist with anti-cholinergic effect. Diphenhydramine HCl Chemical Structure
  89. GC48835 Diphenylpyraline A histamine H1 receptor antagonist Diphenylpyraline Chemical Structure
  90. GC14984 Diphenylpyraline HCl Diphenylpyraline HCl is a potent histamine H1receptor antagonist. Diphenylpyraline HCl Chemical Structure
  91. GC12892 Doxepin (hydrochloride) histamine, serotonin, adrenergic, and muscarinic receptors antagonist Doxepin (hydrochloride) Chemical Structure
  92. GC60791 Doxepin D3 Hydrochloride Doxepin D3 Hydrochloride is a deuterium labeled Doxepin Hydrochloride. Doxepin D3 Hydrochloride Chemical Structure
  93. GC30496 Doxylamine D5 succinate Doxylamine D5 succinate is deuterium labeled Doxylamine, which is a first generation antihistamine. Doxylamine D5 succinate Chemical Structure
  94. GC14051 Doxylamine Succinate Histamine receptor inhibitor Doxylamine Succinate Chemical Structure
  95. GC14742 DPPE fumarate DPPE fumarate (DPPE fumarate), an H1C receptor antagonist, potentiates a wide range of cytotoxics and even to offer some protection of normal cells. DPPE fumarate Chemical Structure
  96. GC15713 Ebastine Histamine receptor antagonist Ebastine Chemical Structure
  97. GC16089 Ebrotidine Ebrotidine Chemical Structure
  98. GC39378 Emedastine Emedastine is an orally active, selective and high affinity histamine H1 receptor antagonist with a Ki value of 1.3 nM. Emedastine Chemical Structure
  99. GC43598 Emedastine (fumarate) Emedastine (fumarate) is an orally active, selective and high affinity histamine H1 receptor antagonist with a Ki value of 1.3 nM. Emedastine (fumarate) Chemical Structure
  100. GC31708 Epinastine (WAL801) Epinastine (WAL801) (WAL801) is an antihistamine and mast cell stabilizer. Epinastine (WAL801) Chemical Structure
  101. GC12030 Epinastine HCl Epinastine HCl (WAL801 hydrochloride) is an antihistamine and mast cell stabilizer. Epinastine HCl Chemical Structure

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