Muscarinic Receptor
Muscarinic receptor is a group of G-protein coupled receptors that binds to acetylcholine and mediates cellular responses, including inhibition of acetylate cyclase, phosphoinositide degradation and regulation of potassium channels. It is involved in the neurological diseases such as Alzheimer's and Parkinson's.
Products for Muscarinic Receptor
- Cat.No. Product Name Information
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GC10736
(+)-Muscarine iodide
Muscarinic acetylcholine receptor agonist
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GC14479
(S)-(+)-Dimethindene maleate
M2 muscarinic receptor antagonist
- GC13348 4-DAMP M3 cholinergic receptor antagonist
- GC14604 5-Methylfurmethiodide muscarinic agonist
- GC12787 Aceclidine (hydrochloride) agonist of muscarinic receptors
- GC14096 Aclidinium Bromide LAMAs antagonist
- GC10219 AF-DX 116 AF-DX 116 (AF-DX 116) is a selective and competitive M2 muscarinic acetylcholine receptor antagonist, with IC50 values of 640 nM and 386 nM for rabbit peripheral lung and rat heart, respectively.
- GC15510 AF-DX 384 M2/M4 selective antagonist
- GC13340 AQ-RA 741 M2 antagonist,selective and high affinity
- GC11415 Arecaidine but-2-ynyl ester tosylate mAChR M2 agonist
- GC16504 Arecaidine propargyl ester tosylate muscarinic receptor agonist
- GC10621 Biperiden HCl Biperiden (KL 373) hydrochloride is a non-selective muscarinic receptor antagonist that competitively binds to M1 muscarinic receptors, thereby inhibiting acetylcholine and enhancing dopamine signaling in the central nervous system.
- GC15758 BQCA positive allosteric modulator of the M1 muscarinic acetylcholine receptor (mAChR)
- GC14215 Cevimeline A muscarinic receptor agonist
- GC17157 Cevimeline hydrochloride hemihydrate
- GC15772 Darifenacin HBr Darifenacin HBr (UK-88525 hydrobromide) is a selective M3 muscarinic receptor antagonist with pKi of 8.9.
- GC10633 DAU 5884 hydrochloride muscarinic M3 receptor antagonist
- GC16087 Fesoterodine Fumarate Muscarinic AChR receptor antagonist
- GC15845 Guvacoline (hydrobromide) full agonist of atrial and ileal muscarinic receptors
- GC12056 J 104129 fumarate M3 muscarinic receptor antagonist
- GC16458 McN-A 343 muscarinic M1 receptor agonist
- GC14619 Milameline hydrochloride Muscarinic receptor agonist
- GC10378 N-Isopropylnoratropine used in the synthesis of ipratropium, a muscarinic antagonist
- GC10525 Nitrocaramiphen hydrochloride M1 muscarinic antagonist
- GC16463 Oxotremorine M Muscarinic receptor agonist
- GC16156 Oxotremorine sesquifumarate Muscarinic agonist
- GC17876 PD 102807 M4 muscarinic receptor antagonist
- GC13403 Pirenzepine dihydrochloride M1 muscarinic receptor selective antagonist
- GC14508 PTAC oxalate muscarinic receptor ligand
- GC17182 Solifenacin succinate Muscarinic receptor antagonist
- GC13174 Telenzepine dihydrochloride muscarinic M1 receptor antagonist
- GC17954 Tolterodine tartrate Competitive muscarinic receptor antagonist
- GC12311 Trihexyphenidyl hydrochloride antiparkinsonian agent of the antimuscarinic class
- GC11831 Umeclidinium bromide A muscarinic acetylcholine receptor antagonist
- GC15990 VU 0238429 positive allosteric modulator of M5 receptors
- GC10464 VU 0255035 muscarinic M1 antagonist
- GC16655 VU 0357017 hydrochloride Positive allosteric modulator of muscarinic M1 receptors
- GC17821 VU 0365114 positive allosteric modulator of M5
- GC10725 VU 10010 allosteric potentiator of M4 acetylcholine receptors
- GC13129 W-84 dibromide M2-receptor selective modulator
- GC18082 Zamifenacin fumarate M3 muscarinic receptor antagonist