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Muscarinic Receptor

Muscarinic receptor is a group of G-protein coupled receptors that binds to acetylcholine and mediates cellular responses, including inhibition of acetylate cyclase, phosphoinositide degradation and regulation of potassium channels. It is involved in the neurological diseases such as Alzheimer's and Parkinson's.

Products for  Muscarinic Receptor

  1. Cat.No. Product Name Information
  2. GC10736 (+)-Muscarine iodide

    Muscarinic acetylcholine receptor agonist

    (+)-Muscarine iodide  Chemical Structure
  3. GC14479 (S)-(+)-Dimethindene maleate

    M2 muscarinic receptor antagonist

    (S)-(+)-Dimethindene maleate  Chemical Structure
  4. GC13348 4-DAMP M3 cholinergic receptor antagonist 4-DAMP  Chemical Structure
  5. GC14604 5-Methylfurmethiodide muscarinic agonist 5-Methylfurmethiodide  Chemical Structure
  6. GC12787 Aceclidine (hydrochloride) agonist of muscarinic receptors Aceclidine (hydrochloride)  Chemical Structure
  7. GC14096 Aclidinium Bromide LAMAs antagonist Aclidinium Bromide  Chemical Structure
  8. GC10219 AF-DX 116 AF-DX 116 (AF-DX 116) is a selective and competitive M2 muscarinic acetylcholine receptor antagonist, with IC50 values of 640 nM and 386 nM for rabbit peripheral lung and rat heart, respectively. AF-DX 116  Chemical Structure
  9. GC15510 AF-DX 384 M2/M4 selective antagonist AF-DX 384  Chemical Structure
  10. GC13340 AQ-RA 741 M2 antagonist,selective and high affinity AQ-RA 741  Chemical Structure
  11. GC11415 Arecaidine but-2-ynyl ester tosylate mAChR M2 agonist Arecaidine but-2-ynyl ester tosylate  Chemical Structure
  12. GC16504 Arecaidine propargyl ester tosylate muscarinic receptor agonist Arecaidine propargyl ester tosylate  Chemical Structure
  13. GC10621 Biperiden HCl Biperiden (KL 373) hydrochloride is a non-selective muscarinic receptor antagonist that competitively binds to M1 muscarinic receptors, thereby inhibiting acetylcholine and enhancing dopamine signaling in the central nervous system. Biperiden HCl  Chemical Structure
  14. GC15758 BQCA positive allosteric modulator of the M1 muscarinic acetylcholine receptor (mAChR) BQCA  Chemical Structure
  15. GC14215 Cevimeline A muscarinic receptor agonist Cevimeline  Chemical Structure
  16. GC17157 Cevimeline hydrochloride hemihydrate Cevimeline hydrochloride hemihydrate  Chemical Structure
  17. GC15772 Darifenacin HBr Darifenacin HBr (UK-88525 hydrobromide) is a selective M3 muscarinic receptor antagonist with pKi of 8.9. Darifenacin HBr  Chemical Structure
  18. GC10633 DAU 5884 hydrochloride muscarinic M3 receptor antagonist DAU 5884 hydrochloride  Chemical Structure
  19. GC16087 Fesoterodine Fumarate Muscarinic AChR receptor antagonist Fesoterodine Fumarate  Chemical Structure
  20. GC15845 Guvacoline (hydrobromide) full agonist of atrial and ileal muscarinic receptors Guvacoline (hydrobromide)  Chemical Structure
  21. GC12056 J 104129 fumarate M3 muscarinic receptor antagonist J 104129 fumarate  Chemical Structure
  22. GC16458 McN-A 343 muscarinic M1 receptor agonist McN-A 343  Chemical Structure
  23. GC14619 Milameline hydrochloride Muscarinic receptor agonist Milameline hydrochloride  Chemical Structure
  24. GC10378 N-Isopropylnoratropine used in the synthesis of ipratropium, a muscarinic antagonist N-Isopropylnoratropine  Chemical Structure
  25. GC10525 Nitrocaramiphen hydrochloride M1 muscarinic antagonist Nitrocaramiphen hydrochloride  Chemical Structure
  26. GC16463 Oxotremorine M Muscarinic receptor agonist Oxotremorine M  Chemical Structure
  27. GC16156 Oxotremorine sesquifumarate Muscarinic agonist Oxotremorine sesquifumarate  Chemical Structure
  28. GC17876 PD 102807 M4 muscarinic receptor antagonist PD 102807  Chemical Structure
  29. GC13403 Pirenzepine dihydrochloride M1 muscarinic receptor selective antagonist Pirenzepine dihydrochloride  Chemical Structure
  30. GC14508 PTAC oxalate muscarinic receptor ligand PTAC oxalate  Chemical Structure
  31. GC17182 Solifenacin succinate Muscarinic receptor antagonist Solifenacin succinate  Chemical Structure
  32. GC13174 Telenzepine dihydrochloride muscarinic M1 receptor antagonist Telenzepine dihydrochloride  Chemical Structure
  33. GC17954 Tolterodine tartrate Competitive muscarinic receptor antagonist Tolterodine tartrate  Chemical Structure
  34. GC12311 Trihexyphenidyl hydrochloride antiparkinsonian agent of the antimuscarinic class Trihexyphenidyl hydrochloride  Chemical Structure
  35. GC11831 Umeclidinium bromide A muscarinic acetylcholine receptor antagonist Umeclidinium bromide  Chemical Structure
  36. GC15990 VU 0238429 positive allosteric modulator of M5 receptors VU 0238429  Chemical Structure
  37. GC10464 VU 0255035 muscarinic M1 antagonist VU 0255035  Chemical Structure
  38. GC16655 VU 0357017 hydrochloride Positive allosteric modulator of muscarinic M1 receptors VU 0357017 hydrochloride  Chemical Structure
  39. GC17821 VU 0365114 positive allosteric modulator of M5 VU 0365114  Chemical Structure
  40. GC10725 VU 10010 allosteric potentiator of M4 acetylcholine receptors VU 10010  Chemical Structure
  41. GC13129 W-84 dibromide M2-receptor selective modulator W-84 dibromide  Chemical Structure
  42. GC18082 Zamifenacin fumarate M3 muscarinic receptor antagonist Zamifenacin fumarate  Chemical Structure

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