Search Site
  • 0
    My Cart

    Click Here to Find How Many Items You Have Added:)

    image loader

    Adding item(s) to cart......

Home >> Signaling Pathways >> Endocrinology and Hormones >> Opioid Receptor

Opioid Receptor

Opioid receptor is a group of G protein-coupled receptors with opioids as ligands.

Products for  Opioid Receptor

  1. Cat.No. Product Name Information
  2. GC60391 β-Casomorphin, bovine TFA β-Casomorphin, bovine TFA Chemical Structure
  3. GC61484 β-Casomorphin, human TFA β-Casomorphin, human TFA Chemical Structure
  4. GC38005 β-Endorphin, equine β-Endorphin, equine is an endogenous opioid peptide, which binds at high affinity to both μ/δ opioid receptors. β-Endorphin, equine Chemical Structure
  5. GC38030 β-Endorphin, equine (TFA) β-Endorphin, equine (TFA) Chemical Structure
  6. GC33736 β-Casomorphin, bovine (β-Casomorphin-7 (bovine)) β-Casomorphin, bovine (β-Casomorphin-7 (bovine)) (β-Casomorphin-7 (bovine) ) is a opioid peptide with an IC50 of 14 μM in an Opioid receptors binding assay. β-Casomorphin, bovine (β-Casomorphin-7 (bovine)) Chemical Structure
  7. GC33784 β-Casomorphin, human (Human β-casomorphin 7) is an opioid peptide, acts as an agonist of opioid receptor. β-Casomorphin, human (Human β-casomorphin 7) Chemical Structure
  8. GC31117 β-Endorphin, human β-Endorphin, human, a prominent endogenous peptide, existing in the hypophysis cerebri and hypothalamus, is an agonist of opioid receptor, with preferred affinity for μ-opioid receptor and δ-opioid receptor; β-Endorphin, human exhibits antinociception activity. β-Endorphin, human Chemical Structure
  9. GC15938 β-Funaltrexamine hydrochloride

    μ opioid receptor antagonist

     β-Funaltrexamine hydrochloride Chemical Structure
  10. GC64007 (±)-U-50488 hydrate hydrochloride (±)-U-50488 hydrate hydrochloride Chemical Structure
  11. GC15885 (±)-U-50488 hydrochloride

    κ-opioid receptor agonist, selective

     (±)-U-50488 hydrochloride Chemical Structure
  12. GC12688 (+)-U-50488 hydrochloride Selective κ-opioid agonist (+)-U-50488 hydrochloride Chemical Structure
  13. GC15944 (-)-U-50488 hydrochloride κ-opioid receptor agonist, selective (-)-U-50488 hydrochloride Chemical Structure
  14. GC70081 (1R,2R)-U-50488 hydrochloride

    (1R,2R)-U-50488 hydrochloride is the absolute configuration of (±)-U-50488 hydrochloride. (±)-U-50488 hydrochloride is a κ opioid receptor agonist.

     (1R,2R)-U-50488 hydrochloride Chemical Structure
  15. GC69798 (Rac)-SNC80

    (Rac)-SNC80 is the racemic form of SNC80. SNC80 (NIH 10815) is an effective and highly selective non-peptide delta-opioid receptor agonist with a Ki of 1.78 nM and IC50 of 2.73 nM. SNC80 has anti-nociceptive, anti-hyperalgesic, and antidepressant-like effects, and can be used in research on various types of headaches.

     (Rac)-SNC80 Chemical Structure
  16. GC66679 2,6-Dimethyl-L-tyrosine 2,6-Dimethyl-L-tyrosine (Dmt) is a tyrosine derivative that enhances receptor affinity, functional bioactivity and in vivo analgesia of opioid peptides. 2,6-Dimethyl-L-tyrosine Chemical Structure
  17. GC64147 Acetyl tetrapeptide-15 Acetyl tetrapeptide-15 is a synthetic peptide used in the cosmetics for sensitive skin. Acetyl tetrapeptide-15 Chemical Structure
  18. GC11829 ADL5859 HCl ADL5859 HCl (compound 20) is a selective and orally active δ opioid receptor (DOR) agonist with an Ki and an EC50 value of 0.84 and 20 nM, respectively. ADL5859 HCl Chemical Structure
  19. GP10109 Adrenorphin Adrenorphin Chemical Structure
  20. GC17623 Alvimopan A μ-opioid receptor antagonist Alvimopan Chemical Structure
  21. GC12619 Alvimopan dihydrate A μ-opioid receptor antagonist Alvimopan dihydrate Chemical Structure
  22. GC35311 Alvimopan monohydrate Alvimopan monohydrate (ADL 8-2698 monohydrate) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan monohydrate Chemical Structure
  23. GC12219 AR-M 1000390 hydrochloride Delta-opioid receptor agonist,low-internalizing AR-M 1000390 hydrochloride Chemical Structure
  24. GC31762 Asimadoline (EMD-61753) Asimadoline (EMD-61753) (EMD-61753) is an orally active, selective and peripherally active κ-opioid agonist with IC50s of 5.6 nM (guinea pig) and 1.2 nM (human recombinant). Asimadoline (EMD-61753) Chemical Structure
  25. GC61397 Asimadoline hydrochloride Asimadoline (EMD-61753) hydrochloride is an orally active, selective and peripherally active κ-opioid agonist with IC50s of 5.6 nM (guinea pig) and 1.2 nM (human recombinant). Asimadoline hydrochloride Chemical Structure
  26. GC11390 BAM 22P Potent endogenous agonist peptide for the newly identified sensory neuron specific receptor (SNSR); BAM 22P Chemical Structure
  27. GC15926 BAN ORL 24 A nociceptin receptor antagonist BAN ORL 24 Chemical Structure
  28. GC30639 Bevenopran (CB-5945) Bevenopran (CB-5945) is a peripheral μ-opioid receptor antagonist. Bevenopran (CB-5945) Chemical Structure
  29. GC38741 BPR1M97 BPR1M97 is a dual-acting mu opioid receptor (MOP) and nociceptin-orphanin FQ peptide (NOP) receptor agonist with Ki values of 1.8 and 4.2 nM, respectively. BPR1M97 Chemical Structure
  30. GC15313 BRL 52537 hydrochloride κ/μ opioid receptor agonist,potent and selective BRL 52537 hydrochloride Chemical Structure
  31. GC16521 BW 373U86 Non-peptide delta agonist,potent and selective BW 373U86 Chemical Structure
  32. GC67907 CCG258747 CCG258747 Chemical Structure
  33. GC35637 Cebranopadol An analgesic NOP and opioid receptor agonist Cebranopadol Chemical Structure
  34. GC35638 Cebranopadol ((1α,4α)stereoisomer) Cebranopadol ((1α,4α)stereoisomer) is a stereoisomer of cebranopadol. Cebranopadol ((1α,4α)stereoisomer) Chemical Structure
  35. GC19229 CERC-501 CERC-501 (CERC-501) is a potent and centrally-penetrant kappa opioid receptor antagonist with a Ki of 0.807 nM. CERC-501 Chemical Structure
  36. GC11535 CTAP Potent and selective μ opioid receptor antagonist CTAP Chemical Structure
  37. GC60730 CTAP TFA CTAP TFA is a potent, highly selective, and BBB penetrant μ opioid receptor antagonist, with an IC50 of 3.5 nM. CTAP TFA Chemical Structure
  38. GC16888 CTOP Potent and selective μ opioid receptor antagonist CTOP Chemical Structure
  39. GC60731 CTOP TFA CTOP TFA is a potent and highly selective μ-opioid receptor antagonist. CTOP TFA Chemical Structure
  40. GC13189 Cyprodime hydrochloride

    μ-opioid receptor antagonist

     Cyprodime hydrochloride Chemical Structure
  41. GC17677 DADLE δ-opioid receptor agonist DADLE Chemical Structure
  42. GC10803 DAMGO μ opioid receptor agonist DAMGO Chemical Structure
  43. GC35805 DAMGO (TFA) DAMGO (TFA) is a μ-opioid receptor (μ-OPR ) selective agonist with a Kd of 3.46 nM for native μ-OPR. DAMGO (TFA) Chemical Structure
  44. GC61954 Deltorphin 2 TFA Deltorphin 2 TFA is a selective peptide agonist for the δ opioid receptor. Deltorphin 2 TFA Chemical Structure
  45. GC12143 Deltorphin I δ-opioid receptor agonist Deltorphin I Chemical Structure
  46. GC31168 Dermorphin

    Dermorphin is a natural heptapeptide μ-opioid receptor (MOR) agonist found in amphibian skin.

     Dermorphin Chemical Structure
  47. GC34223 Dermorphin Analog Dermorphin Analog is an analog of Dermorphin. Dermorphin Analog Chemical Structure
  48. GC17553 DIPPA hydrochloride κ receptor antagonist DIPPA hydrochloride Chemical Structure
  49. GC10333 DPDPE Prototypical selective δ-opioid receptor agonist peptide DPDPE Chemical Structure
  50. GC63431 DPDPE TFA DPDPE TFA, an opioid peptide, is a selective δ-opioid receptor?(DOR) agonist?with anticonvulsant effects. DPDPE TFA Chemical Structure
  51. GC14774 DSLET δ Opioid receptor agonist DSLET Chemical Structure
  52. GC13546 Dynorphin A Endogenous kappa receptor agonist Dynorphin A Chemical Structure
  53. GC35917 Dynorphin A (1-10) TFA Dynorphin A (1-10) TFA Chemical Structure
  54. GA21407 Dynorphin A (1-8) Dynorphin A (1-8) is the predominant opioid peptide identified in placental tissue extracts. Dynorphin A (1-8) Chemical Structure
  55. GC35918 Dynorphin A 1-10 Dynorphin A 1-10 an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor. Dynorphin A 1-10 Chemical Structure
  56. GC15078 Dynorphin B endogenous agonist for the kappa opioid receptor Dynorphin B Chemical Structure
  57. GC35919 Dynorphin B (1-13) (TFA) Dynorphin B (1-13) TFA acts as an agonist on opioid κ-receptor. Dynorphin B (1-13) (TFA) Chemical Structure
  58. GC67956 Endomorphin 1 acetate Endomorphin 1 acetate Chemical Structure
  59. GC35986 Endomorphin 2 TFA Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. Endomorphin 2 TFA Chemical Structure
  60. GP10065 Endomorphin-1 Endomorphin-1 Chemical Structure
  61. GC10059 Endomorphin-2

    μ-opioid receptors agonist

     Endomorphin-2 Chemical Structure
  62. GC15874 FIT δ-opioid agonist, irreversible FIT Chemical Structure
  63. GC60857 Frakefamide TFA Frakefamide TFA is a potent analgesic that acts as a peripheral active μ-selective receptor agonist. Frakefamide TFA Chemical Structure
  64. GC30328 Gluten Exorphin C Gluten exorphin C is an opioid peptide derived from wheat gluten. Gluten Exorphin C Chemical Structure
  65. GC15843 GNTI dihydrochloride κ opioid receptor antagonist GNTI dihydrochloride Chemical Structure
  66. GC14739 GR 89696 fumarate κ-opioid agonist GR 89696 fumarate Chemical Structure
  67. GC68427 GSK1521498 free base GSK1521498 free base Chemical Structure
  68. GA22290 H-D-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr-NH₂ CTAP, an analog of CTOP, is a selective µ-opioid receptor antagonist. H-D-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr-NH₂ Chemical Structure
  69. GC43808 Hecogenin Acetate Hecogenin acetate is a steroid sapogenin and an acetylated form of hecogenin that has anthelmintic and antinociceptive properties. Hecogenin Acetate Chemical Structure
  70. GC32489 Hemorphin-7 Hemorphin-7 is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin. Hemorphin-7 Chemical Structure
  71. GC11639 ICI 154,129 Selective δ opioid antagonist ICI 154,129 Chemical Structure
  72. GC16193 ICI 174,864 Selective δ opioid antagonist ICI 174,864 Chemical Structure
  73. GC12534 ICI 199,441 hydrochloride ICI 199,441 hydrochloride is a potent and selective κ-opioid receptor agonist. ICI 199,441 hydrochloride Chemical Structure
  74. GC13097 ICI 204,448 hydrochloride κ opioid receptor agonist ICI 204,448 hydrochloride Chemical Structure
  75. GC17939 JDTic JDTic Chemical Structure
  76. GC17624 JDTic 2HCl JDTic 2HCl Chemical Structure
  77. GC11826 JTC-801 KOR-3 (NOP) receptor antagonist JTC-801 Chemical Structure
  78. GC31151 Kelatorphan Kelatorphan is a full inhibitor of enkephalin degrading enzymes. Kelatorphan Chemical Structure
  79. GC61003 Loperamide D6 hydrochloride Loperamide D6 hydrochloride (R-18553 D6 hydrochloride) is a deuterium labeled Loperamide hydrochloride. Loperamide D6 hydrochloride Chemical Structure
  80. GC36479 Loperamide hydrochloride Loperamide (hydrochloride) (R-18553 (hydrochloride)) is an opioid receptor agonist. Loperamide hydrochloride Chemical Structure
  81. GC36508 LY-2940094 LY-2940094 (BTRX-246040) is a potent, selective and orally available nociceptin receptor (NOP receptor) antagonist with high affinity (Ki=0.105 nM) and antagonist potency (Kb=0.166 nM). LY-2940094 Chemical Structure
  82. GC39193 LY2444296 LY2444296 is an orally bioavailable, high-affinity and selective short-acting kappa opioid receptor (KOPR) antagonist, with a Ki value of ?1 nM. LY2444296 Chemical Structure
  83. GC19500 LY2795050

    LY2795050 is a novel selective κ-opioid Receptor (KOR) antagonist

     LY2795050 Chemical Structure
  84. GC17874 Matrine An alkaloid with diverse biological activities Matrine Chemical Structure
  85. GC36562 MCOPPB triHydrochloride MCOPPB 3Hcl is a nociceptin receptor agonist with pKi of 10.07; weaker activity at other opioid receptors. MCOPPB triHydrochloride Chemical Structure
  86. GC11016 Meptazinol HCl Partial agonist at the μ1 opioid receptor Meptazinol HCl Chemical Structure
  87. GC63072 Methyl-6-alpha-Naltrexol Methyl-6-alpha-Naltrexol Chemical Structure
  88. GC16177 Methylnaltrexone Bromide Antagonist of peripherally acting μ-opioid Methylnaltrexone Bromide Chemical Structure
  89. GC14525 ML 190 κ opioid receptor (KOP) antagonist ML 190 Chemical Structure
  90. GC12663 N-Benzylnaltrindole hydrochloride δ2 opioid receptor antagonist N-Benzylnaltrindole hydrochloride Chemical Structure
  91. GC16553 N-Desmethylclozapine 5-HT2C serotonin receptor antagonist N-Desmethylclozapine Chemical Structure
  92. GC14979 N-MPPP Hydrochloride High affinity κ agonist N-MPPP Hydrochloride Chemical Structure
  93. GC36778 N-terminally acetylated Leu-enkephalin N-terminally acetylated Leu-enkephalin is the N-terminally acetylated form of Leu-enkephalin. N-terminally acetylated Leu-enkephalin Chemical Structure
  94. GC46182 Naldemedine A peripherally acting opioid receptor antagonist Naldemedine Chemical Structure
  95. GC44312 Nalfurafine

    Nalfurafine is a κ-opioid receptor (KOR) agonist (EC50 = 0.05 nM for human receptors expressed in CHO cell membranes).

     Nalfurafine Chemical Structure
  96. GC30932 Naloxegol (NKTR-118) Naloxegol (NKTR-118) Chemical Structure
  97. GC30881 Naloxegol oxalate (NKTR-118 oxalate)

    A peripherally acting antagonist of the µ-opioid receptor

     Naloxegol oxalate (NKTR-118 oxalate) Chemical Structure
  98. GC16588 Naloxonazine dihydrochloride Naloxonazine dihydrochloride is a specific μ-opioid receptor antagonist with an IC50 of 5.4 nM. Naloxonazine dihydrochloride Chemical Structure
  99. GC11807 Naloxone (hydrochloride) An opioid inverse agonist drug Naloxone (hydrochloride) Chemical Structure
  100. GC63686 Naloxone methiodide Naloxone methiodide Chemical Structure
  101. GC16206 Naltrexone Opioid receptor antagonist Naltrexone Chemical Structure

Items 1 to 100 of 136 total

per page
  1. 1
  2. 2

Set Descending Direction