Thyroid hormone Receptor
Thyroid hormone receptor is a nuclear hormone receptor that activates or represses transcriptioin. It has effects on heart rate, lipid and lipoprotein metabolism.
Products for Thyroid hormone Receptor
- Cat.No. Product Name Information
- GA20164 (D-Trp¹²,Tyr³⁴)-pTH (7-34) amide (bovine) (D-Trp¹²,Tyr³⁴)-pTH (7-34) amide (bovine) is a potent and competitive antagonist of parathyroid hormone (PTH), with a Ki of 69 nM in bovine renal cortical membrane.
- GC52185 (R,S)-Anatabine-d4
- GC62761 1α-Hydroxy-3-epi-vitamin D3 1α-Hydroxy-3-epi-vitamin D3, a natural metabolite of 1alpha,25-dihydroxyvitamin D3, is a potent suppressor of parathyroid hormone (PTH) secretion.
- GC10384 3,3',5'-Triiodo-L-thyronine 3,3',5'-Triiodo-L-thyronine is a thyroid hormone generated by deiodination of the prohormone thyroxine.
- GC48395 3,3',5-Triiodo-L-thyronine (sodium salt hydrate) 3,3',5-Triiodo-L-thyronine (sodium salt hydrate) is an active form of thyroid hormone.
- GC49427 3,5-Diiodo-L-thyronine 3,5-Diiodo-L-thyronine is an endogenous metabolite.
- GC18205 3,5-Diiodothyroacetic Acid 3,5-Diiodothyroacetic acid (diac) is the acetic acid variant of thyroxine.
- GC18696 3,5-Diiodothyropropionic Acid 3,5-Diiodothyropropionic acid (DITPA) is an inotropic thyroid hormone analogue of L-thyroxine that binds to the thyroid hormone receptors TRα and TRβ (Kas = 2.4 and 4.06 x 107 M-1, respectively, for human recombinant receptors).
- GC52129 3-Amino-5-hydroxybenzoic Acid
- GC49180 3-epi-25-hydroxy Vitamin D3 The C-3 epimer of 25-hydroxy vitamin D3
- GC42294 3-Iodothyronamine (hydrochloride) 3-Iodothyronamine is derived from the deiodination and decarboxylation of endogenous thyroxine.
- GC46075 5,6-dimethyl-2-Thiouracil A heterocyclic building block
- GC46768 Abaloparatide (acetate) A synthetic derivative of PTHrP and an agonist of PTHR1
- GC38581 Abaloparatide TFA Abaloparatide TFA (BA 058 TFA) is a parathyroid hormone receptor 1 (PTHR1) analogue selected to be a potent and selective activator of the PTHR1 signaling pathway.
- GC42815 Ansatrienin A Ansatrienin A is an ansamycin antibiotic and antifungal agent first isolated from S.
- GA20967 Boc-D-His-OH An amino acid building block
- GC52351 Citrullinated α-Enolase (R8 + R14) (1-19)-biotin Peptide A biotinylated and citrullinated α-enolase peptide
- GC65587 CO23 CO23 is a selective thyroid hormone receptor (TR) α agonist and used for growth and development regulation.
- GC50178 DPC AJ1951 Potent parathyroid hormone (PTH) receptor agonist
- GC43567 DPC-AJ1951 (trifluoroacetate salt) DPC-AJ1951 is a peptide agonist of the parathyroid hormone (PTH)/PTH-related peptide receptor (PPR; EC50 = 0.15 nM in HEK293 cells expressing human PPR).
- GC64301 DS08210767 DS08210767 is a highly potent, orally bioavailable PTHR1 antagonist with IC50 of 90 nM.
- GC33764 Eprotirome (KB2115) Eprotirome (KB2115) (KB2115) is a liver-selective thyroid hormone receptor (TR) agonist.
- GC62992 Glutaurine Glutaurine containing glutamine and taurine residues is an orally active hormone of the parathyroid.
- GC31616 KAT681 (T0681) KAT681 (T0681) is a liver-selective thyromimetic.
- GC48432 KB-130015 An antiarrhythmic agent
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GC11268
L-Thyroxine
Iodine containing hormone
- GC61010 L-Thyroxine sodium L-Thyroxine sodium (Levothyroxine sodium) is a synthetic hormone for the research of hypothyroidism.
- GC36487 L-Thyroxine sodium salt pentahydrate L-Thyroxine sodium salt pentahydrate (Levothyroxine; T4) is a synthetic hormone for the research of hypothyroidism.
- GC44088 L-Thyroxine-13C9,15N L-Thyroxine-13C9,15N is intended for use as an internal standard for the quantification of L-thyroxine by GC- or LC-MS.
- GC52021 L-Thyroxine-N-methylamide A potential impurity found in commercial preparations of L-thyroxine
- GC48937 L-Tyrosine-13C9,15N An internal standard for the quantification of L-tyrosine
- GC36465 Liothyronine An thyroid hormone which binds to TRβ1, and activates its activity
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GC12409
Liothyronine Sodium
Thyroid hormone (T3) analog
- GC18243 MGL-3196 MGL-3196 (MGL-3196) is a highly selective thyroid hormone receptor β (THR-β) agonist with an EC50 value of 0.21 μM.
- GC49802 N-Acetyl-L-thyroxine A thyroid hormone derivative
- GC49399 N-Desbutyl Dronedarone (hydrochloride) Debutyldronedarone (SR35021) hydrochloride, the main metabolite of Dronedarone, is a selective thyroid hormone receptor α1 (TRα1) inhibitor.
- GC63595 NH-3 NH-3 is an orally active, reversible thyroid hormone receptor (THR) antagonist with an IC50 of 55 nM.
- GC68337 Parathyroid hormone (1-34) (rat) acetate
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GC69654
Parathyroid Hormone (1-34), human, biotinylated
Parathyroid Hormone (1-34), human, biotinylated is a probe for the parathyroid hormone receptor. It can be used to analyze the interaction between parathyroid hormone and its receptor in live cells, and purify the hormone-receptor complex through affinity chromatography.
- GC32415 PCO371 PCO371 is an orally active full agonist of parathyroid hormone receptor 1 (PTHR1), with no effect on PTH type 2 receptor.
- GC47982 Propylthiouracil-d5 An internal standard for the quantification of propylthiouracil
- GC30588 Protirelin (Synthetic thyrotropin-releasing factor) Protirelin (Synthetic thyrotropin-releasing factor) is a highly conserved neuropeptide that exerts the hormonal control of thyroid-stimulating hormone (TSH) levels as well as neuromodulatory functions.
- GC33845 Protirelin Acetate (TRF Acetate) Protirelin Acetate is a highly conserved neuropeptide that exerts the hormonal control of thyroid-stimulating hormone (TSH) levels as well as neuromodulatory functions.
- GA23395 pTH (1-34) (rat) pTH (1-34) (rat) is a parathyroid hormone.
- GC49679 Sauvagine (trifluoroacetate salt) A neuropeptide hormone
- GC12903 Sobetirome An agonist of TRβ
- GC44914 Somatostatin-14 (acetate) Somatostatin-14 is a natural cyclic peptide hormone derived from the preprohormone, somatostatin.
- GC34822 T3-ATA S-isomer T3-ATA S-isomer is the S-isomer of T3-ATA, which is the active form of the thyroid hormone.
- GC34824 T4-ATA S-isomer
- GC17983 Taltirelin novel orally active TRH analogue
- GC37732 Taltirelin acetate Taltirelin acetate (TA-0910 acetate) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release).
- GC48358 Thymulin (acetate hydrate) A peptide hormone
- GC10413 Thyroid Hormone Receptor Antagonist (1-850) Thyroid hormone receptor antagonist
- GC31328 Thyroxine sulfate (T4 Sulfate) Thyroxine sulfate (T4 Sulfate) is a thyroid hormone metabolite.
- GC15001 Tiratricol thyroid hormone analogue
- GC31402 TR antagonist 1 TR antagonist 1 is a high-affinity thyroid hormone receptor (TR) antagonist with IC50s of 36 and 22 nM for TRα and TRβ, respectively.