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Adenosine Receptor

Adenosine receptor (P1 receptors) is a class of purinergic receptors, G protein-coupled receptors with adenosine as endogenous ligand.

Products for  Adenosine Receptor

  1. Cat.No. Product Name Information
  2. GC17413 (±)-5'-Chloro-5'-deoxy-ENBA adenosine A1 receptor agonist, selective and high-affinity (±)-5'-Chloro-5'-deoxy-ENBA  Chemical Structure
  3. GC10600 1,3-Dipropyl-8-phenylxanthine

    A1 adenosine antagonist

    1,3-Dipropyl-8-phenylxanthine  Chemical Structure
  4. GC11112 2'-MeCCPA A1 adenosine receptor agonist 2'-MeCCPA  Chemical Structure
  5. GC10116 2-chloro-3-Deazaadenosine adenosine receptors agonist 2-chloro-3-Deazaadenosine  Chemical Structure
  6. GC11665 2-Chloro-N6-cyclopentyladenosine adenosine A1 receptor agonist, potent and selective 2-Chloro-N6-cyclopentyladenosine  Chemical Structure
  7. GC15111 2-Chloroadenosine adenosine receptor agonist 2-Chloroadenosine  Chemical Structure
  8. GC17503 2-Cl-IB-MECA 2-Cl-IB-MECA (CF-102) is a selective A3 adenosine receptor (A3AR) agonist (Ki=0.33 nM). 2-Cl-IB-MECA displays 2500- and 1400-fold selectivity over A1 and A2A receptors respectively. 2-Cl-IB-MECA  Chemical Structure
  9. GC11002 5'-(N-Cyclopropyl)carboxamidoadenosine adenosine A2 receptor agonist 5'-(N-Cyclopropyl)carboxamidoadenosine  Chemical Structure
  10. GC11199 8-(3-Chlorostyryl)caffeine 8-(3-Chlorostyryl)caffeine is a selective adenosine A2A receptor antagonist. 8-(3-Chlorostyryl)caffeine  Chemical Structure
  11. GC13274 8-Aminoadenine

    Adenine receptor agonist

    8-Aminoadenine  Chemical Structure
  12. GC50354 8-Cyclopentyl-1,3-dimethylxanthine High affinity adenosine A1 receptor antagonist 8-Cyclopentyl-1,3-dimethylxanthine  Chemical Structure
  13. GC30918 A2A receptor antagonist 1 A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Ki values of 4 and 264 nM, respectively. A2A receptor antagonist 1  Chemical Structure
  14. GC30987 A2AR-agonist-1 An agonist of adenosine A2A receptor and inhibitor of ENT1 A2AR-agonist-1  Chemical Structure
  15. GC38104 A2aR/A2bR antagonist-1 A2aR/A2bR antagonist-1 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. A2aR/A2bR antagonist-1  Chemical Structure
  16. GC31974 A2B receptor antagonist 1 A2B receptor antagonist 1 is a potent A2B adenosine receptor antagonist extracted from patent WO 2009157938 A1 EXAMPLE 9B. A2B receptor antagonist 1  Chemical Structure
  17. GC62820 A2B receptor antagonist 2 A2B receptor antagonist 2 (compound 18) is an adenosine receptor A2B antagonist, with Ki values of 2.30 μM, 6.8 μM and 3.44 μM for rA1, rA2A and hA2B, respectively. A2B receptor antagonist 2  Chemical Structure
  18. GC30993 AB-MECA AB-MECA is a high affinity A3 adenosine receptor agonist, has high affinity for recombinant A1 and A3 receptors. AB-MECA  Chemical Structure
  19. GC34143 Acefylline (Theophyllineacetic acid) Acefylline (Theophyllineacetic acid) (Theophyllineacetic acid), a xanthine derivative, is an adenosine receptor antagonist. Acefylline (Theophyllineacetic acid) is a peptidylarginine deiminase (PAD) activator. Acefylline (Theophyllineacetic acid) is also a bronchodilator, which inhibits rat lung cAMP phosphodiesterase isoenzymes. Acefylline (Theophyllineacetic acid)  Chemical Structure
  20. GC19630 Adenosine 2′-monophosphate Adenosine 2′-monophosphate (2'-AMP) is converted by extracellular 2',3'-CAMP. Adenosine 2′-monophosphate  Chemical Structure
  21. GC35248 Adenosine 5'-monophosphate monohydrate Adenosine 5'-monophosphate monohydrate is an adenosine A1 receptor agonist. Adenosine 5'-monophosphate monohydrate  Chemical Structure
  22. GC38733 Adenosine A1 receptor activator T62 Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor. Adenosine A1 receptor activator T62  Chemical Structure
  23. GC38884 Adenosine amine congener An adenosine A1 receptor agonist Adenosine amine congener  Chemical Structure
  24. GC35249 Adenosine antagonist-1 Adenosine antagonist-1 is an adenosine A3 receptor (AA3R) antagonist. Adenosine antagonist-1  Chemical Structure
  25. GC65901 Adenosine receptor antagonist 2 Adenosine receptor antagonist 2 is an orally active A2a/A2b adenosine receptor antagonist with IC50s of 1 nM and 3 nM, respectively. Adenosine receptor antagonist 2 has anti-tumor activity. Adenosine receptor antagonist 2  Chemical Structure
  26. GC66007 Adenosine receptor antagonist 3 Adenosine receptor antagonist 3 is a potent antagonist of adenosine receptor. Adenosine receptor antagonist 3 has the potential for the research of cancer disease (extracted from patent WO2019233994A1, compound 1). Adenosine receptor antagonist 3  Chemical Structure
  27. GC25051 Alloxazine Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor. Alloxazine  Chemical Structure
  28. GC16159 ANR 94 Adenosine A2A-R antagonist ANR 94  Chemical Structure
  29. GC33702 APNEA (N6-[2-(4-Aminophenyl)ethyl]adenosine) APNEA (N6-[2-(4-Aminophenyl)ethyl]adenosine) (N6-[2-(4-Aminophenyl)ethyl]adenosine) is a potent, non-selective A3 adenosine receptor agonist. APNEA (N6-[2-(4-Aminophenyl)ethyl]adenosine)  Chemical Structure
  30. GC38887 Arotinolol Arotinolol is a nonselective α/β-adrenergic receptor blocker and a vasodilating β-blocker. Arotinolol  Chemical Structure
  31. GC19049 AZD4635 AZD4635 (HTL1071) is a potent, selective and orally active adenosine A2A receptor (A2AR) antagonist. AZD4635 binds to human A2AR with a Ki of 1.7 nM and shows >30-fold selectivity over other adenosine receptors. AZD4635  Chemical Structure
  32. GC18114 BAY 60-6583 Potent A2B receptor agonist BAY 60-6583  Chemical Structure
  33. GC19502 BAY-545

    BAY-545 is a potent and selective A2B adenosine receptor antagonist

    BAY-545   Chemical Structure
  34. GC64647 Binodenoson Binodenoson (MRE-0470) is a potent and selective A2A adenosine receptor agonist (KD=270 nM). Binodenoson  Chemical Structure
  35. GC14935 Capadenoson A partial adenosine receptor agonist Capadenoson  Chemical Structure
  36. GC14674 CGH 2466 dihydrochloride adenosine receptor antagonist CGH 2466 dihydrochloride  Chemical Structure
  37. GC10070 CGS 15943 adenosine receptor antagonist CGS 15943  Chemical Structure
  38. GC10172 CGS 21680 A selective agonist of the adenosine A2A receptor CGS 21680  Chemical Structure
  39. GC11978 CGS 21680 HCl CGS 21680 HCl is a selective adenosine A2A receptor agonist with a Ki of 27 nM. CGS 21680 HCl  Chemical Structure
  40. GC32734 CPI-444 (V81444) CPI-444 (V81444) (V81444) is a potent, orally active and selective adenosine A2A receptor (A2AR) antagonist, which induces antitumor responses. CPI-444 (V81444)  Chemical Structure
  41. GC14706 CV 1808 Adenosine A2 receptor agonist CV 1808  Chemical Structure
  42. GC13444 Doxofylline PDE inhibitor Doxofylline  Chemical Structure
  43. GC16099 DPCPX A1 adenosine receptor antagonist DPCPX  Chemical Structure
  44. GC13652 Dyphylline An adenosine receptor antagonist and phosphodiesterase inhibitor Dyphylline  Chemical Structure
  45. GC32675 GP531 GP531 is a potent, second-generation adenosine regulating agent, is pharmacologically silent under basal conditions but increases localized endogenous adenosine during ischemia. GP531  Chemical Structure
  46. GC12315 GR 79236 adenosine A1 receptor agonist GR 79236  Chemical Structure
  47. GC38789 GS-6201 An adenosine A2B receptor antagonist GS-6201  Chemical Structure
  48. GC11493 HEMADO adenosine A3 receptor agonist HEMADO  Chemical Structure
  49. GC19197 IB-MECA IB-MECA (IB-MECA) is a first-in-class, orally active and selective A3 adenosine receptor (A3AR) agonist. IB-MECA  Chemical Structure
  50. GC63022 Inupadenant Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity. Inupadenant  Chemical Structure
  51. GC50679 ISAM 140 ISAM 140 (22b) is a potent and highly selective A2B adenosine receptor antagonist with a Ki of 3.49 nM. ISAM 140  Chemical Structure
  52. GC11590 Istradefylline(KW-6002) Istradefylline(KW-6002) is a very potent, selective and orally active adenosine A2A receptor antagonist with Ki of 2.2 nM in experimental models of Parkinson's disease. Istradefylline(KW-6002)  Chemical Structure
  53. GC31217 KF21213 KF21213 is a highly selective ligand for mapping CNS adenosine A2A receptors. KF21213  Chemical Structure
  54. GC31264 KFM19 KFM19 is a potent, selective Adenosine receptor (A1-receptor) antagonist, with an IC50 of 50 nM. KFM19  Chemical Structure
  55. GC50571 KI-7 Positive allosteric modulator of A2B receptors KI-7  Chemical Structure
  56. GC12417 KW 3902 KW 3902 (KW-3902) is a potent, selective adenosine A1 receptor antagonist that is under development for the treatment of patients with acute congestive heart failure and renal impairment. KW 3902  Chemical Structure
  57. GC33871 LAS101057 A potent adenosine A2B receptor antagonist LAS101057  Chemical Structure
  58. GC17499 Lu AA 47070 adenosine A2A receptor antagonist Lu AA 47070  Chemical Structure
  59. GC11851 LUF 5834 A2A and A2B adenosine receptor partial agonist LUF 5834  Chemical Structure
  60. GC15986 LUF6000 A positive allosteric modulator of adenosine A3 receptors LUF6000  Chemical Structure
  61. GC61872 LUF6096 LUF6096, a potent allosteric enhancer of the adenosine A3 receptor, is able to allosterically enhance agonist binding. LUF6096  Chemical Structure
  62. GC63304 MIPS521 MIPS521 is a positive allosteric modulator of adenosine A1 receptor (A1AR). MIPS521  Chemical Structure
  63. GC12584 MRE 3008F20 adenosine A3 receptor antagonist MRE 3008F20  Chemical Structure
  64. GC11579 MRS 1220 human A3 adenosine receptor antagonist MRS 1220  Chemical Structure
  65. GC10202 MRS 1334 antagonist for the human adenosine A3 receptor MRS 1334  Chemical Structure
  66. GC10320 MRS 1706 adenosine A2B receptor inverse agonist MRS 1706  Chemical Structure
  67. GC13807 MRS 1754

    adenosine A2B receptor antagonist

    MRS 1754  Chemical Structure
  68. GC13021 MRS 3777 hemioxalate adenosine A3 receptor antagonist MRS 3777 hemioxalate  Chemical Structure
  69. GC50162 MRS 5698 High affinity and selective A3 agonist MRS 5698  Chemical Structure
  70. GC38112 MRS-1191 MRS-1191 is a potent and selective A3 adenosine receptor antagonist with a KB value of 92 nM, a Ki value of 31.4 nM for human A3 receptor and an IC50 of 120 nM for CHO cells. MRS-1191  Chemical Structure
  71. GC33652 MRS1177 MRS1177 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 0.3 nM. MRS1177  Chemical Structure
  72. GC33654 MRS1186 MRS1186 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 7.66 nM. MRS1186  Chemical Structure
  73. GC14078 MRS1523 adenosine A3 receptor antagonist MRS1523  Chemical Structure
  74. GC30739 N-0861 racemate N-0861 racemate is the racemate of N-0861. N-0861 racemate  Chemical Structure
  75. GC36676 N-[(4-Aminophenyl)methyl]adenosine N-[(4-Aminophenyl)methyl]adenosine is a adenosine receptor inhibitor, with Ki of 29 nM for Rat ecto-5′-Nucleotidase. N-[(4-Aminophenyl)methyl]adenosine  Chemical Structure
  76. GC36679 N6-(2-Phenylethyl)adenosine N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine), an adenosine derivative, is a potent adenosine receptors (AR) agonist with Ki values of 11.8 nM, 30.1 nM, 0.63 nM for rat A1AR, human A1AR and hA3AR, respectively. N6-(2-Phenylethyl)adenosine  Chemical Structure
  77. GC33667 N6-Cyclohexyladenosine (CHA) N6-Cyclohexyladenosine (CHA) is a selective A1 receptor agonist (EC50 = 8.2 nM). N6-Cyclohexyladenosine (CHA)  Chemical Structure
  78. GC14369 N6-Cyclopentyladenosine

    adenosine A1 receptor agonist

    N6-Cyclopentyladenosine  Chemical Structure
  79. GC34921 N6-Ethyladenosine An adenosine A1 and A3 receptor agonist N6-Ethyladenosine  Chemical Structure
  80. GC15304 NECA NECA (NECA) is a nonselective adenosine receptor agonist. NECA  Chemical Structure
  81. GC16141 Nicergoline vasodilator Nicergoline  Chemical Structure
  82. GN10652 Norisoboldine Norisoboldine  Chemical Structure
  83. GC30916 PD 117519 (CI947) PD 117519 (CI947) (CI947) is an A2A adenosine agonist which has shown oral antihypertensive activity in pharmacological animal models. PD 117519 (CI947)  Chemical Structure
  84. GC10103 PD 81723 Allosteric potentiator at the adenosine A1 receptor PD 81723  Chemical Structure
  85. GC12200 Pentostatin A purine antimetabolite and an ADA inhibitor Pentostatin  Chemical Structure
  86. GC11591 Preladenant An adenosine A2A receptor antagonist Preladenant  Chemical Structure
  87. GC10475 Proxyphylline A1 adenosine receptor antagonist Proxyphylline  Chemical Structure
  88. GC14863 PSB 0777 ammonium salt adenosine A2A receptor full agonist PSB 0777 ammonium salt  Chemical Structure
  89. GC17844 PSB 0788 adenosine A2B receptor antagonist PSB 0788  Chemical Structure
  90. GC12542 PSB 10 hydrochloride human adenosine A3 receptor antagonist PSB 10 hydrochloride  Chemical Structure
  91. GC14702 PSB 11 hydrochloride human adenosine A3 receptor antagonist PSB 11 hydrochloride  Chemical Structure
  92. GC17756 PSB 1115

    human A2B adenosine receptor antagonist

    PSB 1115  Chemical Structure
  93. GC10584 PSB 36

    A1 adenosine receptor antagonist

    PSB 36  Chemical Structure
  94. GC13153 PSB 603 Adenosine A2B receptor antagonist PSB 603  Chemical Structure
  95. GC13082 Regadenoson Highly selective and low affinity A2A adenosine agonist Regadenoson  Chemical Structure
  96. GC12328 SCH 442416 adenosine A2A receptor antagonist SCH 442416  Chemical Structure
  97. GC14565 SCH 58261

    A2A adenosine receptor competitive antagonist

    SCH 58261  Chemical Structure
  98. GC31246 Sch412348

    Sch412348 is a potent competitive antagonist of the human adenosine A2A receptor (Ki=0.6 nM) and has >1000-fold selectivity over all other adenosine receptors.

    Sch412348  Chemical Structure
  99. GC14198 SDZ WAG 994 A1 adenosine receptor agonist SDZ WAG 994  Chemical Structure
  100. GC69893 Sipagladenant

    Sipagladenant (Compound I) is an orally active adenosine receptor A2A inverse agonist that can be used for the study of frontal lobe dysfunction.

    Sipagladenant  Chemical Structure
  101. GC14290 SLV 320 SLV 320 (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. SLV 320  Chemical Structure

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