Home >> Signaling Pathways >> GPCR/G protein >> CaSR

CaSR

CASR (calcium sensing receptor) is a G-protein couple receptor which regulates the calcium homeostasis and involved in proliferation, differentiation and other hormonal secretion.

Products for  CaSR

  1. Cat.No. Product Name Information
  2. GC64905 (Rac)-Upacicalcet (Rac)-Upacicalcet is the racemate of Upacicalcet. (Rac)-Upacicalcet  Chemical Structure
  3. GC50365 AC 265347 Biased allosteric modulator of calcium-sensing receptor (CaSR) AC 265347  Chemical Structure
  4. GC17244 Calcium-Sensing Receptor Antagonists I Calcium-Sensing Receptor Antagonists I  Chemical Structure
  5. GC17697 Calhex 231 hydrochloride

    negative allosteric modulator of Ca2+-sensing receptor (CaSR)

    Calhex 231 hydrochloride  Chemical Structure
  6. GC12620 Calindol (hydrochloride) activator of the calcium-sensing receptor (CaSR) Calindol (hydrochloride)  Chemical Structure
  7. GC13518 Cinacalcet Cinacalcet  Chemical Structure
  8. GC16708 Cinacalcet HCl Cinacalcet HCl (AMG-073 hydrochloride) is an orally active, allosteric agonist of Ca receptor (CaR), used for cardiovascular disease treatment. Cinacalcet HCl  Chemical Structure
  9. GC63745 Cinacalcet-D3 Cinacalcet-D3  Chemical Structure
  10. GC38148 Etelcalcetide Etelcalcetide (AMG 416) is a synthetic peptide as an activator of the calcium sensing receptor (CaSR). Etelcalcetide  Chemical Structure
  11. GC38147 Etelcalcetide hydrochloride A peptide agonist of CaSR Etelcalcetide hydrochloride  Chemical Structure
  12. GC30389 Evocalcet (KHK7580) Evocalcet (KHK7580) has an activating effect on calcium sensing receptor (CaSR) extracted from patent WO 2017061621 A1, compound A. Evocalcet (KHK7580)  Chemical Structure
  13. GN10419 Ligustroflavone Ligustroflavone  Chemical Structure
  14. GC16943 NPS-2143

    NPS-2143?is a calcification drug that acts as an antagonist of the calcium-sensing receptor (CaSR) and consequently stimulates the release of parathyroid hormone.

    NPS-2143  Chemical Structure
  15. GC12240 NPS-2143 hydrochloride An orally-active CaSR antagonist NPS-2143 hydrochloride  Chemical Structure
  16. GC17700 R 568 hydrochloride R 568 hydrochloride (R 568 Hydrochloride), an orally active calcimimetic compound, allosterically and positively modulates the calcium-sensing receptor (CaSR). R 568 hydrochloride  Chemical Structure
  17. GC30095 SB-423562 SB-423562 is a short-acting calcium-sensing receptor (CaR) antagonist. SB-423562  Chemical Structure
  18. GC12442 Strontium chloride Calcium sensing receptor (CaSR) agonist Strontium chloride  Chemical Structure
  19. GC11819 Strontium Ranelate Calcium Channel activator Strontium Ranelate  Chemical Structure
  20. GC64923 Upacicalcet sodium Upacicalcet sodium is an intravenous calcimimetic agent. Upacicalcet sodium  Chemical Structure

19 Item(s)

per page

Set Descending Direction