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GHSR

GHSR (growth hormone secretagogue receptor) is a G protein-coupled receptor that binds ghrelin and plays a role in energy homeostasis and regulation of body weight.

Products for  GHSR

  1. Cat.No. Product Name Information
  2. GC67681 (αR,8aS)-GSK1614343 (αR,8aS)-GSK1614343  Chemical Structure
  3. GC35282 Alexamorelin Met 1 Alexamorelin Met 1  Chemical Structure
  4. GC13253 Anamorelin A small molecule agonist of GHS-R1a Anamorelin  Chemical Structure
  5. GC35337 Anamorelin Fumarate Anamorelin Fumarate is a novel ghrelin receptor agonist with EC50 value of 0.74 nM in the FLIPR assay. Anamorelin Fumarate  Chemical Structure
  6. GC35338 Anamorelin hydrochloride Anamorelin (RC-1291) hydrochloride is a potent ghrelin receptor agonist with EC50 value of 0.74 nM in the FLIPR assay. Anamorelin hydrochloride  Chemical Structure
  7. GC31430 AZP-531 AZP-531 is an analogue of unacylated ghrelin designed to improve glycaemic control and reduce weight. AZP-531  Chemical Structure
  8. GC19087 Capromorelin Tartrate Capromorelin Tartrate is an orally active, potent growth hormone secretagogue receptor (GHSR) agonist, with Ki of 7 nM for hGHS-R1a. Capromorelin Tartrate  Chemical Structure
  9. GC30388 Human growth hormone-releasing factor (Growth Hormone Releasing Factor human) Human growth hormone-releasing factor (Growth Hormone Releasing Factor human) (Growth Hormone Releasing Factor human) is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) on cells in the anterior pituitary. Human growth hormone-releasing factor (Growth Hormone Releasing Factor human)  Chemical Structure
  10. GC61519 Human growth hormone-releasing factor TFA Human growth hormone-releasing factor TFA (Growth Hormone Releasing Factor human TFA) is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) on cells in the anterior pituitary. Human growth hormone-releasing factor TFA  Chemical Structure
  11. GC10287 Ibutamoren Mesylate

    A growth hormone secretagogue and ghrelin receptor agonist

    Ibutamoren Mesylate  Chemical Structure
  12. GC31274 JMV 2959 JMV 2959 is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32 nM. JMV 2959  Chemical Structure
  13. GC34207 JMV 2959 hydrochloride JMV 2959 hydrochloride is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32±3 nM in LLC-PK1 cells. JMV 2959 hydrochloride  Chemical Structure
  14. GC60971 L-692429 L-692429 (MK-0751) is a benzolactam derivative and a nonpeptidyl growth hormone secretagogue (GHS) agonist. L-692429  Chemical Structure
  15. GC34095 ONC212 A GPR132 agonist ONC212  Chemical Structure
  16. GC31478 PF-5190457 PF-5190457 (PF-05190457) is a potent and selective ghrelin receptor inverse agonist with a pKi of 8.36. PF-5190457  Chemical Structure
  17. GC63727 Relamorelin TFA Relamorelin (RM-131) TFA, a pentapeptide ghrelin analog, is a selective ghrelin/growth hormone secretagogue receptor (GHSR) agonist with a Ki of 0.42 nM for GHS-1a receptor. Relamorelin TFA  Chemical Structure
  18. GC19349 TC-G-1008 TC-G-1008 (GPR39-C3) is a potent and orally available GPR39 agonist with EC50 values of 0.4 and 0.8 nM for rat and human receptors respectively. TC-G-1008  Chemical Structure
  19. GC31074 TM-N1324 TM-N1324 is an agonist of G-Protein-Coupled Receptor 39 (GPR39) with EC50s of 9 nM/5 nM in the presence of Zn2+, and 280 nM/180 nM in the absence of Zn2+ for human/murine GPR39. TM-N1324  Chemical Structure

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