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P2Y Receptor

P2Y Receptor is a family of purinergic G protein-coupled receptors, stimulated by nucleotides.

Products for  P2Y Receptor

  1. Cat.No. Product Name Information
  2. GC41668 (±)-Clopidogrel (hydrochloride) Clopidogrel is an antithrombic compound whose active metabolite is a selective, irreversible antagonist of the platelet purinergic P2Y12 receptor (IC50 = 100 nM). (±)-Clopidogrel (hydrochloride)  Chemical Structure
  3. GC64027 2-Methylthio-AMP 2-Methylthio-AMP (2-MeSAMP) is a selective and direct P2Y12 antagonist. 2-Methylthio-AMP  Chemical Structure
  4. GC62783 2-Methylthio-AMP diTEA 2-Methylthio-AMP (2-MeSAMP) diTEA is a selective and direct P2Y12 antagonist. 2-Methylthio-AMP diTEA  Chemical Structure
  5. GC60016 2-Methylthioadenosine diphosphate trisodium An agonist of P2Y receptors 2-Methylthioadenosine diphosphate trisodium  Chemical Structure
  6. GC14753 2-ThioUTP tetrasodium salt P2Y2 agonist 2-ThioUTP tetrasodium salt  Chemical Structure
  7. GC13588 5-OMe-UDP trisodium salt

    Potent P2Y6 agonist

    5-OMe-UDP trisodium salt  Chemical Structure
  8. GC50081 AR-C 118925XX Selective and competitive P2Y2 antagonist AR-C 118925XX  Chemical Structure
  9. GC12914 AR-C 66096 tetrasodium salt P2Y12 antagonist,potent and selective AR-C 66096 tetrasodium salt  Chemical Structure
  10. GC14956 AZD1283 Potent P2Y12 antagonist AZD1283  Chemical Structure
  11. GC19081 BPTU BPTU is a novel P2Y1 allosteric antagonist. BPTU  Chemical Structure
  12. GC43137 Cangrelor (sodium salt) Cangrelor (sodium salt), an adenosine triphosphate analogue, is a reversible and selective platelet P2Y12 antagonist, with prompt and potent antiplatelet effects. Cangrelor (sodium salt)  Chemical Structure
  13. GC35710 Clopidogrel Clopidogrel is an orally active platelet inhibitor that targets P2Y12 receptor. Clopidogrel  Chemical Structure
  14. GC15964 Clopidogrel hydrogen sulfate P2Y12 receptor antagonist Clopidogrel hydrogen sulfate  Chemical Structure
  15. GC35711 Clopidogrel thiolactone Clopidogrel thiolactone is an active metabolites containing thiols resulting from thionolactone transformation of clopidogrel. Clopidogrel thiolactone  Chemical Structure
  16. GC31664 Diquafosol tetrasodium (INS365) Diquafosol tetrasodium (INS365) is a P2Y2 receptor agonist that stimulates fluid and mucin secretion on the ocular surface, as a topical treatment of dry eye disease. Diquafosol tetrasodium (INS365)  Chemical Structure
  17. GC10124 DMNPE-caged ATP diammonium salt DMNPE-caged ATP DMNPE-caged ATP diammonium salt  Chemical Structure
  18. GC18472 Elinogrel Elinogrel is a reversible antagonist of the platelet purinergic P2Y12 receptor (Ki = 23 nM) that inhibits platelet aggregation in a human platelet-rich plasma (hPRP) assay (IC50 = 2.81 nM). Elinogrel  Chemical Structure
  19. GC11311 MRS 2179 tetrasodium salt MRS 2179 tetrasodium salt is a competitive P2Y1 receptor antagonist, with a Kb of 102 nM and a pA2 of 6.99 for turkey P2Y1 receptor. MRS 2179 tetrasodium salt  Chemical Structure
  20. GC15590 MRS 2211 P2Y13 receptor antagonist MRS 2211  Chemical Structure
  21. GC12723 MRS 2279 Selective, high affinity competitive antagonist of the P2Y1 receptor MRS 2279  Chemical Structure
  22. GC14852 MRS 2365 Highly potent, selective P2Y1 receptor agonist MRS 2365  Chemical Structure
  23. GC17476 MRS 2500 tetraammonium salt Highly potent and selective antagonist of the platelet P2Y1 receptor MRS 2500 tetraammonium salt  Chemical Structure
  24. GC11078 MRS 2578 P2Y6 receptor antagonist,potent and selective MRS 2578  Chemical Structure
  25. GC17089 MRS 2690 P2Y14 receptor agonist MRS 2690  Chemical Structure
  26. GC13155 MRS 2693 trisodium salt P2Y6 agonist MRS 2693 trisodium salt  Chemical Structure
  27. GC15919 MRS 2768 tetrasodium salt P2Y2 agonist MRS 2768 tetrasodium salt  Chemical Structure
  28. GC50222 MRS 2905 Potent and selective P2Y14 receptor agonist MRS 2905  Chemical Structure
  29. GC13817 MRS 2957 triethylammonium salt P2Y6 agonist MRS 2957 triethylammonium salt  Chemical Structure
  30. GC39759 MRS2500 tetraammonium MRS2500 tetraammonium is a potent, selective and stable antagonist of the P2Y1 receptor (Ki=0.78 nM for recombinant human P2Y1 receptor). MRS2500 tetraammonium  Chemical Structure
  31. GC36680 N6-(4-Hydroxybenzyl)adenosine N6-(4-Hydroxybenzyl)adenosine is a inhibitor of platelet aggregation induced in vitro by collagen and their activity range was demonstrated (IC50: 6.77-141 μM). N6-(4-Hydroxybenzyl)adenosine  Chemical Structure
  32. GC17320 NF 157 P2Y11/P2X1 antagonist NF 157  Chemical Structure
  33. GC17742 NF 340 P2Y11 antagonist NF 340  Chemical Structure
  34. GC13221 NF 546 P2Y11 agonist NF 546  Chemical Structure
  35. GC67795 P2Y2R/GPR17 antagonist 1 P2Y2R/GPR17 antagonist 1  Chemical Structure
  36. GC10826 PIT Purinergic P2Y receptor ligand PIT  Chemical Structure
  37. GC50080 PPTN hydrochloride High affinity and selective P2Y14 antagonist PPTN hydrochloride  Chemical Structure
  38. GC17464 Prasugrel ADP receptor inhibitor Prasugrel  Chemical Structure
  39. GC14067 Prasugrel hydrochloride P2 Receptor inhibitor Prasugrel hydrochloride  Chemical Structure
  40. GC36957 Prasugrel Maleic acid Prasugrel (PCR 4099) Maleic acid is a thienopyridine and prodrug, inhibits platelet function. Prasugrel Maleic acid  Chemical Structure
  41. GC68419 Prasugrel-d3 Prasugrel-d3  Chemical Structure
  42. GC13095 PSB 0474 P2Y6 receptor agonist PSB 0474  Chemical Structure
  43. GC14468 PSB 0739 P2Y12 receptor antagonist PSB 0739  Chemical Structure
  44. GC15635 PSB 1114 P2Y2 receptor agonist PSB 1114  Chemical Structure
  45. GC50224 SAR 216471 hydrochloride Potent P2Y12 antagonist; orally available SAR 216471 hydrochloride  Chemical Structure
  46. GC37705 Suramin

    Suramin is a reversible and competitive protein-tyrosine phosphatases (PTPases) inhibitor.

    Suramin  Chemical Structure
  47. GC16832 Suramin hexasodium salt Suramin hexasodium salt(Suramin hexasodium salt) is a reversible and competitive protein-tyrosine phosphatases (PTPases) inhibitor. Suramin hexasodium salt  Chemical Structure
  48. GC32594 TAK-024 TAK-024 is a platelet inhibitor with IC50s of 31, 79 and 51 nM in human, monkey and guinea pig, respectively. TAK-024  Chemical Structure
  49. GC15332 Ticagrelor

    P2Y12 receptor antagonist

    Ticagrelor  Chemical Structure
  50. GC11388 UDP disodium salt UDP disodium salt is a potent, selective P2Y6 receptor native agonist (EC50=300 nM; pEC50=6.52 for human P2Y6 receptor). UDP disodium salt  Chemical Structure
  51. GC45111 UDP-α-D-Glucose (sodium salt) UDP-α-D-Glucose (sodium salt) (UDP-D-Glucose disodium salt) is the precursor of glucose-containing oligosaccharides, polysaccharides, glycoproteins, and glycolipids in animal tissues and in some microorganisms. UDP-α-D-Glucose  (sodium salt)  Chemical Structure
  52. GC17171 UTPγS trisodium salt

    P2Y2 and P2Y4 receptor agonist

    UTPγS trisodium salt  Chemical Structure
  53. GC37901 Vicagrel Vicagrel is a potent, safe and orally active antiplatelet agent, which works by irreversibly inhibiting P2Y12 receptor. Vicagrel  Chemical Structure
  54. GC46239 YM-254890 A cyclic depsipeptide Gαq/11 inhibitor YM-254890  Chemical Structure

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