P2Y Receptor
P2Y Receptor is a family of purinergic G protein-coupled receptors, stimulated by nucleotides.
Products for P2Y Receptor
- Cat.No. Product Name Information
- GC41668 (±)-Clopidogrel (hydrochloride) Clopidogrel is an antithrombic compound whose active metabolite is a selective, irreversible antagonist of the platelet purinergic P2Y12 receptor (IC50 = 100 nM).
- GC64027 2-Methylthio-AMP 2-Methylthio-AMP (2-MeSAMP) is a selective and direct P2Y12 antagonist.
- GC62783 2-Methylthio-AMP diTEA 2-Methylthio-AMP (2-MeSAMP) diTEA is a selective and direct P2Y12 antagonist.
- GC60016 2-Methylthioadenosine diphosphate trisodium An agonist of P2Y receptors
- GC14753 2-ThioUTP tetrasodium salt P2Y2 agonist
-
GC13588
5-OMe-UDP trisodium salt
Potent P2Y6 agonist
- GC50081 AR-C 118925XX Selective and competitive P2Y2 antagonist
- GC12914 AR-C 66096 tetrasodium salt P2Y12 antagonist,potent and selective
- GC14956 AZD1283 Potent P2Y12 antagonist
- GC19081 BPTU BPTU is a novel P2Y1 allosteric antagonist.
- GC43137 Cangrelor (sodium salt) Cangrelor (sodium salt), an adenosine triphosphate analogue, is a reversible and selective platelet P2Y12 antagonist, with prompt and potent antiplatelet effects.
- GC35710 Clopidogrel Clopidogrel is an orally active platelet inhibitor that targets P2Y12 receptor.
- GC15964 Clopidogrel hydrogen sulfate P2Y12 receptor antagonist
- GC35711 Clopidogrel thiolactone Clopidogrel thiolactone is an active metabolites containing thiols resulting from thionolactone transformation of clopidogrel.
- GC31664 Diquafosol tetrasodium (INS365) Diquafosol tetrasodium (INS365) is a P2Y2 receptor agonist that stimulates fluid and mucin secretion on the ocular surface, as a topical treatment of dry eye disease.
- GC10124 DMNPE-caged ATP diammonium salt DMNPE-caged ATP
- GC18472 Elinogrel Elinogrel is a reversible antagonist of the platelet purinergic P2Y12 receptor (Ki = 23 nM) that inhibits platelet aggregation in a human platelet-rich plasma (hPRP) assay (IC50 = 2.81 nM).
- GC11311 MRS 2179 tetrasodium salt MRS 2179 tetrasodium salt is a competitive P2Y1 receptor antagonist, with a Kb of 102 nM and a pA2 of 6.99 for turkey P2Y1 receptor.
- GC15590 MRS 2211 P2Y13 receptor antagonist
- GC12723 MRS 2279 Selective, high affinity competitive antagonist of the P2Y1 receptor
- GC14852 MRS 2365 Highly potent, selective P2Y1 receptor agonist
- GC17476 MRS 2500 tetraammonium salt Highly potent and selective antagonist of the platelet P2Y1 receptor
- GC11078 MRS 2578 P2Y6 receptor antagonist,potent and selective
- GC17089 MRS 2690 P2Y14 receptor agonist
- GC13155 MRS 2693 trisodium salt P2Y6 agonist
- GC15919 MRS 2768 tetrasodium salt P2Y2 agonist
- GC50222 MRS 2905 Potent and selective P2Y14 receptor agonist
- GC13817 MRS 2957 triethylammonium salt P2Y6 agonist
- GC39759 MRS2500 tetraammonium MRS2500 tetraammonium is a potent, selective and stable antagonist of the P2Y1 receptor (Ki=0.78 nM for recombinant human P2Y1 receptor).
- GC36680 N6-(4-Hydroxybenzyl)adenosine N6-(4-Hydroxybenzyl)adenosine is a inhibitor of platelet aggregation induced in vitro by collagen and their activity range was demonstrated (IC50: 6.77-141 μM).
- GC17320 NF 157 P2Y11/P2X1 antagonist
- GC17742 NF 340 P2Y11 antagonist
- GC13221 NF 546 P2Y11 agonist
- GC67795 P2Y2R/GPR17 antagonist 1
- GC10826 PIT Purinergic P2Y receptor ligand
- GC50080 PPTN hydrochloride High affinity and selective P2Y14 antagonist
- GC17464 Prasugrel ADP receptor inhibitor
- GC14067 Prasugrel hydrochloride P2 Receptor inhibitor
- GC36957 Prasugrel Maleic acid Prasugrel (PCR 4099) Maleic acid is a thienopyridine and prodrug, inhibits platelet function.
- GC68419 Prasugrel-d3
- GC13095 PSB 0474 P2Y6 receptor agonist
- GC14468 PSB 0739 P2Y12 receptor antagonist
- GC15635 PSB 1114 P2Y2 receptor agonist
- GC50224 SAR 216471 hydrochloride Potent P2Y12 antagonist; orally available
-
GC37705
Suramin
Suramin is a reversible and competitive protein-tyrosine phosphatases (PTPases) inhibitor.
- GC16832 Suramin hexasodium salt Suramin hexasodium salt(Suramin hexasodium salt) is a reversible and competitive protein-tyrosine phosphatases (PTPases) inhibitor.
- GC32594 TAK-024 TAK-024 is a platelet inhibitor with IC50s of 31, 79 and 51 nM in human, monkey and guinea pig, respectively.
-
GC15332
Ticagrelor
P2Y12 receptor antagonist
- GC11388 UDP disodium salt UDP disodium salt is a potent, selective P2Y6 receptor native agonist (EC50=300 nM; pEC50=6.52 for human P2Y6 receptor).
- GC45111 UDP-α-D-Glucose (sodium salt) UDP-α-D-Glucose (sodium salt) (UDP-D-Glucose disodium salt) is the precursor of glucose-containing oligosaccharides, polysaccharides, glycoproteins, and glycolipids in animal tissues and in some microorganisms.
-
GC17171
UTPγS trisodium salt
P2Y2 and P2Y4 receptor agonist
- GC37901 Vicagrel Vicagrel is a potent, safe and orally active antiplatelet agent, which works by irreversibly inhibiting P2Y12 receptor.
- GC46239 YM-254890 A cyclic depsipeptide Gαq/11 inhibitor