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- Cat.No. Product Name Information
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GC10350
TIC10 isomer
Potent Akt/ERK inhibitor
- GC45195 α,β-Methyleneadenosine 5'-triphosphate (sodium salt) α,β-Methyleneadenosine 5'-triphosphate (sodium salt), a phosphonic analog of ATP, is a P2X3 and P2X7 receptor ligand.
- GC40302 α-hydroxy Tamoxifen Tamoxifen is a selective estrogen receptor (ER) modulator that is widely used in the therapeutic and chemopreventive treatment of breast cancer.
- GC37980 α-Tocopherol phosphate α-Tocopherol phosphate is the compound demonstrating the highest vitamin E activity, which is available both in its natural form as RRR-alpha-tocopherol isolated from plant sources.
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GC45224
α-Truxillic Acid
α-Truxillic acid can be formed by the dimerization of two molecules of α-trans-cinnamic acid.
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GC41267
β-cyano-L-Alanine
Hydrogen sulfide (H2S) is a naturally-occurring gasotransmitter with vasodilator and inflammatory modulating activity.
- GA24007 β-Endorphin (30-31) (bovine, camel, mouse, ovine) β-Endorphin (30-31) (bovine, camel, mouse, ovine) (Glycyl-L-glutamine), as a enzymatic cleavage product of β-endorphin, is apparently an endogenous antagonist of beta-endorphin(1-31) in several systems.
- GC31977 α-2,3-sialyltransferase-IN-1 α-2,3-sialyltransferase-IN-1 (Lith-O-Asp analog) is a noncompetitive α-2,3-sialyltransferase inhibitor with an IC50 of 6 μM.
- GC33470 β-Apo-13-carotenone (D'Orenone) β-Apo-13-carotenone (D'Orenone) (D'Orenone) is a naturally occurring β-apocarotenoid functioned as an antagonist of RXRα.
- GC33505 β-Apo-13-carotenone D3 (D'Orenone D3)
- GC30207 γ-L-Glutamyl-L-alanine γ-L-Glutamyl-L-alanine, composed of gamma-glutamate and alanine, is a proteolytic breakdown product of larger proteins.
- GC16005 (±)-CPSI 1306 macrophage inhibitory factor (MIF) inhibitor
- GC32617 (±)-WS75624B (±)-WS75624B is an endothelin converting enzyme (ECE) inhibitor with an IC50 of 0.03 μg/mL.
- GC34953 (+)-BAY-1251152 (+)-BAY-1251152 ((+)-BAY-1251152) is an enanthiomer of BAY-1251152 with rotation (+). (+)-BAY-1251152 is a potent and selective CDK9 inhibitor with an IC50 of 3 nM. (+)-BAY-1251152 has anti-tumour activity.
- GC38119 (+)-Columbianetin (+)-Columbianetin is an isomer of Columbianetin.
- GC38443 (+)-SHIN1 (+)-SHIN1 ((+)-RZ-2994) is an active (+) enantiomer of SHIN1.
- GC17330 (+)-Usniacin (+)-Usniacin is isolated from isolated from lichens, binds at the ATP-binding pocket of mTOR, and inhibits mTORC1/2 activity. (+)-Usniacin inhibits the phosphorylation of mTOR downstream effectors: Akt (Ser473), 4EBP1, S6K, induces autophay, with anti-cancer activity. (+)-Usniacin possesses antimicrobial activity against a number of planktonic gram-positive bacteria, including Staphylococcus aureus, Enterococcus faecalis, and Enterococcus faecium.
- GC34948 (-)-GSK598809 (-)-GSK598809 is an isomer of GSK598809.
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GC14520
(-)-p-Bromotetramisole Oxalate
(-) -P-Bromotetramisole Oxalate is a potent nonspecific alkaline phosphatase inhibitor.
- GC38444 (-)-SHIN1 (-)-SHIN1 ((-)-RZ-2994) is an inactive (?) enantiomer of SHIN1.
- GC12164 (-)-Terreic acid Bruton's tyrosine kinase (BTK) inhibitor
- GC30855 (1R,2R)-2-PCCA(hydrochloride) (1R,2R)-2-PCCA(hydrochloride) is a diastereomer of 2-PCCA, and acts as a potent GPR88 receptor agonist, with an EC50 of 3 nM in cell-free assay, and 603 nM in cell assay.
- GC34440 (1S,2S,3R)-DT-061 (1S,2S,3R)-DT-061 is an enantiomer of DT-061. DT-061 is an orally bioavailable activator of protein phosphatase 2A (PP2A) and could be applied in the therapy of KRAS-mutant and MYC-driven tumorigenesis.
- GC32754 (2R)-Octyl-α-hydroxyglutarate ((2R)-Octyl-2-HG) (2R)-Octyl-α-hydroxyglutarate ((2R)-Octyl-2-HG) ((2R)-Octyl-2-HG) is a modified form of D-isomer 2-Hydroxyglutarate.
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GC19473
(2S)-Octyl-α-hydroxyglutarate
A modified form of S-isomer 2-Hydroxyglutarate
- GC30605 (3β,20E)-24-Norchola-5,20(22)-diene-3,23-diol (3β,20E)-24-Norchola-5,20(22)-diene-3,23-diol is a steroid-based allylic alcohol.
- GC13782 (3S,4S)-3-(Boc-amino)-4-methylpyrrolidine (3S,4S)-3-(Boc-amino)-4-methylpyrrolidine
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GC30701
(5R)-BW-4030W92
(5R)-BW-4030W92 is the R enantiomer of BW-4030W92.
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GC13944
(5Z)-7-Oxozeaenol
TAK1 mitogen-activated protein kinase kinase kinase (MAPKKK) inhibitor
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GC15970
(6-)ε-Aminocaproic acid
antifibrinolytic agent
- GC34975 (9Z,12E)-Tetradecadien-1-yl acetate
- GC34976 (Arg)9 (Arg)9 (Nona-L-arginine;Peptide R9) is a cell-penetrating peptide; exhibits neuroprotective activity with an IC50 of 0.78 μM in the glutamic acid model.
- GC32522 (E)-Alprenoxime (CDDD-1815) (E)-Alprenoxime (CDDD-1815) is the isomer of the Alprenoxime.
- GC34982 (E)-LHF-535 (E)-LHF-535 is the E-isomer of LHF-535.
- GC38229 (R)-(+)-Atenolol An enantiomer of (±)-atenolol
- GC13030 (R)-(-)-Ibuprofen Inhibitor of Cox-1 and Cox-2
- GC33574 (R)-1,2,3,4-Tetrahydro-3-isoquinolinecarboxylic acid (R)-1,2,3,4-Tetrahydro-3-isoquinolinecarboxylic acid is a constrained Phe analogue which can fold into a beta-bend and a helical structure, and to adopt a preferred side-chain disposition in the peptide.
- GC38716 (R)-Apremilast (R)-Apremilast ((R)-CC-10004) is a enantiomer of Apremilast.
- GC34987 (R)-BAY-85-8501 (R)-BAY-85-8501 is the less active Enantiomer of BAY-85-8501.
- GC34988 (R)-CE3F4 (R)-CE3F4 is a potent and selective inhibitor of exchange protein directly activated by cAMP isoform 1 (Epac1), with an IC50 of 4.2 μM, with 10-fold selectivity for Epac1 over Epac2 (IC50, 44 μM).
- GC38717 (R)-CSN5i-3 (R)-CSN5i-3 is the (R)-enantiomer of CSN5i-3. CSN5i-3 is a potent, selective and orally available inhibitor of CSN5.
- GC38718 (R)-FT671 (R)-FT671 is the R-isomer of FT671.
- GC34989 (R)-Ketorolac (R)-Ketorolac is the R-enantiomer of Ketorolac, shows potent analgesic activity, reduces ulcerogenic potential.
- GC38719 (R)-NVS-ZP7-4 (R)-NVS-ZP7-4 is the R-isomer of NVS-ZP7-4.
- GC34991 (R)-Oxiracetam (R)-Oxiracetam is the (R)-enantiomer of the nootropic drug oxiracetam. Oxiracetam (ISF 2522) is a nootropic drug of the racetam family and stimulant.
- GC34992 (R)-Pantetheine (R)-Pantetheine is the biosynthetic precursor to CoA.
- GC34445 (R)-Q-VD-OPh (R)-Q-VD-OPh ((R)-QVD-OPH) is the less active enantiomer of Q-VD-OPha. Q-VD-OPha is an irreversible pan-caspase inhibitor with potent antiapoptotic properties.
- GC34994 (R)-Simurosertib (R)-Simurosertib ((R)-TAK-931) is the (R)-enantiomer of Simurosertib.
- GC38110 (R)-VU 6008667 (R)-VU 6008667, the less active (R)-enantiomer to VU 6008667, is devoid of M5 NAM activity (IC50>10 μM).
- GC38540 (R)-VX-984 (R)-VX-984 ((R)-M9831) is the (R)-enantiomer of VX-984.
- GC33531 (R)-Zanubrutinib ((R)-BGB-3111) (R)-Zanubrutinib ((R)-BGB-3111) is the R enantiomer of Zanubrutinib.
- GC38138 (R,S)-Anatabine A plant alkaloid that reduces Aβ production
- GC38875 (Rac)-ABT-202 dihydrochloride (Rac)-ABT-202 dihydrochloride is a racemate of ABT-202.
- GC34447 (Rac)-BL-918 (Rac)-BL-918 is the racemate of BL-918.
- GC38876 (Rac)-IDO1-IN-5 (Rac)-IDO1-IN-5 (Example 1) is a racemate of IDO1-IN-5. IDO1-IN-5 is a potent, selective and brain penetrated inhibitor of Indoleamine 2,3-Dioxygenase 1 (IDO1) activity, binds to apo-IDO1 lacking heme rather than mature heme-bound IDO1.
- GC38877 (Rac)-LM11A-31 dihydrochloride (Rac)-LM11A-31 dihydrochloride is an isomer of LM11A-31 dihydrochloride.
- GC38722 (Rac)-Telmesteine (Rac)-Telmesteine is a protease inhibitor and is thus a suitable enzyme stabilizer extracted from patent WO 2017220302 A1, compound II-1.
- GC34997 (rel)-Myrislignan (rel)-Myrislignan, a relative configuration of Myrislignan.
- GC38723 (rel)-PROTAC ERRα Degrader-1
- GC30737 (RS)-Carbocisteine (S-(Carboxymethyl)-DL-cysteine) (RS)-Carbocisteine (S-(Carboxymethyl)-DL-cysteine) is the S-carboxymethyl cysteine with no detectable inhibitory effect.
- GC30120 (S)-Dolaphenine hydrochloride (S)-Dolaphenine hydrochloride is a component of Dolastatin 10.
- GC38878 (S)-IDO1-IN-5 (S)-IDO1-IN-5 (Example 1B) is an active S-isomer of IDO1-IN-5. (S)-IDO1-IN-5 binds to IDOL with an IC50 value less than 1.5 ?Μ. IDO1-IN-5 is a potent, selective and brain penetrated inhibitor of Indoleamine 2,3-Dioxygenase 1 (IDO1) activity, binds to apo-IDO1 lacking heme rather than mature heme-bound IDO1.
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GC30264
(S)-Metolachor
(S)-Metolachor, a derivative of aniline, is a major pesticide in use.
- GC35004 (S)-Propafenone (S)-Propafenone ((S)-SA-79) is the S-enantiomer of Propafenone.
- GC35005 (S)-Purvalanol B (S)-Purvalanol B is the S enantiomer of Purvalanol B.
- GC35007 (S)-Tedizolid (S)-Tedizolid is the S-enantiomer of Tedizolid.
- GC38879 (S)-Trolox (S)-Trolox is an analogue of vitamin E, in which the phytyl chain is replaced with a carboxyl group.
- GC35008 (Z)-2-decenoic acid A natural fatty acid which disperses biofilms
- GC38304 (Z)-Aconitic acid (Z)-Aconitic acid (cis-Aconitic acid) is the cis-isomer of Aconitic acid.
- GC30154 (Z)-MDL 105519 (Z)-MDL 105519 is the inactive isoform of MDL 105519.
- GC34202 (Z)2S,4R-Sacubitril (Z)2S,4R-Sacubitril is the impurity of Sacubitril.
- GC34448 1,2,3,6-Tetragalloylglucose 1,2,3,6-Tetragalloylglucose is a potent UDP glucuronosyltransferase 1 family, polypeptide A1 (UGT1A1) inhibitor, with a Ki of 1.68 μM.
- GC35031 1-(3,4-Dimethoxycinnamoyl)piperidine 1-(3,4-Dimethoxycinnamoyl)piperidine, a synthesized piperidine analog, possesses antimicrobial and antioxidant activity.
- GC34189 1-Acetyl-3-o-toluyl-5-fluorouracil (A-OT-Fu) 1-Acetyl-3-o-toluyl-5-fluorouracil (A-OT-Fu) is a potent an antineoplastic agent.
- GC35064 1-Cinnamoylpyrrolidine 1-Cinnamoylpyrrolidine (Compound 3), a crude extract prepared from Piper caninum, is a DNA strand scission agent, induces the relaxation of supercoiled pBR322 plasmid DNA.
- GC10430 1-Deoxygalactonojirimycin (hydrochloride) 1-Deoxygalactonojirimycin (hydrochloride) (GR181413A) is a potent and competitive inhibitor of α-galactosidase A (α-Gal A) with an IC50 of 0.04 μM for human α-Gal A.
- GC30969 11β-HSD1-IN-1 11β-HSD1-IN-1 is an inhibitor of 11β-hydroxydehydrogenase 1 (11β-HSD1), with an IC50 of 52 nM, and used for the treatment of pain.
- GC33899 13-cis-N-[4-(Ethoxycarbonyl)phenyl]retinamide 13-cis-N-[4-(Ethoxycarbonyl)phenyl]retinamide is a derivative of Retinoic acid.
- GC18237 13-Methylberberine (chloride) 13-Methylberberine (13-MB) (chloride) is a 13-methyl-substituted derivative of berberine .
- GC31185 18:0 LYSO-PE (Stearoyl lysophosphatidylethanolamine) 18:0 LYSO-PE (Stearoyl lysophosphatidylethanolamine) is an agent that can induce [Ca2+]i increase.
- GC13452 2'-Deoxycytidine hydrochloride 2'-Deoxycytidine hydrochloride
- GC10897 2'-Deoxyguanosine 2'-Deoxyguanosine
- GC35089 2'-Fluorothymidine 2'-Fluorothymidine (2'-Fluoro-2'-deoxythymidine), a bioisostere of both thymidine (TdR) and methyluridine, is a putative highly selective substrate for thymidine kinase type 2 (TK2).
- GC16996 2,4-Diamino-6-hydroxypyrimidine GTP cyclohydrolase I (GCH1) inhibitor and blocks NO production
- GC33570 2-γ-Linolenoyl-1,3-dilinoleoyl-sn-glycerol 2-γ-Linolenoyl-1,3-dilinoleoyl-sn-glycerol is a triglyceride.
- GC35087 2-Aminoethyl-mono-amide-DOTA-tris(tBu ester) 2-Aminoethyl-mono-amide-DOTA-tris(tBu ester) is a macrocycle DOTA derivative for tumor pretargeting.
- GC30376 2-Aminoheptane (1-Methylhexylamine) 2-Aminoheptane (1-Methylhexylamine) (1-Methylhexylamine) is an isomeric heptylamine commonly used as stimulant.
- GC33542 2-Ethoxybenzamide (Ethenzamide) 2-Ethoxybenzamide (Ethenzamide) is widely used as an antipyretic anodyne.
- GC35091 2-Hydroxy-6-methoxybenzoic acid 2-Hydroxy-6-methoxybenzoic acid can be used for the determination of acetylsalicylic acid and its major metabolite, salicylic acid, in animal plasma.
- GC35092 2-Methoxycinnamic acid 2-Methoxycinnamic acid is a noncompetitive inhibitor of tyrosinase.
- GC35093 2-O-α-D-Glucopyranosyl-L-ascorbic Acid An L-ascorbic acid derivative with antioxidant and radioprotective activities
- GC34382 2-PCCA(hydrochloride)
- GC38692 2-Phenylethylamine hydrochloride
- GC12825 2-Thiouracil antihyperthyroid agent
- GC33412 20-HEDE (WIT 002) 20-HEDE (WIT 002) (WIT 002) is an antagonist of 20-hydroxyeicosatetraenoic acid (20-HETE).
- GC33867 24-Norursodeoxycholic acid (nor-UDCA) 24-norursodeoxycholic acid (Norucholic acid) is a side chain-shortened C23 homologue of UDCA and has shown potent anti-cholestatic, anti-inflammatory and anti-fibrotic properties.
- GC34080 2OH-BNPP1 2OH-BNPP1 is an inhibitor of BUB1 kinase, a Ser/Thr kinase, used for the treatment of cancer.
- GC32645 2R,4R-Sacubitril 2R,4R-Sacubitril is the impurity of Sacubitril.
- GC32651 2R,4S-Sacubitril 2R,4S-Sacubitril is the impurity of Sacubitril.
- GC34201 2S,4R-Sacubitril 2S,4R-Sacubitril is the impurity of Sacubitril.