Selpercatinib |
| Catalog No.GC33192 |
A RET kinase inhibitor
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2152628-33-4
Sample solution is provided at 25 µL, 10mM.
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Selpercatinib is a RET kinase inhibitor extracted from patent WO2018071447A1, Compound Example 163, has an IC50 of 14.0 nM, 24.1 nM, and 530.7 nM for RET (WT), RET (V804M) , and RET (G810R), respectively[1]. Antineoplastic activity[2].
[1]. Steven W. Andrews, et al. Substituted pyrazolo[1,5-a]pyridine compounds as ret kinase inhibitors. WO2018071447A1. [2]. International Nonproprietary Names for Pharmaceutical Substances (INN). WHO Drug Information, Vol. 32, No. 4, 2018.
Average Rating: 5 (Based on Reviews and 10 reference(s) in Google Scholar.)
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