Proteolysis
منتجات لـ نبسب؛ Proteolysis
- القط. رقم اسم المنتج بيانات
-
GC46308
(±)-Sitagliptin-d4 (hydrochloride)
A neuropeptide with diverse biological activities
-
GC41656
(±)2-(14,15-Epoxyeicosatrienoyl) Glycerol
(±)214,15EG
2-Arachidonoyl glycerol (2-AG) is an endogenous central cannabinoid (CB1) receptor agonist that is present at relatively high levels in the central nervous system. -
GC41698
(D)2-Rh 110 (trifluoroacetate salt)
D2R, (Asp)2-Rhodamine 110, Rhodamine 110 bis-(L-aspartic acid amide)
(D)2-Rh 110 is a fluorogenic caspase substrate. -
GC40145
(S)-Laudanosine
(+)-Laudanosine, L-Laudanosine, L-(+)-Laudanosine, NSC 35045
(S)-Laudanosine is the (S) enantiomer of laudanosine, a metabolite of the neuromuscular blocking agents atracurium and cisatracurium. -
GC40121
(Z-DEVD)2-Rh 110 (trifluoroacetate salt)
(Z-Asp-Glu-Val-Asp)2-Rhodamine 110
(Z-DEVD)2-Rh 110 is a fluorogenic substrate for caspase-3. -
GC41742
(Z-IETD)2-Rh 110 (trifluoroacetate salt)
(Z-Ile-Glu-Thr-Asp)2-R110, Rhodamine 110 bis-(N-CBZ-IETD)2
(Z-IETD)2-Rh 110 is a fluorogenic substrate for caspase-8. -
GC49390
13C6-4-Nitroaniline
13C6-p-Nitroaniline
An internal standard for the quantification of 4-nitroaniline -
GC18452
3,4-Dichloroisocoumarin
3,4-DCI
A serine protease inhibitor -
GC18359
4-Epianhydrochlortetracycline (hydrochloride)
4-Epianhydrochlortetracycline is a derivative of tetracycline .
-
GC52227
5-(3',4'-Dihydroxyphenyl)-γ-Valerolactone
(±)-δ-(3,4-Dihydroxyphenyl)-γ-Valerolactone, 5-(3',4'-Dihydroxyphenyl)-γ-VL
An active metabolite of various polyphenols -
GC42548
5-hydroxy Saxagliptin (hydrochloride)
5-hydroxy Saxagliptin is a major active metabolite of saxagliptin.
-
GC41423
5-trans Prostaglandin E2
transDinoprostone, 5,6trans PGE2
5-trans PGE2 occurs naturally in some gorgonian corals and is a common impurity in commercial lots of PGE1. -
GC40202
7α-hydroxy Cholesterol-d7
7α-hydroxycholesterol-d7
7α-hydroxy Cholesterol-d7 is intended for use as an internal standard for the quantification of 7α-hydroxy cholesterol by GC- or LC-MS.
-
GC49443
7α-hydroxy Cholesterol
7β-Hydroxycholesterol, 7β-OHC
7α-hydroxy Cholesterol هو أكسيد كولسترول ويتكون من الأكسدة الأنزيمية وغير الأنزيمية. -
GC42665
AAF-CMK (trifluoroacetate salt)
NAlaAlaPheCMK, Tripeptidyl Peptidase Inhibitor II
Tripeptidyl peptidase II (TPPII) is a serine peptidase of the subtilisin-type which removes tripeptides from the free NH2 terminus of oligopeptides. -
GC42683
Abz-Ala-Pro-Glu-Glu-Ile-Met-Arg-Arg-Gln-EDDnp
Abz-Ala-Pro-Glu-Glu-Ile-Met-Arg-Arg-Gln-EDDnp is a fluorescence-quenched peptide substrate for human neutrophil elastase (kcat/Km = 531 mM-1s-1).
-
GC52499
Abz-Ala-Pro-Glu-Glu-Ile-Met-Arg-Arg-Gln-EDDnp (trifluoroacetate salt)
A sensitive substrate for neutrophil elastase
-
GC42684
Abz-Val-Ala-Asp-Nva-Arg-Asp-Arg-Gln-EDDnp (trifluoroacetate salt)
Abz-Val-Ala-Asp-Nva-Arg-Asp-Arg-Gln-EDDnp is a fluorescence-quenched peptide substrate for human proteinase 3 (kcat/Km = 1,570 mM-1s-1).
-
GC40122
Ac-AAVALLPAVLLALLAP-DEVD-CHO (trifluoroacetate salt)
Ac-Ala-Ala-Val-Ala-Leu-Leu-Pro-Ala-Val-Leu-Leu-Ala-Leu-Leu-Ala-Pro-Asp-Glu-Val-Asp-CHO, Ac-AAVALLPAVLLALLAP-DEVD-aldehyde, Ac-AAVALLPAVLLALLAPDEVD-CHO, Caspase-3 Inhibitor I, DEVD-CHO-CPP 32
Ac-AAVALLPAVLLALLAP-DEVD-CHO is a composite of Ac-DEVD-CHO, a peptide inhibitor of caspase-3 and -7, and a cell-permeable hydrophobic sequence derived from K-FGF. -
GC40118
Ac-AAVALLPAVLLALLAP-IETD-CHO (trifluoroacetate salt)
Ac-Ala-Ala-Val-Ala-Leu-Leu-Pro-Ala-Val-Leu-Leu-Ala-Leu-Leu-Ala-Pro-Ile-Glu-Thr-Asp-CHO, Caspase-8 Inhibitor I
Ac-AAVALLPAVLLALLAP-IETD-CHO is a composite of Ac-IETD-CHO, a peptide inhibitor of caspase-8, and a cell-permeable hydrophobic sequence derived from K-FGF. -
GC40123
Ac-AAVALLPAVLLALLAP-VAD-CHO (trifluoroacetate salt)
Caspase Inhibitor II, Ac-AAVALLPAVLLALLAP-VAD-aldehyde, Ac-AAVALLPAVLLALLAPVAD-CHO
Ac-AAVALLPAVLLALLAP-VAD-CHO is a composite of Ac-VAD-CHO, a non-selective caspase inhibitor, and a cell-permeable hydrophobic sequence derived from K-FGF. -
GA20494
Ac-Asp-Glu-Val-Asp-pNA
Ac-Asp-Glu-Val-Asp-pNA
The cleavage of the chromogenic caspase-3 substrate Ac-DEVD-pNA can be monitored at 405 nm. -
GC48470
Ac-DEVD-CHO (trifluoroacetate salt)
N-Ac-Asp-Glu-Val-Asp-CHO
A dual caspase3/caspase7 inhibitor -
GC48430
Ac-DEVD-CMK (trifluoroacetate salt)
AcAspGluValAspCMK, Caspase3 Inhibitor III
-
GC42687
Ac-DMQD-AMC (trifluoroacetate salt)
Ac-Asp-Met-Gln-Asp-AMC, Ac-Asp-Met-Gln-Asp-7-amino-4-methylcoumarin
Ac-DMQD-AMC is a fluorogenic substrate for caspase-3. -
GC42688
Ac-DMQD-CHO (trifluoroacetate salt)
Ac-Asp-Met-Gln-Asp-CHO, Caspase-3 Inhibitor
Ac-DMQD-CHO is a peptide inhibitor of caspase-3 (IC50 = 39 nM). -
GC42689
Ac-DNLD-AMC
Ac-Asp-Asn-Leu-Asp-MCA, N-Acetyl-Asp-Asn-Leu-Asp-7-amido-Methylcoumarin, Caspase-3 Substrate
Ac-WLA-AMC عبارة عن ركيزة فلوروجينية من caspase-3. -
GC40154
Ac-ESMD-CHO (trifluoroacetate salt)
Ac-Glu-Ser-Met-Asp-CHO
Ac-ESMD-CHO is an inhibitor of caspase-3 maturation. -
GC49704
Ac-FLTD-CMK (trifluoroacetate salt)
Ac-Phe-Leu-Thr-Asp-CMK
An inhibitor of caspase-1, -4, -5, and -11 -
GC42706
Ac-IEPD-AMC (trifluoroacetate salt)
Acetyl-Ile-Glu-Pro-Asp-7-amino-4-Methylcoumarin, Ac-Ile-Glu-Pro-Asp-AMC
Ac-IEPD-AMC is a fluorogenic substrate for granzyme B. -
GC40152
Ac-IEPD-pNA (trifluoroacetate salt)
Ac-Ile-Glu-Pro-Asp-p-nitroanilide, Caspase-8 Chromogenic Substrate, Granzyme B Substrate VIII
Ac-IEPD-pNA is a colorimetric substrate for granzyme B and caspase-8. -
GC40164
Ac-IETD-CHO (trifluoroacetate salt)
Caspase-8 Inhibitor
Ac-IETD-CHO is an inhibitor of caspase-8 (IC50 = 5 nM).
-
GC42708
Ac-LEHD-AFC (trifluoroacetate salt)
N-Acetyl-Leu-Glu-His-Asp-7-amino-4-Trifluoromethylcoumarin, Caspase-9 substrate (Fluorogenic)
Ac-LEHD-AFC is a fluorogenic substrate that can be cleaved by caspase-4, -5, and -9. -
GC18226
Ac-LEHD-AMC (trifluoroacetate salt)
Ac-Leu-Glu-His-Asp-AMC, Caspase-9 Substrate
Ac-LEHD-AMC (ملح ثلاثي فلورو أسيتات) هو ركيزة فلورية لكاسباس 9 (الإثارة: 341 نانومتر ؛ الانبعاث: 441 نانومتر). -
GC46791
Ac-LEHD-pNA (trifluoroacetate salt)
Ac-Leu-Glu-His-Asp-pNA, Caspase-9 Chromogenic Substrate I
A neuropeptide with diverse biological activities -
GC40556
Ac-LETD-AFC
NAcetylLeuGluThrAsp7amino4Trifluoromethylcoumarin, Caspase8 Substrate (Fluorogenic)
Ac-LETD-AFC عبارة عن ركيزة فلورية من كاسباس 8. -
GC42709
Ac-LEVD-CHO (trifluoroacetate salt)
Ac-Leu-Glu-Val-Asp-CHO, Caspase-4 Inhibitor I
Ac-LEVD-CHO is a caspase-4 inhibitor.
-
GC13400
Ac-VDVAD-AFC
N-Acetyl-Val-Asp-Val-Ala-Asp-7-amino-4-Trifluoromethylcoumarin Caspase-2 Substrate (Fluorogenic)
Ac-VDVAD-AFC عبارة عن ركيزة فلورية خاصة بكاسبيز. يمكن لـ Ac-VDVAD-AFC قياس النشاط الشبيه بـ caspase-3 ونشاط caspase-2 ويمكن استخدامه في البحث عن الورم والسرطان. -
GC52372
Ac-VDVAD-AFC (trifluoroacetate salt)
N-Acetyl-Val-Asp-Val-Ala-Asp-AFC, N-Acetyl-Val-Asp-Val-Ala-Asp-7-amino-4-Trifluoromethylcoumarin, Caspase-2 Substrate (Fluorogenic)
A fluorogenic substrate for caspase-2 -
GC42715
Ac-VDVAD-CHO (trifluoroacetate salt)
Ac-Val-Asp-Val-Ala-Asp-CHO
Ac-VDVAD-CHO is an inhibitor of caspase-2, -3, and -7 (Kis = 3.5, 1, and 7.5 nM, respectively). -
GC42716
Ac-VDVAD-pNA (trifluoroacetate salt)
Ac-Val-Asp-Val-Ala-Asp-pNA, Caspase-2 Chromogenic Substrate, acetyl-Val-Asp-Val-Ala-Asp-p-nitroanilide, acetyl-VDVAD-p-nitroanilide
Ac-VDVAD-pNA is a colorimetric substrate for caspase-2. -
GC48974
Ac-VEID-AMC (ammonium acetate salt)
NAcetylValGluIleAsp7amido4Methylcoumarin, Caspase6 Substrate (Fluorogenic)
A caspase-6 fluorogenic substrate -
GC42718
Ac-VEID-CHO (trifluoroacetate salt)
Ac-Val-Glu-Ile-Asp-CHO
Ac-VEID-CHO is an inhibitor of caspase-6 (IC50 = 16.2 nM). -
GC40162
Ac-VEID-pNA (trifluoroacetate salt)
Ac-Val-Glu-Ile-Asp-pNA, Ac-Val-Glu-Ile-Asp-p-nitroanilide, Caspase-6 Chromogenic Substrate
Ac-VEID-pNA is a substrate for caspase-6. -
GC40124
Ac-WEAD-AMC (trifluoroacetate salt)
Ac-Trp-Glu-Ala-Asp-AMC
Ac-WEAD-AMC is a fluorogenic substrate for caspase-1 and caspase-4. -
GC42719
Ac-WEAD-pNA (trifluoroacetate salt)
Ac-Trp-Glu-Ala-Asp-pNA, Ac-Trp-Glu-Ala-Asp-p-nitroanilide, Caspase-1 and Caspase-4 Chromogenic Substrate
Ac-WEAD-pNA is a colorimetric substrate for caspase-1 and caspase-4. -
GC46796
Ac-WEHD-AFC (trifluoroacetate salt)
N-Acetyl-Trp-Glu-His-Asp-7-amino-4-Trifluoromethylcoumarin, Caspase1 Substrate (Fluorogenic), Caspase5 Substrate (Fluorogenic)
A neuropeptide with diverse biological activities -
GC18021
Ac-YVAD-CHO
Caspase-1 Inhibitor I, L 709049, N-Ac-Tyr-Val-Ala-Asp-CHO
Ac-YVAD-CHO (L-709049) هو مثبط إنزيم (ICE) المحول لرباعي الببتيد (ICE) الفعال والقابل للانعكاس مع قيم Ki للإنسان والفأر 3.0 و 0.76 نانومتر. -
GC42721
Ac-YVAD-CMK
N-Ac-Tyr-Val-Ala-Asp-CMK
Ac-YVAD-CMK هو مثبطAc-YVAD-CMK انتقائي لا رجعة فيه لكاسباس 1 (Ki=0.8nM)، والذي يمكن أن يمنع تنشيط السيتوكين IL-1β proinflammatory cytokine. يمكن أن يقلل Ac-YVAD-CMK من الاستجابة الالتهابية ويحفز تأثير الحماية العصبية طويل الأمد. -
GC46841
Amiloride (hydrochloride) (hydrate)
MK-870
A neuropeptide with diverse biological activities -
GC42788
Aminopeptidase N Inhibitor
Aminopeptidase N (AP-N) inhibitor is a reversible inhibitor of AP-N/CD13 (IC50 = 25 μM).
-
GC48509
Apigenin 7-O-Glucuronide (hydrate)
-
GC46867
Apremilast-d5
APR-d5
Apremilast D5 (CC-10004 D5) هو الديوتيريوم المسمى Apremilast -
GC46878
Aranciamycin
NSC 369226
A fungal metabolite with diverse biological activities -
GC46895
Aurintricarboxylic Acid (ammonium salt)
ATA
A protein synthesis inhibitor with diverse biological activities -
GC62711
BAMEA-O16B
BAMEAO16B عبارة عن جسيمات نانوية دهنية
-
GC91898
BI SF3 (hydrochloride)
BI SF3 (hydrochloride) هو وسيط صناعي.
-
GC40155
Biotin-DEVD-CHO (trifluoroacetate salt)
Biotin-Asp-Glu-Val-Asp-CHO
Biotin-DEVD-CHO is a biotin-conjugated form of the caspase-3 and -7 inhibitor Ac-DEVD-CHO. -
GC40149
Boc-AEVD-CHO (trifluoroacetate salt)
Boc-Ala-Glu-Val-Asp-CHO
Boc-AEVD-CHO is an inhibitor of caspase-8 (Ki = 1.6 nM) that also inhibits caspase-1, -3, -6, and -9 (Kis = 10,000, 375, 438, 425, and 320 nM, respectively). -
GC46937
Boc-Glu-OBzl
An amino acid-containing building block
-
GC45394
Bz-IEGR-pNA (acetate)
Bz-Ile-Glu-Gly-Arg-pNA, Bz-Ile-Glu-Gly-Arg-p-nitroanilide, Factor Xa Chromogenic Substrate
-
GC18315
Calpain Inhibitor VI
SJA 6017
Calpain inhibitor VI is an inhibitor of the calcium-dependent cysteine proteases u-calpain (calpain-1; IC50 = 7.5 nM) and m-calpain (calpain-2; IC50 = 78 nM). -
GC47022
Camostat-d6 (hydrochloride)
A neuropeptide with diverse biological activities
-
GC43146
Caspase-9 Inhibitor III (trifluoroacetate salt)
Ac-LEHD-CMK
Caspase-9 inhibitor III is an inhibitor of caspase-9 with cardioprotective effects. -
GC43150
CAY10406
CAY10406 is a trifluoromethyl analog of an isatin sulfonamide compound that selectively inhibits caspases 3 and 7.
-
GC43154
CAY10443
(S)Indan1yl 3,4dichlorobenzylcarbamate
Mitochondrial release of cytochrome c triggers apoptosis via the assembly of a multimeric complex including caspase-9, Apaf-1, and other components, sometimes called the apoptosome. -
GC47079
Chloramine-T (hydrate)
A common reagent
-
GC52360
Chymotrypsin Substrate I, Colorimetric (trifluoroacetate salt)
Suc-GGF-pNA, Suc-Gly-Gly-Phe-pNA, Suc-Gly-Gly-Phe-p-Nitroanilide
A colorimetric chymotrypsin substrate -
GC47164
Dabcyl-GABA-PQGL-Glu(EDANS)-AK-NH2, (trifluoroacetate salt)
MMP Fluorogenic Substrate III
A neuropeptide with diverse biological activities -
GC43369
Dabcyl-GABA-RPKPVE-Nva-WR-Glu(EDANS)-AK-NH2 (trifluoroacetate salt)
Dabcyl-GABA-RPKPVE-Nva-WR-Glu(EDANS)-AK-NH2 is a fluorogenic substrate for matrix metalloproteinase-3 (MMP-3).
-
GC43370
Dabcyl-RGVVNASSRLA-EDANS (trifluoroacetate salt)
Fluorogenic Human CMV Protease Substrate
Dabcyl-RGVVNASSRLA-EDANS is a fluorogenic substrate for human cytomegalovirus (HCMV) protease. -
GC18421
Dabcyl-YVADAPV-EDANS
Dabcyl-ICE-EDANS
Dabcyl-YVADAPV-EDANS is a fluorogenic substrate for caspase-1. -
GC43371
Dabigatran Acyl-β-D-Glucuronide
β-1-O-Acylglucuronide
Dabigatran acyl-β-D-glucuronide is a major active metabolite of the thrombin inhibitor dabigatran.
-
GC47165
Dabigatran etexilate-d13
A neuropeptide with diverse biological activities
-
GC49684
Dabigatran-13C-d3
BIBR 953-13C,d3; BIBR 953ZW-13C,d3
An internal standard for the quantification of dabigatran -
GC49682
Dabigatran-d3
BIBR 953-d3; BIBR 953ZW-d3
An internal standard for the quantification of dabigatran -
GC43407
Demethylwedelolactone
Demethylwedelolactone (DWL) is a coumestan, originally isolated from E.
-
GC47237
Dipyridamole-d16
A neuropeptide with diverse biological activities
-
GC43542
Dnp-GPLGMRGL-NH2 (trifluoroacetate salt)
Dnp-Gly-Pro-Leu-Gly-Met-Arg-Gly-Leu-NH2, Matrix Metalloproteinase-13 Substrate, MMP-13 Substrate
Dnp-GPLGMRGL-NH2 is a peptide substrate for matrix metalloproteinase-13 (MMP-13) with a kcat/Km value of 4,200,000 M-1s-1. -
GC43544
Dnp-P-Cha-Abu-Cys(Me)-HA-K(Nma)-NH2
Dnp-Pro-Cha-Abu-Cys(Me)-His-Ala-Lys(Nma)-NH2, Matrix Metalloproteinase-1 Fluorogenic Substrate III, MMP-1 Fluorogenic Substrate III
Dnp-P-Cha-Abu-Cys(Me)-HA-K(Nma)-NH2 is a fluorogenic substrate for matrix metalloproteinase-1 (MMP-1) and MMP-9. -
GC43545
Dnp-P-Cha-G-Cys(Me)-HA-K(Nma)-NH2
Dnp-Pro-Cha-Gly-Cys(Me)-His-Ala-Lys(Nma)-NH2, Matrix Metalloproteinase-1/Matrix Metalloproteinase-9 Fluorogenic Substrate, MMP-1/MMP-9 Fluorogenic Substrate
Dnp-P-Cha-G-Cys(Me)-HA-K(Nma)-NH2 is a fluorogenic substrate for matrix metalloproteinase-1 (MMP-1) and MMP-9. -
GC43546
Dnp-PLALWAR (trifluoroacetate salt)
Matrix Metalloproteinase-1 Fluorogenic Substrate I, MMP-1 Fluorogenic Substrate I
Dnp-PLALWAR is a fluorogenic substrate for matrix metalloproteinase-1 (MMP-1) and MMP-8. -
GC43547
Dnp-PLAYWAR (trifluoroacetate salt)
Dnp-Pro-Leu-Ala-Tyr-Trp-Ala-Arg-OH, Matrix Metalloproteinase-8/Matrix Metalloproteinase-26 Fluorogenic Substrate, MMP-8/MMP-26 Fluorogenic Substrate
Dnp-PLAYWAR is a fluorogenic substrate for matrix metalloproteinase-8 (MMP-8) and MMP-26. -
GC43548
Dnp-PLG-Cys(Me)-HA-DArg-NH2 (trifluoroacetate salt)
Dnp-Pro-Leu-Gly-Cys(Me)-His-Ala-DArg-NH2, Matrix Metalloproteinase-1 Substrate II, MMP-1 Substrate II
Dnp-PLG-Cys(Me)-HA-DArg-NH2 is a peptide substrate for matrix metalloproteinase-1 (MMP-1). -
GC43549
Dnp-PLGLWA-DArg-NH2 (trifluoroacetate salt)
Dnp-PLGLWA-DArg-NH2 is a fluorogenic substrate for matrix metalloproteinase-1 (MMP-1), MMP-2, MMP-7, and MMP-9.
-
GC43550
Dnp-PLGMWSR (trifluoroacetate salt)
Dnp-Pro-Leu-Gly-Met-Trp-Ser-Arg-OH, Matrix Metalloproteinase-2/Matrix Metalloproteinase-9 Fluorogenic Substrate I, MMP-2/MMP-9 Fluorogenic Substrate I
Dnp-PLGMWSR is a fluorogenic substrate for matrix metalloproteinase-2 (MMP-2) and MMP-9. -
GC43552
Dnp-RPLALWRS (trifluoroacetate salt)
Dnp-Arg-Pro-Leu-Ala-Leu-Trp-Arg-Ser-OH, Matrix Metalloproteinase-7 Fluorogenic Substrate, MMP-7 Fluorogenic Substrate
Dnp-RPLALWRS is a fluorogenic substrate for matrix metalloproteinase-7 (MMP-7). -
GC91782
DPP-9 Inhibitor 42
Dipeptidyl Peptidase 9 Inhibitor 42
DPP-9 inhibitor 42 is an inhibitor of dipeptidyl peptidase 9 (DDP-9; IC50 = 0.0034 µM). -
GC43614
Enteropeptidase Fluorogenic Substrate
Enteropeptidase fluorogenic substrate is a substrate for enteropeptidase that contains a 7-amino-4-trifluoromethylcoumarin (AFC) moiety.
-
GC48995
Enteropeptidase Fluorogenic Substrate (trifluoroacetate salt)
A fluorogenic substrate of enteropeptidase
-
GC43667
FITC-C6-PLALWAR-Lys(Biotin)-NH2 (trifluoroacetate salt)
FITC-C6-Pro-Leu-Ala-Leu-Trp-Ala-Arg-Lys(Biotin)-NH2, MMP-1/MMP-2/MMP-3 Fluorogenic Substrate
FITC-C6-PLALWAR-Lys(Biotin)-NH2 is a substrate for matrix metalloproteinase-1 (MMP-1), MMP-2, and MMP-3 that can be sequestered by streptavidin via its biotin group. -
GC43668
FITC-C6-YVADAP-K(Dnp) (trifluoroacetate salt)
FITC-C6-Tyr-Val-Ala-Asp-Ala-Pro-Lys(Dnp)-OH
FITC-C6-YVADAP-K(Dnp) is a caspase-1 fluorogenic substrate. -
GC91051
Fluostatin A (sodium salt)
مثبط للفلورينون و DPP-3
-
GC90664
Fluostatin B
مثبط للفلورينون و DPP-3
-
GC60871
Gemigliptin tartrate
طرطرات Gemigliptin (LC15-0444 طرطرات) هو مثبط انتقائي للغاية وقابل للعكس وتنافسي ثنائي الببتيداز 4 (DPP-4) ، مع IC 50 من 10.3 نانومتر من أجل DPP-4 المؤتلف البشري
-
GC49322
GGACK (hydrochloride)
Glu-Gly-Arg-Chloromethyl Ketone, Glu-Gly-Arg-CH2Cl
A uPA and factor Xa inhibitor -
GC20007
Ginsenoside CK
Ginsenoside Compound K, Ginsenoside IH901
A metabolite of ginsenoside Rb1 with diverse biological activity -
GC49437
Gliotoxin-13C13
Aspergillin-13C13
An internal standard for the quantification of gliotoxin -
GC45668
Gly-Arg-AMC (hydrochloride)
Gly-Arg-7-amino-4-methylcoumarin, GR-AMC, GR-7-amino-4-methylcoumarin
A fluorogenic substrate for cathepsin C -
GC40758
Gly-Phe-β-naphthylamide
HGlyPheBNA
Gly-Phe-β ؛ -naphthylamide هو الركيزة لـ Cathepsin C.