CK2/ERK8-IN-1 |
| Catalog No.GC39485 |
A dual inhibitor of CK2 and ERK8
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1085822-09-8
Sample solution is provided at 25 µL, 10mM.
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CK2/ERK8-IN-1 is a dual casein kinase 2 (CK2) (Ki of 0.25 µM) and ERK8 inhibitor with IC50s of 0.50 μM. CK2/ERK8-IN-1 also binds to PIM1, HIPK2 (homeodomain-interacting protein kinase 2), and DYRK1A with Kis of 8.65 µM, 15.25 µM, and 11.9 µM, respectively. CK2/ERK8-IN-1 has pro-apoptotic efficacy[1].
[1]. Pagano MA, et al. The selectivity of inhibitors of protein kinase CK2: an update. Biochem J. 2008 Nov 1;415(3):353-65.
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