Btk inhibitor 1 |
Katalog-Nr.GC35561 |
Btk-Inhibitor 1 ist ein Racemat von IBT6A. IBT6A ist eine Verunreinigung von Ibrutinib. IBT6A kann zur Synthese von IBT6A-Ibrutinib-Dimer und IBT6A-Addukt verwendet werden. Ibrutinib ist ein selektiver, irreversibler Btk-Inhibitor mit einer IC50 von 0,5 nM.
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Cas No.: 1412418-47-3
Sample solution is provided at 25 µL, 10mM.
Btk inhibitor 1 is a pyrazolo[3,4-d]pyrimidine derivative as a Btk kinase inhibitor.IC50 value:Target: BtkFrom PCT Int. Appl. (2012), WO 2012158843 A2 20121122.
[1]. PCT Int. Appl. (2012), WO 2012158843 A2 20121122.
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