Phenserine |
| Katalog-Nr.: GC13783 |
Phenserin ((-)-Eserolinphenylcarbamat) ist ein Derivat von Physostigmin und ist ein potenter, nicht kompetitiver, lang wirkender und selektiver AChE-Hemmer.
Sample solution is provided at 25 µL, 10mM.
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Qualitätskontrolle & SDS
- Aktuelle Charge anzeigen:
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Reinheit: >98.00%
- COA (Zertifikat der Analyse)
- SDS (Sicherheitsdatenblatt)
- Datenblatt
(+)-Phenserine is a novel selective cholinesterase noncompetitive inhibitor with an IC50 of 45.3 μM.
References:
[1]. al-Jafari AA, et al. Kinetics of human erythrocyte acetylcholinesterase inhibition by a novel derivative of physostigmine: phenserine. Biochem Biophys Res Commun. 1998 Jul 9; 248(1):180-5.
| Cas No. | 101246-66-6 | SDF | |
| Chemical Name | (3aS,8aR)-1,3a,8-trimethyl-1,2,3,3a,8,8a-hexahydropyrrolo[2,3-b]indol-5-yl phenylcarbamate | ||
| Canonical SMILES | O=C(NC1=CC=CC=C1)OC2=CC3=C(C=C2)N(C)[C@H]4N(C)CC[C@]43C | ||
| Formula | C20H23N3O2 | M.Wt | 337.42 |
| Löslichkeit | DMF: 25 mg/ml,DMSO: 30 mg/ml,DMSO:PBS (pH 7.2)(1:5): 0.16 mg/ml,Ethanol: 25 mg/ml | Storage | Store at -20°C |
| Allgemeine Tipps | Um eine höhere Löslichkeit zu erreichen, erwärmen Sie das Röhrchen auf 37°C und schütteln Sie es eine Weile im Ultraschallbad. Die Stammlösung kann mehrere Monate unter -20°C gelagert werden. | ||
| Versandbedingungen | Probenlösung zur Bewertung: Lieferung mit blauem Eis Alle anderen verfügbaren Größen: Lieferung mit RT , oder blauem Eis auf Anfrage |
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Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.
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