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(S)-MRTX-1719

Katalog-Nr.GC65045

(S)-MRTX-1719 (Beispiel 16-7) ist das S-Enantiomer von MRTX-1719. (S)-MRTX-1719 ist ein PRMT5/MTA-Komplex-Inhibitor mit einem IC50-Wert von 7070 nM.

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(S)-MRTX-1719 Chemische Struktur

Cas No.: 2630904-44-6

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Sample solution is provided at 25 µL, 10mM.

Product Documents

Quality Control & SDS

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Background

(S)-MRTX-1719 (example 16-7) is the S-enantiomer of MRTX-1719. (S)-MRTX-1719 is a PRMT5/MTA complex inhibitor, with an IC50 of 7070 nM[1].

[1]. Thomas P. BOBINSKI, et al. Mta-cooperative prmt5 inhibitors. WO2021050915A1.

Chemical Properties

Cas No. 2630904-44-6 SDF Download SDF
Formula C23H18ClFN6O2 M.Wt 464.88
Löslichkeit Storage Store at -20°C
General tips Please select the appropriate solvent to prepare the stock solution according to the solubility of the product in different solvents; once the solution is prepared, please store it in separate packages to avoid product failure caused by repeated freezing and thawing.Storage method and period of the stock solution: When stored at -80°C, please use it within 6 months; when stored at -20°C, please use it within 1 month.
To increase solubility, heat the tube to 37°C and then oscillate in an ultrasonic bath for some time.
Shipping Condition Evaluation sample solution: shipped with blue ice. All other sizes available: with RT, or with Blue Ice upon request.

Complete Stock Solution Preparation Table

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1 mg 5 mg 10 mg
1 mM 2.1511 mL 10.7555 mL 21.5109 mL
5 mM 0.4302 mL 2.1511 mL 4.3022 mL
10 mM 0.2151 mL 1.0755 mL 2.1511 mL
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