ERAP1-IN-1 |
| Catalog No.GC60811 |
ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 865273-97-8
Sample solution is provided at 25 µL, 10mM.
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ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 competitively inhibits ERAP1 activity towards a nonamer peptide representative of physiological substrates[1].
ERAP1-IN-1 allosterically activates ERAP1's hydrolysis of fluorogenic and chromogenic amino acid substratesv[1].ERAP1-IN-1 (50 µM) exhibits specific inhibition of ERAP1 in the cellular context[1].
[1]. Maben Z, et al. Discovery of Selective Inhibitors of Endoplasmic Reticulum Aminopeptidase 1. J Med Chem. 2019 Dec 30.
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