AST2818 mesylate (Synonyms: AST2818) |
Catalog No.GC33096 |
Le mésylate d'alflutinib (furmonertinib) est un puissant inhibiteur de l'EGFR. Le mésylate d'alflutinib (furmonertinib) inhibe les mutations actives de l'EGFR ainsi que la mutation résistante acquise T790M. Le mésylate d'alflutinib (furmonertinib) a le potentiel pour la recherche sur les maladies cancéreuses, en particulier le cancer du poumon non À petites cellules (NSCLC).
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2130958-55-1
Sample solution is provided at 25 µL, 10mM.
AST2818 mesylate is an EGFR inhibitor.
AST2818 mesylate is designed to inhibit EGFR active mutations as well as the T790M acquired resistant mutation[1].
[1]. Y.Shi, et al. P2.03-028 Third Generation EGFR Inhibitor AST2818 (Alflutinib) in NSCLC Patients with EGFR T790M Mutation: A phase1/2 Multi-Center Clinical Trial. J Thorac Oncol. 2017 Nov, 12(11): S2138.
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