Accueil>>Peptides>>Galanin Receptor Ligand M35

Galanin Receptor Ligand M35

Catalog No.GC36102

Galanin Receptor Ligand M35 est un ligand de haute affinité et un antagoniste du récepteur de la galanine (Kd = 0,1 nM).

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Galanin Receptor Ligand M35 Chemical Structure

Cas No.: 142846-71-7

Taille Prix Stock Qté
1mg
180,00 $US
En stock
5mg
540,00 $US
En stock
10mg
900,00 $US
En stock

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Sample solution is provided at 25 µL, 10mM.

Product has been cited by 1 publications

Product Documents

Quality Control & SDS

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Background

Galanin Receptor Ligand M35 is a high-affinity galanin receptor ligand acting as a galanin receptor antagonist in the rat spinal cord, rat hippocampus and isolated mouse pancreatic islets. Galanin Receptor Ligand M35 exerts a Ki values of 0.11 and 2.0 nM for human GalR1 and GalR2, respectively[1][2]. Ki: 0.11 nM (GalR1), 2.0 nM (GalR2)[2]

[1]. Kask K, et al. Binding and agonist/antagonist actions of M35, galanin(1-13)-bradykinin(2-9)amide chimeric peptide, in Rin m 5F insulinoma cells. Regul Pept. 1995 Nov 10;59(3):341-8. [2]. Webling KE, et al. Galanin receptors and ligands. Front Endocrinol (Lausanne). 2012 Dec 7;3:146.

Chemical Properties

Cas No. 142846-71-7 SDF
Formula C107H153N27O26 M.Wt 2233.6
Solubility Soluble in DMSO Storage Store at -20°C
General tips Please select the appropriate solvent to prepare the stock solution according to the solubility of the product in different solvents; once the solution is prepared, please store it in separate packages to avoid product failure caused by repeated freezing and thawing.Storage method and period of the stock solution: When stored at -80°C, please use it within 6 months; when stored at -20°C, please use it within 1 month.
To increase solubility, heat the tube to 37°C and then oscillate in an ultrasonic bath for some time.
Shipping Condition Evaluation sample solution: shipped with blue ice. All other sizes available: with RT, or with Blue Ice upon request.

Complete Stock Solution Preparation Table

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1 mg 5 mg 10 mg
1 mM 0.4477 mL 2.2385 mL 4.4771 mL
5 mM 0.0895 mL 0.4477 mL 0.8954 mL
10 mM 0.0448 mL 0.2239 mL 0.4477 mL
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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO ( Master liquid concentration mg/mL, Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug. )

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Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

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Review for Galanin Receptor Ligand M35

Average Rating: 5 ★★★★★ (Based on Reviews and 27 reference(s) in Google Scholar.)

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