RVD-Hpα TFA |
Catalog No.GC66413 |
RVD-Hpα ; Le TFA est la forme N-terminale étendue de l'hémopressine humaine qui agit comme un agoniste sélectif des récepteurs CB1. RVD-Hpα ; Le TFA augmente les niveaux intracellulaires de Ca2+ dans les cellules exprimant les récepteurs CB1 in vitro. RVD-Hpα ; TFA également modulateur allostérique positif CB2 À haute affinité (Ki = 50 nM).
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Sample solution is provided at 25 µL, 10mM.
RVD-Hpα TFA is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. RVD-Hpα TFA increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. RVD-Hpα TFA also high affinity CB2 positive allosteric modulator (Ki=50 nM).
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