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GSK2018682

Catalog No.GC31863

An S1P1 and S1P5 receptor agonist

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GSK2018682 Chemical Structure

Cas No.: 1034688-30-6

Size Price Stock Qty
10mM (in 1mL DMSO)
$64.00
In stock
5mg
$59.00
In stock
10mg
$90.00
In stock
25mg
$208.00
In stock
50mg
$378.00
In stock
100mg
$675.00
In stock

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Sample solution is provided at 25 µL, 10mM.

Description Chemical Properties Product Documents Related Products

GSK2018682 is an agonist for S1P1 and S1P5 receptor with pEC50s of 7.7 and 7.2, respectively, and has no agonist activity towards human S1P2, S1P3, or S1P4. GSK2018682 is used in the research of multiple sclerosis.

GSK2018682 is an agonist for S1P1 and S1P5 receptor with pEC50s of 7.7 and 7.2, respectively, and has no agonist activity towards human S1P2, S1P3, or S1P4[1].

[1]. Xu J, et al. Safety, pharmacokinetics, pharmacodynamics, and bioavailability of GSK2018682, a sphingosine-1-phosphate receptor modulator, in healthy volunteers. Clin Pharmacol Drug Dev. 2014 May;3(3):170-8.

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Average Rating: 5 ★★★★★ (Based on Reviews and 25 reference(s) in Google Scholar.)

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