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(±)-Indoxacarb (Synonyms: DPX-JW062, DPX-MP062)

カタログ番号GC45985

(±)-インドキサカルブ ((±)-(±)-インドキサカルブ) は、広域スペクトルのオキサジアジン殺虫剤です。

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(±)-Indoxacarb 化学構造

Cas No.: 144171-61-9

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50mg
$34.00
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100mg
$50.00
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Sample solution is provided at 25 µL, 10mM.

Product Documents

Quality Control & SDS

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Background

(±)-Indoxacarb is a broad-spectrum oxadiazine insecticide.1 It is metabolized in vivo to its active N-decarbomethoxyllated metabolite DCJW. Topical administration of (±)-indoxacarb is lethal to S. frugiperda, H. virescens, L. lineolaris, N. cincticeps, N. lugens, L. decemlineata, A. grandis, and M. domestica (LD50s = 0.03, 0.44, 1.6, 0.72, >7.8, 2.81, 6.45, and 15 ng/mg, respectively). It suppresses voltage-gated sodium channel currents in rat dorsal root ganglion neurons in a concentration-dependent manner.2 Formulations containing (±)-indoxacarb have been used to control various insect pests in tea farming.3

|1. Wing, K.D., Sacher, M., Kagaya, Y., et al. Bioactivation and mode of action of the oxadiazine indoxacarb in insects. Crop Prot. 19(8-10), 537-545 (2000).|2. Nagata, K., Ikeda, T., Honda, H., et al. Suppression of voltage-gated sodium currents by the dihydropyrazole insecticide, DPX-JW062 in rat dorsal root ganglion neurons. J. Pesticide Sci. 23(1), 62-64 (1998).|3. Zhang, X., Luo, F., Lou, Z., et al. Simultaneous and enantioselective determination of cis-epoxiconazole and indoxacarb residues in various teas, tea infusion and soil samples by chiral high performance liquid chromatography coupled with tandem quadrupole-time-of-flight mass spectrometry. J. Chromatogr. A 1359, 212-223 (2014).

Chemical Properties

Cas No. 144171-61-9 SDF
同義語 DPX-JW062, DPX-MP062
Canonical SMILES O=C(N(C1=CC=C(OC(F)(F)F)C=C1)C(OC)=O)N2N=C3C(CC4=C3C=CC(Cl)=C4)(C(OC)=O)OC2
Formula C22H17ClF3N3O7 M.Wt 527.8
溶解度 Ethanol: soluble* Storage Store at -20°C
General tips Please select the appropriate solvent to prepare the stock solution according to the solubility of the product in different solvents; once the solution is prepared, please store it in separate packages to avoid product failure caused by repeated freezing and thawing.Storage method and period of the stock solution: When stored at -80°C, please use it within 6 months; when stored at -20°C, please use it within 1 month.
To increase solubility, heat the tube to 37°C and then oscillate in an ultrasonic bath for some time.
Shipping Condition Evaluation sample solution: shipped with blue ice. All other sizes available: with RT, or with Blue Ice upon request.

Complete Stock Solution Preparation Table

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1 mg 5 mg 10 mg
1 mM 1.8947 mL 9.4733 mL 18.9466 mL
5 mM 0.3789 mL 1.8947 mL 3.7893 mL
10 mM 0.1895 mL 0.9473 mL 1.8947 mL
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Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

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Average Rating: 5 ★★★★★ (Based on Reviews and 36 reference(s) in Google Scholar.)

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