Citrullination
Products for Citrullination
- Cat.No. 상품명 정보
- GC48495 BMS-P5 BMS-P5는 특이적 경구 활성 펩티딜아르기닌 데이미나제 4(PAD4) 억제제입니다. BMS-P5는 동계 마우스 모델에서 MM 유도 NET 형성을 차단하고 MM의 진행을 지연시킵니다.
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GC43202
CAY10723
CAY10723는 강력한 단백질 아르기닌 디미나아제 2 (PAD2) 억제제이며, 우수한 PAD2 선택성을 가지고 있습니다.
- GC47050 CAY10727 A PAD3 inhibitor
- GC52351 Citrullinated α-Enolase (R8 + R14) (1-19)-biotin Peptide A biotinylated and citrullinated α-enolase peptide
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GC52363
Citrullinated Histone H3 (R2 + R8 + R17) (2-22)-biotin Peptide
A biotinylated and citrullinated histone H3 peptide
- GC52367 Citrullinated Vimentin (G146R) (R144 + R146) (139-159)-biotin Peptide A biotinylated and citrullinated mutant vimentin peptide
- GC52370 Citrullinated Vimentin (R144) (139-159)-biotin Peptide A biotinylated and citrullinated vimentin peptide
- GC43275 Citrulline-specific Probe-Rhodamine Protein arginine deiminases (PADs) catalyze the posttranslational modification of arginine residues on proteins to form citrulline, which plays a large role in regulating gene expression.
- GC43651 F-Amidine (trifluoroacetate salt) F-amidine is an inhibitor of protein arginine deiminases (PADs) that is selective for PAD1 and PAD4 (IC50s = 29.5, 350, and 21.6 μM for PAD1, PAD3, and PAD4 in vitro, respectively).
- GC43787 GSK106 (hydrochloride) GSK106(염산염)은 선택적 PAD4 억제제인 GSK484 및 GSK199에 대한 비활성 대조군입니다.
- GC43788 GSK121 (trifluoroacetate salt) GSK-121 트리플루오로아세테이트는 선택적 PAD4 억제제입니다.
- GC43789 GSK199 (hydrochloride) GSK199(염산염)는 칼슘이 없을 때 IC50이 200nM인 가역적이고 선택적 PAD4 억제제입니다.
- GC45548 Photoswitchable PAD Inhibitor (technical grade)
- GC52364 Vimentin (139-159)-biotin Peptide A biotinylated vimentin peptide
- GC52371 Vimentin (G146R) (139-159)-biotin Peptide A biotinylated mutant vimentin peptide