Citrullination
Products for Citrullination
- Cat.No. 상품명 정보
-
GC48495
BMS-P5
BMS-P5는 특이적 경구 활성 펩티딜아르기닌 데이미나제 4(PAD4) 억제제입니다. BMS-P5는 동계 마우스 모델에서 MM 유도 NET 형성을 차단하고 MM의 진행을 지연시킵니다.
-
GC43202
CAY10723
AFM30a, AMF30a
CAY10723는 강력한 단백질 아르기닌 디미나아제 2 (PAD2) 억제제이며, 우수한 PAD2 선택성을 가지고 있습니다.
-
GC90710
CAY10723 (hydrochloride)
PAD2 억제제
-
GC47050
CAY10727
A PAD3 inhibitor
-
GC45402
CAY10729 (trifluoroacetate salt) (technical grade)
-
GC52351
Citrullinated α-Enolase (R8 + R14) (1-19)-biotin Peptide
Citrullinated Enolase-1-biotin, α-Enolase Peptide (Citrulline Residues 8 + 14)
A biotinylated and citrullinated α-enolase peptide -
GC52363
Citrullinated Histone H3 (R2 + R8 + R17) (2-22)-biotin Peptide
Biotin-A-Cit-TKQTA-Cit-KSTGGKAP-Cit-KQLA, Biotin-AXTKQTAXKSTGGKAPXKQLA (X=Citrulline), Citrullinated Histone H3.1-biotin
A biotinylated and citrullinated histone H3 peptide
-
GC52367
Citrullinated Vimentin (G146R) (R144 + R146) (139-159)-biotin Peptide
Biotin-GQGKS(Cit)L(Cit)DLYEEEMRELRRQ, Biotin-GQGKSXLXDLYEEEMRELRRQ (X=Citrulline), Citrullinated VIM (G146R) (R144 + R146)-biotin
A biotinylated and citrullinated mutant vimentin peptide -
GC52370
Citrullinated Vimentin (R144) (139-159)-biotin Peptide
Biotin-GQGKS(Cit)LGDLYEEEMRELRRQ, Biotin-GQGKSXLGDLYEEEMRELRRQ (X=Citrulline), Citrullinated VIM (R144)-biotin
A biotinylated and citrullinated vimentin peptide -
GC40255
Citrulline-specific Probe-biotin
Citrulline-specific probe-biotin is an affinity probe that allows for detection or immobilization of citrullinated proteins through interaction with the biotin ligand.
-
GC43275
Citrulline-specific Probe-Rhodamine
Rhodamine Phenylglyoxal, RhPG
Protein arginine deiminases (PADs) catalyze the posttranslational modification of arginine residues on proteins to form citrulline, which plays a large role in regulating gene expression. -
GC43651
F-Amidine (trifluoroacetate salt)
F-amidine is an inhibitor of protein arginine deiminases (PADs) that is selective for PAD1 and PAD4 (IC50s = 29.5, 350, and 21.6 μM for PAD1, PAD3, and PAD4 in vitro, respectively).
-
GC43787
GSK106 (hydrochloride)
GSK106(염산염)은 선택적 PAD4 억제제인 GSK484 및 GSK199에 대한 비활성 대조군입니다.
-
GC43788
GSK121 (trifluoroacetate salt)
GSK-121 트리플루오로아세테이트는 선택적 PAD4 억제제입니다.
-
GC43789
GSK199 (hydrochloride)
GSK199(염산염)는 칼슘이 없을 때 IC50이 200nM인 가역적이고 선택적 PAD4 억제제입니다.
-
GC91565
GSK199 analog (hydrochloride)
GSK199 analog is an inhibitor of peptidyl arginine deiminase 4 (PAD4) and a derivative of the PAD4 inhibitor GSK199.
-
GC45548
Photoswitchable PAD Inhibitor (technical grade)
-
GC45005
TDFA (trifluoroacetate salt)
Thr-Asp-F-amidine
-
GC52364
Vimentin (139-159)-biotin Peptide
VIM (139-159)-biotin
A biotinylated vimentin peptide -
GC52371
Vimentin (G146R) (139-159)-biotin Peptide
Biotin-GQGKSRLRDLYEEEMRELRRQ, Biotin-GQGKSRLRDLYEEEMRELRRQ (X=Citrulline), VIM (G146R) (139-159)-biotin
A biotinylated mutant vimentin peptide