>> Signaling Pathways >> Chromatin/Epigenetics >> Citrullination

Citrullination

Products for  Citrullination

  1. Cat.No. 상품명 정보
  2. GC48495 BMS-P5 BMS-P5는 특이적 경구 활성 펩티딜아르기닌 데이미나제 4(PAD4) 억제제입니다. BMS-P5는 동계 마우스 모델에서 MM 유도 NET 형성을 차단하고 MM의 진행을 지연시킵니다. BMS-P5  Chemical Structure
  3. GC43202 CAY10723

    AFM30a, AMF30a

    CAY10723는 강력한 단백질 아르기닌 디미나아제 2 (PAD2) 억제제이며, 우수한 PAD2 선택성을 가지고 있습니다.

    CAY10723  Chemical Structure
  4. GC90710 CAY10723 (hydrochloride)

    PAD2 억제제

    CAY10723 (hydrochloride)  Chemical Structure
  5. GC47050 CAY10727 A PAD3 inhibitor CAY10727  Chemical Structure
  6. GC45402 CAY10729 (trifluoroacetate salt) (technical grade)   CAY10729 (trifluoroacetate salt) (technical grade)  Chemical Structure
  7. GC52351 Citrullinated α-Enolase (R8 + R14) (1-19)-biotin Peptide

    Citrullinated Enolase-1-biotin, α-Enolase Peptide (Citrulline Residues 8 + 14)

    A biotinylated and citrullinated α-enolase peptide Citrullinated α-Enolase (R8 + R14) (1-19)-biotin Peptide  Chemical Structure
  8. GC52363 Citrullinated Histone H3 (R2 + R8 + R17) (2-22)-biotin Peptide

    Biotin-A-Cit-TKQTA-Cit-KSTGGKAP-Cit-KQLA, Biotin-AXTKQTAXKSTGGKAPXKQLA (X=Citrulline), Citrullinated Histone H3.1-biotin

    A biotinylated and citrullinated histone H3 peptide

    Citrullinated Histone H3 (R2 + R8 + R17) (2-22)-biotin Peptide  Chemical Structure
  9. GC52367 Citrullinated Vimentin (G146R) (R144 + R146) (139-159)-biotin Peptide

    Biotin-GQGKS(Cit)L(Cit)DLYEEEMRELRRQ, Biotin-GQGKSXLXDLYEEEMRELRRQ (X=Citrulline), Citrullinated VIM (G146R) (R144 + R146)-biotin

    A biotinylated and citrullinated mutant vimentin peptide Citrullinated Vimentin (G146R) (R144 + R146) (139-159)-biotin Peptide  Chemical Structure
  10. GC52370 Citrullinated Vimentin (R144) (139-159)-biotin Peptide

    Biotin-GQGKS(Cit)LGDLYEEEMRELRRQ, Biotin-GQGKSXLGDLYEEEMRELRRQ (X=Citrulline), Citrullinated VIM (R144)-biotin

    A biotinylated and citrullinated vimentin peptide Citrullinated Vimentin (R144) (139-159)-biotin Peptide  Chemical Structure
  11. GC40255 Citrulline-specific Probe-biotin

    Citrulline-specific probe-biotin is an affinity probe that allows for detection or immobilization of citrullinated proteins through interaction with the biotin ligand.

    Citrulline-specific Probe-biotin  Chemical Structure
  12. GC43275 Citrulline-specific Probe-Rhodamine

    Rhodamine Phenylglyoxal, RhPG

    Protein arginine deiminases (PADs) catalyze the posttranslational modification of arginine residues on proteins to form citrulline, which plays a large role in regulating gene expression. Citrulline-specific Probe-Rhodamine  Chemical Structure
  13. GC43651 F-Amidine (trifluoroacetate salt) F-amidine is an inhibitor of protein arginine deiminases (PADs) that is selective for PAD1 and PAD4 (IC50s = 29.5, 350, and 21.6 μM for PAD1, PAD3, and PAD4 in vitro, respectively). F-Amidine (trifluoroacetate salt)  Chemical Structure
  14. GC43787 GSK106 (hydrochloride) GSK106(염산염)은 선택적 PAD4 억제제인 GSK484 및 GSK199에 대한 비활성 대조군입니다. GSK106 (hydrochloride)  Chemical Structure
  15. GC43788 GSK121 (trifluoroacetate salt) GSK-121 트리플루오로아세테이트는 선택적 PAD4 억제제입니다. GSK121 (trifluoroacetate salt)  Chemical Structure
  16. GC43789 GSK199 (hydrochloride) GSK199(염산염)는 칼슘이 없을 때 IC50이 200nM인 가역적이고 선택적 PAD4 억제제입니다. GSK199 (hydrochloride)  Chemical Structure
  17. GC91565 GSK199 analog (hydrochloride) GSK199 analog is an inhibitor of peptidyl arginine deiminase 4 (PAD4) and a derivative of the PAD4 inhibitor GSK199. GSK199 analog (hydrochloride)  Chemical Structure
  18. GC45548 Photoswitchable PAD Inhibitor (technical grade)   Photoswitchable PAD Inhibitor (technical grade)  Chemical Structure
  19. GC45005 TDFA (trifluoroacetate salt)

    Thr-Asp-F-amidine

    TDFA (trifluoroacetate salt)  Chemical Structure
  20. GC52364 Vimentin (139-159)-biotin Peptide

    VIM (139-159)-biotin

    A biotinylated vimentin peptide Vimentin (139-159)-biotin Peptide  Chemical Structure
  21. GC52371 Vimentin (G146R) (139-159)-biotin Peptide

    Biotin-GQGKSRLRDLYEEEMRELRRQ, Biotin-GQGKSRLRDLYEEEMRELRRQ (X=Citrulline), VIM (G146R) (139-159)-biotin

    A biotinylated mutant vimentin peptide Vimentin (G146R) (139-159)-biotin Peptide  Chemical Structure

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