PAK-IN-1 |
| Catalog No.GC33421 |
PAK-IN-1 is a PAK inhibitor that displays group II selectivity. PAK-IN-1 inhibits PAK4, PAK5 and PAK6 with IC50s of 7.5, 36, 126 nM, respectively.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1394121-05-1
Sample solution is provided at 25 µL, 10mM.
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PAK-IN-1 is a PAK inhibitor that displays group II selectivity. PAK-IN-1 inhibits PAK4, PAK5 and PAK6 with IC50s of 7.5, 36, 126 nM, respectively.
PAK-IN-1 is compound 4 from the reference[1].
[1]. Karpov AS, et al. Optimization of a Dibenzodiazepine Hit to a Potent and Selective Allosteric PAK1 Inhibitor. ACS Med Chem Lett. 2015 May 22;6(7):776-81.
Average Rating: 5 (Based on Reviews and 21 reference(s) in Google Scholar.)
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