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Home >> Signaling Pathways >> Angiogenesis >> PAR1

PAR1

PAR1 (protease-activated receptor 1) is a subfamily of related G protein-coupled receptors that are activated by cleavage of part of their extracellular domain.

Products for  PAR1

  1. Cat.No. Product Name Information
  2. GC17368 2-Furoyl-LIGRLO-amide Protease-activated receptor agonist 2-Furoyl-LIGRLO-amide Chemical Structure
  3. GC38731 2-Furoyl-LIGRLO-amide TFA 2-Furoyl-LIGRLO-amide TFA is a potent and selective proteinase-activated receptor 2 (PAR2) agonist with a pD2 value of 7.0. 2-Furoyl-LIGRLO-amide TFA Chemical Structure
  4. GC14831 AC 264613 PAR2 agonist,potent and selective AC 264613 Chemical Structure
  5. GC15290 AC 55541 PAR2 agonist,potent and selective AC 55541 Chemical Structure
  6. GC63658 Atopaxar Atopaxar (E5555) is a potent, orally active, selective and reversible thrombin receptor protease-activated receptor-1 (PAR-1) antagonist. Atopaxar Chemical Structure
  7. GC18152 AZ-3451

    A potent, and selective PAR2 antagonist with Kd of 13.5 nM.

     AZ-3451 Chemical Structure
  8. GC65312 AZ8838 AZ8838 is a potent, competitive, allosteric, orally active non-peptide small molecule antagonist of PAR2 with a pKi of 6.4 for hPAR2. AZ8838 Chemical Structure
  9. GC18717 BMS 986120 A selective PAR4 antagonist BMS 986120 Chemical Structure
  10. GC60807 ENMD-1068 hydrochloride

    6-Amino-1-[4-(3-methyl-1-oxobutyl)-1-piperazinyl]-1-hexanone hydrochloride

     Selective protease-activated receptor 2 (PAR2) anatagonist ENMD-1068 hydrochloride Chemical Structure
  11. GC61501 FSLLRY-NH2 TFA FSLLRY-NH2 TFA is a protease-activated receptor 2 (PAR2) inhibitor. FSLLRY-NH2 TFA Chemical Structure
  12. GC36125 GB-110 GB-110 is a potent, orally active, and nonpeptidic protease activated receptor 2 (PAR2) agonist. GB-110 Chemical Structure
  13. GC38329 GB-110 hydrochloride GB-110 hydrochloride is a potent, orally active, and nonpeptidic protease activated receptor 2 (PAR2) agonist. GB-110 hydrochloride Chemical Structure
  14. GC65439 GB-88 GB-88 is an oral, selective non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 ?M. GB-88 Chemical Structure
  15. GC64979 I-191 I-191 is a potent, selective protease-activated receptor 2 (PAR2) antagonist. I-191 Chemical Structure
  16. GC13227 LRGILS-NH2 Protease-activated receptor agonist LRGILS-NH2 Chemical Structure
  17. GC11951 PAR 4 (1-6)

    GYPGQV

    PAR4 agonist

     PAR 4 (1-6) Chemical Structure
  18. GC62101 PAR-2-IN-1 PAR-2-IN-1 is a protease-activated receptor-2 (PAR2) signaling pathway inhibitor with anti-inflammatory and anticancer effects. PAR-2-IN-1 Chemical Structure
  19. GA23350 PAR-3 (1-6) amide (human) PAR-3 (1-6) amide (human) is a proteinase-activated receptor (PAR-3) agonist peptide. PAR-3 (1-6) amide (human) Chemical Structure
  20. GC33599 PAR-4 Agonist Peptide, amide TFA (PAR-4-AP (TFA))

    PAR-4-AP TFA; AY-NH2 TFA

     PAR-4 agonist peptide, amide TFA (PAR-4-AP (TFA)) is a synthetic peptide primarily used to activate protease-activated receptor 4 (PAR-4) . PAR-4 Agonist Peptide, amide TFA (PAR-4-AP (TFA)) Chemical Structure
  21. GC15817 PAR-4 Agonist Peptide, amide (AY-NH2)

    PAR-4-AP; AY-NH2

     PAR-4 Agonist Peptide, amide(AY-NH2) (PAR-4-AP; AY-NH2) is a proteinase-activated receptor-4 (PAR-4) agonist, which has no effect on either PAR-1 or PAR-2 and whose effects are blocked by a PAR-4 antagonist. PAR-4 Agonist Peptide, amide (AY-NH2) Chemical Structure
  22. GC38134 Parmodulin 2 Reversible inhibitor of PAR1mediated platelet activation Parmodulin 2 Chemical Structure
  23. GC69663 Parstatin(mouse) TFA

    Parstatin (mouse) TFA is a peptide agonist of the PAR-1 thrombin receptor with cell-penetrating properties and an effective inhibitor of angiogenesis.

     Parstatin(mouse) TFA Chemical Structure
  24. GC69768 Protease-Activated Receptor-1, PAR-1 Agonist

    Protease-Activated Receptor-1, PAR-1 Agonist is a selective peptide that activates Protease-Activated Receptor-1 (PAR-1), which corresponds to the PAR1 ligand and selectively mimics the action of thrombin through this receptor.

     Protease-Activated Receptor-1, PAR-1 Agonist Chemical Structure
  25. GC62469 Protease-Activated Receptor-1, PAR-1 Agonist TFA Protease-Activated Receptor-1, PAR-1 Agonist TFA is a selective proteinase-activated receptor1 (PAR-1) agonist peptide. Protease-Activated Receptor-1, PAR-1 Agonist TFA corresponds to PAR1 tethered ligand and which can selectively mimic theactions of thrombin via this receptor. Protease-Activated Receptor-1, PAR-1 Agonist TFA Chemical Structure
  26. GC61456 Protease-Activated Receptor-3 (PAR-3) (1-6), human TFA Protease-Activated Receptor-3 (PAR-3) (1-6), human TFA is a proteinase-activated receptor (PAR-3) agonist peptide. Protease-Activated Receptor-3 (PAR-3) (1-6), human TFA Chemical Structure
  27. GC33429 Protease-Activated Receptor-4 Protease-Activated Receptor-4 is the agonist of proteinase-activated receptor-4 (PAR4). Protease-Activated Receptor-4 Chemical Structure
  28. GC17991 RLLFT-NH2 Protease-activated receptor agonist RLLFT-NH2 Chemical Structure
  29. GC61777 RWJ-56110 dihydrochloride RWJ-56110 dihydrochloride is a potent, selective, peptide-mimetic inhibitor of PAR-1 activation and internalization (binding IC50=0.44 uM) and shows no effect on PAR-2, PAR-3, or PAR-4. RWJ-56110 dihydrochloride Chemical Structure
  30. GC10291 SCH 79797 dihydrochloride PAR1 receptor antagonist SCH 79797 dihydrochloride Chemical Structure
  31. GC63540 SCH79797 SCH79797 is a highly potent, selective nonpeptide protease activated receptor 1 (PAR1) antagonist. SCH79797 Chemical Structure
  32. GC14540 SLIGKV-NH2 SLIGKV-NH2 (SLIGKV-NH2) is a highly potent protease-activated receptor-2 (PAR2) activating peptide. SLIGKV-NH2 Chemical Structure
  33. GC17514 SLIGRL-NH2

    Protease-Activated Receptor-2 Activating Peptide

     PAR2 activator SLIGRL-NH2 Chemical Structure
  34. GC61316 tcY-NH2 TFA

    (trans-Cinnamoyl)-YPGKF-NH2 TFA

     tcY-NH2 ((trans-Cinnamoyl)-YPGKF-NH2) TFA is a potent selective PAR4 antagonist peptide. tcY-NH2 TFA Chemical Structure
  35. GC17444 TFLLR-NH2 PAR1 selective agonist TFLLR-NH2 Chemical Structure
  36. GC37770 TFLLR-NH2(TFA) TFLLR-NH2 (TFA) is a selective PAR1 agonist with an EC50 of 1.9 μM. TFLLR-NH2(TFA) Chemical Structure
  37. GP10085 Thrombin Receptor Activator for Peptide 5 (TRAP-5)

    H2N-Ser-Phe-Leu-Leu-Arg-OH

    Thrombin Receptor Activator for Peptide 5 (TRAP-5) Chemical Structure
  38. GC10140 Thrombin Receptor Agonist Peptide Thrombin Receptor Agonist Peptide is a synthetic thrombin receptor agonist peptide. Thrombin Receptor Agonist Peptide Chemical Structure
  39. GC11662 TRAP-6

    PAR-1 agonist peptide; Thrombin Receptor Activator Peptide 6

    PAR1 agonist

     TRAP-6 Chemical Structure
  40. GC65529 TRAP-6 amide TRAP-6 amide is a PAR-1 thrombin receptor agonist peptide. TRAP-6 amide Chemical Structure
  41. GC37852 UDM-001651 UDM-001651 is a potent, selective, and orally bioavailable protease-activated receptor 4 (PAR4) antagonist (IC50=4 nM; Kd=1.4 nM). UDM-001651 Chemical Structure
  42. GC11727 VKGILS-NH2 control peptide for SLIGKV-NH2, PAR1 agonist VKGILS-NH2 Chemical Structure
  43. GC17545 Vorapaxar PAR-1 antagonist,potent and orally active Vorapaxar Chemical Structure
  44. GC64347 Vorapaxar sulfate Vorapaxar sulfate (SCH 530348 sulfate), an antiplatelet agent, is a selective, orally active, and competitive thrombin receptor protease-activated receptor (PAR-1) antagonist (Ki=8.1 nM). Vorapaxar sulfate Chemical Structure

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