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VDA

VDAs (vascular disrupting agents) target established tumor vasculature and lead to blood vessels shutdown and selective tumor necrosis.

Products for  VDA

  1. Cat.No. Product Name Information
  2. GC10235 Plinabulin (NPI-2358) Plinabulin (NPI-2358) (NPI-2358) is a vascular disrupting agen (VDA) against tubulin-depolymerizing with an IC50 of 9.8 nM against HT-29 cells. Plinabulin (NPI-2358) binds the colchicine binding site of β-tubulin preventing polymerization and has potent inhibitory to tumor cells. Plinabulin (NPI-2358)  Chemical Structure

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