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Home >> Signaling Pathways >> Neuroscience >> GABA Receptor

GABA Receptor

GABA receptors are a class of receptors that respond to the GABA (neurotransmitter gamma-aminobutyric acid), the chief inhibitory neurotransmitter in the vertebrate central nervous system.

Products for  GABA Receptor

  1. Cat.No. Product Name Information
  2. GN10251 Ginkgolide A Ginkgolide A Chemical Structure
  3. GN10254 Ginsenoside Rc Ginsenoside Rc Chemical Structure
  4. GC11303 GS 39783 Positive allosteric modulator of GABAB receptor GS 39783 Chemical Structure
  5. GC60890 Guvacine Guvacine, an alkaloid found in the nut of Areca catechu, is a potent GABA uptakp inhibitor. Guvacine Chemical Structure
  6. GC14659 Guvacine hydrochloride GABA uptake inhibitor Guvacine hydrochloride Chemical Structure
  7. GA10004 H-D-Met-OH H-D-Met-OH Chemical Structure
  8. GA10664 H-Dab?HBr H-Dab?HBr Chemical Structure
  9. GC12359 Hispidulin Partial positive allosteric modulator at the benzodiazepine receptor Hispidulin Chemical Structure
  10. GC63950 Homocarnosine TFA Homocarnosine TFA is a dipeptide of γ-aminobutyric acid (GABA) and histidine unique to brain. Homocarnosine TFA Chemical Structure
  11. GC13567 Isoguvacine hydrochloride

    GABAA receptor agonist

     Isoguvacine hydrochloride Chemical Structure
  12. GC25531 Isonipecotic acid Isonipecotic acid (4-Piperidinecarboxylic acid, 4-Carboxypiperidine, Hexahydroisonicotinic acid) is a heterocyclic compound that mainly acts as a GABAA receptor partial agonist. Isonipecotic acid Chemical Structure
  13. GN10086 Jujuboside A Jujuboside A Chemical Structure
  14. GC17350 L-655,708 inverse agonist for the benzodiazepine site of GABAA receptors containing the α5 subunit L-655,708 Chemical Structure
  15. GC11597 L-838,417 Subtype-selective GABAA receptor partial agonist L-838,417 Chemical Structure
  16. GC30862 L-Cycloserine ((S)-4-Amino-3-isoxazolidone) L-Cycloserine ((S)-4-Amino-3-isoxazolidone) ((S)-4-Amino-3-isoxazolidone) irreversibly inhibits GABA pyridoxal 5′-phosphate-dependent aminitransferase in E. L-Cycloserine ((S)-4-Amino-3-isoxazolidone) Chemical Structure
  17. GC25566 L-DAB HBR L-DAB HBR Chemical Structure
  18. GC44040 LAU159 A positive allosteric modulator of α6β3γ2 subunit-containing GABAA receptors LAU159 Chemical Structure
  19. GC61624 Lesogaberan Lesogaberan (AZD-3355) is a potent and selective GABAB receptor agonist with an EC50 of 8.6 nM for human recombinant GABAB receptors. Lesogaberan Chemical Structure
  20. GC63041 Lesogaberan hydrochloride Lesogaberan (AZD-3355) hydrochloride is a potent and selective GABAB receptor agonist with an EC50 of 8.6 nM for human recombinant GABAB receptor. Lesogaberan hydrochloride Chemical Structure
  21. GC14045 Loreclezole GABAA receptor modulator Loreclezole Chemical Structure
  22. GC18299 Lorediplon Lorediplon is a ligand for α1 subunit-containing GABAA receptors. Lorediplon Chemical Structure
  23. GC65292 Lotilaner Lotilaner is a parasiticide, acts as a potent non-competitive antagonist of insects GABACl receptors, with an IC50 of 23.84 nM for Drosophila melanogaster GABA receptor. Lotilaner Chemical Structure
  24. GC13715 MK 0343 GABAA partial agonist MK 0343 Chemical Structure
  25. GC16528 MRK 016 GABAA receptor inverse agonist MRK 016 Chemical Structure
  26. GC69495 MRK-898

    MRK-898 is an orally effective GABA(A) receptor modulator. MRK-898 binds to the α1, α2, α3 and α5 subunits of the GABA receptor with Ki values of 1.2 nM, 1.0 nM, 0.73 nM and 0.50 nM respectively. However, GABA(A) receptors containing the α1 subunit have been identified as "sedative" receptors while those containing the α2 and/or α3 subunits have been identified as "anxiolytic" subtypes.

     MRK-898 Chemical Structure
  27. GC16353 N-ArachidonylGABA arachidonyl amino acid N-ArachidonylGABA Chemical Structure
  28. GC12169 NCS-382 γ-Hydroxybutyric acid antagonist NCS-382 Chemical Structure
  29. GC11901 Nefiracetam GABA receptor activator Nefiracetam Chemical Structure
  30. GC31018 NEO 376 (SPI-376) NEO 376 (SPI-376) is a selective modulator of 5-HT1 receptor, GABA receptor and dopamine receptor, with anti-psychotic actively. NEO 376 (SPI-376) Chemical Structure
  31. GC16564 Niflumic acid Ca2+-activated Cl- channel blocker Niflumic acid Chemical Structure
  32. GC11821 NNC 05-2090 hydrochloride

    GABA uptake inhibitor

     NNC 05-2090 hydrochloride Chemical Structure
  33. GC11748 NNC 711 NNC-711 (hydrochloride) is a potent and selective inhibitor of GAT-1 ( GABA transporter 1) with an IC50 of 40 nM for hGAT-1. NNC 711 Chemical Structure
  34. GC11143 NS 11394 GABA(A) receptor-positive modulator NS 11394 Chemical Structure
  35. GC16024 Ocinaplon GABAA receptors modulator Ocinaplon Chemical Structure
  36. GC19271 ONO-8590580 ONO-8590580 is a GABAA α5 negative allosteric modulator. ONO-8590580 Chemical Structure
  37. GC14329 Org 20599 GABAA receptor agonist Org 20599 Chemical Structure
  38. GC11963 Oxiracetam cyclic derivative of gamma-aminobutyric acid (GABA) Oxiracetam Chemical Structure
  39. GC31282 p-Hydroxybenzaldehyde p-Hydroxybenzaldehyde is a one of the major components in Dendrocalamus asper bamboo shoots, with antagonistic effect on GABAA receptor of the α1β2γ2S subtype at high concentrations. p-Hydroxybenzaldehyde Chemical Structure
  40. GC12357 Pentylenetetrazole CNS stimulant Pentylenetetrazole Chemical Structure
  41. GC63145 PF-06372865 PF-06372865 is an orally active, α2/α3/α5 subtype-selective GABAA positive allosteric modulator (PAM). PF-06372865 Chemical Structure
  42. GC17691 Phaclofen

    GABAB antagonist

     Phaclofen Chemical Structure
  43. GC63146 Phenibut Phenibut Chemical Structure
  44. GC13557 PHP 501 trifluoroacetate GABAA antagonist PHP 501 trifluoroacetate Chemical Structure
  45. GC61186 Picrotoxinin Picrotoxinin, a potent convulsant, is a chloride channel blocker. Picrotoxinin Chemical Structure
  46. GC30827 Pipequaline (PK-8165) Pipequaline (PK-8165) (PK 8165) is a partial benzodiazepine receptor agonist with anxiolytic activity. Pipequaline (PK-8165) Chemical Structure
  47. GC16569 PK 11195

    peripheral benzodiazepine antagonist

     PK 11195 Chemical Structure
  48. GC17399 Pregnanolone

    GABAA receptor positive allosteric modulator

     Pregnanolone Chemical Structure
  49. GC15960 Primidone anticonvulsant of the pyrimidinedione class Primidone Chemical Structure
  50. GC39424 Propofol

    Propofol potently and directly activates GABAA receptor and inhibits glutamate receptor mediated excitatory synaptic transmission.

     Propofol Chemical Structure
  51. GC65057 Propofol-d18 Propofol-d18 is the deuterium labeled Propofol. Propofol-d18 Chemical Structure
  52. GC50375 PZ-II-029 α6β3γ2-selective GABAA positive allosteric modulator PZ-II-029 Chemical Structure
  53. GC16476 rac BHFF GABAB receptor positive allosteric modulator rac BHFF Chemical Structure
  54. GC65513 Radequinil Radequinil (AC-3933) is a benzodiazepine receptor (BzR) partial inverse agonist. Radequinil Chemical Structure
  55. GC12599 Retigabine dihydrochloride An Analytical Reference Standard Retigabine dihydrochloride Chemical Structure
  56. GC31257 Rilmazafone hydrochloride (450191S) Rilmazafone hydrochloride (450191S) (450191S) is a benzodiazepine (omega) ligand. Rilmazafone hydrochloride (450191S) Chemical Structure
  57. GC13802 Riluzole Sodium channel protein inhibitor Riluzole Chemical Structure
  58. GC44841 Riluzole (hydrochloride) Riluzole is a benzothiazole derivative with anti-excitotoxic effects that acts by blocking the presynaptic release of glutamate, indirectly antagonizing glutamate receptors, and inactivating neuronal voltage-gated Na+ channels (ED50 = 2.3 μM). Riluzole (hydrochloride) Chemical Structure
  59. GC16780 Ro 15-4513 benzodiazepine ligand Ro 15-4513 Chemical Structure
  60. GC12377 Ro 19-4603 Benzodiazepine inverse agonist Ro 19-4603 Chemical Structure
  61. GC37547 Ro 41-3290 Ro 41-3290 is the desethylated derivative of Ro 41-3696, which is a nonbenzodiazepine partial agonist at the benzodiazepine receptor. Ro 41-3290 Chemical Structure
  62. GC30433 Ru-32514 Ru-32514 is an agonist of benzodiazepine receptor. Ru-32514 Chemical Structure
  63. GC11612 RuBi GABA trimethylphosphine GABAB receptor agonist RuBi GABA trimethylphosphine Chemical Structure
  64. GC17321 RuBi-GABA Ruthenium-bipyridine-triphenylphosphine caged GABA RuBi-GABA Chemical Structure
  65. GC13792 Rufinamide voltage-gated sodium channel blocker Rufinamide Chemical Structure
  66. GC31049 RWJ-51204 RWJ-51204 is a partial agonist of GABA(A) receptor, with Ki of 0.2-2 nM to the benzodiazepine site on GABA(A) receptors. RWJ-51204 Chemical Structure
  67. GC31121 S-8510 phosphate (SB-737552 phosphate) S-8510 (phosphate) is an inverse Benzodiazepine (BDZ) receptor agonist, with Kis of 34.6 nM, 36.2 nM for -GABA and +GABA respectively. S-8510 phosphate (SB-737552 phosphate) Chemical Structure
  68. GC17257 Saclofen GABAB receptor antagonist Saclofen Chemical Structure
  69. GC31112 Sarmazenil (Ro 15-3505) Sarmazenil (Ro 15-3505) is a benzodiazepine receptor antagonist. Sarmazenil (Ro 15-3505) Chemical Structure
  70. GC16356 SB 205384 positive GABAA receptor modulator SB 205384 Chemical Structure
  71. GC10888 SCH 50911 GABAB antagonist SCH 50911 Chemical Structure
  72. GC10844 SCS GABAA receptor antagonist SCS Chemical Structure
  73. GC69905 SJM-3

    SJM-3 is a positive allosteric modulator of different subtypes of GABAA receptors. SJM-3 binds with high affinity to the α+/γ- subunit interface of the benzodiazepine binding site.

     SJM-3 Chemical Structure
  74. GC15226 SKF 89976A hydrochloride GABA uptake inhibitor SKF 89976A hydrochloride Chemical Structure
  75. GC14942 SKF 97541 GABAB agonist SKF 97541 Chemical Structure
  76. GC10101 SR 95531 hydrobromide SR 95531 hydrobromide is a selective and competitive antagonist of GABAA receptor, with an IC50 of ~0.2 μM for GABA receptor. SR 95531 hydrobromide Chemical Structure
  77. GC34362 SSD114 hydrochloride SSD114 hydrochloride is a novel GABAB receptor positive allosteric modulator. SSD114 hydrochloride Chemical Structure
  78. GC31196 SX-3228 SX-3228 is a selective benzodiazepine1 (BZ1) receptor agonist with an IC50 of 17 nM. SX-3228 Chemical Structure
  79. GC10967 TACA GABAA agonist TACA Chemical Structure
  80. GC17934 TB 21007 GABAA receptor inverse agonist TB 21007 Chemical Structure
  81. GC15859 TCS 1105 GABAA benzodiazepine receptor (BZR) ligand TCS 1105 Chemical Structure
  82. GC10741 TCS 1205 TCS 1205 (compound 2b) is a potent and selective GABAA agonist. TCS 1205 Chemical Structure
  83. GC63218 Tetrahydrodeoxycorticosterone Tetrahydrodeoxycorticosterone, an neurosteroid, is a potent positive allosteric modulator (PAM) of GABAA receptor. Tetrahydrodeoxycorticosterone Chemical Structure
  84. GC45961 THDOC THDOC (THDOC), an endogenous neurosteroid, is a positive modulator of GABAA receptors. THDOC Chemical Structure
  85. GC39126 Thiocolchicoside Thiocolchicoside is a competitive γ-aminobutyric acid type A (GABAA) receptor antagonist and glycine receptor agonist in the central nervous system. Thiocolchicoside Chemical Structure
  86. GC37784 THIP THIP (Gaboxadol) is a selective extrasynaptic GABAA receptors (eGABARs) agonist (with blood-brain barrier permeability), shows an EC50 value of 13 ?M for δ-GABAAR. THIP Chemical Structure
  87. GC10856 THIP hydrochloride THIP hydrochloride (Lu 02-030 hydrochloride) is a potent agonist of the GABAA receptor and an antagonist of GABAC receptors (IC50=25 μM). THIP hydrochloride Chemical Structure
  88. GC38215 Tiagabine Tiagabine Chemical Structure
  89. GC10186 Tiagabine selective gamma-aminobutyric acid (GABA) reuptake inhibitor Tiagabine Chemical Structure
  90. GC17402 Tiagabine hydrochloride

    GABA uptake inhibitor

     Tiagabine hydrochloride Chemical Structure
  91. GC37788 Tiagabine hydrochloride hydrate Tiagabine hydrochloride hydrate is a potent and selective GABA uptake inhibitor, used as an anticonvulsant agent, with IC50s of 67, 446 and 182 nM for [3H]GABA uptake in Synaptosomes, Neurons and Glia, respectively. Tiagabine hydrochloride hydrate Chemical Structure
  92. GC16149 Topiramate An anticonvulsant Topiramate Chemical Structure
  93. GC50198 Topiramate - d12 Deuterated topiramate Topiramate - d12 Chemical Structure
  94. GC16360 TP 003 GABAA receptor (α3 subtype) partial agonist TP 003 Chemical Structure
  95. GC30865 TPA 023 TPA 023 is a GABAA α2/α3 subtype-selective agonist, with Ki of 0.19-0.41 nM. TPA 023 Chemical Structure
  96. GC67996 TPA-023B TPA-023B Chemical Structure
  97. GC10183 TPMPA GABAA-ρ antagonist TPMPA Chemical Structure
  98. GC10262 Tracazolate hydrochloride GABAA receptor modulator Tracazolate hydrochloride Chemical Structure
  99. GC17381 trans-4-Hydroxycrotonic acid ligand of γ-hydroxybutyric acid (GHB) receptor trans-4-Hydroxycrotonic acid Chemical Structure
  100. GC14933 U 89843A Positive allosteric modulator of GABAA receptors U 89843A Chemical Structure
  101. GC13509 U 90042 GABAA receptor ligand U 90042 Chemical Structure

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