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GluR

GluR (glutamate receptor) is a group of synaptic receptors located primarily on the membranes of neuronal cells.

Products for  GluR

  1. Cat.No. Product Name Information
  2. GC18033 γDGG γDGG is a competitive AMPA receptor blocker. γDGG  Chemical Structure
  3. GC12699 (±)-LY 395756 ligand for mGlu2 and mGlu3 receptor (±)-LY 395756  Chemical Structure
  4. GC12394 (±)-trans-ACPD

    metabotropic glutamate receptors agonist

    (±)-trans-ACPD  Chemical Structure
  5. GC16207 (1S,3R)-ACPD group I and II mGlu receptor agonist (1S,3R)-ACPD  Chemical Structure
  6. GC11379 (2R,4R)-APDC group II metabotropic glutamate receptor agonist (2R,4R)-APDC  Chemical Structure
  7. GC17722 (R)-3,4-DCPG AMPA receptor antagonist with weak activity at NMDA receptors and little activity at kainate receptors (R)-3,4-DCPG  Chemical Structure
  8. GC14124 (R)-3-Carboxy-4-hydroxyphenylglycine NMDA and AMPA/kainate receptor antagonist (R)-3-Carboxy-4-hydroxyphenylglycine  Chemical Structure
  9. GC16542 (RS)-3,4-DCPG antagonist of AMPA receptors and agonist of mGluR8 (RS)-3,4-DCPG  Chemical Structure
  10. GC15342 (RS)-3,5-DHPG

    DHPG ((RS)-3,5-DHPG) is an amino acid that is a selective potent agonist for group I mGluR (mGluR 1 and mGluR 5) and has no effect on Group II and III mGluR.

    (RS)-3,5-DHPG  Chemical Structure
  11. GC12985 (RS)-3-Hydroxyphenylglycine PI-linked metabotropic glutamate receptors agonist (RS)-3-Hydroxyphenylglycine  Chemical Structure
  12. GC13288 (RS)-4-Carboxy-3-hydroxyphenylglycine broad spectrum EAA agonist/antagonist (RS)-4-Carboxy-3-hydroxyphenylglycine  Chemical Structure
  13. GC13773 (RS)-4-Carboxyphenylglycine broad spectrum EAA ligand (RS)-4-Carboxyphenylglycine  Chemical Structure
  14. GC11771 (RS)-APICA group II metabotropic glutamate receptor antagonist (RS)-APICA  Chemical Structure
  15. GC12279 (RS)-MCPG mGluR antagonist (RS)-MCPG  Chemical Structure
  16. GC11997 (RS)-MCPG disodium salt group I/group II metabotropic glutamate receptor antagonist (RS)-MCPG disodium salt  Chemical Structure
  17. GC11433 (RS)-PPG group III metabotropic glutamate receptor agonist (RS)-PPG  Chemical Structure
  18. GC14639 (S)-3,4-DCPG mGlu8a agonist (S)-3,4-DCPG  Chemical Structure
  19. GC16858 (S)-3,5-DHPG group I mGlu receptor agonist (S)-3,5-DHPG  Chemical Structure
  20. GC11536 (S)-3-Carboxy-4-hydroxyphenylglycine group I metabotropic glutamate receptor antagonist and group II mGlu agonist (S)-3-Carboxy-4-hydroxyphenylglycine  Chemical Structure
  21. GC16234 (S)-3-Hydroxyphenylglycine group I metabotropic glutamate receptors agonist (S)-3-Hydroxyphenylglycine  Chemical Structure
  22. GC12012 (S)-4-Carboxy-3-hydroxyphenylglycine group I mGlu1a/1a receptor antagonist and mGluR2 agonist (S)-4-Carboxy-3-hydroxyphenylglycine  Chemical Structure
  23. GC14176 (S)-4-Carboxyphenylglycine group I metabotropic glutamate receptor antagonist (S)-4-Carboxyphenylglycine  Chemical Structure
  24. GC10739 (S)-HexylHIBO Group I mGlu receptor antagonist (S)-HexylHIBO  Chemical Structure
  25. GC16349 (S)-MCPG mGluR antagonist (S)-MCPG  Chemical Structure
  26. GC14752 2,4-Dihydroxyphenylacetyl-L-asparagine glutamate receptors blocker 2,4-Dihydroxyphenylacetyl-L-asparagine  Chemical Structure
  27. GC11223 3-MATIDA mGlu1 receptor antagonist 3-MATIDA  Chemical Structure
  28. GC16068 A 841720 mGluR1 antagonist, non-competitive A 841720  Chemical Structure
  29. GC17079 ACDPP hydrochloride mGlu5 receptor antagonist ACDPP hydrochloride  Chemical Structure
  30. GC12435 ACPT-I Agonist for group III mGlu receptors ACPT-I  Chemical Structure
  31. GC12460 ADX 10059 hydrochloride Negative allosteric modulator at mGlu5 ADX 10059 hydrochloride  Chemical Structure
  32. GC10494 ADX-47273 mGluR5 receptor positive allosteric modulator, potent and selective ADX-47273  Chemical Structure
  33. GC14146 AIDA AIDA (AIDA), a rigid (carboxyphenyl) glycine derivative, is a relatively potent and selective antagonist of group I metabotropic glutamate receptors (mGlu1a) with an IC50 of 214 μM. AIDA  Chemical Structure
  34. GC11287 AMN 082 dihydrochloride AMN 082 dihydrochloride, a selective, orally active, and brain penetrant mGluR7 agonist, directly activates receptor signaling via an allosteric site in the transmembrane domain. AMN 082 dihydrochloride  Chemical Structure
  35. GC10141 Bay 36-7620 Selective mGlu1 receptor non-competitive antagonist Bay 36-7620  Chemical Structure
  36. GC12510 BINA BINA (BINA) is a selective human mGluR2 (hmGluR2) potentiator for the treatment of many neurological disorders. BINA  Chemical Structure
  37. GC12899 CBiPES hydrochloride positive allosteric modulator of the mGlu2 receptor CBiPES hydrochloride  Chemical Structure
  38. GC10422 CDPPB positive allosteric modulator of the mGlu5 receptor CDPPB  Chemical Structure
  39. GC12532 CHPG mGlu5 metabotropic glutamate receptor agonist CHPG  Chemical Structure
  40. GC17963 CHPG Sodium salt mGlu5 agonist CHPG Sodium salt  Chemical Structure
  41. GC12705 Cinnabarinic acid

    A mGlu4 receptor agonist

    Cinnabarinic acid  Chemical Structure
  42. GC18134 CPCCOEt hmGlu1 subtype-selective antagonist CPCCOEt  Chemical Structure
  43. GC12100 CPPG group III mGlu receptor antagonist CPPG  Chemical Structure
  44. GC12063 D-AP4 broad spectrum excitatory amino acid receptor antagonist D-AP4  Chemical Structure
  45. GC15385 DCB Allosteric ligand for mGlu5 DCB  Chemical Structure
  46. GC16247 DCG IV highly potent agonist for group II mGlu receptors DCG IV  Chemical Structure
  47. GC13120 Desmethyl-YM 298198 mGlu1-selective antagonist Desmethyl-YM 298198  Chemical Structure
  48. GC11246 DFB DFB (DFB) is a selective positive allosteric modulator of mGluR5. DFB  Chemical Structure
  49. GC14687 DL-AP4 broad spectrum EAA antagonist DL-AP4  Chemical Structure
  50. GC12960 DL-AP4 Sodium salt Broad spectrum EAA ligand DL-AP4 Sodium salt  Chemical Structure
  51. GC13126 DMeOB Negative allosteric modulator of mGlu5 DMeOB  Chemical Structure
  52. GC13192 E4CPG group I/group II metabotropic glutamate receptor antagonist E4CPG  Chemical Structure
  53. GC17326 EGLU

    group II mGlu receptor antagonist

    EGLU  Chemical Structure
  54. GC11766 Fenobam mGlu5 antagonist Fenobam  Chemical Structure
  55. GC17446 HexylHIBO

    Group I mGlu receptor antagonist

    HexylHIBO  Chemical Structure
  56. GC12198 IEM 1754 dihydrobroMide IEM 1754 dihydrobroMide, a dicationic adamantane derivative, is a potent blocker of open channels of native ionotropic glutamate receptors including quisqualate-sensitive receptors in insect muscles, NMDAR in cultured rat cortical neurons, and AMPAR in freshly isolated hippocampal cells. IEM 1754 dihydrobroMide  Chemical Structure
  57. GC12521 Ifenprodil Tartrate NMDA receptor antagonist Ifenprodil Tartrate  Chemical Structure
  58. GC17217 JNJ 16259685 mGlu1 antagonist JNJ 16259685  Chemical Structure
  59. GC17932 L-AP4

    group III metabotropic glutamate receptor agonist

    L-AP4  Chemical Structure
  60. GC15136 L-AP6 selective agonist for 'quis'-sensitized site L-AP6  Chemical Structure
  61. GC12224 L-BMAA hydrochloride L-BMAA hydrochloride (BMAA hydrochloride) is a neurotoxin produced by cyanobacteria. L-BMAA hydrochloride  Chemical Structure
  62. GC13881 L-CCG-l

    group II metabotropic glutamate receptor agonist

    L-CCG-l  Chemical Structure
  63. GC17974 Latrepirdine dihydrochloride Latrepirdine is a neuroactive compound with antagonist activity at histaminergic, α-adrenergic, and serotonergic receptors. Latrepirdine dihydrochloride  Chemical Structure
  64. GC18309 LSN2463359 LSN2463359 is a positive allosteric modulator of the metabotropic glutamate receptor 5 (mGluR5; EC50 = 24 nM). LSN2463359  Chemical Structure
  65. GC14722 LY 2389575 hydrochloride negative allosteric modulator of mGlu3 LY 2389575 hydrochloride  Chemical Structure
  66. GC10605 LY 354740 LY 354740 (LY354740) is a highly potent and selective group II (mGlu2/3) receptor agonist with IC50s of 5 and 24 nM on transfected human mGlu2 and mGlu3 receptors, respectively. LY 354740  Chemical Structure
  67. GC12831 LY 367385 mGlu1a receptor antagonist LY 367385  Chemical Structure
  68. GC14861 LY 379268 Group II mGlu receptor agonist, highly selective LY 379268  Chemical Structure
  69. GC16557 LY 379268 disodium salt group II mGlu receptor agonist LY 379268 disodium salt  Chemical Structure
  70. GC17492 LY 456236 hydrochloride mGlu1 receptor antagonist LY 456236 hydrochloride  Chemical Structure
  71. GC14097 LY 487379 hydrochloride Positive allosteric modulator of mGlu2 receptors LY 487379 hydrochloride  Chemical Structure
  72. GC11571 MAP4 metabotropic glutamate receptor modulator MAP4  Chemical Structure
  73. GC10045 MFZ 10-7 negative allosteric modulator of the mGlu5 receptor MFZ 10-7  Chemical Structure
  74. GC14869 ML 289 negative allosteric modulator of mGlu3 receptors ML 289  Chemical Structure
  75. GC17095 ML 337 negative allosteric modulator of mGlu3 ML 337  Chemical Structure
  76. GC17950 MMPIP hydrochloride allosteric mGlu7-selective receptor antagonist MMPIP hydrochloride  Chemical Structure
  77. GC10238 MNI 137 negative allosteric modulator of group II mGlu receptors MNI 137  Chemical Structure
  78. GC14227 MNI-caged-L-glutamate rapidly and efficiently releases glutamate MNI-caged-L-glutamate  Chemical Structure
  79. GC15769 MPPG mGlu receptor antagonist MPPG  Chemical Structure
  80. GC17185 MSOP group III metabotropic glutamate receptor antagonist MSOP  Chemical Structure
  81. GC13548 MSPG

    mGlu receptor antagonist

    MSPG  Chemical Structure
  82. GC11428 MTPG Group II/group III metabotropic glutamate receptor antagonist MTPG  Chemical Structure
  83. GC13222 N-Acetylglycyl-D-glutamic acid Excitatory peptide that induces seizures N-Acetylglycyl-D-glutamic acid  Chemical Structure
  84. GC17456 NMDA (N-Methyl-D-aspartic acid) NMDA (N-Methyl-D-aspartic acid) is a specific agonist forNMDA (N-Methyl-D-aspartic acid)receptor mimicking the action of glutamate, the neurotransmitter which normally acts at that receptor. NMDA (N-Methyl-D-aspartic acid)  Chemical Structure
  85. GC17604 NPEC-caged-(1S,3R)-ACPD group I and II mGlu receptor agonist NPEC-caged-(1S,3R)-ACPD  Chemical Structure
  86. GC11554 NPEC-caged-(S)-3,4-DCPG mGlu8a agonist NPEC-caged-(S)-3,4-DCPG  Chemical Structure
  87. GC10784 NPEC-caged-LY 379268 group II mGlu receptor agonist NPEC-caged-LY 379268  Chemical Structure
  88. GC11563 NPS 2390 group I mGlu antagonist NPS 2390  Chemical Structure
  89. GC10123 O-Phospho-L-serine group III metabotropic glutamate receptor agonist O-Phospho-L-serine  Chemical Structure
  90. GC17383 PHCCC Group I metabotropic glutamate receptor antagonist PHCCC  Chemical Structure
  91. GC14383 Ro 01-6128 Positive allosteric modulator of mGlu1 receptors Ro 01-6128  Chemical Structure
  92. GC11704 Ro 64-5229 mGlu2 antagonist Ro 64-5229  Chemical Structure
  93. GC14172 Ro 67-4853 Positive allosteric modulator of mGlu group I receptors Ro 67-4853  Chemical Structure
  94. GC12485 Ro 67-7476 positive allosteric modulator of mGlu1 receptors Ro 67-7476  Chemical Structure
  95. GC15435 RuBi-Glutamate Ruthenium-bipyridine-trimethylphosphine caged glutamate RuBi-Glutamate  Chemical Structure
  96. GC10026 S-Sulfo-L-cysteine sodium salt EAA receptor agonist S-Sulfo-L-cysteine sodium salt  Chemical Structure
  97. GC11269 Salsolinol-1-carboxylic acid amino acid that occurs naturally in the CNS Salsolinol-1-carboxylic acid  Chemical Structure
  98. GC11233 SIB 1757 mGlu5 antagonist SIB 1757  Chemical Structure
  99. GC10452 SIB 1893 SIB 1893 is a racemic compound of (E)-SIB-1893 and (Z)-SIB-1893 isomers. SIB 1893  Chemical Structure
  100. GC14301 Spaglumic acid mGlu3 receptor agonist and NMDA receptor activator Spaglumic acid  Chemical Structure
  101. GC11750 TC-N 22A mGlu4 receptor positive allosteric modulator TC-N 22A  Chemical Structure

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