GluR
GluR (glutamate receptor) is a group of synaptic receptors located primarily on the membranes of neuronal cells.
Products for GluR
- Cat.No. Product Name Information
- GC18033 γDGG γDGG is a competitive AMPA receptor blocker.
- GC12699 (±)-LY 395756 ligand for mGlu2 and mGlu3 receptor
-
GC12394
(±)-trans-ACPD
metabotropic glutamate receptors agonist
- GC16207 (1S,3R)-ACPD group I and II mGlu receptor agonist
- GC11379 (2R,4R)-APDC group II metabotropic glutamate receptor agonist
- GC17722 (R)-3,4-DCPG AMPA receptor antagonist with weak activity at NMDA receptors and little activity at kainate receptors
- GC14124 (R)-3-Carboxy-4-hydroxyphenylglycine NMDA and AMPA/kainate receptor antagonist
- GC16542 (RS)-3,4-DCPG antagonist of AMPA receptors and agonist of mGluR8
-
GC15342
(RS)-3,5-DHPG
DHPG ((RS)-3,5-DHPG) is an amino acid that is a selective potent agonist for group I mGluR (mGluR 1 and mGluR 5) and has no effect on Group II and III mGluR.
- GC12985 (RS)-3-Hydroxyphenylglycine PI-linked metabotropic glutamate receptors agonist
- GC13288 (RS)-4-Carboxy-3-hydroxyphenylglycine broad spectrum EAA agonist/antagonist
- GC13773 (RS)-4-Carboxyphenylglycine broad spectrum EAA ligand
- GC11771 (RS)-APICA group II metabotropic glutamate receptor antagonist
- GC12279 (RS)-MCPG mGluR antagonist
- GC11997 (RS)-MCPG disodium salt group I/group II metabotropic glutamate receptor antagonist
- GC11433 (RS)-PPG group III metabotropic glutamate receptor agonist
- GC14639 (S)-3,4-DCPG mGlu8a agonist
- GC16858 (S)-3,5-DHPG group I mGlu receptor agonist
- GC11536 (S)-3-Carboxy-4-hydroxyphenylglycine group I metabotropic glutamate receptor antagonist and group II mGlu agonist
- GC16234 (S)-3-Hydroxyphenylglycine group I metabotropic glutamate receptors agonist
- GC12012 (S)-4-Carboxy-3-hydroxyphenylglycine group I mGlu1a/1a receptor antagonist and mGluR2 agonist
- GC14176 (S)-4-Carboxyphenylglycine group I metabotropic glutamate receptor antagonist
- GC10739 (S)-HexylHIBO Group I mGlu receptor antagonist
- GC16349 (S)-MCPG mGluR antagonist
- GC14752 2,4-Dihydroxyphenylacetyl-L-asparagine glutamate receptors blocker
- GC11223 3-MATIDA mGlu1 receptor antagonist
- GC16068 A 841720 mGluR1 antagonist, non-competitive
- GC17079 ACDPP hydrochloride mGlu5 receptor antagonist
- GC12435 ACPT-I Agonist for group III mGlu receptors
- GC12460 ADX 10059 hydrochloride Negative allosteric modulator at mGlu5
- GC10494 ADX-47273 mGluR5 receptor positive allosteric modulator, potent and selective
- GC14146 AIDA AIDA (AIDA), a rigid (carboxyphenyl) glycine derivative, is a relatively potent and selective antagonist of group I metabotropic glutamate receptors (mGlu1a) with an IC50 of 214 μM.
- GC11287 AMN 082 dihydrochloride AMN 082 dihydrochloride, a selective, orally active, and brain penetrant mGluR7 agonist, directly activates receptor signaling via an allosteric site in the transmembrane domain.
- GC10141 Bay 36-7620 Selective mGlu1 receptor non-competitive antagonist
- GC12510 BINA BINA (BINA) is a selective human mGluR2 (hmGluR2) potentiator for the treatment of many neurological disorders.
- GC12899 CBiPES hydrochloride positive allosteric modulator of the mGlu2 receptor
- GC10422 CDPPB positive allosteric modulator of the mGlu5 receptor
- GC12532 CHPG mGlu5 metabotropic glutamate receptor agonist
- GC17963 CHPG Sodium salt mGlu5 agonist
-
GC12705
Cinnabarinic acid
A mGlu4 receptor agonist
- GC18134 CPCCOEt hmGlu1 subtype-selective antagonist
- GC12100 CPPG group III mGlu receptor antagonist
- GC12063 D-AP4 broad spectrum excitatory amino acid receptor antagonist
- GC15385 DCB Allosteric ligand for mGlu5
- GC16247 DCG IV highly potent agonist for group II mGlu receptors
- GC13120 Desmethyl-YM 298198 mGlu1-selective antagonist
- GC11246 DFB DFB (DFB) is a selective positive allosteric modulator of mGluR5.
- GC14687 DL-AP4 broad spectrum EAA antagonist
- GC12960 DL-AP4 Sodium salt Broad spectrum EAA ligand
- GC13126 DMeOB Negative allosteric modulator of mGlu5
- GC13192 E4CPG group I/group II metabotropic glutamate receptor antagonist
-
GC17326
EGLU
group II mGlu receptor antagonist
- GC11766 Fenobam mGlu5 antagonist
-
GC17446
HexylHIBO
Group I mGlu receptor antagonist
- GC12198 IEM 1754 dihydrobroMide IEM 1754 dihydrobroMide, a dicationic adamantane derivative, is a potent blocker of open channels of native ionotropic glutamate receptors including quisqualate-sensitive receptors in insect muscles, NMDAR in cultured rat cortical neurons, and AMPAR in freshly isolated hippocampal cells.
- GC12521 Ifenprodil Tartrate NMDA receptor antagonist
- GC17217 JNJ 16259685 mGlu1 antagonist
-
GC17932
L-AP4
group III metabotropic glutamate receptor agonist
- GC15136 L-AP6 selective agonist for 'quis'-sensitized site
- GC12224 L-BMAA hydrochloride L-BMAA hydrochloride (BMAA hydrochloride) is a neurotoxin produced by cyanobacteria.
-
GC13881
L-CCG-l
group II metabotropic glutamate receptor agonist
- GC17974 Latrepirdine dihydrochloride Latrepirdine is a neuroactive compound with antagonist activity at histaminergic, α-adrenergic, and serotonergic receptors.
- GC18309 LSN2463359 LSN2463359 is a positive allosteric modulator of the metabotropic glutamate receptor 5 (mGluR5; EC50 = 24 nM).
- GC14722 LY 2389575 hydrochloride negative allosteric modulator of mGlu3
- GC10605 LY 354740 LY 354740 (LY354740) is a highly potent and selective group II (mGlu2/3) receptor agonist with IC50s of 5 and 24 nM on transfected human mGlu2 and mGlu3 receptors, respectively.
- GC12831 LY 367385 mGlu1a receptor antagonist
- GC14861 LY 379268 Group II mGlu receptor agonist, highly selective
- GC16557 LY 379268 disodium salt group II mGlu receptor agonist
- GC17492 LY 456236 hydrochloride mGlu1 receptor antagonist
- GC14097 LY 487379 hydrochloride Positive allosteric modulator of mGlu2 receptors
- GC11571 MAP4 metabotropic glutamate receptor modulator
- GC10045 MFZ 10-7 negative allosteric modulator of the mGlu5 receptor
- GC14869 ML 289 negative allosteric modulator of mGlu3 receptors
- GC17095 ML 337 negative allosteric modulator of mGlu3
- GC17950 MMPIP hydrochloride allosteric mGlu7-selective receptor antagonist
- GC10238 MNI 137 negative allosteric modulator of group II mGlu receptors
- GC14227 MNI-caged-L-glutamate rapidly and efficiently releases glutamate
- GC15769 MPPG mGlu receptor antagonist
- GC17185 MSOP group III metabotropic glutamate receptor antagonist
-
GC13548
MSPG
mGlu receptor antagonist
- GC11428 MTPG Group II/group III metabotropic glutamate receptor antagonist
- GC13222 N-Acetylglycyl-D-glutamic acid Excitatory peptide that induces seizures
- GC17456 NMDA (N-Methyl-D-aspartic acid) NMDA (N-Methyl-D-aspartic acid) is a specific agonist forNMDA (N-Methyl-D-aspartic acid)receptor mimicking the action of glutamate, the neurotransmitter which normally acts at that receptor.
- GC17604 NPEC-caged-(1S,3R)-ACPD group I and II mGlu receptor agonist
- GC11554 NPEC-caged-(S)-3,4-DCPG mGlu8a agonist
- GC10784 NPEC-caged-LY 379268 group II mGlu receptor agonist
- GC11563 NPS 2390 group I mGlu antagonist
- GC10123 O-Phospho-L-serine group III metabotropic glutamate receptor agonist
- GC17383 PHCCC Group I metabotropic glutamate receptor antagonist
- GC14383 Ro 01-6128 Positive allosteric modulator of mGlu1 receptors
- GC11704 Ro 64-5229 mGlu2 antagonist
- GC14172 Ro 67-4853 Positive allosteric modulator of mGlu group I receptors
- GC12485 Ro 67-7476 positive allosteric modulator of mGlu1 receptors
- GC15435 RuBi-Glutamate Ruthenium-bipyridine-trimethylphosphine caged glutamate
- GC10026 S-Sulfo-L-cysteine sodium salt EAA receptor agonist
- GC11269 Salsolinol-1-carboxylic acid amino acid that occurs naturally in the CNS
- GC11233 SIB 1757 mGlu5 antagonist
- GC10452 SIB 1893 SIB 1893 is a racemic compound of (E)-SIB-1893 and (Z)-SIB-1893 isomers.
- GC14301 Spaglumic acid mGlu3 receptor agonist and NMDA receptor activator
- GC11750 TC-N 22A mGlu4 receptor positive allosteric modulator