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Home >> Signaling Pathways >> Neuroscience >> Histamine Receptor

Histamine Receptor

Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.

Products for  Histamine Receptor

  1. Cat.No. Product Name Information
  2. GC17299 Famotidine Histamine H2-receptor antagonist Famotidine Chemical Structure
  3. GC31750 Fenspiride Hydrochloride Fenspiride Hydrochloride Chemical Structure
  4. GC33499 Fexofenadine D6 (MDL-16455 D6) Fexofenadine D6 (MDL-16455 D6) is deuterium labeled is Fexofenadine, which is an antihistamine pharmaceutical agent. Fexofenadine D6 (MDL-16455 D6) Chemical Structure
  5. GC10966 Fexofenadine HCl Fexofenadine (MDL-16455) hydrochloride is an orally active and nonsedative H1 receptor antagonist. Fexofenadine HCl Chemical Structure
  6. GC32050 FRG8701 FRG-8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM. FRG8701 Chemical Structure
  7. GC19178 GSK189254A GSK189254A (GSK189254) is a novel, potent and selective histamine H3 receptor antagonist with pKi values of 9.59-9.90 and 8.51-9.17 for human and rat H3, respectively. GSK189254A Chemical Structure
  8. GC16180 GT 2016 H3 receptor antagonist GT 2016 Chemical Structure
  9. GC31310 H3 receptor antagonist 1 H3 receptor antagonist 1 Chemical Structure
  10. GC30759 H3 receptor-MO-1 H3 receptor-MO-1 is a modulator of histamine H3 receptor. H3 receptor-MO-1 Chemical Structure
  11. GC64661 H3R antagonist 1 hydrochloride H3R antagonist 1 hydrochloride is a histamine receptor 3 (H3R) inverse agonist extracted from patent WO2013107336A1, compound example 2. H3R antagonist 1 hydrochloride Chemical Structure
  12. GC34338 H3R-IN-1 Hydrochloride H3R-IN-1 Hydrochloride Chemical Structure
  13. GC31232 H4 Receptor antagonist 1 H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM. H4 Receptor antagonist 1 Chemical Structure
  14. GC31884 H4R antagonist 1

    H4R antagonist 1 is a potent and highly selective histamine H4 receptor (H4R) antagonist with an IC50 of 27 nM.

     H4R antagonist 1 Chemical Structure
  15. GC30775 Histamine (Ergamine) Histamine (Ergamine) is an organic nitrogenous compound involved in local immune responses as well as regulating physiological function in the gut and acting as a neurotransmitter. Histamine (Ergamine) Chemical Structure
  16. GC10806 Histamine 2HCl Histamine 2HCl is an endogenous metabolite. Histamine 2HCl Chemical Structure
  17. GC17869 Histamine Phosphate Histamine receptor agonist Histamine Phosphate Chemical Structure
  18. GC68330 Histamine-α,α,β,β-d4 dihydrochloride Histamine-α,α,β,β-d4 dihydrochloride Chemical Structure
  19. GC17429 HTMT dimaleate H1 and H2 receptor agonist HTMT dimaleate Chemical Structure
  20. GC16122 Hydroxyzine histamine H1-receptor antagonist Hydroxyzine Chemical Structure
  21. GC10306 Hydroxyzine 2HCl Hydroxyzine 2HCl, a benzodiazepine antihistamine agent, acts as a orally active histamineH1-receptor and serotonin antagonist. Hydroxyzine 2HCl Chemical Structure
  22. GC36278 Hydroxyzine D4 dihydrochloride Hydroxyzine D4 dihydrochloride is deuterium labeled Hydroxyzine. Hydroxyzine D4 dihydrochloride Chemical Structure
  23. GC60924 Hydroxyzine D8 Hydroxyzine D8 is deuterium labeled Hydroxyzine. Hydroxyzine D8 Chemical Structure
  24. GC36279 Hydroxyzine pamoate Hydroxyzine pamoate is a histamine H1-receptor antagonist. Hydroxyzine pamoate Chemical Structure
  25. GC16162 ICI 162,846 histamine H2 receptor antagonist ICI 162,846 Chemical Structure
  26. GC11220 Imetit dihydrobromide H3 and H4 receptors agonist Imetit dihydrobromide Chemical Structure
  27. GC12966 Immepip dihydrobromide histamine H3 receptor agonist Immepip dihydrobromide Chemical Structure
  28. GC14260 Immethridine dihydrobromide histamine H3 receptor agonist Immethridine dihydrobromide Chemical Structure
  29. GC10241 Impentamine dihydrobromide histamine H3 receptor antagonist Impentamine dihydrobromide Chemical Structure
  30. GC65937 INCB38579 INCB38579 is an orally active, highly brain penetrable, and selective histamine H4 receptor (HH4R) antagonist (hH4R IC50=4.8 nM, mH4R IC50=42 nM, rH4R IC50=32 nM). INCB38579 shows anti-inflammatory pain and anti-pruritic activities. INCB38579 Chemical Structure
  31. GC12265 Iodophenpropit dihydrobromide H3 antagonist Iodophenpropit dihydrobromide Chemical Structure
  32. GC12371 JNJ 10181457 dihydrochloride Histamine H3 receptor antagonist JNJ 10181457 dihydrochloride Chemical Structure
  33. GC14429 JNJ 10191584 maleate histamine H4 receptor silent antagonist JNJ 10191584 maleate Chemical Structure
  34. GC50405 JNJ 39758979 dihydrochloride High affinity and selective histamine H4 antagonist; orally bioavailable JNJ 39758979 dihydrochloride Chemical Structure
  35. GC11046 JNJ 5207852 dihydrochloride JNJ 5207852 dihydrochloride is a selective and potent histamine H3 receptor (H3R) antagonist, with pKis of 8.9, 9.24 for rat and human H3R, respectively. JNJ 5207852 dihydrochloride Chemical Structure
  36. GC30821 JNJ-39758979 JNJ-39758979 is a selective, orally active, and high-affinity histamine H4 receptor antagonist with Kis of 12.5, 5.3, and 25 nM for human, mouse, and monkey histamine H4 receptor, respectively. JNJ-39758979 Chemical Structure
  37. GC10400 JNJ-7777120 Histamine H4 receptor antagonist JNJ-7777120 Chemical Structure
  38. GC17733 Ketotifen Fumarate Histamine H1 receptor antagonist Ketotifen Fumarate Chemical Structure
  39. GC67995 Ketotifen-d3 fumarate Ketotifen-d3 fumarate Chemical Structure
  40. GC32001 KP136 (AL136) KP136 (AL136) (AL136) is an orally effective antiallergic agent. KP136 (AL136) Chemical Structure
  41. GC16085 Lafutidine Histamine H2-receptor antagonist Lafutidine Chemical Structure
  42. GC17974 Latrepirdine dihydrochloride Latrepirdine is a neuroactive compound with antagonist activity at histaminergic, α-adrenergic, and serotonergic receptors. Latrepirdine dihydrochloride Chemical Structure
  43. GC19441 Levocabastine (hydrochloride) Levocabastine is a potent and selective histamine H1 receptor antagonist with an IC50 value of 8.32 nM (Kis = 62.5, 23,500, and 1,937 nM for H1, H2, and H3, respectively) for inhibition of phosphoinositide turnover on human conjunctival epithelial cells. Levocabastine (hydrochloride) Chemical Structure
  44. GC25571 Levocetirizine Levocetirizine (LCZ, (R)-Cetirizine), the R-enantiomer of cetirizine, is an antagonist of histamine H(1) receptor. Levocetirizine Chemical Structure
  45. GC15214 Levodropropizine Histamine receptor inhibitor,cough suppressant Levodropropizine Chemical Structure
  46. GC17608 Lidocaine Anasthetic and class Ib antiarrhythmic agent Lidocaine Chemical Structure
  47. GC38450 LML134 LML134 (compound 18b) is an orally active and high selective Histamine 3 receptor (H3R) inverse agonist with Kis of 0.3 nM and 12 nM for hH3R cAMP and hH3R bdg. LML134 Chemical Structure
  48. GC18282 Lodoxamide

    Lodoxamide is a potent agonist of GPR35 with an EC50 value of 1.61 nM in a β-arrestin-2 interaction assay using CHO-K1 cells expressing the human receptor.

     Lodoxamide Chemical Structure
  49. GC36476 Lodoxamide tromethamine Lodoxamide tromethamine (U-42585E) is a medication for the treatment of prophylaxis of mast cell-mediated allergic disease. Lodoxamide tromethamine Chemical Structure
  50. GC15252 Loratadine

    Loratadine is a non- sedating antihistamine that acts as a selective inverse agonist of peripheral histamine H 1 receptors (K i = 35 nM).

     Loratadine Chemical Structure
  51. GC31787 Mebhydrolin Mebhydrolin is a specific histamine H1 receptor antagonist. Mebhydrolin Chemical Structure
  52. GC31848 Mebhydrolin napadisylate (Mebhydroline 1,5-naphthalenedisulfonate salt) Mebhydrolin napadisylate (Mebhydroline 1,5-naphthalenedisulfonate salt) is a specific histamine H1 receptor antagonist. Mebhydrolin napadisylate (Mebhydroline 1,5-naphthalenedisulfonate salt) Chemical Structure
  53. GC11291 Mepyramine maleate

    inverse agonist for the H1 receptor

     Mepyramine maleate Chemical Structure
  54. GC31743 Mequitazine (LM-209) Mequitazine (LM-209) is a potent, and long-acting histamine H1 antagonist. Mequitazine (LM-209) Chemical Structure
  55. GC17010 Methimepip dihydrobromide histamine H3 receptor agonist Methimepip dihydrobromide Chemical Structure
  56. GC13024 Metiamide Metiamide Chemical Structure
  57. GC15518 Mianserin

    H1 receptor inverse agonist

     Mianserin Chemical Structure
  58. GC14726 Mianserin HCl Mianserin HCl (Org GB 94) is a H1 receptor inverse agonist and is a psychoactive agent of the tetracyclic antidepressant. Mianserin HCl Chemical Structure
  59. GC48855 Mirtazapine (CRM) A Certified Reference Material Mirtazapine (CRM) Chemical Structure
  60. GC12549 Mizolastine Histamine H1-receptor antagonist Mizolastine Chemical Structure
  61. GC10478 Mizolastine dihydrochloride Histamine H1-receptor antagonist Mizolastine dihydrochloride Chemical Structure
  62. GC31027 MK-0249 MK-0249 (Compound 1) is a potent, selective and orally active histamine H3 receptor antagonist, with an IC50 of 1.7 nM for human H3. MK-0249 Chemical Structure
  63. GC16487 Nα-Methylhistamine dihydrochloride

    histamine H3 receptor agonist

     Nα-Methylhistamine dihydrochloride Chemical Structure
  64. GC18463 N-acetyl Histamine N-acetyl Histamine is a histamine metabolite that is formed via acetyl-CoA-dependent N-acetylation of histamine by AANATL7 in D. N-acetyl Histamine Chemical Structure
  65. GC17000 Nedocromil anti-inflammatory agent Nedocromil Chemical Structure
  66. GC44360 Nedocromil (sodium salt) Nedocromil (sodium salt) suppresses the action or formation of multiple mediators, including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2). Nedocromil (sodium salt) Chemical Structure
  67. GC61467 Niaprazine Niaprazine is a histamine H1-receptor antagonist. Niaprazine Chemical Structure
  68. GC46185 Nimbin A limonoid with diverse biological activities Nimbin Chemical Structure
  69. GC31455 Niperotidine Niperotidine is a histamine H2-receptor antagonist. Niperotidine Chemical Structure
  70. GC12794 Nizatidine Histamine H2 receptor antagonist Nizatidine Chemical Structure
  71. GC48892 NSC 19005 NSC 19005 (NSC19005) is an impurity of Betahistine. NSC 19005 Chemical Structure
  72. GC10511 Olopatadine HCl Olopatadine HCl (ALO4943A) is a histamine blocker used to treat allergic conjunctivitis. Olopatadine HCl Chemical Structure
  73. GN10333 Osthole Osthole Chemical Structure
  74. GC61401 Oxatomide Oxatomide is a potent and orally active dual H1-histamine receptor and P2X7 receptor antagonist with antihistamine and anti-allergic activity. Oxatomide Chemical Structure
  75. GC12238 Oxomemazine NULL Oxomemazine Chemical Structure
  76. GC17892 Pemirolast potassium Histamine H1 receptor antagonist Pemirolast potassium Chemical Structure
  77. GC31767 Peptide 401 Peptide 401, a potent mast cell degranulating factor from bee venom, suppresses the increased vascular permeability due to intradermal injection of various smooth muscle spasmogens (histamine, and 5-HT). Peptide 401 Chemical Structure
  78. GC12293 Perphenazine dopamine antagonist Perphenazine Chemical Structure
  79. GC36875 Perphenazine D8 Dihydrochloride Perphenazine D8 Dihydrochloride is the deuterium labeled Perphenazine, which is a typical antipsychotic drug(5-HT, Dopamine receptor ligand). Perphenazine D8 Dihydrochloride Chemical Structure
  80. GC36878 PF-03654746 PF-03654746 is a potent and selective histamine H3 receptor antagonist with high brain penetration. PF-03654746 Chemical Structure
  81. GC38558 PF-03654746 Tosylate PF-03654746 Tosylate is a potent and selective histamine H3 receptor antagonist with high brain penetration. PF-03654746 Tosylate Chemical Structure
  82. GC31790 PF-3893787 hydrochloride PF-3893787 hydrochloride (PF-3893787 hydrochloride) is a novel histamine H4 receptor antagonist binding affinity (Ki=2.4 nM) and is also a functional (Ki=1.56 nM) antagonist. PF-3893787 hydrochloride Chemical Structure
  83. GC16787 Pheniramine Maleate Histamine receptor antagonist Pheniramine Maleate Chemical Structure
  84. GC30999 Pimethixene (Pimetixene) Pimethixene (Pimetixene) is antihistamine and antiserotonergic compound, acts as an antimigraine agent. Pimethixene (Pimetixene) Chemical Structure
  85. GC65296 Pimethixene maleate Pimethixene maleate is antihistamine and antiserotonergic compound, acts as an antimigraine agent. Pimethixene maleate Chemical Structure
  86. GC31897 Pirolate (CP-32387) Pirolate (CP-32387) is a histamine H1 receptor antagonist. Pirolate (CP-32387) Chemical Structure
  87. GC36931 Pitolisant A histamine H3 receptor antagonist and inverse agonist Pitolisant Chemical Structure
  88. GC11382 Pitolisant hydrochloride A histamine H3 receptor antagonist and inverse agonist Pitolisant hydrochloride Chemical Structure
  89. GC36932 Pitolisant oxalate Pitolisant oxalate is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM). Pitolisant oxalate Chemical Structure
  90. GC25785 Promethazine Promethazine is a potent histamine H1 receptor antagonist. Promethazine is a medication used in the management and treatment of allergic conditions, nausea and vomiting, motion sickness, and sedation. Promethazine exhibits antiparasitic properties. Promethazine Chemical Structure
  91. GC10814 Promethazine HCl Promethazine HCl is the first-generation antihistamine; strong antagonist of the H1 receptor and moderate mACh receptor antagonist, moderate affinity for 5-HT2A, 5-HT2C, D2 and α1-adrenergic receptors. Promethazine HCl Chemical Structure
  92. GC69738 Promethazine-d4 hydrochloride

    Promethazine-d4 (hydrochloride) is the deuterated form of Promethazine hydrochloride. Promethazine hydrochloride is a first-generation antihistamine with H1 receptor potent antagonism and mAChR antagonism, as well as some affinity for 5-HT2A, 5-HT2C, D2, and alpha-1 adrenergic receptors.

     Promethazine-d4 hydrochloride Chemical Structure
  93. GC63312 Promethazine-d6 hydrochloride Promethazine-d6 hydrochloride Chemical Structure
  94. GC15957 Proxyfan oxalate histamine H3 receptor ligand Proxyfan oxalate Chemical Structure
  95. GC64646 Psoralenoside Psoralenoside is a benzofuran glycoside from Psoralea corylifolia. Psoralenoside Chemical Structure
  96. GC31820 Quinotolast sodium (FR71021) Quinotolast sodium (FR71021) in the concentration range of 1-100 μg/mL inhibits histamine, LTC4 and PGD2 release in a concentration-dependent manner. Quinotolast sodium (FR71021) Chemical Structure
  97. GC12365 Ranitidine hydrochloride Histamine H2-receptor antagonist Ranitidine hydrochloride Chemical Structure
  98. GC31812 ReN-1869 hydrochloride (NNC-05-1869 hydrochloride) ReN 1869 hydrochloride is a novel, selective histamine H1 receptor antagonist, which demonstrates affinity to the histamine H1 receptor (guinea pig brain) with Ki of 0.19±0.04 μM and the non-selective σ site (guinea pig brain) with Ki of 0.45 μM. ReN-1869 hydrochloride (NNC-05-1869 hydrochloride) Chemical Structure
  99. GC30455 Rocastine (AHR-11325) Rocastine (AHR-11325) is a selective, nonsedating H1 antagonist, acting as an antihistamine. Rocastine (AHR-11325) Chemical Structure
  100. GC12085 ROS 234 dioxalate ROS 234 dioxalate is a potent H3 antagonist, with a pKB of 9.46 for Guinea-pig ileum H3-receptor, a pKi of 8.90 for Rat cerebral cortex H3-receptor, and a ED50 of 19.12 mg/kg (ip) in ex vivo of Rat cerebral cortex. ROS 234 dioxalate Chemical Structure
  101. GC10369 Roxatidine Acetate HCl Roxatidine Acetate HCl is a potent, selective, competitive and orally active histamine H2-receptor antagonist. Roxatidine Acetate HCl Chemical Structure

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