Search Site
  • 0
    My Cart

    Click Here to Find How Many Items You Have Added:)

    image loader

    Adding item(s) to cart......

Home >> Signaling Pathways >> Endocrinology and Hormones >> Androgen Receptor

Androgen Receptor

AR (androgen receptor) is a member of steroid hormone receptor and ligand-activated transcription factor. It plays a crucial role in prostate cellular proliferation and male sexual differentiation.

Products for  Androgen Receptor

  1. Cat.No. Product Name Information
  2. GC45239 δ4-Abiraterone

    CB 7627, D4A

     δ4-Abiraterone is a major metabolite of abiraterone. δ4-Abiraterone is an inhibitor of CYP17A1, 3b-hydroxysteroid dehydrogenase (3βHSD) and steroid-5a-reductase (SRD5A) and also an antagonist of androgen receptor. δ4-Abiraterone Chemical Structure
  3. GC61491 (R)-Bicalutamide (R)-Bicalutamide is the (R)-enantiomer of Bicalutamide. (R)-Bicalutamide is an androgen receptor (AR) antagonist, with antineoplastic activity. (R)-Bicalutamide is widely used for the research of prostate cancer. (R)-Bicalutamide Chemical Structure
  4. GC73509 (R)-SKBG-1 (R)-SKBG-1 is an RNA-binding protein NONO inhibitor. (R)-SKBG-1 Chemical Structure
  5. GC30710 (R)-UT-155 (R)-UT-155 (compound 11) is a selective androgen receptor degrader (SARD) ligand. Less active than the S-isomer. (R)-UT-155 Chemical Structure
  6. GC63292 (rac)-PF-998425 (Rac)-PF-998425 is a potent, selective, nonsteroidal androgen receptor (AR) antagonist. (rac)-PF-998425 Chemical Structure
  7. GC49520 (S)-Equol

    4',7Dihydroxyisoflavan, (-)Equol, 4',7Isoflavandiol

    An estrogen receptor β agonist

     (S)-Equol Chemical Structure
  8. GC40528 11α-hydroxy Testosterone 11α-hydroxy Testosterone is a metabolite of testosterone, produced by the cytochrome P450 (CYP) isoform CYP3A. 11α-hydroxy Testosterone Chemical Structure
  9. GC46456 16α-Hydroxyetiocholanolone A metabolite of 16α-DHEA and androstenedione 16α-Hydroxyetiocholanolone Chemical Structure
  10. GC17557 17 alpha-propionate

    CB-03-01

     A peripherally selective androgen receptor antagonist 17 alpha-propionate Chemical Structure
  11. GC41300 17β-hydroxy Exemestane 17β-hydroxy Exemestane is the primary active metabolite of exemestane. 17β-hydroxy Exemestane Chemical Structure
  12. GC46471 17β-hydroxy Exemestane-d3 A neuropeptide with diverse biological activities 17β-hydroxy Exemestane-d3 Chemical Structure
  13. GC35069 2,2,5,7,8-Pentamethyl-6-Chromanol 2,2,5,7,8-Pentamethyl-6-Chromanol (PMC) is the anti-oxidant moiety of vitamin E (α-tocopherol). 2,2,5,7,8-Pentamethyl-6-Chromanol has potent androgen receptor (AR) signaling modulation and anti-cancer activity against prostate cancer cell lines. 2,2,5,7,8-Pentamethyl-6-Chromanol Chemical Structure
  14. GC17160 2-hydroxy Flutamide

    Hydroxyniphtholide,SCH 16423

     2-hydroxy Flutamide (HF), an active metabolite of Flutamide, is a potent androgen receptor antagonist (IC50=700 nM). 2-hydroxy Flutamide can be used for the research of prostate cancer. 2-hydroxy Flutamide Chemical Structure
  15. GC12791 3,3'-Diindolylmethane

    DIM

     A phytochemical with antiradiation and chemopreventative effects 3,3'-Diindolylmethane Chemical Structure
  16. GC49542 5α-Androstan-3β-ol

    NSC 50887

     A steroidal androgen 5α-Androstan-3β-ol Chemical Structure
  17. GC48808 5β-Androstane-3α,17β-diol

    5β-Adiol, 5β-Androstanediol, β-Androstane-3α,17β-diol, Etiocholanediol

     A metabolite of testosterone 5β-Androstane-3α,17β-diol Chemical Structure
  18. GC49827 5-Androstenetriol

    Δ5-AT

     An active metabolite of DHEA 5-Androstenetriol Chemical Structure
  19. GC15774 5α-dihydro-11-keto Testosterone

    5α-Androstane-3,11-dione-17β-ol,11-keto Dihydrotestosterone,17β-hydroxy-5α-Androstane-3,11-dione

     5α-dihydro-11-keto Testosterone (11-KDHT; 5α-Dihydro-11-keto testosterone) is an endogenous steroid and a metabolite of 11β-Hydroxyandrostenedione. 5α-dihydro-11-keto Testosterone Chemical Structure
  20. GC19458 6β-hydroxy Testosterone

    4-Androsten-6β,17β-diol-3-one, 6β, 17β,-Dihydroxyandrost-4-en-3-one

     CYP3A4 and CYP3A5 are cytochrome P450 enzymes whose expression is induced by glucocorticoids and certain xenobiotics, including many drugs and chemical carcinogens. 6β-hydroxy Testosterone Chemical Structure
  21. GC49391 7α-Thiospironolactone

    Deacetylspironolactone, Mercaptospironolactone, SC-24813, 7α-Thio-SL

     An active metabolite of spironolactone 7α-Thiospironolactone Chemical Structure
  22. GC63764 7-α-Methylthio Spironolactone-D3 7-α-Methylthio Spironolactone-D3 Chemical Structure
  23. GC48880 7-Methoxyflavone A flavone with diverse biological activities 7-Methoxyflavone Chemical Structure
  24. GC46775 Abiraterone Acetate-d4

    CB-7630-d4

     A neuropeptide with diverse biological activities Abiraterone Acetate-d4 Chemical Structure
  25. GC46777 AC-262536 A selective androgen receptor modulator AC-262536 Chemical Structure
  26. GC31738 ACP-105 ACP-105 is an orally available, selective amd potent androgen receptor modulator (SARM), with pEC50s of 9.0 and 9.3 for AR wild type and T877A mutant, respectively. ACP-105 Chemical Structure
  27. GC67703 Adrenocorticotropic hormone TFA

    ACTH TFA; Adrenocorticotrophic hormone TFA

     Adrenocorticotropic hormone TFA Chemical Structure
  28. GC68630 AH3960

    AH3960 (compound 16c) is a androgen receptor antagonist. AH3960 can bind to both wild-type and T877 mutant androgen receptors, selectively inhibiting T877 (IC50=0.82 μM). AH3960 is also an agonist of the parathyroid hormone receptor PTHR1.

     AH3960 Chemical Structure
  29. GC31742 Ailanthone (δ13-Dehydrochaparrinone)

    Δ13-Dehydrochaparrinone

     Ailanthone (δ13-Dehydrochaparrinone) (δ13-Dehydrochaparrinone) is a potent inhibitor of both full-length androgen receptor (AR) (IC50=69nM) and constitutively active truncated AR splice variants (AR1-651 IC50=309nM). Ailanthone (δ13-Dehydrochaparrinone) Chemical Structure
  30. GC13685 Andarine

    Andarine, S-4, SARM S-4

     Andarine (S-4) is an orally active and selective nonsteroidal androgen receptor (AR) modulator (SARM) and a partial agonist, with Ki of 4 nM. Andarine (S-4) is identified as SARMs with potent and tissue-selective in vivo pharmacological activity. Andarine Chemical Structure
  31. GC67698 Androgen receptor-IN-2 Androgen receptor-IN-2 Chemical Structure
  32. GC73577 Androgen receptor-IN-6 Androgen receptor-IN-6 (compound 16) is an orally available androgen receptor (Androgen Receptor) potent inhibitor (IC50=0.12 μM in vitro), targeting the disordered N-terminal domain (NTD). Androgen receptor-IN-6 Chemical Structure
  33. GC31254 Androst-4-ene-3,17-diol, dipropanoate, (3β,17β)- (Androst-4-ene-3β,17β-diol, dipropionate) Androst-4-ene-3,17-diol, dipropanoate, (3β,17β)- (Androst-4-ene-3β,17β-diol, dipropionate) Chemical Structure
  34. GC34887 Androstanolone acetate Androstanolone acetate Chemical Structure
  35. GC60589 Apalutamide D4

    ARN-509-d4

     Apalutamide D4 (ARN-509 D4) is a deuterium labeled Apalutamide. Apalutamide is a potent and competitive androgen receptor (AR) antagonist, binding AR with an IC50 of 16 nM. Apalutamide D4 Chemical Structure
  36. GC64540 Ar-V7-IN-1 Ar-V7-IN-1 is a potent inhibitor of Ar-V7. AR-V7 is a hormone-independent splice variant of the androgen receptor. Ar-V7-IN-1 has the potential for the research of various indications, in particular cancers such as prostate cancer (extracted from patent WO2018114781A1, compound 43). Ar-V7-IN-1 Chemical Structure
  37. GC73613 ARD-1676 ARD-1676 is an orally available androgen receptor (AR) PROTAC degrader, consisting of AR ligand and cereblon ligand. ARD-1676 Chemical Structure
  38. GC73277 ARD-2051 ARD-2051 is a potent and orally active androgen receptor (AR) proteolysis-targeting chimera degrader. ARD-2051 Chemical Structure
  39. GC72850 ARD-69 ARD-69 (compound 34) is a potent PROTAC androgen receptor degrader. ARD-69 Chemical Structure
  40. GC16840 ARN-509

    ARN 509; ARN509

     ARN-509 (ARN-509) is a potent and competitive androgen receptor (AR) antagonist, binding AR with an IC50 of 16 nM. ARN-509 Chemical Structure
  41. GC62118 ARV-110

    ARV-110

     ARV-110 (ARV-110) is an orally active, specific androgen receptor (AR) PROTAC degrader. ARV-110 promotes ubiquitination and degradation of AR. ARV-110 can be used for the research of prostate cancer. ARV-110 Chemical Structure
  42. GC10547 ASC-J9 A selective enhancer of AR degradation ASC-J9 Chemical Structure
  43. GC66207 Atraric acid

    Methyl atrarate

     Atraric acid (Methyl atrarate) is a specific androgen receptor (AR) antagonist with anti-inflammatory and anticancer effects. Atraric acid represses the expression of the endogenous prostate specific antigen gene in both LNCaP and C4-2 cells. Atraric acid can also inhibit the synthesis of NO and cytokine, and suppress the MAPK-NFκB signaling pathway. Atraric acid can be used to research prostate diseases and inflammatory diseases. Atraric acid Chemical Structure
  44. GC10372 AZD3514 Androgen receptor downregulator AZD3514 Chemical Structure
  45. GC12271 Bicalutamide

    ICI 176334, ZD 176334

     Androgen receptor antagonist Bicalutamide Chemical Structure
  46. GC46925 Bicalutamide-d4 An internal standard for the quantification of bicalutamide Bicalutamide-d4 Chemical Structure
  47. GC31577 Bifluranol (BX341)

    BX341

     Bifluranol (BX341) (BX341) is an anti-androgen. Bifluranol (BX341) Chemical Structure
  48. GC35534 BMS-564929 BMS-564929 is an androgen receptor (AR) agonist, binds to androgen receptor (AR) with a Ki of 2.11±0.16 nM. BMS-564929 Chemical Structure
  49. GC41187 Boldenone Cypionate Boldenone is an anabolic androgenic steroid and synthetic derivative of testosterone that was originally developed for veterinary use. Boldenone Cypionate Chemical Structure
  50. GC35541 Boldenone Undecylenate

    Boldenone 10-Undecenoate

     Boldenone Undecylenate Chemical Structure
  51. GC73237 BWA-522 BWA-522 is an orally available small molecule protein-targeting chimera (PROTACs) with significant degradation effect on AR-FL and AR-V7. BWA-522 Chemical Structure
  52. GC17491 CITCO

    Constitutive androstane receptor (CAR) agonist

     CITCO Chemical Structure
  53. GC14560 Cl-4AS-1 steroidal androgen receptor agonist Cl-4AS-1 Chemical Structure
  54. GC62209 CLP-3094 CLP-3094 is a potent BF3 (binding function 3)-directed inhibitor of the androgen receptor (AR). CLP-3094 Chemical Structure
  55. GC47159 Cyprodinil An anilinopyrimidine fungicide Cyprodinil Chemical Structure
  56. GC13971 Cyproterone Acetate

    CPA, Cyprostat, NSC 81430, SH 714

     Androgen receptor antagonist Cyproterone Acetate Chemical Structure
  57. GC10785 Danazol

    Danocrine,Ladogal,NSC 270916,WIN 17,757

     A derivative of testosterone and ethisterone Danazol Chemical Structure
  58. GC11070 Dehydroepiandrosterone (DHEA)

    Androstenolone, trans-Dehydroandrosterone, DHEA, Diandrone, NSC 9896, Prasterone, Psicosterone

     Dehydroepiandrosterone (DHEA) and its sulfate ester, DHEAS, together represent the most abundant steroid hormones in the human body . Dehydroepiandrosterone (DHEA) Chemical Structure
  59. GC34005 Dehydroisoandrosterone 3-acetate (Dehydroepiandrosterone 3-acetate) Dehydroepiandrosterone 3-acetate is a testosterone/estrogen precursor and known modulator of vertebrate aggression. Dehydroisoandrosterone 3-acetate (Dehydroepiandrosterone 3-acetate) Chemical Structure
  60. GC47215 Dienogest-d8 An internal standard for the quantification of dienogest Dienogest-d8 Chemical Structure
  61. GC47231 Dimethomorph A morpholine fungicide Dimethomorph Chemical Structure
  62. GC31441 DJ-V-159 DJ-V-159 is an agonist for G protein-coupled receptor family C group 6 member A (GPRC6A). DJ-V-159 Chemical Structure
  63. GC49648 Enobosarm-d4

    (S)-Enobosarm-d4

     An internal standard for the quantification of enobosarm Enobosarm-d4 Chemical Structure
  64. GC64854 Enzalutamide-d3 Enzalutamide D3 is a deuterium labeled Enzalutamide (MDV3100). Enzalutamide is an androgen receptor (AR) antagonist with an IC50 of 36 nM in LNCaP prostate cells. Enzalutamide-d3 Chemical Structure
  65. GC69072 Enzalutamide-d6

    MDV3100-d6

    Enzalutamide-d6 is a deuterium-labeled Enzalutamide (MDV3100). Enzalutamide is an androgen receptor (AR) antagonist with an IC50 of 36 nM in LNCaP prostate cancer cells.

     Enzalutamide-d6 Chemical Structure
  66. GC16631 EPI-001 AR antagonist EPI-001 Chemical Structure
  67. GC73291 EPI-7170 EPI-7170, a ralaniten analogue, is a potent androgen receptor N-terminal structural domain antagonist that blocks the transcriptional activity of full-length AR (FL-AR) and AR splice variants (AR-Vs). EPI-7170 Chemical Structure
  68. GC13072 Epiandrosterone

    5α-Androstan-3β-ol-17-one, Isoandrosterone, trans-Androsterone, NSC 93996

     steroid hormone with weak androgenic activity Epiandrosterone Chemical Structure
  69. GC11796 Estradiol valerate

    Estradiol 17β-valerate, NSC 17590

     Estradiol valerate (β-estradiol 17-valerate) is a synthetic estrogen widely used in combination with other steroid hormones in hormone replacement therapy drugs. Estradiol valerate Chemical Structure
  70. GC49563 Fenhexamid

    KBR 2738

     Fenhexamid, a botryticide, is a sterol biosynthesis inhibitor. Fenhexamid Chemical Structure
  71. GC10618 Fluoxymesterone

    NSC 10704, NSC 12165

     androgen receptor agonist Fluoxymesterone Chemical Structure
  72. GC12126 Flutamide

    Niftolide, NSC 147834, NSC 251876, SCH 13521

     Androgen receptor antagonists Flutamide Chemical Structure
  73. GC48831 Flutamide-d7

    SCH 13521-d7

     An internal standard for the quantification of flutamide Flutamide-d7 Chemical Structure
  74. GC90891 Furosine (hydrochloride)

    An L-lysine derivative

     Furosine (hydrochloride) Chemical Structure
  75. GC74031 GA32 GA32 (compound 58r) is potent androgen receptor (AR)/glucocorticoid receptor (GR) dual inhibitor with IC50 values of 0.13 μM and 0.83 μM for AR and GR, respectively. GA32 Chemical Structure
  76. GC49303 Ganoderic Acid DM A triterpenoid with diverse biological activities Ganoderic Acid DM Chemical Structure
  77. GC30086 GLPG0492 A selective androgen receptor modulator GLPG0492 Chemical Structure
  78. GC30101 GLPG0492 R enantiomer GLPG0492 R enantiomer is the R enantiomer of GLPG-0492, which is a novel selective androgen receptor modulator. GLPG0492 R enantiomer Chemical Structure
  79. GC17679 GSK2881078 selective androgen receptor modulator (SARM) GSK2881078 Chemical Structure
  80. GC69200 Gumelutamide

    Gumelutamide is a tetrahydropyridine and pyrimidine compound that acts as an anti-androgen and anti-tumor agent. Gumelutamide is an androgen receptor antagonist.

     Gumelutamide Chemical Structure
  81. GC14221 HE-3235

    Apoptone,17α-Ethynyl-5α-androstane-3α,17ß-diol

     HE-3235, synthetic analogue of 3β-androstanediol, is an orally bioavailable anticancer agent. HE-3235 is active in rodent models of prostate and breast cancer. HE-3235 Chemical Structure
  82. GC62249 Honokiol DCA

    Honokiol dichloroacetate

     Honokiol DCA Chemical Structure
  83. GC36344 Isosilybin B Isosilybin B, a flavonolignan isolated from silymarin, has anti-prostate cancer (PCA) activity via inhibiting proliferation and inducing G1 phase arrest and apoptosis. Isosilybin B causes androgen receptor (AR) degradation. Isosilybin B Chemical Structure
  84. GC62106 JNJ-63576253

    TRC-253

     JNJ-63576253 (TRC-253) is a potent and orally active full antagonist of androgen receptor (AR), with IC50s of 37 and 54 nM for F877L mutant AR and wild-type AR in LNCaP cells. JNJ-63576253 can be used for the research of castration-resistant prostate cancer (CRPC). JNJ-63576253 Chemical Structure
  85. GC92094 KISS1-305 (trifluoroacetate salt)

    D-Tyr-D-Pya(4)-Asn-Ser-Phe-azaGly-Leu-Arg(Me)-Phe-NH2

     KISS1-305 is a peptide agonist of the kisspeptin receptor. KISS1-305 (trifluoroacetate salt) Chemical Structure
  86. GC18496 Leelamine (hydrochloride)

    Dehydroabietylamine

     Leelamine is a diterpene molecule whose name derives from the Sanskrit word leela which means 'play'- It has weak affinity for the human central cannabinoid (CB1) and peripheral cannabinoid (CB2) receptors, exhibiting 20% displacement of [3H]-CP55940 at a concentration of 10 uM. Leelamine (hydrochloride) Chemical Structure
  87. GC47554 Letrozole-d4 An internal standard for the quantification of letrozole Letrozole-d4 Chemical Structure
  88. GC32403 LGD-3303

    LGD-3303 is a selective androgen receptor modulator (SARM).

     LGD-3303 Chemical Structure
  89. GC32408 LGD-4033 An Analytical Reference Standard LGD-4033 Chemical Structure
  90. GC61971 Liarozole

    R 75251

     Liarozole (R75251; R85246) is an imidazole derivative and orally active retinoic acid (RA) metabolism-blocking agent (RAMBA). Liarozole Chemical Structure
  91. GC63579 Linuron Linuron is a phenylurea herbicide that is widely used to control the growth of grass and weeds in various agriculture crops and in orchards. Linuron Chemical Structure
  92. GN10142 Lupeol

    Clerodol, Fagarasterol, Lupenol, Monogynol B, NSC 90487, βViscol

     Lupeol Chemical Structure
  93. GC31380 LY2452473

    LY2452473 is an orally bioavailable, selective androgen receptor modulator (SARM).

     LY2452473 Chemical Structure
  94. GC12385 MDV3100 (Enzalutamide)

    Enzalutamide

     MDV3100(enzalutamide) is a second-generation AR antagonist with an IC50 of 36nM in LNCaP prostate cells. MDV3100 (Enzalutamide) Chemical Structure
  95. GC12974 Medroxyprogesterone acetate

    NSC 21171, NSC 26386, U-8839

     Medroxyprogesterone acetate (MPA) is a synthetic progestin. Medroxyprogesterone acetate Chemical Structure
  96. GC61850 Medroxyprogesterone acetate D3 Medroxyprogesterone acetate D3 Chemical Structure
  97. GC62061 Melengestrol acetate

    MGA, NSC 70968

     Melengestrol acetate is a progesterone derivative, acts as an orally active corticosteroid hormone to promote endometrial proliferation, pregnancy maintenance, and delay of menstrual activity. Melengestrol acetate Chemical Structure
  98. GC63066 Methenolone acetate Methenolone acetate Chemical Structure
  99. GC11837 MI-136 menin-MLL interaction inhibitor MI-136 Chemical Structure
  100. GC47674 Mifepristone-d3

    RU486-d3; RU 38486-d3

     A neuropeptide with diverse biological activities Mifepristone-d3 Chemical Structure
  101. GC36621 MK-0773

    PF-05314882

     MK-0773 is a selective androgen receptor modulators (SARMs) that binds to AR with an IC50 of 6.6 nM. MK-0773 Chemical Structure

Items 1 to 100 of 149 total

per page
  1. 1
  2. 2

Set Descending Direction