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Home >> Signaling Pathways >> Endocrinology and Hormones >> Estrogen/progestogen Receptor

Estrogen/progestogen Receptor

The estrogen/progestogen receptors are activated by the hormone estrogen/progesterone and regulate the gene transcription.

Products for  Estrogen/progestogen Receptor

  1. Cat.No. Product Name Information
  2. GC11282 β-Estradiol

    β-Estradiol, Estradiol, 17β-Oestradiol, E2

    Sex hormone

     β-Estradiol Chemical Structure
  3. GC45226 β-BHC

    β-HCH, β-Hexachlorocyclohexane, β-Lindane

     β-BHC is an isomer of the organochlorine pesticide γ-lindane that is a potential impurity found in commercial preparations of lindane. β-BHC Chemical Structure
  4. GC15975 α-Estradiol

    Alfatradiol, α-Estradiol, 17-epi Estradiol, NSC 20293, 17α-Oestradiol

     α-Estradiol is a weak estrogen and a 5α-reductase inhibitor which is used as a topical medication in the treatment of androgenic alopecia. α-Estradiol Chemical Structure
  5. GC41671 (±)-Equol 4'-sulfate (sodium salt)

    R,S-Equol 4'-Sulfate

    (±)-Equol 4'-sulfate is a gut-mediated phase II metabolite of the isoflavonoid phytoestrogen (±)-equol.

     (±)-Equol 4'-sulfate (sodium salt) Chemical Structure
  6. GC15373 (E)-2-Decenoic acid

    trans-2-Decylenic Acid

     An unsaturated fatty acid found in royal jelly (E)-2-Decenoic acid Chemical Structure
  7. GC49189 (E/Z)-4-hydroxy Tamoxifen-d5

    Afimoxifene-d5, 4-OHT-d5

     An internal standard for the quantification of (E/Z)-4-hydroxy tamoxifen (E/Z)-4-hydroxy Tamoxifen-d5 Chemical Structure
  8. GC91543 (E/Z)-Droloxifene

    3-Hydroxytamoxifen

     (E/Z)-Droloxifene is a mixture of (E)-droloxifene, a selective estrogen receptor modulator (SERM), and (Z)-droloxifene. (E/Z)-Droloxifene Chemical Structure
  9. GC40833 (E/Z)-Endoxifen

    (E/Z)-N-desmethyl-4-hydroxy Tamoxifen

     (E/Z)-Endoxifen is an active metabolite of tamoxifen produced by the sequential action of cytochrome P450 (CYP) isoforms, including CYP2D6. (E/Z)-Endoxifen Chemical Structure
  10. GC13373 (R)-DPN estrogen receptor (ER) β agonist (R)-DPN Chemical Structure
  11. GC18003 (R,R)-THC ERα receptor agonist (R,R)-THC Chemical Structure
  12. GC49520 (S)-Equol

    4',7Dihydroxyisoflavan, (-)Equol, 4',7Isoflavandiol

    An estrogen receptor β agonist

     (S)-Equol Chemical Structure
  13. GC16372 (Z)-4-Hydroxytamoxifen

    ICI 79280, trans-4-hydroxy Tamoxifen

     (Z)-4-Hydroxytamoxifen is a selective estrogen receptor modulator (SERM) that influences the binding of [3H]oestradiol to the estrogen receptor with an IC50 value of 3.3 nM. (Z)-4-Hydroxytamoxifen Chemical Structure
  14. GC91226 10-Chloroestra-1,4-diene-3,17-dione

    A sterone ERα agonist

     10-Chloroestra-1,4-diene-3,17-dione Chemical Structure
  15. GC49161 16α-hydroxy Dehydroepiandrosterone

    16α-hydroxy DHEA

     A metabolite of dehydroepiandrosterone 16α-hydroxy Dehydroepiandrosterone Chemical Structure
  16. GC41950 16α-hydroxy Estrone

    16α-hydroxy E1, 16αOHE1

     The naturally-occurring estrogens are estrone, estradiol, and estriol. 16α-hydroxy Estrone Chemical Structure
  17. GC49068 16-Epiestriol

    16-epi Estriol, 16-EpiE3, 16β-hydroxy-17α-Estradiol, NSC 26646

     A metabolite of estrone 16-Epiestriol Chemical Structure
  18. GC49848 16-Ketoestradiol

    16-keto E2, NSC 51169, 16-Oxoestradiol

     An active metabolite of estrone 16-Ketoestradiol Chemical Structure
  19. GC91109 17β-Estradiol 3-O-Sulfate (sodium salt)

    An inactive metabolite of 17β-estradiol

     17β-Estradiol 3-O-Sulfate (sodium salt) Chemical Structure
  20. GC90945 17β-Estradiol-2,4,16,16-d4 3-sulfate (sodium salt)

    An internal standard for the quantification of 17β-estradiol-3-sulfate

     17β-Estradiol-2,4,16,16-d4 3-sulfate (sodium salt) Chemical Structure
  21. GC46470 17β-Estradiol-d2

    2,4-Dideuteriostradiol, E2-d2, Estradiol-d2, β-Estradiol-d2, 17β-Oestradiol-d2

     17β-Estradiol-d2 (β-17β-Estradiol-d2) is the deuterium labeled Estradiol. 17β-Estradiol-d2 Chemical Structure
  22. GC41300 17β-hydroxy Exemestane 17β-hydroxy Exemestane is the primary active metabolite of exemestane. 17β-hydroxy Exemestane Chemical Structure
  23. GC48819 17-Epiestriol

    16α-hydroxy-17α-Estradiol, 16α,17α-Estriol, 17α-Estriol, 17-epi-Estriol, NSC 84051

     A metabolite of estrone 17-Epiestriol Chemical Structure
  24. GC17475 17-Hydroxyprogesterone

    NSC 15468, 17-OHP, 17-hydroxy Progesterone

     An endogenous progestogen and chemical intermediate 17-Hydroxyprogesterone Chemical Structure
  25. GC18635 18-hydroxy-11-deoxy Corticosterone

    18-Hydroxydeoxycorticosterone, 18-OH-DOC

     18-hydroxy-11-deoxy Corticosterone (18-OH-DOC) is a mineralocorticoid secreted by the zona fasciculata of the adrenal gland. 18-hydroxy-11-deoxy Corticosterone Chemical Structure
  26. GC49609 2-bromo 17β-Estradiol

    2-bromo E2, 2-bromo β-Estradiol, 2-bromo Estradiol, NSC 105460, 2-bromo 17β-Oestradiol

     A synthetic steroid and inhibitor of estrogen 2-hydroxylase 2-bromo 17β-Estradiol Chemical Structure
  27. GC49172 2-hydroxy Estrone

    Catecholestrone, 2-hydroxy E1, 2-OHE1

     An active metabolite of estrone 2-hydroxy Estrone Chemical Structure
  28. GC48910 2-Hydroxyanthraquinone

    2-hydroxy-9,10-Anthraquinone, 2-hATQ, β-Hydroxyanthraquinone, NSC 2595

     An anthraquinone with antibacterial and estrogenic activities 2-Hydroxyanthraquinone Chemical Structure
  29. GC18462 3-Formylsalicylic Acid

    NSC 55753

     3-Formylsalicylic acid is a non-competitive inhibitor of estrone sulfatase (IC50 = 150 nM; Ki = 120 nM), the enzyme that converts estrone sulfate to estrone. 3-Formylsalicylic Acid Chemical Structure
  30. GC48824 4-hydroxy Estrone

    4-hydroxy E1, 4-OHE1

     A metabolite of estrone 4-hydroxy Estrone Chemical Structure
  31. GC19552 4-Hydroxyestradiol

    4-Hydroxy-17β-estradiol

    4-Hydroxyestradiol, an metabolite of estradiol, forms adducts with adenine (3) and guanine (N7) by depurinating sites in DNA of cultured human breast epithelial cells.

     4-Hydroxyestradiol Chemical Structure
  32. GC17803 4-Hydroxytamoxifen

    Afimoxifene, 4-OHT

     4-hydroxytamoxifen is a major metabolite of tamoxifen and selective estrogen receptor antagonist. 4-Hydroxytamoxifen Chemical Structure
  33. GC49562 4-methoxy Estrone

    4-MeOE1, 4-methoxy E1

     An active metabolite of estrone 4-methoxy Estrone Chemical Structure
  34. GC11606 4-Methylbenzylidene camphor

    Enzacamene|Eusolex 6300|4-MBC|Neo Heliopan MBC|Parsol 500|Uvinul MBC 95

     ultraviolet light blocker used in cosmetics and sunscreen preparations that also has estrogenic activities. 4-Methylbenzylidene camphor Chemical Structure
  35. GC42473 4-tert-Octylphenol diethoxylate

    OP2EO

     4-tert-Octylphenol diethoxylate is a degradation product of the multi-purpose surfactant, Triton X. 4-tert-Octylphenol diethoxylate Chemical Structure
  36. GC52365 4-tert-Octylphenol monoethoxylate

    NSC 5259, OP1EO

     An alkylphenolethoxylate and a degradation product of non-ionic surfactants 4-tert-Octylphenol monoethoxylate Chemical Structure
  37. GC13917 4’-hydroxy Tamoxifen metabolite of tamoxifen, an estrogen receptor modulator 4’-hydroxy Tamoxifen Chemical Structure
  38. GC49326 5β-Dihydroprogesterone

    5β-DHP, NSC 82868, 5β-Pregnanedione

     A progesterone receptor agonist and metabolite of progesterone 5β-Dihydroprogesterone Chemical Structure
  39. GC90889 5-(3'-Hydroxyphenyl)-γ-Valerolactone

    A metabolite of various polyphenols

     5-(3'-Hydroxyphenyl)-γ-Valerolactone Chemical Structure
  40. GC90492 5-Dibromomethyl Anastrozole

    A synthetic intermediate of anastrozole

     5-Dibromomethyl Anastrozole Chemical Structure
  41. GC49391 7α-Thiospironolactone

    Deacetylspironolactone, Mercaptospironolactone, SC-24813, 7α-Thio-SL

     An active metabolite of spironolactone 7α-Thiospironolactone Chemical Structure
  42. GC17119 8-Prenylnaringenin

    Flavaprenin,8-PN

     estrogen receptor inhibitor 8-Prenylnaringenin Chemical Structure
  43. GC50091 AC 186 Potent and selective ERβ agonist; neuroprotective AC 186 Chemical Structure
  44. GC13297 Altrenogest

    Allyltrenbolone, DRC 6246, RU 2267

     Progestogen receptor agonist Altrenogest Chemical Structure
  45. GC14405 AZD9496 estrogen receptor inhibitor, orally active AZD9496 Chemical Structure
  46. GC17588 Bavachin

    Corylifolin

     estrogen receptors ERα and ERβ activator Bavachin Chemical Structure
  47. GC14883 Bazedoxifene Bazedoxifene Chemical Structure
  48. GC10852 Bazedoxifene acetate

    TSE 424

     A selective estrogen receptor modulator Bazedoxifene acetate Chemical Structure
  49. GC10245 Bazedoxifene HCl Bazedoxifene HCl (TSE-424 hydrochloride) is an oral active, BBB-penetrant nonsteroidal selective estrogen receptor modulator (SERM), with IC50s of 23 nM and 99 nM for ERα and ERβ, respectively. Bazedoxifene HCl can be used for the research of osteoporosis. Bazedoxifene HCl acts as an inhibitor of IL-6/GP130 protein-protein interactions. Bazedoxifene HCl can be used for the research of pancreatic cancer. Bazedoxifene HCl Chemical Structure
  50. GC49757 Bazedoxifene N-oxide An oxidative degradation product of bazedoxifene Bazedoxifene N-oxide Chemical Structure
  51. GC46907 Bazedoxifene-d4 An internal standard for the quantification of bazedoxifene Bazedoxifene-d4 Chemical Structure
  52. GC11144 Chlormadinone acetate

    NSC 92338

     steroidal progestin with additional antiandrogen and antigonadotropic effects Chlormadinone acetate Chemical Structure
  53. GC10012 Chlorotrianisene

    NSC 10108, TACE, Tri-p-anisylchloroethylene

     Estrogen agonist Chlorotrianisene Chemical Structure
  54. GC15366 Clomiphene citrate

    Clomifene, Omifin, NSC 35770

     Selective estrogen receptor modulator Clomiphene citrate Chemical Structure
  55. GC10002 Coumestrol

    NSC 22842

     competitive binder of the estrogen receptors ERα Coumestrol Chemical Structure
  56. GC45413 Cridanimod (sodium salt)

    10-Carboxymethyl-9-Acridanone

       Cridanimod (sodium salt) Chemical Structure
  57. GC10180 Cyclofenil

    ICI 48213, NSC 86464

     Non-steroidal selective estrogen receptor modulator (SERM) Cyclofenil Chemical Structure
  58. GC47168 Daidzein-d4 An internal standard for the quantification of daidzein Daidzein-d4 Chemical Structure
  59. GC49025 Desogestrel-13C2-d2 An internal standard for the quantification of desogestrel Desogestrel-13C2-d2 Chemical Structure
  60. GC17688 Diarylpropionitrile(DPN)

    diarylpropionitrile

     Diarylpropionitrile(DPN) (Diarylpropionitrile) is a non-steroidal estrogen receptor β (ERβ) selective ligand, with an EC50 of 0.85 nM. Diarylpropionitrile(DPN) Chemical Structure
  61. GC15578 Dienogest

    STS 557

     Orally active synthetic progesterone Dienogest Chemical Structure
  62. GC47215 Dienogest-d8 An internal standard for the quantification of dienogest Dienogest-d8 Chemical Structure
  63. GC10663 Dihydrodaidzein

    (±)-Dihydrodaidzein,4',7-dihydroxy Isoflavanone

     estrogen receptor agonist Dihydrodaidzein Chemical Structure
  64. GC12379 Drospirenone

    1,2-dihydro Spirorenone, ZK 30595

     Synthetic progestin Drospirenone Chemical Structure
  65. GC52420 Drospirenone-13C3

    1,2-dihydro Spirorenone-13C3, ZK 30595-13C3

     An internal standard for the quantification of drospirenone Drospirenone-13C3 Chemical Structure
  66. GC12140 Endoxifen Endoxifen Z-isomer is the most important Tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha (ERα). Endoxifen Chemical Structure
  67. GC18333 Equilenin

    (+)-Equilenin, d-Equilenin, NSC 9901

     Equilenin is an equine estrogen found in the urine of pregnant mares. Equilenin Chemical Structure
  68. GC16292 Equol non-steroidal estrogen Equol Chemical Structure
  69. GC10389 ERB 041 ERB 041 (ERB-041) is a potent and selective estrogen receptor (ER) β agonist with IC50s of 5.4, 3.1 and 3.7 nM for human, rat and mouse ERβ, respectively. ERB 041 displays >200-fold selectivity for ERβ over ERα. ERB 041 is a potent skin cancer chemopreventive agent that acts by dampening the WNT/β-catenin signaling pathway. ERB 041 induces ovarian cancer apoptosis. ERB 041 Chemical Structure
  70. GC11822 Erteberel (LY500307)

    LY500307

     Erteberel (LY500307) (LY500307) is a potent and selective estrogen receptor beta (ERβ) agonist with Ki and EC50 of 1.54 nM and 3.61 nM, respectively. Erteberel (LY500307) Chemical Structure
  71. GC47309 Estetrol (hydrate)

    E4, 15α-Hydroxyestriol

     A naturally occurring estrogen Estetrol (hydrate) Chemical Structure
  72. GC48979 Estradiol 17-(β-D-Glucuronide) (sodium salt hydrate)

    E217G, βEstradiol 17(βDGlucuronide), 17βEstradiol 17(βDGlucuronide), 17βOestradiol 17(βDGlucuronide)

     A substrate of multidrug resistance protein 2 Estradiol 17-(β-D-Glucuronide) (sodium salt hydrate) Chemical Structure
  73. GC43629 Estradiol 3-sulfate 17β-Glucuronide (potassium salt) Estradiol 3-sulfate is a sulfated form of the steroid hormone 17β-estradiol, and is common in fetal plasma and in the breast tissues of patients with mammary carcinoma. Estradiol 3-sulfate 17β-Glucuronide (potassium salt) Chemical Structure
  74. GC10139 Estradiol Cypionate

    Estradiol 17β-Cyclopentanepropionate, Estradiol 17-Cypionate, NSC 3354

     Estrogen receptor inhibitor Estradiol Cypionate Chemical Structure
  75. GC12182 Estriol

    E3, 16α-hydroxy-17β-Estradiol, 1,3,5(10)-Estratriene-3,16α,17β-triol

     Estrogen receptor antagonist Estriol Chemical Structure
  76. GC45450 Estriol-d2

    E3-d2, 16αhydroxy17βEstradiol-d2, 1,3,5(10)Estratriene3,16α,17βtriol-d2

     Estriol-d2 is the deuterium labeled Estriol. Estriol is an antagonist of the G-protein coupled estrogen receptor in estrogen receptor-negative breast cancer cells. Estriol-d2 Chemical Structure
  77. GC14385 Estrone

    E1

     Estrone is one of the three major endogenous estrogens, the others being estradiol and estriol. Estrone Chemical Structure
  78. GC45451 Estrone 3-methyl ether

    (+)-Estrone methyl ether, 3-O-methyl Estrone, NSC 88911

       Estrone 3-methyl ether Chemical Structure
  79. GC49254 Estrone-3-Glucuronide (sodium salt hydrate)

    E1G, Estrone Glucuronide, Estrone β-D-Glucuronide

     A metabolite of 17β-estradiol Estrone-3-Glucuronide (sodium salt hydrate) Chemical Structure
  80. GC45452 Estrone-d2

    E1-d2

       Estrone-d2 Chemical Structure
  81. GC16852 Estropipate

    Piperazine Estrone Sulfate

     Estrogen receptor agonist Estropipate Chemical Structure
  82. GC12148 Ethinyl Estradiol

    Ethynyl βEstradiol, Ethynyl 17βEstradiol, Ethynyl 17βOestradiol, Ethynyl E2

     Ethinyl Estradiol (17α-Ethynylestradiol;Ethynylestradiol) is an orally bio-active estrogen used in almost all modern formulations of combined oral contraceptive pills. Ethinyl Estradiol Chemical Structure
  83. GC11436 Ethisterone Progestogen hormone Ethisterone Chemical Structure
  84. GC12000 Ethynodiol diacetate

    SC-11800

     Progestogen receptor agonist Ethynodiol diacetate Chemical Structure
  85. GC47320 Ethynyl Estradiol 3-β-D-Glucuronide (hydrate)

    17α-Ethynylestradiol 3-Glucuronide

     A metabolite of ethynyl estradiol Ethynyl Estradiol 3-β-D-Glucuronide (hydrate) Chemical Structure
  86. GC13303 Etonogestrel

    ORG 3236, 3-keto Desogestrel, 3-oxo Desogestrel

     steroidal progestin Etonogestrel Chemical Structure
  87. GC49563 Fenhexamid

    KBR 2738

     Fenhexamid, a botryticide, is a sterol biosynthesis inhibitor. Fenhexamid Chemical Structure
  88. GC14131 FERb 033 ERβ receptor agonist FERb 033 Chemical Structure
  89. GC18641 Ferutinin Ferutinin is a plant-derived ester of a sesquiterpenic alcohol that acts as an agonist for estrogen receptor (ER) α (IC50 = 33.1 nM) and an agonist/antagonist for ERβ (IC50 = 180.5 nM). Ferutinin Chemical Structure
  90. GC18000 Fulvestrant (ICI 182,780)

    ICI 182780

     Fulvestrant is a selective estrogen receptor (ER) antagonist. It binds, blocks and degrades estrogen receptor, then inhibits estrogen receptor(ER)-mediated transcriptional activity with an IC50 of 9.4 nM . Fulvestrant (ICI 182,780) Chemical Structure
  91. GC49878 Fulvestrant 9-sulfone An estrogen receptor antagonist and a derivative of fulvestrant Fulvestrant 9-sulfone Chemical Structure
  92. GC40241 Fulvestrant-d3

    ICI 182780-d3; ZD 9238-d3; ZM 182780-d3

     Fulvestrant-d3 is intended for use as an internal standard for the quantification of fulvestrant by GC- or LC-MS. Fulvestrant-d3 Chemical Structure
  93. GC12766 G-1 G-1 is a selective and potent agonist of GPR30 with EC50 value about 2 nM. G-1 Chemical Structure
  94. GC16618 G-15

    A GPER receptor antagonist

     G-15 Chemical Structure
  95. GC14902 G-36

    GPER activator

     G-36 Chemical Structure
  96. GC10017 Gestodene Progestogen hormonal contraceptive Gestodene Chemical Structure
  97. GC48763 Gestodene-d6

    SHB 331-d6; WL 70-d6

     An internal standard for the quantification of gestodene Gestodene-d6 Chemical Structure
  98. GC10558 GSK 4716 estrogen-related receptors ERRβ and ERRγ agonist GSK 4716 Chemical Structure
  99. GC15324 Hexestrol

    Hexoestrol, meso-Hexestrol, NSC 9894

     Estrogen receptor agonist Hexestrol Chemical Structure
  100. GC15599 Hydroxyprogesterone caproate

    17-Caproxyprogesterone, HPC, Hormofort, Hydroxyprogesterone Hexanoate, NSC 17592, Progesterone Caproate, 17α-hydroxy Progesterone Caproate

     synthetic progestational agent Hydroxyprogesterone caproate Chemical Structure
  101. GC44036 Lasofoxifene

    CP 336,156

     Lasofoxifene is a third-generation, non-steroidal selective estrogen receptor modulator (SERM). Lasofoxifene Chemical Structure

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