Home >> Signaling Pathways >> Endocrinology and Hormones >> Estrogen/progestogen Receptor

Estrogen/progestogen Receptor

The estrogen/progestogen receptors are activated by the hormone estrogen/progesterone and regulate the gene transcription.

Products for  Estrogen/progestogen Receptor

  1. Cat.No. Product Name Information
  2. GC11282 β-Estradiol

    Sex hormone

     β-Estradiol  Chemical Structure
  3. GC15975 α-Estradiol α-Estradiol is a weak estrogen and a 5α-reductase inhibitor which is used as a topical medication in the treatment of androgenic alopecia. α-Estradiol  Chemical Structure
  4. GC41671 (±)-Equol 4'-sulfate (sodium salt)

    (±)-Equol 4'-sulfate is a gut-mediated phase II metabolite of the isoflavonoid phytoestrogen (±)-equol.

    (±)-Equol 4'-sulfate (sodium salt)  Chemical Structure
  5. GC15373 (E)-2-Decenoic acid An unsaturated fatty acid found in royal jelly (E)-2-Decenoic acid  Chemical Structure
  6. GC49189 (E/Z)-4-hydroxy Tamoxifen-d5 An internal standard for the quantification of (E/Z)-4-hydroxy tamoxifen (E/Z)-4-hydroxy Tamoxifen-d5  Chemical Structure
  7. GC40833 (E/Z)-Endoxifen (E/Z)-Endoxifen is an active metabolite of tamoxifen produced by the sequential action of cytochrome P450 (CYP) isoforms, including CYP2D6. (E/Z)-Endoxifen  Chemical Structure
  8. GC13373 (R)-DPN estrogen receptor (ER) β agonist (R)-DPN  Chemical Structure
  9. GC18003 (R,R)-THC ERα receptor agonist (R,R)-THC  Chemical Structure
  10. GC49520 (S)-Equol

    An estrogen receptor β agonist

    (S)-Equol  Chemical Structure
  11. GC16372 (Z)-4-Hydroxytamoxifen (Z)-4-Hydroxytamoxifen is a metabolite of Tamoxifen. (Z)-4-Hydroxytamoxifen shows higher affinity for the ER than Tamoxifen. (Z)-4-Hydroxytamoxifen induces a non-apoptotic cytotoxic effect in human endometrial adenocarcinoma cells. (Z)-4-Hydroxytamoxifen  Chemical Structure
  12. GC49161 16α-hydroxy Dehydroepiandrosterone A metabolite of dehydroepiandrosterone 16α-hydroxy Dehydroepiandrosterone  Chemical Structure
  13. GC41950 16α-hydroxy Estrone The naturally-occurring estrogens are estrone, estradiol, and estriol. 16α-hydroxy Estrone  Chemical Structure
  14. GC49068 16-Epiestriol A metabolite of estrone 16-Epiestriol  Chemical Structure
  15. GC49848 16-Ketoestradiol An active metabolite of estrone 16-Ketoestradiol  Chemical Structure
  16. GC46470 17β-Estradiol-d2 17β-Estradiol-d2 (β-17β-Estradiol-d2) is the deuterium labeled Estradiol. 17β-Estradiol-d2  Chemical Structure
  17. GC41300 17β-hydroxy Exemestane 17β-hydroxy Exemestane is the primary active metabolite of exemestane. 17β-hydroxy Exemestane  Chemical Structure
  18. GC48819 17-Epiestriol A metabolite of estrone 17-Epiestriol  Chemical Structure
  19. GC17475 17-Hydroxyprogesterone An endogenous progestogen and chemical intermediate 17-Hydroxyprogesterone  Chemical Structure
  20. GC18635 18-hydroxy-11-deoxy Corticosterone 18-hydroxy-11-deoxy Corticosterone (18-OH-DOC) is a mineralocorticoid secreted by the zona fasciculata of the adrenal gland. 18-hydroxy-11-deoxy Corticosterone  Chemical Structure
  21. GC49609 2-bromo 17β-Estradiol A synthetic steroid and inhibitor of estrogen 2-hydroxylase 2-bromo 17β-Estradiol  Chemical Structure
  22. GC49172 2-hydroxy Estrone An active metabolite of estrone 2-hydroxy Estrone  Chemical Structure
  23. GC48910 2-Hydroxyanthraquinone An anthraquinone with antibacterial and estrogenic activities 2-Hydroxyanthraquinone  Chemical Structure
  24. GC18462 3-Formylsalicylic Acid 3-Formylsalicylic acid is a non-competitive inhibitor of estrone sulfatase (IC50 = 150 nM; Ki = 120 nM), the enzyme that converts estrone sulfate to estrone. 3-Formylsalicylic Acid  Chemical Structure
  25. GC48824 4-hydroxy Estrone A metabolite of estrone 4-hydroxy Estrone  Chemical Structure
  26. GC17803 4-Hydroxytamoxifen 4-Hydroxytamoxifen (Afimoxifene) is a racemic compound of (Z)-4-Hydroxytamoxifen and (E)-4-Hydroxytamoxifen isomers. 4-Hydroxytamoxifen is an estrogen receptor modulator. 4-Hydroxytamoxifen  Chemical Structure
  27. GC49562 4-methoxy Estrone An active metabolite of estrone 4-methoxy Estrone  Chemical Structure
  28. GC11606 4-Methylbenzylidene camphor ultraviolet light blocker used in cosmetics and sunscreen preparations that also has estrogenic activities. 4-Methylbenzylidene camphor  Chemical Structure
  29. GC42473 4-tert-Octylphenol diethoxylate 4-tert-Octylphenol diethoxylate is a degradation product of the multi-purpose surfactant, Triton X. 4-tert-Octylphenol diethoxylate  Chemical Structure
  30. GC52365 4-tert-Octylphenol monoethoxylate An alkylphenolethoxylate and a degradation product of non-ionic surfactants 4-tert-Octylphenol monoethoxylate  Chemical Structure
  31. GC13917 4’-hydroxy Tamoxifen metabolite of tamoxifen, an estrogen receptor modulator 4’-hydroxy Tamoxifen  Chemical Structure
  32. GC49326 5β-Dihydroprogesterone A progesterone receptor agonist and metabolite of progesterone 5β-Dihydroprogesterone  Chemical Structure
  33. GC49391 7α-Thiospironolactone An active metabolite of spironolactone 7α-Thiospironolactone  Chemical Structure
  34. GC17119 8-Prenylnaringenin estrogen receptor inhibitor 8-Prenylnaringenin  Chemical Structure
  35. GC50091 AC 186 Potent and selective ERβ agonist; neuroprotective AC 186  Chemical Structure
  36. GC13297 Altrenogest Progestogen receptor agonist Altrenogest  Chemical Structure
  37. GC14405 AZD9496 estrogen receptor inhibitor, orally active AZD9496  Chemical Structure
  38. GC17588 Bavachin estrogen receptors ERα and ERβ activator Bavachin  Chemical Structure
  39. GC14883 Bazedoxifene Bazedoxifene  Chemical Structure
  40. GC10852 Bazedoxifene acetate A selective estrogen receptor modulator Bazedoxifene acetate  Chemical Structure
  41. GC10245 Bazedoxifene HCl Bazedoxifene HCl (TSE-424 hydrochloride) is an oral active, BBB-penetrant nonsteroidal selective estrogen receptor modulator (SERM), with IC50s of 23 nM and 99 nM for ERα and ERβ, respectively. Bazedoxifene HCl can be used for the research of osteoporosis. Bazedoxifene HCl acts as an inhibitor of IL-6/GP130 protein-protein interactions. Bazedoxifene HCl can be used for the research of pancreatic cancer. Bazedoxifene HCl  Chemical Structure
  42. GC49757 Bazedoxifene N-oxide An oxidative degradation product of bazedoxifene Bazedoxifene N-oxide  Chemical Structure
  43. GC46907 Bazedoxifene-d4 An internal standard for the quantification of bazedoxifene Bazedoxifene-d4  Chemical Structure
  44. GC11144 Chlormadinone acetate steroidal progestin with additional antiandrogen and antigonadotropic effects Chlormadinone acetate  Chemical Structure
  45. GC10012 Chlorotrianisene Estrogen agonist Chlorotrianisene  Chemical Structure
  46. GC15366 Clomiphene citrate Selective estrogen receptor modulator Clomiphene citrate  Chemical Structure
  47. GC10002 Coumestrol competitive binder of the estrogen receptors ERα Coumestrol  Chemical Structure
  48. GC45413 Cridanimod (sodium salt)   Cridanimod (sodium salt)  Chemical Structure
  49. GC10180 Cyclofenil Non-steroidal selective estrogen receptor modulator (SERM) Cyclofenil  Chemical Structure
  50. GC47168 Daidzein-d4 An internal standard for the quantification of daidzein Daidzein-d4  Chemical Structure
  51. GC49025 Desogestrel-13C2-d2 An internal standard for the quantification of desogestrel Desogestrel-13C2-d2  Chemical Structure
  52. GC17688 Diarylpropionitrile(DPN) Diarylpropionitrile(DPN) (Diarylpropionitrile) is a non-steroidal estrogen receptor β (ERβ) selective ligand, with an EC50 of 0.85 nM. Diarylpropionitrile(DPN)  Chemical Structure
  53. GC15578 Dienogest Orally active synthetic progesterone Dienogest  Chemical Structure
  54. GC47215 Dienogest-d8 An internal standard for the quantification of dienogest Dienogest-d8  Chemical Structure
  55. GC10663 Dihydrodaidzein estrogen receptor agonist Dihydrodaidzein  Chemical Structure
  56. GC12379 Drospirenone Synthetic progestin Drospirenone  Chemical Structure
  57. GC52420 Drospirenone-13C3 An internal standard for the quantification of drospirenone Drospirenone-13C3  Chemical Structure
  58. GC12140 Endoxifen Endoxifen Z-isomer is the most important Tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha (ERα). Endoxifen  Chemical Structure
  59. GC18333 Equilenin Equilenin is an equine estrogen found in the urine of pregnant mares. Equilenin  Chemical Structure
  60. GC16292 Equol non-steroidal estrogen Equol  Chemical Structure
  61. GC10389 ERB 041 ERB 041 (ERB-041) is a potent and selective estrogen receptor (ER) β agonist with IC50s of 5.4, 3.1 and 3.7 nM for human, rat and mouse ERβ, respectively. ERB 041 displays >200-fold selectivity for ERβ over ERα. ERB 041 is a potent skin cancer chemopreventive agent that acts by dampening the WNT/β-catenin signaling pathway. ERB 041 induces ovarian cancer apoptosis. ERB 041  Chemical Structure
  62. GC11822 Erteberel (LY500307) Erteberel (LY500307) (LY500307) is a potent and selective estrogen receptor beta (ERβ) agonist with Ki and EC50 of 1.54 nM and 3.61 nM, respectively. Erteberel (LY500307)  Chemical Structure
  63. GC47309 Estetrol (hydrate) A naturally occurring estrogen Estetrol (hydrate)  Chemical Structure
  64. GC48979 Estradiol 17-(β-D-Glucuronide) (sodium salt hydrate) A substrate of multidrug resistance protein 2 Estradiol 17-(β-D-Glucuronide) (sodium salt hydrate)  Chemical Structure
  65. GC43629 Estradiol 3-sulfate 17β-Glucuronide (potassium salt) Estradiol 3-sulfate is a sulfated form of the steroid hormone 17β-estradiol, and is common in fetal plasma and in the breast tissues of patients with mammary carcinoma. Estradiol 3-sulfate 17β-Glucuronide (potassium salt)  Chemical Structure
  66. GC10139 Estradiol Cypionate Estrogen receptor inhibitor Estradiol Cypionate  Chemical Structure
  67. GC12182 Estriol Estrogen receptor antagonist Estriol  Chemical Structure
  68. GC45450 Estriol-d2 Estriol-d2 is the deuterium labeled Estriol. Estriol is an antagonist of the G-protein coupled estrogen receptor in estrogen receptor-negative breast cancer cells. Estriol-d2  Chemical Structure
  69. GC14385 Estrone Estrogenic hormone Estrone  Chemical Structure
  70. GC45451 Estrone 3-methyl ether   Estrone 3-methyl ether  Chemical Structure
  71. GC43631 Estrone 3-sulfate (sodium salt) Estrone sulfate, a biologically inactive form of estrogen, is a major circulating plasma estrogen that is converted into the biologically active estrogen, estrone (E1) by steroid sulfatase (STS). strone sulfate can be used for the research of breast cancer. Estrone 3-sulfate (sodium salt)  Chemical Structure
  72. GC49254 Estrone-3-Glucuronide (sodium salt hydrate) A metabolite of 17β-estradiol Estrone-3-Glucuronide (sodium salt hydrate)  Chemical Structure
  73. GC45452 Estrone-d2   Estrone-d2  Chemical Structure
  74. GC16852 Estropipate Estrogen receptor agonist Estropipate  Chemical Structure
  75. GC12148 Ethinyl Estradiol Ethinyl Estradiol (17α-Ethynylestradiol;Ethynylestradiol) is an orally bio-active estrogen used in almost all modern formulations of combined oral contraceptive pills. Ethinyl Estradiol  Chemical Structure
  76. GC11436 Ethisterone Progestogen hormone Ethisterone  Chemical Structure
  77. GC12000 Ethynodiol diacetate Progestogen receptor agonist Ethynodiol diacetate  Chemical Structure
  78. GC47320 Ethynyl Estradiol 3-β-D-Glucuronide (hydrate) A metabolite of ethynyl estradiol Ethynyl Estradiol 3-β-D-Glucuronide (hydrate)  Chemical Structure
  79. GC13303 Etonogestrel steroidal progestin Etonogestrel  Chemical Structure
  80. GC49563 Fenhexamid Fenhexamid, a botryticide, is a sterol biosynthesis inhibitor. Fenhexamid  Chemical Structure
  81. GC14131 FERb 033 ERβ receptor agonist FERb 033  Chemical Structure
  82. GC18641 Ferutinin Ferutinin is a plant-derived ester of a sesquiterpenic alcohol that acts as an agonist for estrogen receptor (ER) α (IC50 = 33.1 nM) and an agonist/antagonist for ERβ (IC50 = 180.5 nM). Ferutinin  Chemical Structure
  83. GC18000 Fulvestrant (ICI 182,780)

    Fulvestrant is a selective estrogen receptor (ER) antagonist. It binds, blocks and degrades ER, then inhibits ER-mediated transcriptional activity with an IC50 of 9.4 nM.

    Fulvestrant (ICI 182,780)  Chemical Structure
  84. GC49878 Fulvestrant 9-sulfone An estrogen receptor antagonist and a derivative of fulvestrant Fulvestrant 9-sulfone  Chemical Structure
  85. GC12766 G-1

    G-1 is a selective and potent agonist of GPR30 with EC50 value about 2 nM.

    G-1  Chemical Structure
  86. GC16618 G-15

    A GPER receptor antagonist

    G-15  Chemical Structure
  87. GC14902 G-36

    GPER activator

    G-36  Chemical Structure
  88. GC10017 Gestodene Progestogen hormonal contraceptive Gestodene  Chemical Structure
  89. GC48763 Gestodene-d6 An internal standard for the quantification of gestodene Gestodene-d6  Chemical Structure
  90. GC10558 GSK 4716 estrogen-related receptors ERRβ and ERRγ agonist GSK 4716  Chemical Structure
  91. GC15324 Hexestrol Estrogen receptor agonist Hexestrol  Chemical Structure
  92. GC15599 Hydroxyprogesterone caproate synthetic progestational agent Hydroxyprogesterone caproate  Chemical Structure
  93. GC44036 Lasofoxifene Lasofoxifene is a third-generation, non-steroidal selective estrogen receptor modulator (SERM). Lasofoxifene  Chemical Structure
  94. GC11425 Lasofoxifene (tartrate) third-generation, non-steroidal selective estrogen receptor modulator (SERM) Lasofoxifene (tartrate)  Chemical Structure
  95. GC47554 Letrozole-d4 An internal standard for the quantification of letrozole Letrozole-d4  Chemical Structure
  96. GC14704 Levonorgestrel Estrogen/progestogen receptor agonist Levonorgestrel  Chemical Structure
  97. GC11781 Medroxyprogesterone potent progesterone receptor agonist Medroxyprogesterone  Chemical Structure
  98. GC12974 Medroxyprogesterone acetate

    Steroidal progestin

    Medroxyprogesterone acetate  Chemical Structure
  99. GC11688 Megestrol Acetate Anti-estrogen agent Megestrol Acetate  Chemical Structure
  100. GC25627 Menotropin Menotropin (Human Menopausal Gonadotrophin) is a hormonally active medication for the treatment of fertility disturbances, which are extracted from the urine of postmenopausal women. Menotropin  Chemical Structure
  101. GC17161 Methylpiperidino pyrazole

    ERα selective antagonist

    Methylpiperidino pyrazole  Chemical Structure

Items 1 to 100 of 138 total

per page
  1. 1
  2. 2

Set Descending Direction