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Home >> Signaling Pathways >> Endocrinology and Hormones >> Opioid Receptor

Opioid Receptor

Opioid receptor is a group of G protein-coupled receptors with opioids as ligands.

Products for  Opioid Receptor

  1. Cat.No. Product Name Information
  2. GC60391 β-Casomorphin, bovine TFA

    β-Casomorphin-7 (bovine) (TFA); Bovine β-casomorphin-7 TFA

     β-Casomorphin, bovine TFA Chemical Structure
  3. GC61484 β-Casomorphin, human TFA

    Human β-casomorphin 7 TFA

     β-Casomorphin, human TFA Chemical Structure
  4. GC38005 β-Endorphin, equine β-Endorphin, equine is an endogenous opioid peptide, which binds at high affinity to both μ/δ opioid receptors. β-Endorphin, equine Chemical Structure
  5. GC38030 β-Endorphin, equine (TFA) β-Endorphin, equine (TFA) Chemical Structure
  6. GC72132 β-Endorphin, equine TFA β-Endorphin, equine TFA is an endogenous opioid peptide, which binds at high affinity to both μ/δ opioid receptors. β-Endorphin, equine TFA Chemical Structure
  7. GC33736 β-Casomorphin, bovine (β-Casomorphin-7 (bovine)) β-Casomorphin, bovine (β-Casomorphin-7 (bovine)) (β-Casomorphin-7 (bovine) ) is a opioid peptide with an IC50 of 14 μM in an Opioid receptors binding assay. β-Casomorphin, bovine (β-Casomorphin-7 (bovine)) Chemical Structure
  8. GC33784 β-Casomorphin, human (Human β-casomorphin 7)

    Human β-casomorphin 7

     is an opioid peptide, acts as an agonist of opioid receptor. β-Casomorphin, human (Human β-casomorphin 7) Chemical Structure
  9. GC31117 β-Endorphin, human β-Endorphin, human, a prominent endogenous peptide, existing in the hypophysis cerebri and hypothalamus, is an agonist of opioid receptor, with preferred affinity for μ-opioid receptor and δ-opioid receptor; β-Endorphin, human exhibits antinociception activity. β-Endorphin, human Chemical Structure
  10. GC15938 β-Funaltrexamine hydrochloride

    μ opioid receptor antagonist

     β-Funaltrexamine hydrochloride Chemical Structure
  11. GC64007 (±)-U-50488 hydrate hydrochloride

    (±)-Trans-(1R,2R)-U-50488 hydrate hydrochloride

     (±)-U-50488 hydrate hydrochloride Chemical Structure
  12. GC15885 (±)-U-50488 hydrochloride

    (±)-Trans-(1R,2R)-U-50488 hydrochloride

    κ-opioid receptor agonist, selective

     (±)-U-50488 hydrochloride Chemical Structure
  13. GC12688 (+)-U-50488 hydrochloride

    (+)-Trans-(1R,2R)-U-50488 hydrochloride

     Selective κ-opioid agonist (+)-U-50488 hydrochloride Chemical Structure
  14. GC15944 (-)-U-50488 hydrochloride

    (-)-Trans-(1S,2S)-U-50488 hydrochloride

     (-)-U-50488 hydrochloride is a selective agonist of the kappa opioid receptor (KOR) with an IC50 value of 0.25μM. (-)-U-50488 hydrochloride Chemical Structure
  15. GC70081 (1R,2R)-U-50488 hydrochloride

    (1R,2R)-U-50488 hydrochloride is the absolute configuration of (±)-U-50488 hydrochloride. (±)-U-50488 hydrochloride is a κ opioid receptor agonist.

     (1R,2R)-U-50488 hydrochloride Chemical Structure
  16. GC69798 (Rac)-SNC80

    (Rac)-NIH 10815

    (Rac)-SNC80 is the racemic form of SNC80. SNC80 (NIH 10815) is an effective and highly selective non-peptide delta-opioid receptor agonist with a Ki of 1.78 nM and IC50 of 2.73 nM. SNC80 has anti-nociceptive, anti-hyperalgesic, and antidepressant-like effects, and can be used in research on various types of headaches.

     (Rac)-SNC80 Chemical Structure
  17. GC66679 2,6-Dimethyl-L-tyrosine

    Dmt

     2,6-Dimethyl-L-tyrosine (Dmt) is a tyrosine derivative that enhances receptor affinity, functional bioactivity and in vivo analgesia of opioid peptides. 2,6-Dimethyl-L-tyrosine Chemical Structure
  18. GC48735 2-methyl AP-237-d7 (hydrochloride)

    2-methyl Buccinazine-d7

     2-methyl AP-237-d7 (hydrochloride) Chemical Structure
  19. GC18432 6α-Naloxol

    6-hydroxy Naloxone, NLL

     An Analytical Reference Material 6α-Naloxol Chemical Structure
  20. GC64147 Acetyl tetrapeptide-15 Acetyl tetrapeptide-15 is a synthetic peptide used in the cosmetics for sensitive skin. Acetyl tetrapeptide-15 Chemical Structure
  21. GC11829 ADL5859 HCl ADL5859 HCl (compound 20) is a selective and orally active δ opioid receptor (DOR) agonist with an Ki and an EC50 value of 0.84 and 20 nM, respectively. ADL5859 HCl Chemical Structure
  22. GP10109 Adrenorphin

    H2N-Tyr-Gly-Gly-Phe-Met-Arg-Arg-Val-amide

    Adrenorphin Chemical Structure
  23. GC17623 Alvimopan

    ADL 8-2698, LY246736

     A μ-opioid receptor antagonist Alvimopan Chemical Structure
  24. GC12619 Alvimopan dihydrate A μ-opioid receptor antagonist Alvimopan dihydrate Chemical Structure
  25. GC35311 Alvimopan monohydrate Alvimopan monohydrate (ADL 8-2698 monohydrate) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan monohydrate Chemical Structure
  26. GC46860 AP-238 (hydrochloride)

    2,6-dimethyl Propionyl AP-237

     A neuropeptide with diverse biological activities AP-238 (hydrochloride) Chemical Structure
  27. GC12219 AR-M 1000390 hydrochloride Delta-opioid receptor agonist,low-internalizing AR-M 1000390 hydrochloride Chemical Structure
  28. GC31762 Asimadoline (EMD-61753)

    EMD 61753

     Asimadoline (EMD-61753) (EMD-61753) is an orally active, selective and peripherally active κ-opioid agonist with IC50s of 5.6 nM (guinea pig) and 1.2 nM (human recombinant). Asimadoline (EMD-61753) Chemical Structure
  29. GC61397 Asimadoline hydrochloride Asimadoline (EMD-61753) hydrochloride is an orally active, selective and peripherally active κ-opioid agonist with IC50s of 5.6 nM (guinea pig) and 1.2 nM (human recombinant). Asimadoline hydrochloride Chemical Structure
  30. GC11390 BAM 22P

    Bovine adrenal medulla-22P

     Potent endogenous agonist peptide for the newly identified sensory neuron specific receptor (SNSR); BAM 22P Chemical Structure
  31. GC15926 BAN ORL 24 A nociceptin receptor antagonist BAN ORL 24 Chemical Structure
  32. GC30639 Bevenopran (CB-5945)

    CB-5945; ADL-5945

     Bevenopran (CB-5945) is a peripheral μ-opioid receptor antagonist. Bevenopran (CB-5945) Chemical Structure
  33. GC68785 BMS-986121

    BMS-986121 is a positive allosteric modulator (PAM) of the μ opioid receptor, derived from patent WO2014107344. BMS-986121 is built on a chemical scaffold and represents a new chemical type of μ receptor PAMs.

     BMS-986121 Chemical Structure
  34. GC38741 BPR1M97 BPR1M97 is a dual-acting mu opioid receptor (MOP) and nociceptin-orphanin FQ peptide (NOP) receptor agonist with Ki values of 1.8 and 4.2 nM, respectively. BPR1M97 Chemical Structure
  35. GC15313 BRL 52537 hydrochloride κ/μ opioid receptor agonist,potent and selective BRL 52537 hydrochloride Chemical Structure
  36. GC16521 BW 373U86

    SNC86

     Non-peptide delta agonist,potent and selective BW 373U86 Chemical Structure
  37. GC67907 CCG258747 CCG258747 Chemical Structure
  38. GC35637 Cebranopadol

    GRT6005

     An analgesic NOP and opioid receptor agonist Cebranopadol Chemical Structure
  39. GC35638 Cebranopadol ((1α,4α)stereoisomer)

    GRT6005 (1α,4α)stereoisomer

     Cebranopadol ((1α,4α)stereoisomer) is a stereoisomer of cebranopadol. Cebranopadol ((1α,4α)stereoisomer) Chemical Structure
  40. GC19229 CERC-501

    CERC-501, JNJ-67953964, LY2456302

     CERC-501 (CERC-501) is a potent and centrally-penetrant kappa opioid receptor antagonist with a Ki of 0.807 nM. CERC-501 Chemical Structure
  41. GC11535 CTAP Potent and selective μ opioid receptor antagonist CTAP Chemical Structure
  42. GC60730 CTAP TFA CTAP TFA is a potent, highly selective, and BBB penetrant μ opioid receptor antagonist, with an IC50 of 3.5 nM. CTAP TFA Chemical Structure
  43. GC16888 CTOP Potent and selective μ opioid receptor antagonist CTOP Chemical Structure
  44. GC60731 CTOP TFA CTOP TFA is a potent and highly selective μ-opioid receptor antagonist. CTOP TFA Chemical Structure
  45. GC13189 Cyprodime hydrochloride

    μ-opioid receptor antagonist

     Cyprodime hydrochloride Chemical Structure
  46. GC17677 DADLE

    D-Ala2, D-Leu5-Enkephalin

     δ-opioid receptor agonist DADLE Chemical Structure
  47. GC72209 DALDA acetate DALDA acetate is a potent and highly selective μ-opioid receptor agonist with a Ki of 1.69 nM. DALDA acetate Chemical Structure
  48. GC10803 DAMGO μ opioid receptor agonist DAMGO Chemical Structure
  49. GC35805 DAMGO (TFA) DAMGO (TFA) is a μ-opioid receptor (μ-OPR ) selective agonist with a Kd of 3.46 nM for native μ-OPR. DAMGO (TFA) Chemical Structure
  50. GC61954 Deltorphin 2 TFA

    [D-Ala2]-Deltorphin II TFA

     Deltorphin 2 TFA is a selective peptide agonist for the δ opioid receptor. Deltorphin 2 TFA Chemical Structure
  51. GC12143 Deltorphin I

    Deltorphin 1; Deltorphin C

     δ-opioid receptor agonist Deltorphin I Chemical Structure
  52. GC31168 Dermorphin

    Dermorphin is a natural heptapeptide μ-opioid receptor (MOR) agonist found in amphibian skin.

     Dermorphin Chemical Structure
  53. GC34223 Dermorphin Analog Dermorphin Analog is an analog of Dermorphin. Dermorphin Analog Chemical Structure
  54. GC17553 DIPPA hydrochloride κ receptor antagonist DIPPA hydrochloride Chemical Structure
  55. GC10333 DPDPE Prototypical selective δ-opioid receptor agonist peptide DPDPE Chemical Structure
  56. GC63431 DPDPE TFA DPDPE TFA, an opioid peptide, is a selective δ-opioid receptor?(DOR) agonist?with anticonvulsant effects. DPDPE TFA Chemical Structure
  57. GC14774 DSLET δ Opioid receptor agonist DSLET Chemical Structure
  58. GC13546 Dynorphin A Endogenous kappa receptor agonist Dynorphin A Chemical Structure
  59. GC35917 Dynorphin A (1-10) TFA Dynorphin A (1-10) TFA Chemical Structure
  60. GA21407 Dynorphin A (1-8) Dynorphin A (1-8) is the predominant opioid peptide identified in placental tissue extracts. Dynorphin A (1-8) Chemical Structure
  61. GC35918 Dynorphin A 1-10 Dynorphin A 1-10 an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor. Dynorphin A 1-10 Chemical Structure
  62. GC15078 Dynorphin B

    Dynorphin B-13, Rimorphin

     endogenous agonist for the kappa opioid receptor Dynorphin B Chemical Structure
  63. GC35919 Dynorphin B (1-13) (TFA) Dynorphin B (1-13) TFA acts as an agonist on opioid κ-receptor. Dynorphin B (1-13) (TFA) Chemical Structure
  64. GC67956 Endomorphin 1 acetate Endomorphin 1 acetate Chemical Structure
  65. GC35986 Endomorphin 2 TFA Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. Endomorphin 2 TFA Chemical Structure
  66. GP10065 Endomorphin-1 Endomorphin-1 Chemical Structure
  67. GC10059 Endomorphin-2

    μ-opioid receptors agonist

     Endomorphin-2 Chemical Structure
  68. GC15874 FIT

    δ-opioid agonist, irreversible

     FIT Chemical Structure
  69. GC60857 Frakefamide TFA Frakefamide TFA is a potent analgesic that acts as a peripheral active μ-selective receptor agonist. Frakefamide TFA Chemical Structure
  70. GC30328 Gluten Exorphin C Gluten exorphin C is an opioid peptide derived from wheat gluten. Gluten Exorphin C Chemical Structure
  71. GC15843 GNTI dihydrochloride

    5'-Guanidinonaltrindole

     κ opioid receptor antagonist GNTI dihydrochloride Chemical Structure
  72. GC14739 GR 89696 fumarate κ-opioid agonist GR 89696 fumarate Chemical Structure
  73. GC68427 GSK1521498 free base GSK1521498 free base Chemical Structure
  74. GC43808 Hecogenin Acetate

    NSC 15489

     Hecogenin acetate is a steroid sapogenin and an acetylated form of hecogenin that has anthelmintic and antinociceptive properties. Hecogenin Acetate Chemical Structure
  75. GC32489 Hemorphin-7 Hemorphin-7 is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin. Hemorphin-7 Chemical Structure
  76. GC11639 ICI 154,129 Selective δ opioid antagonist ICI 154,129 Chemical Structure
  77. GC16193 ICI 174,864 Selective δ opioid antagonist ICI 174,864 Chemical Structure
  78. GC12534 ICI 199,441 hydrochloride ICI 199,441 hydrochloride is a potent and selective κ-opioid receptor agonist. ICI 199,441 hydrochloride Chemical Structure
  79. GC13097 ICI 204,448 hydrochloride κ opioid receptor agonist ICI 204,448 hydrochloride Chemical Structure
  80. GC70385 J-113397 J-113397 is the first potent and selective nonpeptidyl ORL1 receptor antagonist (Ki: cloned human ORL1=1.8 nM) without any agonistic effects on other opioid receptors. J-113397 Chemical Structure
  81. GC17939 JDTic JDTic Chemical Structure
  82. GC17624 JDTic 2HCl JDTic 2HCl Chemical Structure
  83. GC11826 JTC-801 KOR-3 (NOP) receptor antagonist JTC-801 Chemical Structure
  84. GC31151 Kelatorphan Kelatorphan is a full inhibitor of enkephalin degrading enzymes. Kelatorphan Chemical Structure
  85. GC69337 KNT-127

    KNT-127 is an effective selective δ opioid receptor agonist that works effectively through systemic administration. KNT-127 has selectivity for the δ receptor (with Ki values of 21.3, 0.16, and 153 nM for opioid receptors μ, δ, and κ, respectively). It can increase dopamine and L-glutamate release in the striatum, ventral pallidum, and anterior cingulate cortex. It also exhibits antidepressant-like effects.

     KNT-127 Chemical Structure
  86. GC61003 Loperamide D6 hydrochloride Loperamide D6 hydrochloride (R-18553 D6 hydrochloride) is a deuterium labeled Loperamide hydrochloride. Loperamide D6 hydrochloride Chemical Structure
  87. GC36479 Loperamide hydrochloride

    NSC 696356, PJ 185, R 18553

     Loperamide (hydrochloride) (R-18553 (hydrochloride)) is an opioid receptor agonist. Loperamide hydrochloride Chemical Structure
  88. GC36508 LY-2940094

    BTRX-246040

     LY-2940094 (BTRX-246040) is a potent, selective and orally available nociceptin receptor (NOP receptor) antagonist with high affinity (Ki=0.105 nM) and antagonist potency (Kb=0.166 nM). LY-2940094 Chemical Structure
  89. GC39193 LY2444296

    FP3FBZ

     LY2444296 is an orally bioavailable, high-affinity and selective short-acting kappa opioid receptor (KOPR) antagonist, with a Ki value of ?1 nM. LY2444296 Chemical Structure
  90. GC70466 LY255582 LY255582 is a pan-opioid antagonist and has high affinity for mu, delta, and kappa receptors (Ki: 0.4 nM, 5.2, 2.0 nM respectively). LY255582 Chemical Structure
  91. GC19500 LY2795050

    LY2795050 is a novel selective κ-opioid Receptor (KOR) antagonist

     LY2795050 Chemical Structure
  92. GC17874 Matrine

    NSC 146051, NSC 318810

     Matrine is an alkaloid found in Sophora japonica plants that acts as a kappa opioid receptor and µ-receptor agonist. Matrine Chemical Structure
  93. GC36562 MCOPPB triHydrochloride

    MCOPPB 3HCl

     MCOPPB 3Hcl is a nociceptin receptor agonist with pKi of 10.07; weaker activity at other opioid receptors. MCOPPB triHydrochloride Chemical Structure
  94. GC11016 Meptazinol HCl Partial agonist at the μ1 opioid receptor Meptazinol HCl Chemical Structure
  95. GC63072 Methyl-6-alpha-Naltrexol Methyl-6-alpha-Naltrexol Chemical Structure
  96. GC16177 Methylnaltrexone Bromide

    MRZ 2663BR, Naltrexone methylbromide

     Antagonist of peripherally acting μ-opioid Methylnaltrexone Bromide Chemical Structure
  97. GC14525 ML 190 κ opioid receptor (KOP) antagonist ML 190 Chemical Structure
  98. GC70268 MT-7716 hydrochloride MT-7716 hydrochloride (W-212393 hydrochloride) is a selective non-peptide nociceptin receptor (NOP) agonist and promising potential treatment drug for alcohol abuse and relapse prevention. MT-7716 hydrochloride Chemical Structure
  99. GC12663 N-Benzylnaltrindole hydrochloride δ2 opioid receptor antagonist N-Benzylnaltrindole hydrochloride Chemical Structure
  100. GC16553 N-Desmethylclozapine

    Norclozapine

     5-HT2C serotonin receptor antagonist N-Desmethylclozapine Chemical Structure
  101. GC14979 N-MPPP Hydrochloride High affinity κ agonist N-MPPP Hydrochloride Chemical Structure

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