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Home >> Signaling Pathways >> GPCR/G protein

GPCR/G protein

Products for  GPCR/G protein

  1. Cat.No. Product Name Information
  2. GC31974 A2B receptor antagonist 1 A2B receptor antagonist 1 is a potent A2B adenosine receptor antagonist extracted from patent WO 2009157938 A1 EXAMPLE 9B. A2B receptor antagonist 1 Chemical Structure
  3. GC62820 A2B receptor antagonist 2 A2B receptor antagonist 2 (compound 18) is an adenosine receptor A2B antagonist, with Ki values of 2.30 μM, 6.8 μM and 3.44 μM for rA1, rA2A and hA2B, respectively. A2B receptor antagonist 2 Chemical Structure
  4. GC32674 A81988 (Abbott81988) A81988 (Abbott81988) is a potent, competitive, non-peptidic antagonist of angiotensin AT1 receptors. A81988 (Abbott81988) Chemical Structure
  5. GC41327 Aaptamine Aaptamine is a marine sponge alkaloid originally isolated from A. Aaptamine Chemical Structure
  6. GC30993 AB-MECA AB-MECA is a high affinity A3 adenosine receptor agonist, has high affinity for recombinant A1 and A3 receptors. AB-MECA Chemical Structure
  7. GC67702 Abanoquil Abanoquil Chemical Structure
  8. GC31055 Abaperidone Abaperidone is a potent antagonist of 5-HT2A?receptor and dopamine D2 receptor with IC50s of 6.2 and 17 nM. Abaperidone Chemical Structure
  9. GC64356 Ablukast Ablukast (Ro 23-3544) is a specific and active leukotriene receptor antagonist. Ablukast Chemical Structure
  10. GC12728 Abn-CBD GPR55 cannabinoid receptor agonist Abn-CBD Chemical Structure
  11. GC50125 ABP 688 High affinity human mGlu5 antagonist ABP 688 Chemical Structure
  12. GC13416 ABT 702 dihydrochloride Adenosine kinase inhibitor ABT 702 dihydrochloride Chemical Structure
  13. GC50695 ABT 702 hydrochloride ABT 702 hydrochloride Chemical Structure
  14. GC10097 AC 187 Amylin receptor antagonist, Potent and selective AC 187 Chemical Structure
  15. GC50365 AC 265347 Biased allosteric modulator of calcium-sensing receptor (CaSR) AC 265347 Chemical Structure
  16. GC10014 Ac-RYYRIK-NH2 High affinity ligand for the NOP site Ac-RYYRIK-NH2 Chemical Structure
  17. GC15444 Ac-RYYRWK-NH2 selective partial agonist peptide for the NOP receptor Ac-RYYRWK-NH2 Chemical Structure
  18. GC30859 AC260584 AC260584 is an M1 muscarinic receptor allosteric agonist with a pEC50 of 7.6. AC260584 Chemical Structure
  19. GC15522 Ac9-25 formyl peptide receptor 1 (FPR1) ligand Ac9-25 Chemical Structure
  20. GC60552 Acebutolol D7 Acebutolol D7 is a deuterium labeled Acebutolol. Acebutolol D7 Chemical Structure
  21. GC13000 Acebutolol HCl Acebutolol HCl is an orally active β1 adrenergic receptor (β1AR) antagonist. Acebutolol HCl Chemical Structure
  22. GC64332 Aceclidine Aceclidine is a modulator of M3 muscarinic acetylcholine receptor. Aceclidine Chemical Structure
  23. GC34143 Acefylline (Theophyllineacetic acid) Acefylline (Theophyllineacetic acid) (Theophyllineacetic acid), a xanthine derivative, is an adenosine receptor antagonist. Acefylline (Theophyllineacetic acid) is a peptidylarginine deiminase (PAD) activator. Acefylline (Theophyllineacetic acid) is also a bronchodilator, which inhibits rat lung cAMP phosphodiesterase isoenzymes. Acefylline (Theophyllineacetic acid) Chemical Structure
  24. GC62825 ACH-000143 ACH-000143 is a potent and orally active melatonin receptor agonist, with EC50 values of 0.06 nM and 0.32 nM for MT1 and MT2, respectively. ACH-000143 Chemical Structure
  25. GC15791 Acifran HM74A/GPR109A and GPR109B agonist,hypolipidemic agent Acifran Chemical Structure
  26. GC14096 Aclidinium Bromide LAMAs antagonist Aclidinium Bromide Chemical Structure
  27. GC14036 ACPT-II metabotropic receptor antagonist ACPT-II Chemical Structure
  28. GC10623 ACS 67 analog of latanoprost (free acid),prostaglandin (PG) analog ACS 67 Chemical Structure
  29. GC16336 ACT 335827 Orexin receptor 1 antagonist,potent and selective ACT 335827 Chemical Structure
  30. GC50142 ACT 462206 Potent, dual orexin receptor antagonist ACT 462206 Chemical Structure
  31. GC13236 ACT-132577 ACT-132577 (ACT-132577) is the major and pharmacologically active metabolite of Macitentan. ACT-132577 Chemical Structure
  32. GC35243 ACTH (1-14) TFA ACTH (1-14) TFA Chemical Structure
  33. GC35244 ACTH (1-17) TFA ACTH (1-17) TFA Chemical Structure
  34. GC12239 ACTH (1-39) ACTH (1-39) is a melanocortin receptor agonist. ACTH (1-39) Chemical Structure
  35. GC66383 ACTH (11-24) (acetate) ACTH (11-24) (acetate) is an adrenocorticotropic hormone (ACTH) receptor antagonist. ACTH (11-24) is a fragment of adrenocorticotropic and induces cortisol release. ACTH (11-24) can be used for the research of central nervous system. ACTH (11-24) (acetate) Chemical Structure
  36. GC30547 ACTH 1-14 (Adrenocorticotropic Hormone Fragment 1-14) ACTH 1-14 (Adrenocorticotropic Hormone Fragment 1-14) is a fragment of adrenocorticotrophin, which regulates cortisol and androgen production. ACTH 1-14 (Adrenocorticotropic Hormone Fragment 1-14) Chemical Structure
  37. GC31109 ACTH 1-17 (α1-17-ACTH) ACTH 1-17 (α1-17-ACTH), an adrenocorticotropin analogue, is a potent human melanocortin 1 (MC1) receptor agonist with a Ki of 0.21 nM. ACTH 1-17 (α1-17-ACTH) Chemical Structure
  38. GC31954 ACTH 11-24 (Adrenocorticotropic Hormone (11-24)) ACTH 11-24 (Adrenocorticotropic Hormone (11-24)) is an adrenocorticotropic hormone (ACTH) receptor antagonist. ACTH 11-24 (Adrenocorticotropic Hormone (11-24)) Chemical Structure
  39. GC19630 Adenosine 2′-monophosphate Adenosine 2′-monophosphate (2'-AMP) is converted by extracellular 2',3'-CAMP. Adenosine 2′-monophosphate Chemical Structure
  40. GC35248 Adenosine 5'-monophosphate monohydrate Adenosine 5'-monophosphate monohydrate is an adenosine A1 receptor agonist. Adenosine 5'-monophosphate monohydrate Chemical Structure
  41. GC38733 Adenosine A1 receptor activator T62 Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor. Adenosine A1 receptor activator T62 Chemical Structure
  42. GC38884 Adenosine amine congener An adenosine A1 receptor agonist Adenosine amine congener Chemical Structure
  43. GC35249 Adenosine antagonist-1 Adenosine antagonist-1 is an adenosine A3 receptor (AA3R) antagonist. Adenosine antagonist-1 Chemical Structure
  44. GC35250 Adenosine deaminase

    Involved in metabolism of purines

     Adenosine deaminase Chemical Structure
  45. GC16930 Adenosine Kinase Inhibitor (hydrate) inhibitor of adenosine kinase Adenosine Kinase Inhibitor (hydrate) Chemical Structure
  46. GC65901 Adenosine receptor antagonist 2 Adenosine receptor antagonist 2 is an orally active A2a/A2b adenosine receptor antagonist with IC50s of 1 nM and 3 nM, respectively. Adenosine receptor antagonist 2 has anti-tumor activity. Adenosine receptor antagonist 2 Chemical Structure
  47. GC66007 Adenosine receptor antagonist 3 Adenosine receptor antagonist 3 is a potent antagonist of adenosine receptor. Adenosine receptor antagonist 3 has the potential for the research of cancer disease (extracted from patent WO2019233994A1, compound 1). Adenosine receptor antagonist 3 Chemical Structure
  48. GC10254 AdipoRon AdipoR1 and AdipoR2 agonist, first orally active AdipoRon Chemical Structure
  49. GC35251 AdipoRon hydrochloride AdipoRon hydrochloride is an orally active and specific AdipoR agonist, binding to AdipoR1 and AdipoR2, with Kds of 1.8 and 3.1 μM, respectively. AdipoRon hydrochloride Chemical Structure
  50. GC31322 Adomeglivant (LY2409021) Adomeglivant (LY2409021) (LY2409021) is a potent, selective glucagon receptor (GluR) allosteric antagonist. Adomeglivant (LY2409021) Chemical Structure
  51. GC35252 Adoprazine Adoprazine (SLV313) is a full 5-HT1A receptor agonist with a pEC50 of 9 at cloned h5-HT1A receptors. Adoprazine Chemical Structure
  52. GC13814 Adrenalone HCl Decoyinine (Angustmycin A), a specific inhibitor of bacterial GMPS, has been isolated from Streptomyces . Adrenalone HCl Chemical Structure
  53. GC35254 Adrenocorticotropic Hormone (ACTH) (1-39), rat Adrenocorticotropic Hormone (ACTH) (1-39), rat is a potent melanocortin 2 (MC2) receptor agonist. Adrenocorticotropic Hormone (ACTH) (1-39), rat Chemical Structure
  54. GC35255 Adrenocorticotropic Hormone (ACTH) (1-39), rat TFA Adrenocorticotropic Hormone (ACTH) (1-39), rat (TFA) is a potent melanocortin 2 (MC2) receptor agonist. Adrenocorticotropic Hormone (ACTH) (1-39), rat TFA Chemical Structure
  55. GC10494 ADX-47273 mGluR5 receptor positive allosteric modulator, potent and selective ADX-47273 Chemical Structure
  56. GC30793 ADX88178 ADX88178 is a potent metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) with an EC50 of 4 nM for human mGluR4. ADX88178 Chemical Structure
  57. GC10219 AF-DX 116 AF-DX 116 (AF-DX 116) is a selective and competitive M2 muscarinic acetylcholine receptor antagonist, with IC50 values of 640 nM and 386 nM for rabbit peripheral lung and rat heart, respectively. AF-DX 116 Chemical Structure
  58. GC19023 AF38469 AF38469 is a novel, selective, orally bioavailable Sortilin inhibitor with an IC50 value of 330 nM. AF38469 Chemical Structure
  59. GC38586 AF40431 AF40431, the first reported small-molecule ligand of sortilin, has an IC50 of 4.4 ?M and a Kd of 0.7 ?M . AF40431 Chemical Structure
  60. GC15147 AG 045572 GnRH antagonist AG 045572 Chemical Structure
  61. GC11603 AG-041R gastrin/cholecystokinin-2 (CCKB) receptor antagonist AG-041R Chemical Structure
  62. GC30572 Aganepag (AGN 210937) Aganepag (AGN 210937) is a potent Prostanoid EP2 receptor agonist, with an EC50 of 0.19 nM, and shows no activity at EP4 receptor. Aganepag (AGN 210937) Chemical Structure
  63. GC64435 Aganepag isopropyl Aganepag isopropyl (AGN-210961) is an EP2 agonist. Aganepag isopropyl Chemical Structure
  64. GC64665 AGI-41998 AGI-41998 is a potent inhibitor of methionine adenosyltransferase 2A (MAT2A). AGI-41998 Chemical Structure
  65. GC64635 AGI-43192 AGI-43192 is a potent inhibitor of methionine adenosyltransferase 2A (MAT2A). AGI-43192 Chemical Structure
  66. GC16831 Agmatine sulfate α2-adrenergic receptor ligand Agmatine sulfate Chemical Structure
  67. GC32599 AGN 192836 AGN 192836 is a potent and selective α2 adrenergic agonist with EC50s of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively. AGN 192836 Chemical Structure
  68. GC31972 AGN 210676 (Simenepag) AGN 210676 (Simenepag) is a selective prostaglandin EP2 agonist extracted from patent US20070203222A1, Compound example 23, has an EC50 of 5 nM. AGN 210676 (Simenepag) Chemical Structure
  69. GC40750 Agnuside Agnuside is an iridoid glycoside originally isolated from V. Agnuside Chemical Structure
  70. GC17981 Agomelatine MT1/MT2 / 5-HT2C agonist Agomelatine Chemical Structure
  71. GC35269 Agomelatine hydrochloride Agomelatine hydrochloride (S-20098 hydrochloride) is a specific agonist of MT1 and MT2 receptors with Kis of 0.1, 0.06, 0.12, and 0.27 nM for CHO-hMT1, HEK-hMT1, CHO-hMT2, and HEK-hMT2, respectively. Agomelatine hydrochloride Chemical Structure
  72. GC35270 Agomelatine L(+)-Tartaric acid Agomelatine L(+)-Tartaric acid (S-20098 L(+)-Tartaric acid) is a specific agonist of MT1 and MT2 receptors with Kis of 0.1, 0.06, 0.12, and 0.27 nM for CHO-hMT1, HEK-hMT1, CHO-hMT2, and HEK-hMT2, respectively. Agomelatine L(+)-Tartaric acid Chemical Structure
  73. GC10197 AH 11110 hydrochloride α1B-AR ligand,subtype-selective AH 11110 hydrochloride Chemical Structure
  74. GC17224 AH 23848 (calcium salt) dual antagonist of TP1 and EP4 receptors AH 23848 (calcium salt) Chemical Structure
  75. GC14879 AH 6809 An EP and DP receptor antagonist AH 6809 Chemical Structure
  76. GC17753 AH 7614

    FFA4/GPR120 antagonist

     AH 7614 Chemical Structure
  77. GC10146 AHU-377(Sacubitril) AHU-377(Sacubitril) (AHU-377) is a potent and orally active NEP (neprilysin) inhibitor with an IC50 of 5 nM. AHU-377(Sacubitril) Chemical Structure
  78. GC35272 Ajmalicine A terpenoid indole alkaloid Ajmalicine Chemical Structure
  79. GC32405 AL 082D06 (D06) AL 082D06 (D06) is a selective, nonsteroidal glucocorticoid receptor (GR) antagonist with Ki of 210 nM. AL 082D06 (D06) Chemical Structure
  80. GC16895 AL 8810

    Antagonist of prostaglandin F2α (FP) receptor.

     AL 8810 Chemical Structure
  81. GC16566 AL 8810 isopropyl ester lipid soluble, esterified prodrug form of AL 8810, a FP receptor antagonist AL 8810 isopropyl ester Chemical Structure
  82. GC31388 ALB-127158(a) ALB-127158(a) is a potent and selective melanin concentrating hormone 1 (MCH1) receptor antagonist. ALB-127158(a) Chemical Structure
  83. GC25046 Albiglutide Fragment Albiglutide fragment is one copy of a 30-amino-acid sequence of modified human GLP-1 (fragment 7-36). Albiglutide Fragment Chemical Structure
  84. GC35282 Alexamorelin Met 1 Alexamorelin Met 1 Chemical Structure
  85. GC16740 Alfuzosin alpha-adrenergic blocker Alfuzosin Chemical Structure
  86. GC13730 Alfuzosin HCl Alfuzosin (SL 77499-10) hydrochloride is an orally active, selective and competitive α1-adrenoceptor antagonist. Alfuzosin HCl Chemical Structure
  87. GC32558 Aligeron Aligeron is a non-selective prostaglandin (PG) antagonist, and has vasodilatory properties. Aligeron Chemical Structure
  88. GC62833 ALK4290 ALK4290 (AKST4290) is a potent and orally actively CCR3 inhibitor extracted from patent US20130261153A1, compound Example 2, with a Ki of 3.2 nM for hCCR3. ALK4290 Chemical Structure
  89. GC25051 Alloxazine Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor. Alloxazine Chemical Structure
  90. GC10717 Almorexant OX1R/OX2R antagonist Almorexant Chemical Structure
  91. GC10050 Almorexant hydrochloride OX1R/OX2R antagonist Almorexant hydrochloride Chemical Structure
  92. GC15153 Almotriptan Malate 5-HT1B/1D-receptor agonist Almotriptan Malate Chemical Structure
  93. GC31054 Alniditan (Alnitidan) Alniditan (Alnitidan) (Alnitidan) is a potent 5-HT1B and 5-HT1D receptors agonist, with IC50s of 1.7 nM and 1.3 nM for h5-HT1B and h5-HT1D receptors in HEK293 cells, respectively. Alniditan (Alnitidan) Chemical Structure
  94. GC35301 Alosetron ((Z)-2-butenedioate) Alosetron (GR 68755) (Z)-2-butenedioate is a potent and highly selective serotonin 5-HT3 receptor antagonist. Alosetron ((Z)-2-butenedioate) Chemical Structure
  95. GC35302 Alosetron (Hydrochloride(1:X)) Alosetron (GR 68755) Hydrochloride(1:X) is a potent and highly selective serotonin 5-HT3 receptor antagonist. Alosetron (Hydrochloride(1:X)) Chemical Structure
  96. GC35303 Alosetron D3 Hydrochloride Alosetron D3 Hydrochloride (GR-68755C D3) is deuterium labeled Alosetron, which is a serotonin 5HT3-receptor antagonist. Alosetron D3 Hydrochloride Chemical Structure
  97. GC64265 Alosetron-13C,d3 Alosetron-13C,d3 Chemical Structure
  98. GC32905 Alprenolol ((RS)-Alprenolol) Alprenolol ((RS)-Alprenolol) ((RS)-Alprenolol ((RS)-Alprenolol); dl-Alprenolol ((RS)-Alprenolol)) is an orally active non-selective β-adrenoceptor antagonist and an antagonist of 5-HT1A and 5-HT1B receptors. Alprenolol ((RS)-Alprenolol) is used as an anti-hypertensive, anti-anginal and anti-arrhythmic agent. Alprenolol ((RS)-Alprenolol) Chemical Structure
  99. GC14105 Alprenolol hydrochloride β-adrenoceptor and 5-HT1A receptor antagonist. Alprenolol hydrochloride Chemical Structure
  100. GC17347 Alprostadil Alprostadil (Alprostadil) is a prostanoid receptor ligand, with Kis of 1.1 nM, 2.1 nM, 10 nM, 33 nM and 36 nM for mouse EP3, EP4, EP2, IP and EP1, respectively. Alprostadil Chemical Structure
  101. GC14030 Altanserin hydrochloride 5-HT2A receptor antagonist Altanserin hydrochloride Chemical Structure

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