Adrenergic Receptor
Adrenergic receptor is a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine and epinephrine.
Products for Adrenergic Receptor
- Cat.No. Product Name Information
- GC37983 β3-AR agonist 1 β3-AR agonist 1 (compound 15) is a highly potent, selective, and orally available β3-adrenergic receptor (β3-AR) agonist (EC50=18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold).
- GC31237 α1 adrenoceptor-MO-1 α1 adrenoceptor-MO-1, an S enantiomer, has affinity at alpha 1 adrenergic receptor, shows alphalytic activity, and possesses analgesic action; more active than R enantiomer.
- GC31573 β3-AR agonist 2 β3-AR agonist 2 is a potent and selective β3-adrenergic receptor (β3-AR) agonist with an EC50 of 8 nM.
- GC46283 (±)-Clorprenaline-d7 A neuropeptide with diverse biological activities
- GC62727 (±)-Penbutolol-d9 hydrochloride (±)-Penbutolol-d9 ((Rac)-Penbutolol-d9) hydrochloride is a deuterium labeled (±)-Penbutolol hydrochloride.
- GC32523 (±)-Befunolol (±)-Befunolol is a β-adrenoceptor blocking agent.
- GC31597 (+)-Penbutolol ((R)-Penbutolol) (+)-Penbutolol ((R)-Penbutolol) is a β-adrenoceptor antagonist, with an IC50 of 0.74 μM.
- GC10675 (+,-)-Octopamine HCl Octopamine ((±)-p-Octopamine) hydrochloride, a biogenic monoamine structurally related to noradrenaline, acts as a neurohormone, a neuromodulator and a neurotransmitter in invertebrates.
- GC32644 (4E)-SUN9221 (4E)-SUN9221 is a potent antagonist of α1-adrenergic receptor and 5-HT2 receptor, with antihypertensive and anti-platelet aggregation activities.
- GC11952 (R)-(+)-Atenolol less active enantiomer of the racemic β1-adrenergic receptor antagonist, (R,S)-atenolol.
- GC11937 (R)-(+)-m-Nitrobiphenyline oxalate α2C-AR (adrenoceptor) agonist
-
GC10608
(R)-(+)-Propranolol hydrochloride
β-adrenoceptor antagonist
- GC12144 (R)-(-)-Niguldipine hydrochloride L-type Ca2+ channel blocker and α1A-adrenoceptor antagonist
- GC60001 (R)-Carvedilol (R)-Carvedilol ((R)-BM 14190), the R-enantiomer of Carvedilol, is a non-selective β/α-1 blocker.
- GC39298 (R)-Terazosin (R)-Terazosin is an active R-enantiomer of Terazosin.
- GC14145 (R,R)-Formoterol β2-selective adrenergic agonist
- GC12823 (R,S)-Atenolol (R,S)-Atenolol ((RS)-(R,S)-Atenolol) is a cardioselective β1-adrenergic receptor blocker, with a Ki of 697 nM atβ1-adrenoceptor in guine pig left ventricle membrane.
- GC64481 (rac)-Dobutamine-d4 hydrochloride
- GC62642 (rac)-Dobutamine-d6 hydrochloride
- GC62228 (rac)-Nebivolol-d4 (Rac)-Nebivolol-d4 ((Rac)-R 065824-d4) is a labelled racemic Nebivolol.
- GC34367 (RS)-Butyryltimolol (RS)-Butyryltimolol is the racemate of Butyryltimolol.
- GC15292 (S)-(+)-Niguldipine hydrochloride L-type Ca2+ channel blocker and α1A-adrenoceptor antagonist
-
GC12463
(S)-(-)-Atenolol
β-adrenergic blocker
- GC15039 (S)-(-)-Pindolol beta-adrenergic antagonist
- GC16637 (S)-(-)-Propranolol hydrochloride β-adrenoceptor antagonist
- GC60006 (S)-Carvedilol (S)-Carvedilol, the S-enantiomer of Carvedilol, is a non-selective β/α-1 blocker.
- GC39249 (S)-Terazosin (S)-Terazosin is an active S-enantiomer of Terazosin.
- GC16663 (±)-4-hydroxy Propranolol (hydrochloride) β1- and β2-adrenergic receptors inhibitor
- GC15087 (±)-Talinolol β1-selective adrenoceptor antagonist
- GC16412 2-MPMDQ α1-adrenoceptor antagonist,potent and selective
- GC13695 2-PMDQ α1-adrenoceptor antagonist
- GN10169 3-Hydroxy-4-methoxycinnamic acid
- GC10073 3-MPPI ligand for adrenergic α1 receptor
- GC68327 4-Hydroxyatomoxetine-d3
- GC64116 4-Hydroxypropranolol-d7
- GC32655 5-HT2 antagonist 1 5-HT2 antagonist 1 is a potent antagonist of 5-HT2 receptor, with weak α1 adrenoceptor blocking activity.
- GC14527 A 61603 hydrobromide A 61603 hydrobromide is a selective α1A-adrenergic receptor agonist.
- GC13027 A 80426 mesylate α2-adrenoceptor antagonist and 5-HT uptake inhibitor
- GC41327 Aaptamine Aaptamine is a marine sponge alkaloid originally isolated from A.
- GC67702 Abanoquil
- GC60552 Acebutolol D7 Acebutolol D7 is a deuterium labeled Acebutolol.
- GC13000 Acebutolol HCl Acebutolol HCl is an orally active β1 adrenergic receptor (β1AR) antagonist.
- GC35243 ACTH (1-14) TFA
- GC30547 ACTH 1-14 (Adrenocorticotropic Hormone Fragment 1-14) ACTH 1-14 (Adrenocorticotropic Hormone Fragment 1-14) is a fragment of adrenocorticotrophin, which regulates cortisol and androgen production.
- GC13814 Adrenalone HCl Decoyinine (Angustmycin A), a specific inhibitor of bacterial GMPS, has been isolated from Streptomyces .
- GC16831 Agmatine sulfate α2-adrenergic receptor ligand
- GC32599 AGN 192836 AGN 192836 is a potent and selective α2 adrenergic agonist with EC50s of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively.
- GC10197 AH 11110 hydrochloride α1B-AR ligand,subtype-selective
- GC35272 Ajmalicine A terpenoid indole alkaloid
- GC16740 Alfuzosin alpha-adrenergic blocker
- GC13730 Alfuzosin HCl Alfuzosin (SL 77499-10) hydrochloride is an orally active, selective and competitive α1-adrenoceptor antagonist.
- GC14105 Alprenolol hydrochloride β-adrenoceptor and 5-HT1A receptor antagonist.
- GC32516 Amezinium methylsulfate (Amezinium metilsulfate) Amezinium metilsulfate has multiple mechanisms, including stimulation of alpha and beta-1 receptors and inhibition ofnoradrenaline and tyramine uptake.
- GC33983 Amitraz (BTS-27419) Amitraz (BTS-27419) is a non-systemic acaricide and insecticide, with alpha-adrenergic agonist activity, interaction with octopamine receptors of the central nervous system and inhibition of monoamine oxidases and prostaglandin synthesis.
- GC32582 Ancarolol Ancarolol is a beta-adrenergic blocking agent.
-
GC17736
Anisodamine
weak antagonist of α1-adrenoceptors
- GC60593 Arbutamine Arbutamine is a short-acting, potent and nonselective β-adrenoceptor agonist.
- GC10965 ARC 239 dihydrochloride α2B adrenoceptor antagonist
- GC42851 Arformoterol (tartrate) Aformoterol is the (R,R)-enantiomer of the β2-adrenergic receptor (β2-AR) agonist formoterol.
- GC11824 Asenapine Inhibits adrenergic receptor/5-HT receptor
- GC30791 Atipamezole (MPV 1248) Atipamezole (MPV 1248) (MPV 1248) is a potent α2-adrenoceptor antagonist with a Ki of 1.6 nM.
- GC16106 Atipamezole hydrochloride α2-adrenergic receptor antagonist
- GC14491 B-HT 920 A potent agonist of D2 receptors
- GC14514 B-HT 933 dihydrochloride Azepexole (B-HT 933) dihydrochloride is a potent and selective alpha 2-adrenoceptor agonist with pKis of 8.3, 7.6, and 7.5 for α2A-, α2B- and α2C-adrenoceptor subtypes, resepctively.
- GC13577 Bambuterol long acting beta-adrenoceptor agonist
- GC42896 Bambuterol (hydrochloride) Bambuterol is a prodrug for terbutaline, a long-acting β-adrenoceptor agonist (Ki = 15.4 μM for human β2-adrenergic receptor).
- GC63433 Bambuterol-d9 hydrochloride
- GC31690 Batefenterol (GSK961081) Batefenterol (GSK961081) (GSK961081;TD-5959) is a novel muscarinic receptor antagonist and β2-adrenoceptor agonist; displays high affinity for hM2, hM3 muscarinic and hβ2-adrenoceptor with Ki values of 1.4, 1.3 and 3.7 nM, respectively.
- GC65252 Benoxathian hydrochloride Benoxathian hydrochloride is a potent α1 adrenoceptor antagonist, can be used for researching anorexia.
- GC30474 Benzquinamide (P2647)
- GC14021 Betaxolol βadrenergic receptor blocker
- GC17731 Betaxolol HCl Betaxolol Hydrochloride is a selective beta1 adrenergic receptor blocker that can be used for the research of hypertension and glaucoma.
- GC39546 Bevantolol hydrochloride A β1-AR antagonist
- GC38378 BI-167107 BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR) with a dissociation constant Kd of 84 pM.
- GC25140 Bisoprolol Bisoprolol is a cardioselective β1-adrenergic blocking agent used for secondary prevention of myocardial infarction (MI), heart failure, angina pectoris and mild to moderate hypertension.
- GC14818 Bisoprolol fumarate Bisoprolol fumarate is a potent, selective and orally active β1-adrenergic receptor blocker with little activity on β2-receptor.
- GC32665 Bometolol Hydrochloride Bometolol Hydrochloride is a beta-adrenergic blocking agent, used for the research of cardiovascular disease.
- GC10738 Brimonidine Tartrate Highly selective α-adrenergic receptor agonist
- GC13785 BRL 37344, sodium salt BRL 37344, sodium salt (BRL 37344A) is a specific β3-adrenergic receptor agonist.
- GC13996 BRL 44408 maleate Selective α2A-AR antagonist
- GC15328 Bucindolol beta adrenergic blocker
- GC67692 Bufuralol
- GC15347 Bufuralol (hydrochloride) non-specific β-adrenergic blocker
- GC64450 Bunazosin Bunazosin is a potent and selective α1-adrenoceptor antagonist.
- GC62648 Bupranolol Bupranolol is an orally active, competitive and non-selective β-adrenoceptor antagonist without intrinsic sympathomimetic activity.
- GC64504 Butyryltimolol Butyryltimolol, an effective prodrug of Timolol, improves the corneal penetration of Timolol.
- GC13180 Carazolol high-affinity, lipophilic, non-selective ligand of the β-adrenergic receptors
- GC15243 Carbazochrome sodium sulfonate (AC-17) Carbazochrome sodium sulfonate (AC-17) (AC-17) is a capillary stabiliser and used for the research of haemorrhage.
- GC16395 Carteolol HCl Carteolol HCl (OPC-1085 hydrochloride) is a non-selective beta blocker used to treat glaucoma.
- GC14769 Carvedilol Potent β-adrenoceptor and α1-adrenoceptor antagonist
- GC25197 Carvedilol EP IMpurity E Carvedilol is a nonselective beta blocker/alpha-1 blocker and used in management of congestive heart failure (CHF).
- GC35613 Carvedilol phosphate hemihydrate Carvedilol phosphate hemihydrate (BM 14190 phosphate hemihydrate) is a non-selective β/α-1 blocker.
- GC64003 Carvedilol-d4
- GC12023 Celiprolol (hydrochloride) β1 adrenergic receptor antagonist and β2 adrenergic receptor partial agonist
- GC31283 Centanafadine (EB-1020) Centanafadine (EB-1020) is dual norepinephrine (NE)/dopamine (DA) transporter inhibitor, also inhibits serotonin transporter, with IC50s of 6 nM, 38 nM and 83 nM for human NE, DA and serotonin transporter , respectively.
- GC31175 Centanafadine hydrochloride (EB-1020 (hydrochloride)) Centanafadine (hydrochloride) is dual norepinephrine (NE)/dopamine (DA) transporter inhibitor, also inhibits serotonin transporter, with IC50s of 6 nM, 38 nM and 83 nM for human NE, DA and serotonin transporter , respectively.
- GC17717 CGP 12177 hydrochloride β1/β2-AR antagonist,β3 AR partial agonist
- GC38752 CGP 20712 A CGP 20712 A (CGP 20712 mesylate) is a highly selective β1-adrenoceptor antagonist with an IC50 of 0.7 nM.
- GC15354 CGP 20712 dihydrochloride β1 antagonist,highly potent and selective
- GC32542 Cicloprolol hydrochloride Cicloprolol is a partial β 1-adrenoceptor agonist .