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Home >> Signaling Pathways >> GPCR/G protein >> Adrenergic Receptor

Adrenergic Receptor

Adrenergic receptor is a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine and epinephrine.

Products for  Adrenergic Receptor

  1. Cat.No. Product Name Information
  2. GC37983 β3-AR agonist 1 β3-AR agonist 1 (compound 15) is a highly potent, selective, and orally available β3-adrenergic receptor (β3-AR) agonist (EC50=18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold). β3-AR agonist 1 Chemical Structure
  3. GC31237 α1 adrenoceptor-MO-1 α1 adrenoceptor-MO-1, an S enantiomer, has affinity at alpha 1 adrenergic receptor, shows alphalytic activity, and possesses analgesic action; more active than R enantiomer. α1 adrenoceptor-MO-1 Chemical Structure
  4. GC31573 β3-AR agonist 2 β3-AR agonist 2 is a potent and selective β3-adrenergic receptor (β3-AR) agonist with an EC50 of 8 nM. β3-AR agonist 2 Chemical Structure
  5. GC46283 (±)-Clorprenaline-d7

    Isoprophenamine-d7

     A neuropeptide with diverse biological activities (±)-Clorprenaline-d7 Chemical Structure
  6. GC62727 (±)-Penbutolol-d9 hydrochloride (±)-Penbutolol-d9 ((Rac)-Penbutolol-d9) hydrochloride is a deuterium labeled (±)-Penbutolol hydrochloride. (±)-Penbutolol-d9 hydrochloride Chemical Structure
  7. GC32523 (±)-Befunolol (±)-Befunolol is a β-adrenoceptor blocking agent. (±)-Befunolol Chemical Structure
  8. GC31597 (+)-Penbutolol ((R)-Penbutolol)

    (R)-Penbutolol; (+)-Isopenbutolol

     (+)-Penbutolol ((R)-Penbutolol) is a β-adrenoceptor antagonist, with an IC50 of 0.74 μM. (+)-Penbutolol ((R)-Penbutolol) Chemical Structure
  9. GC10675 (+,-)-Octopamine HCl

    β,4-Dihydroxyphenethylamine, Epirenor, Norfen, NSC 108685, (±)-4-Octopamine, (±)-p-Octopamine

     Octopamine ((±)-p-Octopamine) hydrochloride, a biogenic monoamine structurally related to noradrenaline, acts as a neurohormone, a neuromodulator and a neurotransmitter in invertebrates. (+,-)-Octopamine HCl Chemical Structure
  10. GC74197 (-)-Isoproterenol hydrochloride

    Levisoprenaline hydrochloride; Proternol L hydrochloride

     (-)-Isoproterenol (Levisoprenaline; Proternol L) drochloride is a β-adrenoceptor agonist. (-)-Isoproterenol hydrochloride Chemical Structure
  11. GC32644 (4E)-SUN9221 (4E)-SUN9221 is a potent antagonist of α1-adrenergic receptor and 5-HT2 receptor, with antihypertensive and anti-platelet aggregation activities. (4E)-SUN9221 Chemical Structure
  12. GC11952 (R)-(+)-Atenolol

    (R)-Atenolol

     less active enantiomer of the racemic β1-adrenergic receptor antagonist, (R,S)-atenolol. (R)-(+)-Atenolol Chemical Structure
  13. GC11937 (R)-(+)-m-Nitrobiphenyline oxalate α2C-AR (adrenoceptor) agonist (R)-(+)-m-Nitrobiphenyline oxalate Chemical Structure
  14. GC10608 (R)-(+)-Propranolol hydrochloride

    β-adrenoceptor antagonist

     (R)-(+)-Propranolol hydrochloride Chemical Structure
  15. GC12144 (R)-(-)-Niguldipine hydrochloride L-type Ca2+ channel blocker and α1A-adrenoceptor antagonist (R)-(-)-Niguldipine hydrochloride Chemical Structure
  16. GC60001 (R)-Carvedilol (R)-Carvedilol ((R)-BM 14190), the R-enantiomer of Carvedilol, is a non-selective β/α-1 blocker. (R)-Carvedilol Chemical Structure
  17. GC39298 (R)-Terazosin (R)-Terazosin is an active R-enantiomer of Terazosin. (R)-Terazosin Chemical Structure
  18. GC14145 (R,R)-Formoterol

    (-)-Formoterol;Arformoterol;Formoterol

     β2-selective adrenergic agonist (R,R)-Formoterol Chemical Structure
  19. GC12823 (R,S)-Atenolol

    Duraatenol,IC I66082,Tenormin®

     (R,S)-Atenolol ((RS)-(R,S)-Atenolol) is a cardioselective β1-adrenergic receptor blocker, with a Ki of 697 nM atβ1-adrenoceptor in guine pig left ventricle membrane. (R,S)-Atenolol Chemical Structure
  20. GC64481 (rac)-Dobutamine-d4 hydrochloride (rac)-Dobutamine-d4 hydrochloride Chemical Structure
  21. GC62642 (rac)-Dobutamine-d6 hydrochloride (rac)-Dobutamine-d6 hydrochloride Chemical Structure
  22. GC62228 (rac)-Nebivolol-d4 (Rac)-Nebivolol-d4 ((Rac)-R 065824-d4) is a labelled racemic Nebivolol. (rac)-Nebivolol-d4 Chemical Structure
  23. GC34367 (RS)-Butyryltimolol (RS)-Butyryltimolol is the racemate of Butyryltimolol. (RS)-Butyryltimolol Chemical Structure
  24. GC15292 (S)-(+)-Niguldipine hydrochloride L-type Ca2+ channel blocker and α1A-adrenoceptor antagonist (S)-(+)-Niguldipine hydrochloride Chemical Structure
  25. GC12463 (S)-(-)-Atenolol (S)-(-)-Atenolol is a potent β-adrenergic receptor blocker. (S)-(-)-Atenolol is the S(-) enantiomer of Atenolol, while the R(+) enantiomer of Atenolol has almost no β-receptor blocker activity. (S)-(-)-Atenolol Chemical Structure
  26. GC15039 (S)-(-)-Pindolol beta-adrenergic antagonist (S)-(-)-Pindolol Chemical Structure
  27. GC16637 (S)-(-)-Propranolol hydrochloride β-adrenoceptor antagonist (S)-(-)-Propranolol hydrochloride Chemical Structure
  28. GC60006 (S)-Carvedilol (S)-Carvedilol, the S-enantiomer of Carvedilol, is a non-selective β/α-1 blocker. (S)-Carvedilol Chemical Structure
  29. GC39249 (S)-Terazosin (S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin Chemical Structure
  30. GC16663 (±)-4-hydroxy Propranolol (hydrochloride) β1- and β2-adrenergic receptors inhibitor (±)-4-hydroxy Propranolol (hydrochloride) Chemical Structure
  31. GC15087 (±)-Talinolol

    Cordanum

     β1-selective adrenoceptor antagonist (±)-Talinolol Chemical Structure
  32. GC91055 2,6-Xylidine-d6 (hydrochloride)

    An Analytical Reference Standard

     2,6-Xylidine-d6 (hydrochloride) Chemical Structure
  33. GC16412 2-MPMDQ α1-adrenoceptor antagonist,potent and selective 2-MPMDQ Chemical Structure
  34. GC13695 2-PMDQ α1-adrenoceptor antagonist 2-PMDQ Chemical Structure
  35. GN10169 3-Hydroxy-4-methoxycinnamic acid

    3-methoxy Caffeic Acid, 3-hydroxy-4-Methoxycinnamic Acid, NSC 51987

     3-Hydroxy-4-methoxycinnamic acid Chemical Structure
  36. GC10073 3-MPPI ligand for adrenergic α1 receptor 3-MPPI Chemical Structure
  37. GC68327 4-Hydroxyatomoxetine-d3 4-Hydroxyatomoxetine-d3 Chemical Structure
  38. GC64116 4-Hydroxypropranolol-d7

    (±)-4-Hydroxy Propranolol-d7

     4-Hydroxypropranolol-d7 Chemical Structure
  39. GC70207 4-Hydroxypropranolol-d7 hydrochloride 4-Hydroxypropranolol-d7 (hydrochloride) is a deuterium labeled 4-Hydroxypropranolol hydrochloride. 4-Hydroxypropranolol-d7 hydrochloride Chemical Structure
  40. GC32655 5-HT2 antagonist 1 5-HT2 antagonist 1 is a potent antagonist of 5-HT2 receptor, with weak α1 adrenoceptor blocking activity. 5-HT2 antagonist 1 Chemical Structure
  41. GC14527 A 61603 hydrobromide A 61603 hydrobromide is a selective α1A-adrenergic receptor agonist. A 61603 hydrobromide Chemical Structure
  42. GC13027 A 80426 mesylate α2-adrenoceptor antagonist and 5-HT uptake inhibitor A 80426 mesylate Chemical Structure
  43. GC41327 Aaptamine Aaptamine is a marine sponge alkaloid originally isolated from A. Aaptamine Chemical Structure
  44. GC67702 Abanoquil

    U-K52046; Albanoquil

     Abanoquil Chemical Structure
  45. GC60552 Acebutolol D7 Acebutolol D7 is a deuterium labeled Acebutolol. Acebutolol D7 Chemical Structure
  46. GC13000 Acebutolol HCl

    M&B 17803A

     Acebutolol HCl is an orally active β1 adrenergic receptor (β1AR) antagonist. Acebutolol HCl Chemical Structure
  47. GC35243 ACTH (1-14) TFA

    Adrenocorticotropic Hormone Fragment 1-14 TFA

     ACTH (1-14) TFA Chemical Structure
  48. GC30547 ACTH 1-14 (Adrenocorticotropic Hormone Fragment 1-14) ACTH 1-14 (Adrenocorticotropic Hormone Fragment 1-14) is a fragment of adrenocorticotrophin, which regulates cortisol and androgen production. ACTH 1-14 (Adrenocorticotropic Hormone Fragment 1-14) Chemical Structure
  49. GC68627 ADRA1D receptor antagonist 1

    ADRA1D receptor antagonist 1 is a highly efficient, selective, orally active α1D adrenergic receptor antagonist with a Ki value of 1.6 nM.

     ADRA1D receptor antagonist 1 Chemical Structure
  50. GC13814 Adrenalone HCl Decoyinine (Angustmycin A), a specific inhibitor of bacterial GMPS, has been isolated from Streptomyces . Adrenalone HCl Chemical Structure
  51. GC16831 Agmatine sulfate

    NIH 11035

     α2-adrenergic receptor ligand Agmatine sulfate Chemical Structure
  52. GC32599 AGN 192836 AGN 192836 is a potent and selective α2 adrenergic agonist with EC50s of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively. AGN 192836 Chemical Structure
  53. GC70735 Agroclavine Agroclavine is a natural, clavine type of ergot alkaloid. Agroclavine Chemical Structure
  54. GC10197 AH 11110 hydrochloride α1B-AR ligand,subtype-selective AH 11110 hydrochloride Chemical Structure
  55. GC35272 Ajmalicine

    (-)-Ajmalicine, NSC 72133, NSC 95087, Raubasine

     A terpenoid indole alkaloid Ajmalicine Chemical Structure
  56. GC16740 Alfuzosin alpha-adrenergic blocker Alfuzosin Chemical Structure
  57. GC13730 Alfuzosin HCl

    SL 7749910, Uroxatral

     Alfuzosin (SL 77499-10) hydrochloride is an orally active, selective and competitive α1-adrenoceptor antagonist. Alfuzosin HCl Chemical Structure
  58. GC14105 Alprenolol hydrochloride β-adrenoceptor and 5-HT1A receptor antagonist. Alprenolol hydrochloride Chemical Structure
  59. GC32516 Amezinium methylsulfate (Amezinium metilsulfate) Amezinium metilsulfate has multiple mechanisms, including stimulation of alpha and beta-1 receptors and inhibition ofnoradrenaline and tyramine uptake. Amezinium methylsulfate (Amezinium metilsulfate) Chemical Structure
  60. GC33983 Amitraz (BTS-27419)

    NSC 324552

     Amitraz (BTS-27419) is a non-systemic acaricide and insecticide, with alpha-adrenergic agonist activity, interaction with octopamine receptors of the central nervous system and inhibition of monoamine oxidases and prostaglandin synthesis. Amitraz (BTS-27419) Chemical Structure
  61. GC70259 Amosulalol Amosulalol (YM 09538) is an orally active and dual inhibitor of α1/β1-Adrenergic Receptor. Amosulalol Chemical Structure
  62. GC70475 Ampreloxetine Ampreloxetine (TD-9855) is a potent and orally active norepinephrine (NE) and serotonin 5-HT inhibitor. Ampreloxetine Chemical Structure
  63. GC70476 Ampreloxetine TFA Ampreloxetine (TD-9855) TFA is a potent and orally active norepinephrine (NE) and serotonin 5-HT inhibitor. Ampreloxetine TFA Chemical Structure
  64. GC32582 Ancarolol Ancarolol is a beta-adrenergic blocking agent. Ancarolol Chemical Structure
  65. GC17736 Anisodamine

    6-hydroxy Hyoscyamine

    weak antagonist of α1-adrenoceptors

     Anisodamine Chemical Structure
  66. GC60593 Arbutamine Arbutamine is a short-acting, potent and nonselective β-adrenoceptor agonist. Arbutamine Chemical Structure
  67. GC68683 ARC 239

    ARC 239 is an α2B/C-adrenergic receptor antagonist, with pKi values of 7.06 and 6.95 for rat kidney α2B and human kidney α2C, respectively. ARC 239 also inhibits the 5-HT1A receptor with a Ki value of 63.1 nM.

     ARC 239 Chemical Structure
  68. GC10965 ARC 239 dihydrochloride α2B adrenoceptor antagonist ARC 239 dihydrochloride Chemical Structure
  69. GC42851 Arformoterol (tartrate)

    (R,R)-Formoterol

     Aformoterol is the (R,R)-enantiomer of the β2-adrenergic receptor (β2-AR) agonist formoterol. Arformoterol (tartrate) Chemical Structure
  70. GC11824 Asenapine Inhibits adrenergic receptor/5-HT receptor Asenapine Chemical Structure
  71. GC30791 Atipamezole (MPV 1248)

    MPV 1248

     Atipamezole (MPV 1248) (MPV 1248) is a potent α2-adrenoceptor antagonist with a Ki of 1.6 nM. Atipamezole (MPV 1248) Chemical Structure
  72. GC16106 Atipamezole hydrochloride α2-adrenergic receptor antagonist Atipamezole hydrochloride Chemical Structure
  73. GC14491 B-HT 920 A potent agonist of D2 receptors B-HT 920 Chemical Structure
  74. GC14514 B-HT 933 dihydrochloride

    Azepexole, Oxazoloazepin

     Azepexole (B-HT 933) dihydrochloride is a potent and selective alpha 2-adrenoceptor agonist with pKis of 8.3, 7.6, and 7.5 for α2A-, α2B- and α2C-adrenoceptor subtypes, resepctively. B-HT 933 dihydrochloride Chemical Structure
  75. GC13577 Bambuterol long acting beta-adrenoceptor agonist Bambuterol Chemical Structure
  76. GC42896 Bambuterol (hydrochloride)

    KWD 2183

     Bambuterol is a prodrug for terbutaline, a long-acting β-adrenoceptor agonist (Ki = 15.4 μM for human β2-adrenergic receptor). Bambuterol (hydrochloride) Chemical Structure
  77. GC63433 Bambuterol-d9 hydrochloride Bambuterol-d9 hydrochloride Chemical Structure
  78. GC31690 Batefenterol (GSK961081)

    GSK961081, TD-5959

     Batefenterol (GSK961081) (GSK961081;TD-5959) is a novel muscarinic receptor antagonist and β2-adrenoceptor agonist; displays high affinity for hM2, hM3 muscarinic and hβ2-adrenoceptor with Ki values of 1.4, 1.3 and 3.7 nM, respectively. Batefenterol (GSK961081) Chemical Structure
  79. GC65252 Benoxathian hydrochloride Benoxathian hydrochloride is a potent α1 adrenoceptor antagonist, can be used for researching anorexia. Benoxathian hydrochloride Chemical Structure
  80. GC30474 Benzquinamide (P2647) Benzquinamide (P2647) Chemical Structure
  81. GC74632 Benzquinamide hydrochloride

    P2647 hydrochloride; BZQ hydrochloride; Benzoquinamide hydrochloride

     Benzquinamide (P2647) is an antiemetic which can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) with Ki values of 1,365, 691, and 545 nM, respectively. Benzquinamide hydrochloride Chemical Structure
  82. GC14021 Betaxolol βadrenergic receptor blocker Betaxolol Chemical Structure
  83. GC17731 Betaxolol HCl

    SL 75212

     Betaxolol Hydrochloride is a selective beta1 adrenergic receptor blocker that can be used for the research of hypertension and glaucoma. Betaxolol HCl Chemical Structure
  84. GC71649 Betaxolol-d5 Betaxolol-d5 is the deuterium labeled Betaxolol. Betaxolol-d5 Chemical Structure
  85. GC39546 Bevantolol hydrochloride

    CI-755, DL-Bevantolol, NC-1400

     A β1-AR antagonist Bevantolol hydrochloride Chemical Structure
  86. GC38378 BI-167107 BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR) with a dissociation constant Kd of 84 pM. BI-167107 Chemical Structure
  87. GC25140 Bisoprolol Bisoprolol is a cardioselective β1-adrenergic blocking agent used for secondary prevention of myocardial infarction (MI), heart failure, angina pectoris and mild to moderate hypertension. Bisoprolol Chemical Structure
  88. GC14818 Bisoprolol fumarate

    EMD 33512

     Bisoprolol fumarate is a potent, selective and orally active β1-adrenergic receptor blocker with little activity on β2-receptor. Bisoprolol fumarate Chemical Structure
  89. GC70620 Bisoprolol-d5 Bisoprolol-d5 is the deuterium labeled Bisoprolol. Bisoprolol-d5 Chemical Structure
  90. GC68786 BMY 14802

    BMY 14802 is an antagonist of the sigma-1 receptor (σ1R) and an agonist of the serotonin 1A receptor (5-HT 1A Receptor) and alpha-1 adrenergic receptor (α-1 adrenergic receptor). In a rat model of Parkinson's disease (PD), BMY 14802 can inhibit abnormal involuntary movements (AIM) and downregulate AIM expression.

     BMY 14802 Chemical Structure
  91. GC32665 Bometolol Hydrochloride Bometolol Hydrochloride is a beta-adrenergic blocking agent, used for the research of cardiovascular disease. Bometolol Hydrochloride Chemical Structure
  92. GC10738 Brimonidine Tartrate

    AGN 190342LF, Alphagan P

     Highly selective α-adrenergic receptor agonist Brimonidine Tartrate Chemical Structure
  93. GC13785 BRL 37344, sodium salt

    BRL 37344A

     BRL 37344, sodium salt (BRL 37344A) is a specific β3-adrenergic receptor agonist. BRL 37344, sodium salt Chemical Structure
  94. GC13996 BRL 44408 maleate Selective α2A-AR antagonist BRL 44408 maleate Chemical Structure
  95. GC72764 BRL-37344 BRL-37344 (Fosigotifator (THAM sodium)) is a specific β3-adrenergic receptor agonist. BRL-37344 Chemical Structure
  96. GC70761 Bromchlorbuterol hydrochloride Bromchlorbuterol hydrochloride is an active β-adrenergic agonist (β-agonist) and can be used for the research of pulmonary disease and asthma. Bromchlorbuterol hydrochloride Chemical Structure
  97. GC15328 Bucindolol

    DL-Bucindolol, MJ13105-1

     beta adrenergic blocker Bucindolol Chemical Structure
  98. GC67692 Bufuralol Bufuralol Chemical Structure
  99. GC15347 Bufuralol (hydrochloride)

    Ro 3-4787

     non-specific β-adrenergic blocker Bufuralol (hydrochloride) Chemical Structure
  100. GC64450 Bunazosin Bunazosin is a potent and selective α1-adrenoceptor antagonist. Bunazosin Chemical Structure
  101. GC62648 Bupranolol

    (±)-Bupranolol

     Bupranolol is an orally active, competitive and non-selective β-adrenoceptor antagonist without intrinsic sympathomimetic activity. Bupranolol Chemical Structure

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