Adrenergic Receptor
Adrenergic receptor is a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine and epinephrine.
Products for Adrenergic Receptor
- Cat.No. Product Name Information
- GC12626 Cimaterol β-Adrenergic agonist
- GC45826 Cimaterol-d7 An internal standard for the quantification of cimaterol
- GC62897 Cimbuterol-D9 Cimbuterol-D9 is the deuterium labeled Cimbuterol.
- GC15218 Cirazoline hydrochloride α1 agonist
- GC12226 Cisatracurium Besylate Neuromuscular-blocking drug
-
GC43276
CL 316,243 (disodium salt)
A murine-selective β3 adrenoceptor agonist
- GC12778 Clenbuterol (hydrochloride) sympathomimetic β2-adrenoceptor agonist used as a bronchodilator in the treatment of pulmonary diseases
- GC68418 Clenbuterol-d9
- GC62900 Clenproperol-D7 Clenproperol-D7 is the deuterium labeled Clenproperol.
- GC60717 Clonidine Clonidine is an alpha 2-adrenergic agonist.
- GC14032 Clonidine HCl Clonidine HCl is an agonist of α2-adrenoceptor and potent antihypertensive agent.
- GC12949 Clorprenaline HCL Clorprenaline HCL is a β2-adrenergic receptor agonist that is implicated in bronchial expansion.
- GC30665 D2343 D2343 is a β2-adrenoceptor agonist and also is an α1- adrenoceptor inhibitor.
- GC38762 Dabuzalgron Dabuzalgron (Ro 115-1240) is an orally active and selective α-1A adrenergic receptor agonist for the treatment of urinary incontinence.
- GC30188 Dapiprazole hydrochloride An α-adrenergic receptor antagonist
- GC65955 Denopamine Denopamine ((R)-(-)-Denopamine) is an orally active, selective β1-adrenergic agonist. Denopamine prolongs survival in a murine model of congestive heart failure induced by viral myocarditis: suppression of tumor necrosis factor-α production in the heart. Cardiovascular effects.
- GC31468 Deriglidole (SL 86-0715) Deriglidole (SL 86-0715) is a peripheral adrenoceptor antagonist with a high affinity for α2-adrenoceptors.
- GC17197 Detomidine α2-adrenergic agonist
- GC17081 Detomidine HCl Detomidine HCl, an imidazole derivative, is a potent α2-adrenergic agonist.
-
GC17494
Dexmedetomidine
An α2-adrenergic receptor agonist
- GC10750 Dexmedetomidine HCl Dexmedetomidine HCl ((+)-Medetomidine hydrochloride) is a potent, selective and orally active agonist of α2-adrenoceptor, with a Ki of 1.08 nM.
- GC60764 Diacetolol D7 Diacetolol D7 is a deuterium labeled Diacetolol.
- GC60767 Dibenamine hydrochloride Dibenamine hydrochloride is a competitive and irreversible?adrenergic blocking agent and?is known to modify the pharmacological effects of epinephrine.
- GC38527 Dicentrine Dicentrine is a natural product isolated from the plant Lindera megaphylla with antihypertensive effect.
- GC13256 Dihydroergocristine mesylate 5-HT receptor antagonist and partial agonist of adrenergic and dopaminergic receptors
- GC13378 DL-Adrenaline Adrenergic receptor agonist
- GC39257 DL-Norepinephrine hydrochloride DL-Norepinephrine hydrochloride is a synthetic phenylethylamine that mimics the sympathomimetic actions of the endogenous norepinephrine.DL-Norepinephrine hydrochloride is a neurotransmitter targets α1 and β1 adrenoceptors, has an increasing effect on subendocardial oxygen tension.
- GC35891 Dobutamine hydrochloride Dobutamine hydrochloride is a synthetic catecholamine that acts on α1-AR, β1-AR, β2-AR (α-1, β-1 andβ-2 adrenoceptors).
- GC32627 Dopexamine hydrochloride (FPL60278AR) Dopexamine hydrochloride (FPL60278AR) is a β2 adrenergic receptor agonist.
- GC13447 Doxazosin Quinazoline-derivative that selectively antagonizes postsynaptic α1-adrenergic receptors
- GC60790 Doxazosin D8 Doxazosin D8 (UK 33274 D8) is a deuterium labeled Doxazosin (UK 33274).
- GC13443 Doxazosin Mesylate α1-adrenergic receptor antagonist
- GC12042 DSP-4 DSP-4 is a highly and selective adrenergic neurotoxin.
- GC32547 Ecastolol Ecastolol is a beta adrenergic receptor antagonist, with antianginal activities.
- GC15672 Efaroxan hydrochloride α2 adrenoceptor antagonist and imidazoline I1 receptor ligand
- GC31378 Epanolol (Visacor) Epanolol (Visacor) (Visacor; ICI141292) is a potent β-adrenoceptor partial agonist with a greater affinity for β1- than β2-adrenoceptors.
- GC13393 Epinephrine Bitartrate Adrenergic receptor agonist
- GC15698 Epinephrine HCl Adrenergic receptor agonist
- GC25385 Esmolol Esmolol is a cardioselective beta1 receptor blocker with rapid onset, a very short duration of action, and no significant intrinsic sympathomimetic or membrane stabilising activity at therapeutic dosages.
- GC14968 Esmolol HCl Esmolol HCl is a beta adrenergic receptor blocker.
- GC32418 Falintolol, (Z)- Falintolol, (Z)-, a new β-adrenergic antagonist, is characterized by the presence of an oxime function.
- GC18086 Fendiline (hydrochloride) α2-adrenergic receptor antagonist
- GC31271 Fenmetozole Tosylate Fenmetozole Tosylate is an antagonist of the actions of ethanol, also antagonizes α2-adrenergic receptor, and acts as an antidepressant drug.
- GC25412 Fenoterol Fenoterol (Phenoterol) is a β2 adrenoreceptor agonist with bronchodilator activity.
- GC43661 Fenoterol (hydrobromide) Fenoterol is an analytical reference standard categorized as a β2-adrenergic receptor agonist.
- GC31750 Fenspiride Hydrochloride
- GC30679 Fiduxosin Fiduxosin is a potent α1-adrenoceptor antagonist, with Ki of 0.160 nM, 24.9 nM, and 0.920 nM for α1a-, α1b-, and α1d-adrenoceptors, respectively.
- GC15918 Formoterol Hemifumarate Potent, selective and long-acting β2-adrenoceptor agonist
- GC11385 G-Protein antagonist peptide Inhibits G protein activation by GPCRs
- GC41486 Glaucine Glaucine is an alkaloid originally isolated from G.
- GN10104 Gramine
- GC25484 Guanabenz Guanabenz (GBZ, GA, Wytensin, Wy-8678,BR-750) is an orally active central alpha 2-adrenoceptor (α2 adrenergic receptor) agonist with antihypertensive action.
- GC13302 Guanabenz (hydrochloride) α2-adrenergic receptor agonist
- GC16839 Guanabenz Acetate α2-adrenergic receptor agonist
- GC14813 Guanfacine selective α2A receptor agonist
- GC12132 Guanfacine hydrochloride An α2-adrenergic receptor agonist
- GC32662 Guanoxabenz (Hydroxyguanabenz) Guanoxabenz (Hydroxyguanabenz) is an α2 adrenergic receptor agonist, with a Ki of 4000 nM and the fully activated form 40 nM for an α2A adrenoceptor.
- GC61882 Guanoxabenz hydrochloride Guanoxabenz (Hydroxyguanabenz) hydrochloride is an α2 adrenergic receptor agonist, with a Ki of 4000 nM and the fully activated form 40 nM for an α2A adrenoceptor.
- GC15384 Harmane endogenous ligand for imidazoline binding sites
- GC12206 HEAT hydrochloride α1-adrenoceptor antagonist
- GC38099 Higenamine Higenamine (Norcoclaurine), a β2-AR agonist, is a key component of the Chinese herb aconite root that prescribes for treating symptoms of heart failure in the oriental Asian countries.
- GC38237 Higenamine hydrochloride Higenamine hydrochloride (Norcoclaurine hydrochloride), a β2-AR agonist, is a key component of the Chinese herb aconite root that prescribes for treating symptoms of heart failure in the oriental Asian countries.
- GC12243 HOKU-81
- GC36266 Hydrocortisone 17-butyrate Hydrocortisone 17-butyrate is an adrenocortico hormone
- GC43877 Hydroxy Bupropion Buproprion is an inhibitor of the reuptake of dopamine and norepinephrine and is also an antagonist of neuronal acetylcholine nicotinic receptors.
-
GC14033
ICI 118,551 hydrochloride
Highly selective β2 adrenergic receptor antagonist
- GC16547 ICI 215,001 hydrochloride active metabolite of ZD 7114
- GC12761 ICI 89406 β-adrenergic antagonist
- GC38192 Idazoxan hydrochloride
-
GC15813
Idazoxan hydrochloride
Idazoxan hydrochloride (RX 781094 hydrochloride) is an α2-adrenoceptor antagonist and also an antagonist of imidazoline receptors (IRs).
- GC11077 Imiloxan hydrochloride α2-adrenoceptor antagonist
- GC33705 Imoxiterol (RP 58802B) Imoxiterol (RP 58802B) (RP 58802B) is a β-adrenergic agonist.
- GC13808 Indacaterol A long-acting β2-adrenergic receptor agonist
- GC11130 Indacaterol Maleate Ultra-long-acting β-adrenoceptor agonist
- GC32512 Indanidine Indanidine is an alpha-adrenergic agonist.
- GC30391 Indoramin D5 (Indoramine D5) Indoramin D5 (Indoramine D5) is deuterium labeled Indoramin, which is a piperidine antiadrenergic agent.
- GC64514 Isometheptene mucate
- GC11029 Isoprenaline HCl Isoprenaline (Isoproterenol) hydrochloride is a non-selective, orally active β-adrenergic receptor agonist.
- GC17998 Isoxsuprine (hydrochloride) β-adrenergic receptor modulator
- GC30434 Ivabradine D3 Hydrochloride An internal standard for the quantification of ivabradine
- GC34289 Ivabradine D6 hydrochloride
- GC10194 Ivabradine HCl Ivabradine HCl is a potent and orally active HCN (hyperpolarization-activated cyclic nucleotide-gated) channel blocker that inhibits the cardiac pacemaker current (If).
- GC17884 JP 1302 dihydrochloride α2C-adrenoceptor antagonist
- GC43932 JP-1302 (hydrochloride) JP-1302 (hydrochloride) is a selective, high affinity antagonist of the alpha2C-adrenoceptor (α2C-adrenoceptor), with a Kb value (antagonist activity) of 16 nM and a Ki (binding affinity) value of 28 nM.
- GC31329 Ko-3290 Ko-3290 is an antagonist of β-adrenoceptor, with cardioselectivity and antilipolytic effects in animals.
- GC36413 L-(-)-α-Methyldopa hydrate L-(-)-α-Methyldopa hydrate (L-(-)-α-L-(-)-α-Methyldopa hydrate), a potent antihyoertensive agent, is an alpha-adrenergic agonist (selective for α2-adrenergic receptors).
- GC16401 L-(-)-α-Methyldopa hydrochloride L-(-)-α-Methyldopa hydrochloride (L-(-)-α-L-(-)-α-Methyldopa hydrochloride) hydrochloride, a potent antihyoertensive agent, is an alpha-adrenergic agonist (selective for α2-adrenergic receptors).
- GC16939 L-748,337 Competitive β3-adrenoceptor antagonist
- GC15743 L-755,507 β3 adrenergic receptor agonist
- GC32670 L-765314 L-765314 is a potent and selective α1b adrenergic receptor antagonist with Kis of 5.4 nM and 2.0 nM for rat and human α1b adrenergic receptor, respectively.
- GC33410 L-771688 L-771688 is a highly selective α1A-Adrenoceptor antagonist with a Ki of 0.43±0.02 nM.
- GC14816 L-Adrenaline An adrenergic receptor agonist
- GC17319 L-Phenylephrine (R)-(-)-L-Phenylephrine is a selective α1-adrenoceptor agonist primarily used as a decongestant.
- GC64143 Labetalol Labetalol (AH5158) is an orally active selective α1- and non-selective β-adrenergic receptors competitive antagonist.
- GC10887 Labetalol HCl Labetalol HCl is a mixed alpha/beta adrenergic antagonist that is used to treat high blood pressure.
- GC36422 Landiolol hydrochloride Landiolol hydrochloride (ONO1101 hydrochloride) is a highly beta1 selective ultra-short acting beta-blocker (β1/β2 selectivity?=?255:1, a half-life of 4?min), acts as an adrenoceptor antagonist.
- GC17974 Latrepirdine dihydrochloride Latrepirdine is a neuroactive compound with antagonist activity at histaminergic, α-adrenergic, and serotonergic receptors.
- GC36441 Levalbuterol tartrate Levosalbutamol tartrate(levalbuterol) is the R-enantiomer of the short-acting β2-adrenergic receptor agonist salbutamol.
- GC17653 Levobetaxolol HCl Levobetaxolol HCl is a beta-adrenergic receptor inhibitor (beta blocker) that can lower the pressure in the eye.
- GC30972 Lidanserin (ZK-33839) Lidanserin (ZK-33839) (ZK-33839) acts as a 5-HT2A and α1-adrenergic receptor antagonist.