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Home >> Signaling Pathways >> GPCR/G protein >> Adrenergic Receptor

Adrenergic Receptor

Adrenergic receptor is a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine and epinephrine.

Products for  Adrenergic Receptor

  1. Cat.No. Product Name Information
  2. GC36477 Lofexidine Lofexidine is a selective α2-receptor agonist, commonly used to alleviate the physical symptoms of heroin and other types of opioid withdrawal. Lofexidine Chemical Structure
  3. GC17064 Lofexidine (hydrochloride) α2-adrenergic receptor agonist Lofexidine (hydrochloride) Chemical Structure
  4. GC67977 Lubabegron Lubabegron Chemical Structure
  5. GC31266 Lusaperidone (R107474) Lusaperidone (R107474) (R107474) is an α2 adrenergic receptor antagonist with Kis of 0.13 and 0.15 nM for α2A and α2C, respectively. Lusaperidone (R107474) Chemical Structure
  6. GC63054 Mabuterol-D9 Mabuterol-D9 is a deuterium labeled Mabuterol. Mabuterol-D9 Chemical Structure
  7. GC12376 Maprotiline HCl Maprotiline HCl is a selective noradrenalin re-uptake inhibitor and a tetracyclic antidepressant. Maprotiline HCl Chemical Structure
  8. GC13144 Medetomidine Medetomidine Chemical Structure
  9. GC12983 Medetomidine HCl Medetomidine (hydrochloride) is a potent, selective, and specific α2-adrenoceptor agonist in both the peripheral and central nervous systems. Medetomidine HCl Chemical Structure
  10. GC65874 Medroxalol Medroxalol (RMI81968) is an orally active adrenergic receptor antagonist, blocks α- and β-adrenergic receptors. Medroxalol shows antihypertensive and vasodilating effects. Medroxalol Chemical Structure
  11. GC60243 Meranzin Meranzin is an absorbed bioactive compound from the Traditional Chinese Medicine (TCM) Chaihu-Shugan-San (CSS). Meranzin Chemical Structure
  12. GC44169 Metaproterenol (hemisulfate) Metaproterenol is a β2-adrenergic receptor (β2-AR) agonist with bronchodilator actions. Metaproterenol (hemisulfate) Chemical Structure
  13. GC63067 Methoxyphenamine Methoxyphenamine Chemical Structure
  14. GC63068 Methoxyphenamine hydrochloride Methoxyphenamine hydrochloride Chemical Structure
  15. GC16490 Methyldopa alpha-2 adrenergic receptor agonist Methyldopa Chemical Structure
  16. GC17888 Metipranolol A β-AR antagonist Metipranolol Chemical Structure
  17. GC44185 Metipranolol (hydrochloride) Metipranolol is a non-selective β-adrenergic receptor (β-AR) antagonist. Metipranolol (hydrochloride) Chemical Structure
  18. GC36603 Metoprolol Metoprolol is an orally active, selective β1-adrenoceptor antagonist. Metoprolol Chemical Structure
  19. GC17945 Metoprolol Succinate beta-1 selective adrenergic receptor antagonist Metoprolol Succinate Chemical Structure
  20. GC14536 Metoprolol Tartrate β1-adrenergic blocking agent Metoprolol Tartrate Chemical Structure
  21. GC34048 MG 1 MG 1 is an α1 adrenergic receptor antagonist. MG 1 Chemical Structure
  22. GC67691 Midaglizole Midaglizole Chemical Structure
  23. GC31615 Midaglizole hydrochloride ((±)-DG5128) Midaglizole hydrochloride ((±)-DG5128) (DG5128) is a preferential α2-adrenoceptor antagonist. Midaglizole hydrochloride ((±)-DG5128) Chemical Structure
  24. GC11239 Midodrine (hydrochloride) prodrug of the α1-adrenergic receptor agonist Midodrine (hydrochloride) Chemical Structure
  25. GC11915 Mirabegron (YM178) Mirabegron (YM178) is a selective β3-adrenoceptor agonist with EC50 of 22.4 nM. Mirabegron (YM178) Chemical Structure
  26. GC48855 Mirtazapine (CRM) A Certified Reference Material Mirtazapine (CRM) Chemical Structure
  27. GC32485 Moxisylyte hydrochloride (Thymoxamine hydrochloride) Moxisylyte (hydrochloride) is (alpha 1-blocker) antagonist, it can vasodilates cerebral vessels without reducing blood pressure. Moxisylyte hydrochloride (Thymoxamine hydrochloride) Chemical Structure
  28. GC39740 Nadolol Nadolol (SQ-11725) is a non-selective and orally active β-adrenergic receptors blocker and is a substrate of organic anion transporting polypeptide 1A2 (OATP1A2). Nadolol Chemical Structure
  29. GC36687 Nadolol D9 Nadolol D9 (SQ-11725 D9) is the deuterium labeled Nadolol. Nadolol D9 Chemical Structure
  30. GC16836 Naftopidil α1-adrenergic receptor antagonist Naftopidil Chemical Structure
  31. GC44311 Naftopidil (hydrochloride) Naftopidil is an α1-adrenergic receptor antagonist that competitively inhibits α-adrenoceptor-mediated contractions induced by noradrenaline with pA2 values of 6.73-8.15 in various blood vessels from dog, rabbit, guinea pig, and rat. Naftopidil (hydrochloride) Chemical Structure
  32. GC17765 Naftopidil DiHCl Naftopidil DiHCl (KT-611 dihydrochloride) is a selective alpha1-adrenoceptor antagonist, with Kis of 3.7 nM, 20 nM and 1.2 nM for the cloned human α1a-, α1b- and α1d-adrenoceptor subtypes, respectively. Naftopidil DiHCl has antiproliferative effects. Naftopidil DiHCl can be used for the research of prostate hyperplasia. Naftopidil DiHCl Chemical Structure
  33. GC14988 Naphazoline HCl Naphazoline (Naphthazoline) hydrochloride is a potent α-adrenergic receptor agonist. Naphazoline HCl Chemical Structure
  34. GC25663 Nebivolol Nebivolol (Bystolic,R 065824) is a β1 receptor blocker with nitric oxide-potentiating vasodilatory effect used in treatment of hypertension and also for left ventricular failure. Nebivolol Chemical Structure
  35. GC13906 Nebivolol hydrochloride Highly selective β1-adrenoceptor antagonist Nebivolol hydrochloride Chemical Structure
  36. GC15786 Nedaplatin DNA synthesis inhibitor Nedaplatin Chemical Structure
  37. GC16324 Nefazodone hydrochloride 5-HT2A receptor antagonist Nefazodone hydrochloride Chemical Structure
  38. GC16141 Nicergoline vasodilator Nicergoline Chemical Structure
  39. GC14919 Niguldipine (hydrochloride) α1A-adrenoceptor antagonist Niguldipine (hydrochloride) Chemical Structure
  40. GC50113 Noradrenaline bitartrate Norepinephrine (Levarterenol; L-Noradrenaline) tartrate is a potent adrenergic receptor (AR) agonist. Noradrenaline bitartrate Chemical Structure
  41. GC10976 Noradrenaline bitartrate monohydrate Norepinephrine (Levarterenol; L-Noradrenaline) bitartrate monohydrate is a potent adrenergic receptor (AR) agonist. Noradrenaline bitartrate monohydrate Chemical Structure
  42. GC30744 Norepinephrine (Adrenor) Norepinephrine (Adrenor) (Levarterenol; L-Noradrenaline) is a potent adrenergic receptor (AR) agonist. Norepinephrine (Adrenor) Chemical Structure
  43. GC36758 Norepinephrine hydrochloride Norepinephrine (Levarterenol; L-Noradrenaline) hydrochloride is a potent adrenergic receptor (AR) agonist. Norepinephrine hydrochloride Chemical Structure
  44. GC15704 NPEC-caged-noradrenalin Adrenergic receptor agonist NPEC-caged-noradrenalin Chemical Structure
  45. GC31015 NRA-0160 NRA-0160 is a selective dopamine D4 receptor antagonist, with a Ki value of 0.48 nM and with negligible affinity for dopamine D2 receptor (Ki: >10000 nM), D3 receptor (Ki: 39 nM), rat 5-HT2A receptor (Ki: 180 nM) and rat α1 adrenoceptor (Ki: 237 nM). NRA-0160 Chemical Structure
  46. GC61813 O-Desmethyl Mebeverine alcohol hydrochloride O-Desmethyl Mebeverine alcohol hydrochloride is a metabolite of Mebeverine, which is a potent α1 repector inhibitor, causing relaxation of the gastrointestinal tract. O-Desmethyl Mebeverine alcohol hydrochloride Chemical Structure
  47. GC61809 Olanzapine D3 Olanzapine D3 (LY170053-d3) is the deuterium labeled Olanzapine. Olanzapine D3 Chemical Structure
  48. GC62219 Olodaterol hydrochloride Olodaterol (BI1744) hydrochloride is a selective, long acting β2-adrenoceptor (β2-AR) agonist (EC50=0.1 nM and pKi= 9.14 for human β2-adrenoceptor, respectively). Olodaterol hydrochloride Chemical Structure
  49. GC32543 OPC-28326 OPC-28326 is a selective peripheral vasodilator and an angatonist of α2-adrenergic receptor, with Ki of 2040, 285, and 55?nM for α2A-, α2B- and α2C-adrenoceptors, respectively. OPC-28326 Chemical Structure
  50. GC10818 Oxprenolol hydrochloride β-adrenergic inhibitor Oxprenolol hydrochloride Chemical Structure
  51. GC13844 p-iodo-Clonidine (hydrochloride) partial agonist of the α2-adrenergic receptor p-iodo-Clonidine (hydrochloride) Chemical Structure
  52. GC32532 Pamatolol Pamatolol is a cardioselective beta-adrenoceptor antagonist without sympathomimetic activity. Pamatolol Chemical Structure
  53. GC31069 Pardoprunox (SLV-308) Pardoprunox (SLV-308) (SLV-308) is a partial dopamine D2 and D3 receptor partial agonist and a serotonin 5-HT1A receptor agonist, with pEC50s of 8, 9.2, and 6.3, respectively. Pardoprunox (SLV-308) Chemical Structure
  54. GC30980 Pardoprunox hydrochloride (SLV-308 hydrochloride) Pardoprunox (SLV-308) hydrochloride is a partial dopamine D2 and D3 receptor partial agonist and a serotonin 5-HT1A receptor agonist, with pEC50s of 8, 9.2, and 6.3, respectively. Pardoprunox hydrochloride (SLV-308 hydrochloride) Chemical Structure
  55. GC31009 Pargolol hydrochloride (Ko 1400 hydrochloride) Pargolol hydrochloride (Ko 1400 hydrochloride) is a β adrenergic receptor antagonist. Pargolol hydrochloride (Ko 1400 hydrochloride) Chemical Structure
  56. GC32494 Penbutolol sulfate ((-)-Terbuclomine) Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both beta-1 adrenergic receptors and beta-2 adrenergic receptors (the two subtypes), thus making it a non-selective β blocker. Penbutolol sulfate ((-)-Terbuclomine) Chemical Structure
  57. GC12293 Perphenazine dopamine antagonist Perphenazine Chemical Structure
  58. GC36875 Perphenazine D8 Dihydrochloride Perphenazine D8 Dihydrochloride is the deuterium labeled Perphenazine, which is a typical antipsychotic drug(5-HT, Dopamine receptor ligand). Perphenazine D8 Dihydrochloride Chemical Structure
  59. GC12724 Phenoxybenzamine HCl Phenoxybenzamine HCl is a nonselective, irreversible, orally active α-adrenoceptor antagonist that is commonly used for the research of hypertension, specifically caused by pheochromocytoma. Phenoxybenzamine HCl Chemical Structure
  60. GC16291 Phentolamine Mesylate Alpha 1/2-blocking agent Phentolamine Mesylate Chemical Structure
  61. GC11272 Phenylephrine HCl (R)-(-)-Phenylephrine HCl is a selective α1-adrenoceptor agonist with pKis of 5.86, 4.87 and 4.70 for α1D, α1B and α1A receptors respectively. Phenylephrine HCl Chemical Structure
  62. GC69700 Phenylephrine-2,4,6-d3 hydrochloride

    Phenylephrine-2,4,6-d3 (hydrochloride) is the deuterated form of Phenylephrine hydrochloride. (R)-(-)-Phenylephrine hydrochloride is a selective α1-adrenergic receptor agonist with pKis values of 5.86, 4.87 and 4.70 for α1D, α1B and α1A receptors respectively.

     Phenylephrine-2,4,6-d3 hydrochloride Chemical Structure
  63. GC63947 Phenylephrine-d3 hydrochloride Phenylephrine-d3 hydrochloride Chemical Structure
  64. GC68407 Phenylethanolamine A-d3 Phenylethanolamine A-d3 Chemical Structure
  65. GC10643 Pimozide dopamine receptors inhibitor Pimozide Chemical Structure
  66. GC45756 Pimozide-d4 An internal standard for the quantification of pimozide Pimozide-d4 Chemical Structure
  67. GC17734 Pindolol

    β-adrenoceptor antagonist with partial agonist activity

     Pindolol Chemical Structure
  68. GC31782 Piperoxan hydrochloride (Benodaine hydrochloride) Piperoxan (Benodaine) hydrochloride is an α2 adrenoceptor antagonist. Piperoxan hydrochloride (Benodaine hydrochloride) Chemical Structure
  69. GC36929 Piribedil A dopamine receptor agonist Piribedil Chemical Structure
  70. GC30396 Piribedil D8 (ET-495 D8) Piribedil D8 (ET-495 D8) (ET-495 D8) is the deuterium labeled Piribedil, which is an antiparkinsonian agent. Piribedil D8 (ET-495 D8) Chemical Structure
  71. GC61789 Practolol Practolol is a potent and selective β1-adrenergic receptor antagonist. Practolol Chemical Structure
  72. GC16785 Prazosin alpha-adrenergic blocker Prazosin Chemical Structure
  73. GC18072 Prazosin HCl Prazosin HCl is a well-tolerated, CNS-active α1-adrenergic receptor antagonist for the research of high blood pressure and alcohol use disorders. Prazosin HCl Chemical Structure
  74. GC64843 Prenalterol Prenalterol is a selective β1-adrenergic receptor agonist. Prenalterol Chemical Structure
  75. GC17085 Procaterol hydrochloride β2 agonist Procaterol hydrochloride Chemical Structure
  76. GC32538 Pronethalol ((±)-Pronethalo) Pronethalol ((±)-Pronethalo) ((±)-Pronethalo) is a non-selective β-adrenergic antagonist. Pronethalol ((±)-Pronethalo) Chemical Structure
  77. GC10536 Pronethalol hydrochloride

    β-adrenergic antagonist

     Pronethalol hydrochloride Chemical Structure
  78. GC25786 Propafenone Propafenone (SA-79) is an orally active sodium channel blocking agent and a beta-adrenoceptor (β-adrenergic receptor) antagonist. Propafenone offers a broad spectrum of activity in the treatment of cardiac arrhythmias. Propafenone Chemical Structure
  79. GC36980 Propranolol Propranolol is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with Ki values of 1.8 nM and 0.8 nM, respectively. Propranolol Chemical Structure
  80. GC61208 Propranolol D7 hydrochloride Propranolol D7 hydrochloride is a deuterium labeled Propranolol hydrochloride. Propranolol D7 hydrochloride Chemical Structure
  81. GC11343 Propranolol HCl Propranolol HCl is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with Ki values of 1.8 nM and 0.8 nM, respectively. Propranolol HCl Chemical Structure
  82. GC32631 QF0301B QF0301B is an α1 adrenergic receptor antagonist and a low α2 adrenoceptor, 5-HT2A, and histamine H1 receptor blocker. QF0301B Chemical Structure
  83. GC16250 Rauwolscine hydrochloride α2-adrenergic antagonist Rauwolscine hydrochloride Chemical Structure
  84. GC46212 Rec 15/2615 (hydrochloride) An α1B-AR antagonist Rec 15/2615 (hydrochloride) Chemical Structure
  85. GC17812 Rec 15/2615 dihydrochloride α1B-adrenoceptor antagonist Rec 15/2615 dihydrochloride Chemical Structure
  86. GC60325 Rilmenidine An antihypertensive agent Rilmenidine Chemical Structure
  87. GC15657 Rilmenidine (hemifumarate) I1-imidazoline binding site selective ligand and α2-adrenoceptor agonist Rilmenidine (hemifumarate) Chemical Structure
  88. GC15063 Ritodrine HCl Ritodrine (DU21220) hydrochloride is a β-adrenergic agonist, also an effective smooth muscle and uterine relaxant. Ritodrine HCl Chemical Structure
  89. GC61871 Ro 363 hydrochloride Ro 363 hydrochloride, an effective inotropic stimulant, is a potent and highly selective β1-adrenoceptor agonist. Ro 363 hydrochloride Chemical Structure
  90. GC67683 Romifidine Romifidine Chemical Structure
  91. GC10614 Rotigotine A non-selective dopamine receptor agonist Rotigotine Chemical Structure
  92. GC16017 Rotigotine hydrochloride A non-selective dopamine receptor agonist Rotigotine hydrochloride Chemical Structure
  93. GC13069 RS 100329 hydrochloride Subtype-selective α1A-adrenoceptor antagonist RS 100329 hydrochloride Chemical Structure
  94. GC17070 RS 17053 hydrochloride α1A-adrenoceptor antagonist, novel and selective RS 17053 hydrochloride Chemical Structure
  95. GC10723 RS 79948 hydrochloride α2-adrenoreceptor antagonist RS 79948 hydrochloride Chemical Structure
  96. GC10514 RWJ 52353 α2D adrenergic receptor agonist RWJ 52353 Chemical Structure
  97. GC14463 RX 821002 hydrochloride RX 821002 hydrochloride (RX821002 hydrochloride) is a highly selective alpha 2-adrenoceptor antagonist with little or no imidazoline antagonist effect. RX 821002 hydrochloride Chemical Structure
  98. GC31059 Salbutamol (Albuterol) Salbutamol (Albuterol) is a short-acting β2-adrenergic receptor agonist used for the relief of bronchospasm in conditions such as asthma and chronic obstructive pulmonary disease (COPD). Salbutamol (Albuterol) Chemical Structure
  99. GC13974 Salbutamol Sulfate Salbutamol Hemisulfate (Albuterol hemisulfate) is a short-acting β2 adrenergic receptor agonistTarget: β2 Adrenergic ReceptorSalbutamol Hemisulfate (Albuterol hemisulfate) is a short-acting, selective beta2-adrenergic receptor agonist used in the treatment of asthma and COPD. Salbutamol Sulfate Chemical Structure
  100. GC12188 Salmefamol β2-adrenergic receptor agonist Salmefamol Chemical Structure
  101. GC30092 Salmeterol (GR33343X) Salmeterol (GR33343X) (GR33343X) is a potent and selective human β2 adrenoceptor agonist. Salmeterol (GR33343X) Chemical Structure

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