Adrenergic Receptor
Adrenergic receptor is a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine and epinephrine.
Products for Adrenergic Receptor
- Cat.No. Product Name Information
- GC11531 Salmeterol xinafoate A long-acting β2-adrenergic receptor agonist
- GC48067 Salmeterol-d3 An internal standard for the quantification of salmeterol
- GC14220 Scopine α1-adrenergic receptor agonist
- GC11373 Scopine HCl Scopine HCl (6,7-Epoxytropine hydrochloride) is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.
- GC13623 SDZ 21009 β-adrenoceptor and 5-HT1A/1B receptor antagonist
- GC13990 Setiptiline
- GC13549 Setiptiline maleate
- GC15719 Silodosin α1-adrenoceptor antagonist
- GC12856 SKF 86466 hydrochloride α2-adrenoceptor antagonist
- GC15426 SNAP 5089 α1A-adrenoceptor antagonist
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GC34808
Solabegron
Solabegron (GW 427353) is a selective β3-adrenergic receptor agonist, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR, with an EC50 value of 22 nM.
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GC13173
Sotalol
Adrenergic receptor antagonist
- GC15631 Sotalol hydrochloride β-adrenergic receptor antagonist
- GC45893 Sotalol-d6 (hydrochloride) An internal standard for the quantification of sotalol
- GC31005 Spirendolol (Li 32-468) Spirendolol (Li 32-468) is a β adrenergic receptor antagonist.
- GC13338 Spiroxatrine 5-HT1A antagonist and α2C adrenergic receptor antagonist
- GC16091 SR 58611A hydrochloride SR 58611A hydrochloride is a selective β3-adrenoceptor agonist, with an EC50 of 3.5 nM for β-adrenoceptor in rat colon; SR 58611A hydrochloride has anxiolytic and antidepressant activity.
- GC12227 SR 59230A hydrochloride β3 adrenoceptor antagonist
- GC39725 SR59230A SR59230A is a potent, selective, and blood-brain barrier penetrating β3-adrenergic receptor antagonist with IC50s of 40, 408, and 648 nM for β3, β1, and β2 receptors, respectively.
- GC11913 ST 91 α2-adrenoceptor agonist
- GC38438 Synephrine
- GC12715 Synephrine HCl Synephrine (Oxedrine) hydrochloride, an alkaloid, is an α-adrenergic and β-adrenergic agonist derived from the Citrus aurantium.
- GC39449 Tamsulosin Tamsulosin ((R)-(-)-YM12617 free base) is an inhibitor of α1-adrenergic receptor.
- GC50035 Tamsulosin hydrochloride Selective α1A antagonist
- GC65276 Tasipimidine sulfate Tasipimidine sulfate is an orally active and selective α2A-adrenoceptor agonist with a pEC50 of 7.57 against human α2A-adrenoceptor.
- GC16217 TC-G 1000 α2D-adrenoceptor agonist
- GC31453 TD-5471 hydrochloride TD-5471 hydrochloride is a potent and selective full agonist of the human β2-adrenoceptor.
- GC30273 Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) Tedatioxetine (Lu AA24530) hydrobromide acts as a serotonin and norepinephrine (NE)-preferring triple reuptake inhibitor (TRI) and 5-HT2A, 5-HT2C, 5-HT3 and α1A-adrenergic receptor antagonist.
- GC30458 Teoprolol Teoprolol is a β-adrenergic receptor blocker.
- GC13085 Terazosin α1-adrenergic receptor antagonist
- GC61320 Terazosin dimer impurity dihydrochloride Terazosin dimer impurity dihydrochloride, a dimer of Terazosin, is an impurity of Terazosin.
- GC13993 Terazosin HCl Terazosin HCl is a quinazoline derivative and a competitive and orally active α1-adrenoceptor antagonist.
- GC50017 Terazosin hydrochloride α1 and α2B antagonist (α1 > α2B). Orally active
- GC11211 Terbutaline Sulfate Selective β2-adrenergic receptor agonist
- GC32637 Tertatolol ((±)-Tertatolol) Tertatolol ((±)-Tertatolol) is a potent antagonist of beta-adrenoceptor and 5-HT receptor, with unique renal vasodilatatory effects.
- GC39016 Tetrahydroalstonine Tetrahydroalstonine, a indole alkaloid isolated from the fruits of Rhazya stricta, is a selective alpha 2-adrenoceptor antagonist.
- GC14962 Tetrahydrozoline HCl Tetrahydrozoline HCl (Tetryzoline hydrochloride), a derivative of imidazoline, is an α-adrenergic agonist that causes vasoconstriction.
- GC12468 Timolol Maleate Timolol Maleate (L-714,465 Maleate) is a non-cardioselective hydrophilic β-adrenoceptor blocker.
- GC31150 Tiodazosin (BL-5111) Tiodazosin (BL-5111) is a potent competitive postsynaptic alpha adrenergic receptor antagonist.
- GC15629 Tizanidine α2 adrenergic agonist
- GC17891 Tizanidine HCl Tizanidine HCl is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.
- GC63310 Tizanidine-d4
- GC32574 Todralazine (Ecarazine) Todralazine (Ecarazine) (Ecarazine) is an anti-hypertensive agent, acts as a β2AR blocker, with antioxidant and free radical scavenging activity.
- GC18327 Todralazine (hydrochloride) Todralazine (hydrochloride) is a β2-adrenergic receptor antagonist with peripheral vasodilator activity.
- GC30405 Tolazoline (Imidaline) Tolazoline (Imidaline)(Imidaline) is a non-selective competitive α-adrenergic receptor antagonist.
- GC18092 Tolazoline HCl Tolazoline (hydrochloride)(Imidaline (hydrochloride)) Hcl is a non-selective competitive α-adrenergic receptor antagonist.
- GC13031 Trifluoperazine 2HCl Dopamine D2 receptor inhibitor
- GC63241 Trifluoperazine D8
- GC32642 Tropodifene (Tropaphen) Tropodifene (Tropaphen) (Tropaphen) is an α-Adrenergic receptor inhibitor.
- GC62650 Tulobuterol Tulobuterol (C-78 free base) is a long-acting β2-adrenoceptor agonist, which reduces the frequency of exacerbations of chronic obstructive pulmonary disease and bronchial asthma.
- GC31730 Tulobuterol hydrochloride Tulobuterol hydrochloride (C-78) is a long-acting β2-adrenoceptor agonist, which reduces the frequency of exacerbations of chronic obstructive pulmonary disease and bronchial asthma.
- GC63349 Tulobuterol-D9 hydrochloride
- GC13552 UK 14,304 UK 14,304 (UK 14304) is a full α2-adrenergic receptor (α2-AR) agonist.
- GC67715 Upidosin
- GC37861 Urapidil Urapidil is an α1 adrenoreceptor antagonist and a 5-HT1A receptor agonist.
- GC15829 Urapidil HCl Urapidil HCl is an orally active α1-adrenoceptor antagonist and 5-HT1A receptor agonist with a pIC50 of 6.13 and 4.38 against α1- and α2-adrenoceptor, respectively.
- GC30994 Vanilpyruvic acid (Vanylpyruvic acid) Vanilpyruvic acid (Vanylpyruvic acid) is a catecholamine metabolite and precursor to vanillactic acid.
- GC30938 Vatinoxan hydrochloride (MK-467 hydrochloride) Vatinoxan hydrochloride (MK-467 hydrochloride) (MK-467 hydrochloride;L-659066 hydrochloride) is a peripheral α2 adrenergic receptor antagonist.
- GC63254 Vibegron Vibegron (MK-4618) is a potent, highly selective β3-adrenoceptor agonist (EC50=1.1 nM).
- GC13747 Vilanterol β2-AR agonist
- GC14950 Vilanterol trifenatate β2-AR agonist
- GC17740 WB 4101 hydrochloride α1A-adrenergic antagonist
- GC17666 Xamoterol hemifumarate β1-adrenoceptor partial agonist
- GC12073 Xylazine α2-adrenoceptor agonist
- GC17296 Xylazine HCl α2 Adrenoceptor agonist
- GC11479 Xylometazoline HCl Xylometazoline HCl is an α-adrenergic receptor agonist (Ki=0.05-1.7 μM).
- GC37952 Yohimbine Yohimbine is a potent and relatively nonselective alpha 2-adrenergicreceptor (AR) antagonist, with IC50 of 0.6 μM.
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GN10606
Yohimbine Hydrochloride
An α2-adrenoceptor antagonist
- GC37954 YS-49 YS-49 is a PI3K/Akt (a downstream target of RhoA) activator, to reduce RhoA/PTEN activation in the 3-methylcholanthrene-treated cells.
- GC37955 YS-49 monohydrate YS-49 (monohydrate) is a PI3K/Akt (a downstream target of RhoA) activator, to reduce RhoA/PTEN activation in the 3-methylcholanthrene-treated cells.
- GC11174 ZD 2079 ZD 2079 (ZD2079 hydrochloride) is a potent β3-adrenoceptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery.
- GC17543 ZD 7114 hydrochloride β3-adrenoceptor agonist
- GC13333 Zilpaterol β-adrenergic receptor agonist
- GC48269 Zilpaterol-d7 An internal standard for the quantification of zilpaterol
- GC16111 Zinterol hydrochloride Zinterol hydrochloride (MJ 9184) is a potent and selective β2-adrenoceptor agonist.
- GC32034 ZK-90055 hydrochloride ZK-90055 hydrochloride is a β2 adrenergic receptor agonist.