Search Site
  • 0
    My Cart

    Click Here to Find How Many Items You Have Added:)

    image loader

    Adding item(s) to cart......

Home >> Signaling Pathways >> GPCR/G protein >> Angiotensin Receptor

Angiotensin Receptor

The angiotensin receptors are seven-membrane G-protein-coupled receptors. They mediate the cardiovascular and other effects of angiotensin II which is a bioactive peptide of the renin–angiotensin system.

Products for  Angiotensin Receptor

  1. Cat.No. Product Name Information
  2. GA20291 (Sar¹)-Angiotensin II (Sar¹)-Angiotensin II, an analogue of Angiotensin II, is a specific agonist of angiotensin AT1 receptor. (Sar¹)-Angiotensin II Chemical Structure
  3. GC17757 1H-1-ethyl Candesartan Cilexetil selective angiotensin II type 1 receptor (AT1) antagonist 1H-1-ethyl Candesartan Cilexetil Chemical Structure
  4. GC14445 2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine nonpeptidic angiotensin II receptor antagonist 2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine Chemical Structure
  5. GC11004 A 779 angiotensin-(1-7)/ Mas receptor antagonist A 779 Chemical Structure
  6. GC32674 A81988 (Abbott81988) A81988 (Abbott81988) is a potent, competitive, non-peptidic antagonist of angiotensin AT1 receptors. A81988 (Abbott81988) Chemical Structure
  7. GC10146 AHU-377(Sacubitril) AHU-377(Sacubitril) (AHU-377) is a potent and orally active NEP (neprilysin) inhibitor with an IC50 of 5 nM. AHU-377(Sacubitril) Chemical Structure
  8. GP10077 Angiotensin (1-7)

    Ang-(1-7) (H - Asp - Arg - Val - Tyr - Ile - His - Pro - OH) is an endogenous peptide fragment that can be produced from Ang I or Ang II via endo- or carboxy-peptidases respectively[1].

     Angiotensin (1-7) Chemical Structure
  9. GC61496 Angiotensin (1-7) (acetate) Angiotensin 1-7 (Ang-(1-7)) acetate is an endogenous heptapeptide from the renin-angiotensin system (RAS) with a cardioprotective role due to its anti-inflammatory and anti-fibrotic activities in cardiac cells. Angiotensin (1-7) (acetate) Chemical Structure
  10. GA20760 Angiotensin A (1-7) Angiotensin A (1-7), a member of the renin-angiotensin system (RAS), a vasoactive peptide, is an endogenous ligand of the G protein-coupled receptor MrgD. Angiotensin A (1-7) Chemical Structure
  11. GC12671 Angiotensin Fragment 1-7 (acetate) type 1 angiotensin II receptor agonist Angiotensin Fragment 1-7 (acetate) Chemical Structure
  12. GC61952 Angiotensin I/II (1-6) (TFA) Angiotensin I/II (1-6) TFA contains the amino acids 1-6 and is converted from Angiotensin I/II peptide. Angiotensin I/II (1-6) (TFA) Chemical Structure
  13. GC35351 Angiotensin II (1-4), human

    Angiotensin II (1-4), human is an endogenous peptide produced from AT I by angiotensin-converting-enzyme (ACE).

     Angiotensin II (1-4), human Chemical Structure
  14. GC35352 Angiotensin II (3-8), human

    Angiotensin II (3-8), human is a less effective agonist at the angiotensin AT1 receptor.

     Angiotensin II (3-8), human Chemical Structure
  15. GC35353 Angiotensin II (3-8), human TFA

    Angiotensin II (3-8), human (TFA) is a less effective agonist at the angiotensin AT1 receptor.

     Angiotensin II (3-8), human TFA Chemical Structure
  16. GC42810 Angiotensin II (5-8) (human, rat, mouse) Angiotensin II (5-8) (human, rat, mouse) is an endogenous C-terminal fragment of the peptide vasoconstrictor angiotensin II. Angiotensin II (5-8) (human, rat, mouse) Chemical Structure
  17. GC35354 Angiotensin II 5-valine

    Angiotensin II 5-valine is an agonist of angiotensin receptor.

     Angiotensin II 5-valine Chemical Structure
  18. GC60584 Angiotensin II human acetate

    Angiotensin II human (Angiotensin II) acetate is a vasoconstrictor and a major bioactive peptide of the renin/angiotensin system.

     Angiotensin II human acetate Chemical Structure
  19. GC62844 Angiotensin II human TFA

    Angiotensin II human (Angiotensin II) TFA is a vasoconstrictor and a major bioactive peptide of the renin/angiotensin system.

     Angiotensin II human TFA Chemical Structure
  20. GC35355 Angiotensin III Angiotensin III Chemical Structure
  21. GP10110 Angiotensin III (human, mouse) An agonist at AT1 and AT2 receptors Angiotensin III (human, mouse) Chemical Structure
  22. GC35356 Angiotensin III TFA Angiotensin III TFA Chemical Structure
  23. GC66025 Angiotensin III, human, mouse TFA Angiotensin III, human, mouse (TFA) is an angiotensin. Angiotensin III, human, mouse TFA Chemical Structure
  24. GC12065 AVE 0991 AVE 0991 is a Nonpeptide Mimic of the Effects of Angiotensin-(1-7) on the Endothelium. AVE 0991 Chemical Structure
  25. GC17686 AVE 0991 sodium salt Ang-(1-7) receptor Mas agonist AVE 0991 sodium salt Chemical Structure
  26. GC13277 Azilsartan Potent angiotensin II type 1 (AT1) receptor inverse agonist Azilsartan Chemical Structure
  27. GC35452 Azilsartan D5 Azilsartan D5 (TAK-536 D5) is the deuterium labeled Azilsartan(TAK-536), which is a specific and potent angiotensin II type 1 receptor antagonist. Azilsartan D5 Chemical Structure
  28. GC11407 Azilsartan Medoxomil

    Angiotensin II receptor type 1 antagonist

     Azilsartan Medoxomil Chemical Structure
  29. GC10642 Azilsartan medoxomil monopotassium

    Angiotensin II receptor type 1 antagonist

     Azilsartan medoxomil monopotassium Chemical Structure
  30. GC66468 Azilsartan mepixetil Azilsartan mepixetil is the antagonist of angiotensin II receptor. Azilsartan mepixetil has stronger and longer blood pressure effect, more abvious and longer lasting heart rate lowering effect and high safety. Azilsartan mepixetil achieves ideal protective effect for heart and kidney functions. Azilsartan mepixetil has the potential for the research of hypertension, chronic heart failure and diabetic nephropathy (extracted from patent CN107400122A). Azilsartan mepixetil Chemical Structure
  31. GC66440 Azilsartan mopivabil Azilsartan mopivabil is the potent antagonist of angiotensin II receptor. Azilsartan mopivabil Chemical Structure
  32. GC46913 Benazepril-d5 (hydrochloride) An internal standard for the quantification of benazapril Benazepril-d5 (hydrochloride) Chemical Structure
  33. GC19071 BIBS 39 BIBS 39 is a new nonpeptide angiotensin II (AII) receptor antagonist. BIBS 39 Chemical Structure
  34. GC60095 Brain Natriuretic Peptide (1-32), rat acetate Brain Natriuretic Peptide (1-32), rat acetate (BNP (1-32), rat acetate) is a 32 amino acid polypeptide secreted by the ventricles of the heart in response to excessive stretching of heart muscle cells (cardiomyocytes). Brain Natriuretic Peptide (1-32), rat acetate Chemical Structure
  35. GC32589 Brain Natriuretic Peptide (BNP) (1-32), rat Brain Natriuretic Peptide (BNP) (1-32), rat (BNP (1-32), rat) is a 32 amino acid polypeptide secreted by the ventricles of the heart in response to excessive stretching of heart muscle cells (cardiomyocytes). Brain Natriuretic Peptide (BNP) (1-32), rat Chemical Structure
  36. GC12034 C-type natriuretic peptide (1-22) (human, rat, swine) C-type natriuretic peptide (1-22) (human, rat, swine), a 1-22 fragment of CNP, is a natriuretic peptide receptor B (NPR-B) agonist. C-type natriuretic peptide (1-22) (human, rat, swine) Chemical Structure
  37. GC35756 C-Type Natriuretic Peptide (1-53), human C-Type Natriuretic Peptide (1-53), human is the 1-53 fragment of C-Type Natriuretic Peptide. C-Type Natriuretic Peptide (1-53), human Chemical Structure
  38. GC68908 C-Type Natriuretic Peptide (1-53), human TFA

    C-Type Natriuretic Peptide (1-53), human TFA is a fragment of C-type natriuretic peptide consisting of amino acids 1 to 53. C-Type Natriuretic Peptide TFA belongs to the family of natriuretic peptides and is involved in maintaining electrolyte-fluid balance and vascular tone.

     C-Type Natriuretic Peptide (1-53), human TFA Chemical Structure
  39. GC16978 Candesartan Angiotensin II receptor 1 (AT1) antagonist Candesartan Chemical Structure
  40. GC12318 Candesartan Cilexetil Prodrug of the angiotensin II receptor 1 (AT1) antagonist candesartan Candesartan Cilexetil Chemical Structure
  41. GC40238 Candesartan-d4 Candesartan-d4 is intended for use as an internal standard for the quantification of candesartan by GC- or LC-MS. Candesartan-d4 Chemical Structure
  42. GC15406 CGP 42112 angiotensin AT2 receptor ligand CGP 42112 Chemical Structure
  43. GC32561 CGP48369 CGP48369 is a nonpeptidic angiotensin II receptor antagonist, used for anti-hypertensive research. CGP48369 Chemical Structure
  44. GC60748 Dehydro Olmesartan Dehydro Olmesartan is a derivative of Olmesartan. Dehydro Olmesartan Chemical Structure
  45. GC43580 DX600 DX600 is a potent and selective peptide inhibitor of angiotensin-converting enzyme 2 (ACE2; Kis = 2.8, 200, and 1,200 nM for recombinant, human, and murine ACE2, respectively). DX600 Chemical Structure
  46. GC49566 DX600 (trifluoroacetate salt) A peptide inhibitor of ACE2 DX600 (trifluoroacetate salt) Chemical Structure
  47. GC32536 Elisartan (HN 65021) Elisartan (HN 65021) is an orally active non-peptide pro-drug of angiotensin II AT1 receptor antagonist HN-12206, and shows anti-hypertension activities. Elisartan (HN 65021) Chemical Structure
  48. GC19137 EMA401 EMA401 (EMA401) is a highly selective, orally active, peripherally restricted angiotensin II type 2 receptor (AT2R) antagonist. EMA401 Chemical Structure
  49. GC13436 EMD 66684 angiotensin AT1 receptor antagonist EMD 66684 Chemical Structure
  50. GC16297 Eprosartan Mesylate Angiotensin AT1 receptor antagonists Eprosartan Mesylate Chemical Structure
  51. GC36046 Fimasartan Fimasartan(BR-A-657) is a non-peptide angiotensin II receptor antagonist used for the treatment of hypertension and heart failure. Fimasartan Chemical Structure
  52. GC47371 Fosinopril-d7 (sodium salt) An internal standard for the quantification of fosinopril Fosinopril-d7 (sodium salt) Chemical Structure
  53. GC49228 Ganoderol B A triterpenoid with diverse biological activities Ganoderol B Chemical Structure
  54. GC31529 H-Val-Pro-Pro-OH H-Val-Pro-Pro-OH, a milk-derived proline peptides derivative, is an inhibitor of Angiotensin I converting enzyme (ACE), with an IC50 of 9 μM. H-Val-Pro-Pro-OH Chemical Structure
  55. GC34326 H-Val-Pro-Pro-OH TFA H-Val-Pro-Pro-OH (TFA), a milk-derived proline peptides derivative, is an inhibitor of Angiotensin I converting enzyme (ACE), with an IC50 of 9 μM. H-Val-Pro-Pro-OH TFA Chemical Structure
  56. GC10467 Irbesartan Angiotensin II inhibitor Irbesartan Chemical Structure
  57. GC40208 Irbesartan-d4 Irbesartan-d4 is intended for use as an internal standard for the quantification of irbesartan by GC- or LC-MS. Irbesartan-d4 Chemical Structure
  58. GC32569 L-159282 (MK 996) L-159282 (MK 996) is a highly potent, orally active, nonpeptide angiotensin II receptor antagonist, with anti-hypertensive activity. L-159282 (MK 996) Chemical Structure
  59. GC30443 L162389 L162389 is a potent antagonist of angiotensin AT1 receptor with Ki of 28 nM. L162389 Chemical Structure
  60. GC31567 L162441 L162441 is an Angiotensin type 1 receptor antagonist. L162441 Chemical Structure
  61. GC11784 LCZ696 LCZ696 (LCZ696), comprised Valsartan and Sacubitril (AHU377) in 1:1 molar ratio, is a first-in-class, orally bioavailable, and dual-acting angiotensin receptor-neprilysin (ARN) inhibitor for hypertension and heart failure. LCZ696 Chemical Structure
  62. GC45501 Lisinopril-d5   Lisinopril-d5 Chemical Structure
  63. GC10249 Losartan

    Angiotensin II receptor antagonist

     Losartan Chemical Structure
  64. GC12512 Losartan Carboxylic Acid AT1 antagonist Losartan Carboxylic Acid Chemical Structure
  65. GC36480 Losartan D4 An internal standard for the quantification of losartan Losartan D4 Chemical Structure
  66. GC36481 Losartan D4 Carboxylic Acid Losartan D4 Carboxylic Acid (E-3174 D4) is the deuterium labeled Losartan(EXP-3174), which is an angiotensin II receptor antagonist. Losartan D4 Carboxylic Acid Chemical Structure
  67. GC10257 Losartan Potassium (DuP 753) Losartan Potassium (DuP 753) (DuP-753 potassium) is an angiotensin II receptor type 1 (AT1) antagonist, competing with the binding of angiotensin II to AT1 with an IC50 of 20 nM. Losartan Potassium (DuP 753) Chemical Structure
  68. GC32632 LY285434 LY285434 is a suitable angiotensin II receptor antagonist. LY285434 Chemical Structure
  69. GC64604 Mopivabil Mopivabil is the antagonist of angiotensin II receptor. Mopivabil Chemical Structure
  70. GC10024 Novokinin Angiotensin AT2 receptor agonist Novokinin Chemical Structure
  71. GC16936 Olmesartan An AT1 receptor antagonist and active metabolite of olmesartan medoxomil Olmesartan Chemical Structure
  72. GC36802 Olmesartan D4 Olmesartan D4 (RNH-6270 D4) is the deuterium labeled Olmesartan. Olmesartan D4 Chemical Structure
  73. GC16752 Olmesartan medoxomil A prodrug form of olmesartan Olmesartan medoxomil Chemical Structure
  74. GC61153 Olmesartan medoxomil impurity C Olmesartan medoxomil impurity C is an Olmesartan medoxomil impurity. Olmesartan medoxomil impurity C Chemical Structure
  75. GC61154 Olmesartan methyl ester Olmesartan methyl ester is an intermediate in the synthesis of Olmesartan medoxomil. Olmesartan methyl ester Chemical Structure
  76. GC17384 PD 123319 ditrifluoroacetate A selective angiotensin II type 2 receptor antagonist PD 123319 ditrifluoroacetate Chemical Structure
  77. GC16394 PD123319

    PD123319 is a non-peptide inhibitor of angiotensin II receptor with IC50 value of 34nM .

     PD123319 Chemical Structure
  78. GC16871 Perindopril ACE inhibitor Perindopril Chemical Structure
  79. GC32530 Pratosartan (FW 7203) Pratosartan (FW 7203) is a selective angiotensin II receptor antagonist. Pratosartan (FW 7203) Chemical Structure
  80. GC48513 Quinapril-d5 An internal standard for the quantification of quinapril Quinapril-d5 Chemical Structure
  81. GC49653 Ramipril Diketopiperazine A potential impurity found in commercial preparations of ramipril Ramipril Diketopiperazine Chemical Structure
  82. GC49408 Ramipril Diketopiperazine Acid A potential impurity found in commercial preparations of ramipril Ramipril Diketopiperazine Acid Chemical Structure
  83. GC39821 Saralasin TFA Saralasin ([Sar1,Ala8] Angiotensin II) TFA is an octapeptide analog of angiotensin II. Saralasin TFA Chemical Structure
  84. GC32591 SL910102 SL910102 is a nonpeptide angiotensin AT1 receptor antagonist. SL910102 Chemical Structure
  85. GC32479 Sparsentan (RE-021) Sparsentan (RE-021) (RE-021) is a highly potent dual angiotensin II and endothelin A receptor antagonist with Kis of 0.8 and 9.3 nM, respectively. Sparsentan (RE-021) Chemical Structure
  86. GC32507 Tasosartan (WAY-ANA 756) Tasosartan (WAY-ANA 756) is a long-acting angiotensin II (AngII) receptor antagonist. Tasosartan (WAY-ANA 756) Chemical Structure
  87. GC38856 TD-0212 TFA TD-0212 TFA is an orally active dual pharmacology angiotensin II type 1 receptor (AT1) antagonist and neprilysin (NEP) inhibitor, with a pKi of 8.9 for AT1 and a pIC50 of 9.2 for NEP. TD-0212 TFA Chemical Structure
  88. GC15023 Telmisattan Telmisattan is a potent, long lasting antagonist of angiotensin II type 1 receptor (AT1), selectively inhibiting the binding of 125I-AngII to AT1 receptors with IC50 of 9.2 nM. Telmisattan Chemical Structure
  89. GC18202 Temocaprilat An ACE inhibitor Temocaprilat Chemical Structure
  90. GC46233 Trandolaprilat (hydrate) Trandolaprilat (hydrate) is a potent angiotensin-converting enzyme (ACE) inhibitor. Trandolaprilat (hydrate) Chemical Structure
  91. GC13389 Tranilast Angiogenesis inhibitor Tranilast Chemical Structure
  92. GC12443 Tranilast Sodium Antiallergic agent Tranilast Sodium Chemical Structure
  93. GC37819 trans-Tranilast trans-Tranilast (trans-MK-341) is an antiallergic drug, used to treat bronchial asthma, allergic rhinitis and atopic dermatitis. trans-Tranilast Chemical Structure
  94. GC70070 TRV-120027

    TRV120027 is a β-arrestin-1 agonist for angiotensin II type 1 receptor (AT1R). TRV120027 induces acute catecholamine secretion through coupling with the cation channel subfamily C3 (TRPC3), promoting the formation of a large molecular complex consisting of AT1R-β-arrestin-1-TRPC3-PLCγ on the plasma membrane. TRV120027 inhibits angiotensin II-mediated vasoconstriction and increases myocardial contractility. It has potential for use in research on acute decompensated heart failure (ADHF).

     TRV-120027 Chemical Structure
  95. GC70068 TRV055

    TRV055 is a G protein-biased agonist that selectively targets the type 1 angiotensin II receptor (AT1R) through Gq signaling. It effectively stimulates intracellular signal transduction mediated by Gq.

     TRV055 Chemical Structure
  96. GC67768 TRV055 hydrochloride TRV055 hydrochloride Chemical Structure
  97. GC70069 TRV056

    TRV056 is a ligand for the Gq-biased type 1 angiotensin II receptor (AT1R). TRV056 effectively stimulates cell signaling mediated by Gq. TRV056 can be used to develop Gq-biased AT1R agonists.

     TRV056 Chemical Structure
  98. GC10765 Valsartan

    Angiotensin II AT1 receptor antagonist

     Valsartan Chemical Structure
  99. GC37884 Valsartan D9 Valsartan D9 (CGP 48933-d9) is deuterium labeled valsartan. Valsartan D9 Chemical Structure
  100. GC37954 YS-49 YS-49 is a PI3K/Akt (a downstream target of RhoA) activator, to reduce RhoA/PTEN activation in the 3-methylcholanthrene-treated cells. YS-49 Chemical Structure
  101. GC37955 YS-49 monohydrate YS-49 (monohydrate) is a PI3K/Akt (a downstream target of RhoA) activator, to reduce RhoA/PTEN activation in the 3-methylcholanthrene-treated cells. YS-49 monohydrate Chemical Structure

Items 1 to 100 of 102 total

per page
  1. 1
  2. 2

Set Descending Direction