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OX Receptor

OX receptor (orexin receptor) is a G-protein coupled receptor that is involved in the regulation of feeding behaviour.

Products for  OX Receptor

  1. Cat.No. Product Name Information
  2. GC16336 ACT 335827 Orexin receptor 1 antagonist,potent and selective ACT 335827  Chemical Structure
  3. GC50142 ACT 462206 Potent, dual orexin receptor antagonist ACT 462206  Chemical Structure
  4. GC10717 Almorexant OX1R/OX2R antagonist Almorexant  Chemical Structure
  5. GC10050 Almorexant hydrochloride OX1R/OX2R antagonist Almorexant hydrochloride  Chemical Structure
  6. GC65550 Danavorexton Danavorexton is an orexin receptor agonist. Danavorexton  Chemical Structure
  7. GC13741 EMPA OX2 receptor antagonist EMPA  Chemical Structure
  8. GC30832 GSK1059865 GSK1059865 is a potent orexin 1 receptor antagonist. GSK1059865  Chemical Structure
  9. GC30829 IPSU An orexin receptor 2 antagonist IPSU  Chemical Structure
  10. GC14809 JNJ 10397049 OX2 receptor antagonist JNJ 10397049  Chemical Structure
  11. GC63415 JNJ-54717793 JNJ-54717793, as a brain penetrant, is an orally active, selective and high affinity orexin-1 receptor (OX1R) antagonist (plasma EC50=85 ng/mL). JNJ-54717793  Chemical Structure
  12. GC19220 Lemborexant

    Lemborexant (E2006) is an oral active diorexin receptor antagonist (DORA) and has been approved by the US Food and Drug Administration for the treatment of insomnia.

    Lemborexant  Chemical Structure
  13. GC12242 MK 6096 MK 6096 (MK-6096) is an orally bioavailable potent and selective reversible antagonist of OX1 and OX2 receptor(<3 nM in binding). MK 6096  Chemical Structure
  14. GC19249 MK-1064 MK-1064 is a selective orexin 2 receptor antagonist (2-SORA) for the research of insomnia. MK-1064  Chemical Structure
  15. GC19250 MK-3697 MK-3697 is an isonicotinamide small molecule, acting as a potent and selective Orexin 2 receptor antagonist with Ki = 0.95 nM. MK-3697  Chemical Structure
  16. GC30941 Nemorexant (ACT-541468) Nemorexant (ACT-541468)  Chemical Structure
  17. GC19272 Orexin 2 Receptor Agonist Orexin 2 Receptor Agonist is a potent (EC50 on OX2R is 23 nM) and OX2R-selective (OX1R/OX2R EC50 ratio is 70) agonist. Orexin 2 Receptor Agonist  Chemical Structure
  18. GC67929 Orexin 2 Receptor Agonist 2

    Orexin 2 Receptor Agonist 2 is a selective orexin 2 receptor agonist.

    Orexin 2 Receptor Agonist 2  Chemical Structure
  19. GC67957 Orexin A (human, rat, mouse) (acetate) Orexin A (human, rat, mouse) (acetate)  Chemical Structure
  20. GC38352 Orexin A (human, rat, mouse) (TFA) Orexin A human, rat, mouse TFA, a 33 amino acid excitatory neuropeptide, orchestrates diverse central and peripheral processes. Orexin A (human, rat, mouse) (TFA)  Chemical Structure
  21. GC14887 Orexin B (human) Endogenous agonist at orexin receptors Orexin B (human)  Chemical Structure
  22. GC16745 Orexin B (mouse) Orexin B (mouse) (Rat orexin B) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively. Orexin B (mouse)  Chemical Structure
  23. GC36812 Orexin B, human TFA Orexin B, human (TFA) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively. Orexin B, human TFA  Chemical Structure
  24. GC64021 Orexin B, rat, mouse TFA Orexin B, rat, mouse (Rat orexin B) TFA is an endogenous orexin receptor agonist. Orexin B, rat, mouse TFA  Chemical Structure
  25. GC61770 Orexin receptor antagonist 2 Orexin receptor antagonist 2 (compound 30) is a potent orexin receptor antagonist with pKis of 7.69 and 9.78. Orexin receptor antagonist 2  Chemical Structure
  26. GC65382 Orexin receptor antagonist 5 Orexin receptor antagonist 5  Chemical Structure
  27. GC11818 OXA (17-33) orexin OX1 receptor agonist OXA (17-33)  Chemical Structure
  28. GC13539 SB-334867 Orexin-1 receptor antagonist SB-334867  Chemical Structure
  29. GC15034 SB-334867 free base orexin-1 receptor antagonist, selective SB-334867 free base  Chemical Structure
  30. GC16540 SB-408124 Hydrochloride A potent orexin 1 receptor antagonist SB-408124 Hydrochloride  Chemical Structure
  31. GC19323 SB-649868 SB-649868 is a potent and selective orally active orexin (OX) 1 and OX2 receptor antagonist (pKi =9.4 and 9.5 at the OX1 and OX2 receptor, respectively). SB-649868  Chemical Structure
  32. GC15534 SB-674042 A potent and selective orexin 1 receptor antagonist SB-674042  Chemical Structure
  33. GC15317 SB408124 OX(1)receptor antagonist SB408124  Chemical Structure
  34. GC37623 Seltorexant Seltorexant (JNJ-42847922) is an orally active, high-affinity, and selective orexin-2 receptor (OX2R) antagonist (pKi values of 8.0 and 8.1 for human and rat OX2R). Seltorexant  Chemical Structure
  35. GC17807 TCS 1102 Antagonist for OX2 and OX1 receptors TCS 1102  Chemical Structure
  36. GC10549 TCS OX2 29

    OX2 receptor antagonist

    TCS OX2 29  Chemical Structure
  37. GC64826 Vornorexant Vornorexant (ORN-0829; TS-142) is a potent dual OX1R and OX2R antagonist with IC50 values of 1.05 nM and 1.27 nM, respectively. Vornorexant  Chemical Structure
  38. GC50559 YNT 185 YNT 185 is a nonpeptide, selective orexin type-2 receptor (OX2R) agonist, with EC50s of 0.028 and 2.75 μM for OX2R and OX1R, respectively. YNT 185  Chemical Structure
  39. GC17992 [Ala11,D-Leu15]-Orexin B [Ala11,D-Leu15]-Orexin B is a potent and selective orexin-2 receptor (OX2) agonist. [Ala11,D-Leu15]-Orexin B  Chemical Structure

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