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Home >> Signaling Pathways >> GPCR/G protein >> Vasopressin Receptor

Vasopressin Receptor

Vasopressin receptors are G-protein coupled receptors that mediate coagulation factor release, platelet aggregation, vasoconstriction, release of antidiuresis and ACTH release etc.

Products for  Vasopressin Receptor

  1. Cat.No. Product Name Information
  2. GC72235 (Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin acetate (Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin is a potent vasopressin V1 receptor (VP V1R) antagonist. (Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin acetate Chemical Structure
  3. GC66678 2-(3-Trifluoromethylphenyl)glycine hydrochloride 2-(3-Trifluoromethylphenyl)glycine hydrochloride is a precursor of substituted 2-acetamido-5-aryl-l, 2,4-triazolones. Substituted 2-acetamido-5-aryl-l, 2,4-triazolones are dual V1a/V2 receptor antagonists and can be used in cardiovascular disease research. 2-(3-Trifluoromethylphenyl)glycine hydrochloride Chemical Structure
  4. GC30764 Argipressin (Vasopressin) Arginine-vasopressin, as an important hormone in the regulation of plasma osmolality and blood volume/pressure, always is used in the treatment of septic shock and decompensated cirrhosis. Argipressin (Vasopressin) Chemical Structure
  5. GC12194 Atosiban

    RW22164; RWJ22164

    mixed antagonist of oxytocin and vasopressin receptors

     Atosiban Chemical Structure
  6. GC39849 Atosiban acetate Atosiban acetate (RW22164 acetate;RWJ22164 acetate) is a nonapeptide competitive vasopressin/oxytocin receptor antagonist, and is a desamino-oxytocin analogue. Atosiban acetate Chemical Structure
  7. GC31295 Balovaptan (RG7314)

    RG7314

     Balovaptan (RG7314) (RG7314) is an orally available, selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors, and is used for the research of autism. Balovaptan (RG7314) Chemical Structure
  8. GA20807 Big Endothelin-1 (1-38), human Big Endothelin-1 (1-38), human is the precursor of endothelin-1. Big Endothelin-1 (1-38), human Chemical Structure
  9. GA20808 Big Endothelin-1 (1-39), porcine Big Endothelin-1 (1-39), porcine is the precursor of endothelin-1. Big Endothelin-1 (1-39), porcine Chemical Structure
  10. GC12627 Conivaptan HCl

    YM-087

     Conivaptan (hydrochloride) is a non-peptide antagonist of vasopressin receptor, with Ki values of 0.48 and 3.04 nM for rat liver V1A receptor and rat kidney V2 receptor respectively. Conivaptan HCl Chemical Structure
  11. GC12303 Desmopressin A vasopressin receptor agonist Desmopressin Chemical Structure
  12. GC11265 Desmopressin Acetate Desmopressin Acetate (DDAVP), a synthetic peptide analog of vasopressin, is a safe antidiuretic and hemostatic compound that acts as a selective agonist at the vasopressin V2 membrane receptor (V2R). Desmopressin Acetate Chemical Structure
  13. GC16591 d[Cha4]-AVP human vasopressin V1B receptor agonist d[Cha4]-AVP Chemical Structure
  14. GC15154 d[Leu4,Lys8]-VP Selective vasopressin V1B receptor agonist d[Leu4,Lys8]-VP Chemical Structure
  15. GC61959 D[LEU4,LYS8]-VP TFA D[LEU4,LYS8]-VP TFA is a selective agonist of vasopressin V1b receptor, with the Kis of 0.16 nM, 0.52 nM, and 0.1.38 nM for rat, human and mouse V1b receptor, respectively. D[LEU4,LYS8]-VP TFA Chemical Structure
  16. GC72087 F992 TFA F992 TFA is an antidiuretic peptide and vasopressin (antidiuretic hormone) analogue. F992 TFA Chemical Structure
  17. GC65415 Felypressin acetate Felypressin acetate (PLV-2 acetate) is a non-catecholamine vasoconstrictor and a vasopressin 1 agonist. Felypressin acetate Chemical Structure
  18. GC11991 L-371,257 human oxytocin (OT) receptor antagonist L-371,257 Chemical Structure
  19. GC32453 Lixivaptan (VPA-985)

    VPA-985, WAY-VPA-985

     Lixivaptan (VPA-985) (VPA-985, WAY-VPA 985) is an orally active and selective vasopressin receptor V2 antagonist, with IC50 values of 1.2 and 2.3 nM for human and rat V2, respectively. Lixivaptan (VPA-985) Chemical Structure
  20. GC14880 Mozavaptan novel competitive vasopressin receptor antagonist Mozavaptan Chemical Structure
  21. GC44247 Mozavaptan (hydrochloride)

    OPC 31260

     Mozavaptan is a benzazepine derivative that antagonizes the binding of arginine vasopressin (AVP) to vasopressin receptors located in the liver (V1; IC50 = 1.2 μM) and kidney (V2; IC50 = 14 nM). Mozavaptan (hydrochloride) Chemical Structure
  22. GC10622 OPC 21268 OPC 21268 (OPC-21268) is an orally effective, nonpeptide, vasopressin V1 receptor antagonist with an IC50 of 0.4 μM. OPC 21268 Chemical Structure
  23. GC30890 RG7713 (RO5028442)

    RO5028442

     RG7713 (RO5028442) (RO5028442) is a highly potent and selective Brain-Penetrant Vasopressin 1a (V1a) receptor antagonist with Kis of 1 nM (hV1a) and 39 nM (mV1a). RG7713 (RO5028442) Chemical Structure
  24. GC69875 Selepressin acetate

    FE 202158 acetate

    Selepressin (FE 202158) acetate is a selective vasopressin V1A receptor agonist. Selepressin acetate is an effective vasoconstrictor and can be used in the research of septic shock.

     Selepressin acetate Chemical Structure
  25. GC72171 SKF 100398 SKF 100398 (d(CH2)5Tyr(Et)VAVP), an arginine vasopressin (AVP) analogue, is a specific antagonist of the antidiuretic effect of exogenous and endogenous AVP. SKF 100398 Chemical Structure
  26. GC12462 SR 49059

    Relcovaptan

     vasopressin V1A receptor antagonist SR 49059 Chemical Structure
  27. GC38948 SRX246 SRX246 is a potent, CNS-penetrant, highly selective, orally bioavailable vasopressin 1a (V1a) receptor antagonist (Ki=0.3 nM for human V1a). SRX246 Chemical Structure
  28. GC50376 SSR 149415 Potent and selective vasopressin V1B antagonist SSR 149415 Chemical Structure
  29. GC50246 TASP 0390325 Potent and selective V1B receptor antagonist; orally bioavailable TASP 0390325 Chemical Structure
  30. GC32463 Terlipressin Terlipressin is a vasopressin analogue with potent vasoactive properties. Terlipressin Chemical Structure
  31. GC39830 Terlipressin acetate

    Glycylpressin, Remestyp

     A prodrug form of lysipressin Terlipressin acetate Chemical Structure
  32. GC70580 Terlipressin diacetate Terlipressin diacetate is a vasopressin analogue with potent vasoactive properties. Terlipressin diacetate Chemical Structure
  33. GC15575 Tolvaptan

    OPC 41061

     AVP V2-receptor antagonist Tolvaptan Chemical Structure
  34. GC74398 Vasopressin Dimer (parallel) (TFA) Vasopressin Dimer (parallel) TFA is a parallel dimer of Vasopressin. Vasopressin Dimer (parallel) (TFA) Chemical Structure
  35. GC31475 WAY-151932 (VNA-932)

    VNA-932; WAY-VNA 932

     WAY-151932 (VNA-932) is a vasopressin V2-receptor agonist with IC50 of 80.3 nM and 778 nM in human-V2 binding and V1a binding assay. WAY-151932 (VNA-932) Chemical Structure

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