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Home >> Signaling Pathways >> GPCR/G protein >> Vasopressin Receptor

Vasopressin Receptor

Vasopressin receptors are G-protein coupled receptors that mediate coagulation factor release, platelet aggregation, vasoconstriction, release of antidiuresis and ACTH release etc.

Products for  Vasopressin Receptor

  1. Cat.No. Product Name Information
  2. GA20084 (Deamino-Cys¹,β-cyclohexyl-Ala⁴,Arg⁸)-Vasopressin Studies revealed that this specific vasopressin agonist exhibited a nanomolar affinity for V-1b receptors from various mammalian species (bovine, human, rat). It exhibited high V-1b/V-1a and V-1b/oxytocin selectivity for rat, human, and bovine receptors. Furthermore, it showed a high V-1b/V-2 specificity for both bovine and human vasopressin receptors. Therefore, d(Cha?)-AVP is a promising tool for research of V-1b receptor structure-function relationships. (Deamino-Cys¹,β-cyclohexyl-Ala⁴,Arg⁸)-Vasopressin Chemical Structure
  3. GC66678 2-(3-Trifluoromethylphenyl)glycine hydrochloride 2-(3-Trifluoromethylphenyl)glycine hydrochloride is a precursor of substituted 2-acetamido-5-aryl-l, 2,4-triazolones. Substituted 2-acetamido-5-aryl-l, 2,4-triazolones are dual V1a/V2 receptor antagonists and can be used in cardiovascular disease research. 2-(3-Trifluoromethylphenyl)glycine hydrochloride Chemical Structure
  4. GC30764 Argipressin (Vasopressin) Argipressin (Vasopressin) (Arg8-vasopressin) binds to the V1, V2, V3-vascular arginine vasopressin receptor, with a Kd value of 1.31 nM in A7r5 rat aortic smooth muscle cells for V1. Argipressin (Vasopressin) Chemical Structure
  5. GC12194 Atosiban

    mixed antagonist of oxytocin and vasopressin receptors

     Atosiban Chemical Structure
  6. GC39849 Atosiban acetate Atosiban acetate (RW22164 acetate;RWJ22164 acetate) is a nonapeptide competitive vasopressin/oxytocin receptor antagonist, and is a desamino-oxytocin analogue. Atosiban acetate Chemical Structure
  7. GC31295 Balovaptan (RG7314) Balovaptan (RG7314) (RG7314) is an orally available, selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors, and is used for the research of autism. Balovaptan (RG7314) Chemical Structure
  8. GA20807 Big Endothelin-1 (1-38), human Big Endothelin-1 (1-38), human is the precursor of endothelin-1. Big Endothelin-1 (1-38), human Chemical Structure
  9. GA20808 Big Endothelin-1 (1-39), porcine Big Endothelin-1 (1-39), porcine is the precursor of endothelin-1. Big Endothelin-1 (1-39), porcine Chemical Structure
  10. GC12627 Conivaptan HCl Conivaptan (hydrochloride) is a non-peptide antagonist of vasopressin receptor, with Ki values of 0.48 and 3.04 nM for rat liver V1A receptor and rat kidney V2 receptor respectively. Conivaptan HCl Chemical Structure
  11. GC12303 Desmopressin A vasopressin receptor agonist Desmopressin Chemical Structure
  12. GC11265 Desmopressin Acetate Desmopressin Acetate Chemical Structure
  13. GC16591 d[Cha4]-AVP human vasopressin V1B receptor agonist d[Cha4]-AVP Chemical Structure
  14. GC15154 d[Leu4,Lys8]-VP Selective vasopressin V1B receptor agonist d[Leu4,Lys8]-VP Chemical Structure
  15. GC61959 D[LEU4,LYS8]-VP TFA D[LEU4,LYS8]-VP TFA is a selective agonist of vasopressin V1b receptor, with the Kis of 0.16 nM, 0.52 nM, and 0.1.38 nM for rat, human and mouse V1b receptor, respectively. D[LEU4,LYS8]-VP TFA Chemical Structure
  16. GC65415 Felypressin acetate Felypressin acetate (PLV-2 acetate) is a non-catecholamine vasoconstrictor and a vasopressin 1 agonist. Felypressin acetate Chemical Structure
  17. GC11991 L-371,257 human oxytocin (OT) receptor antagonist L-371,257 Chemical Structure
  18. GC32453 Lixivaptan (VPA-985) Lixivaptan (VPA-985) (VPA-985, WAY-VPA 985) is an orally active and selective vasopressin receptor V2 antagonist, with IC50 values of 1.2 and 2.3 nM for human and rat V2, respectively. Lixivaptan (VPA-985) Chemical Structure
  19. GC14880 Mozavaptan novel competitive vasopressin receptor antagonist Mozavaptan Chemical Structure
  20. GC44247 Mozavaptan (hydrochloride) Mozavaptan is a benzazepine derivative that antagonizes the binding of arginine vasopressin (AVP) to vasopressin receptors located in the liver (V1; IC50 = 1.2 μM) and kidney (V2; IC50 = 14 nM). Mozavaptan (hydrochloride) Chemical Structure
  21. GC10622 OPC 21268 OPC 21268 (OPC-21268) is an orally effective, nonpeptide, vasopressin V1 receptor antagonist with an IC50 of 0.4 μM. OPC 21268 Chemical Structure
  22. GC30890 RG7713 (RO5028442) RG7713 (RO5028442) (RO5028442) is a highly potent and selective Brain-Penetrant Vasopressin 1a (V1a) receptor antagonist with Kis of 1 nM (hV1a) and 39 nM (mV1a). RG7713 (RO5028442) Chemical Structure
  23. GC69875 Selepressin acetate

    Selepressin (FE 202158) acetate is a selective vasopressin V1A receptor agonist. Selepressin acetate is an effective vasoconstrictor and can be used in the research of septic shock.

     Selepressin acetate Chemical Structure
  24. GC12462 SR 49059 vasopressin V1A receptor antagonist SR 49059 Chemical Structure
  25. GC38948 SRX246 SRX246 is a potent, CNS-penetrant, highly selective, orally bioavailable vasopressin 1a (V1a) receptor antagonist (Ki=0.3 nM for human V1a). SRX246 Chemical Structure
  26. GC50376 SSR 149415 Potent and selective vasopressin V1B antagonist SSR 149415 Chemical Structure
  27. GC50246 TASP 0390325 Potent and selective V1B receptor antagonist; orally bioavailable TASP 0390325 Chemical Structure
  28. GC32463 Terlipressin Terlipressin is a vasopressin analogue with potent vasoactive properties. Terlipressin Chemical Structure
  29. GC39830 Terlipressin acetate A prodrug form of lysipressin Terlipressin acetate Chemical Structure
  30. GC15575 Tolvaptan AVP V2-receptor antagonist Tolvaptan Chemical Structure
  31. GC31475 WAY-151932 (VNA-932) WAY-151932 (VNA-932) is a vasopressin V2-receptor agonist with IC50 of 80.3 nM and 778 nM in human-V2 binding and V1a binding assay. WAY-151932 (VNA-932) Chemical Structure

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