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Membrane Transporter/Ion Channel

Products for  Membrane Transporter/Ion Channel

  1. Cat.No. Product Name Information
  2. GC13733 A 438079 hydrochloride An antagonist of the nucleotide receptor P2X7 A 438079 hydrochloride  Chemical Structure
  3. GC17091 A 784168 TRPV1 antagonist,potent and selective A 784168  Chemical Structure
  4. GC17870 A 804598 P2X7 antagonist,potent and selective A 804598  Chemical Structure
  5. GC15434 A 839977 P2X7 antagonist,potent and selective A 839977  Chemical Structure
  6. GC50088 A 85380 dihydrochloride High affinity and selective α4β2 nAChR agonist A 85380 dihydrochloride  Chemical Structure
  7. GC14481 A 887826 voltage-dependent Nav1.8 sodium channel blocker A 887826  Chemical Structure
  8. GC11701 A 967079 Selective TRPA1 channel blocker A 967079  Chemical Structure
  9. GC30837 A-1165442 A-1165442 is a potent, competitive and orally available TRPV1 antagonist with an IC50 of 9 nM for human TRPV1. A-1165442  Chemical Structure
  10. GC17710 A-317491 A P2X3 and P2X2/3 receptor antagonist A-317491  Chemical Structure
  11. GC35211 A-317491 sodium salt hydrate A-317491 sodium salt hydrate is a potent, selective and non-nucleotide antagonist of P2X3 and P2X2/3 receptors, with Kis of 22, 22, 9, and 92 nM for hP2X3, rP2X3, hP2X2/3, and rP2X2/3, respectively. A-317491 sodium salt hydrate  Chemical Structure
  12. GC11178 A-7 hydrochloride calmodulin antagonist A-7 hydrochloride  Chemical Structure
  13. GC11842 A-740003 A selective P2X7 antagonist A-740003  Chemical Structure
  14. GC15701 A-803467 NaV1.8 channel blocker,potent and selective A-803467  Chemical Structure
  15. GC15014 A-867744 A positive allosteric modulator of α7 nAChRs A-867744  Chemical Structure
  16. GC11200 A23187

    A23187, free acid is a Ca2+ ionophore

    A23187  Chemical Structure
  17. GC39335 A2764 dihydrochloride A2764 dihydrochloride is a highly selective inhibitor of TRESK (TWIK-related spinal cord K+ channel, K2P18.1), which has moderate inhibitory effects on TREK-1 and TALK-1. A2764 dihydrochloride  Chemical Structure
  18. GC60545 A2793 A2793 is an efficient dual TWIK-related acid-sensitive K+ channel (TASK)-1/TRESK inhibitor, with an IC50 of 6.8 μM for mTRESK. A2793  Chemical Structure
  19. GC10641 AA 29504 GABAA receptor modulator AA 29504  Chemical Structure
  20. GC50167 AAQ chloride Photoswitchable Kv channel blocker AAQ chloride  Chemical Structure
  21. GC62823 Abeprazan Abeprazan (DWP14012) is a potassium-competitive acid blocker. Abeprazan  Chemical Structure
  22. GC65377 Abeprazan hydrochloride Abeprazan hydrochloride (DWP14012 hydrochloride) is a potassium-competitive acid blocker. Abeprazan hydrochloride  Chemical Structure
  23. GC35222 ABT-239 ABT-239 is a novel, highly efficacious, non-imidazole?class of H3R antagonist and a transient receptor potential vanilloid type 1 (TRPV1) antagonist. ABT-239  Chemical Structure
  24. GC60549 ABT-418 hydrochloride ABT-418 hydrochloride is a potent and selective agonist of nAChRs with cognitive enhancing and anxiolytic activities. ABT-418 hydrochloride  Chemical Structure
  25. GC19016 ABT-639 ABT-639 is a novel, peripherally acting, selective T-type Ca2+ channel blocker. ABT-639  Chemical Structure
  26. GC33720 ABT-639 hydrochloride ABT-639 hydrochloride is a novel, peripherally acting, selective T-type Ca2+ channel blocker. ABT-639 hydrochloride  Chemical Structure
  27. GC40860 AC1903 AC1903 is an inhibitor of transient receptor potential canonical channel 5 (TRPC5; IC50 = 14.7 μM). AC1903  Chemical Structure
  28. GN10812 Acacetin Acacetin  Chemical Structure
  29. GC11286 ACBC ACBC is a NMDA receptor partial agonist acting at the glycine site, NR1. ACBC  Chemical Structure
  30. GC14712 ACET ACET (ACET) is a highly potent and selective kainate receptor GluK1 (GluR5) antagonist, with a Kb value of 1.4 nM. ACET  Chemical Structure
  31. GC18262 Acetamiprid A neonicotinoid insecticide Acetamiprid  Chemical Structure
  32. GC14142 Acetylcholine Chloride Major transmitter at many nervous sites Acetylcholine Chloride  Chemical Structure
  33. GC18474 Acetyldigitoxin Acetyldigitoxin is cardiac glycoside and an inhibitor of the Na+/K+ ATPase with an IC50 value of 5 nM in isolated rat pinealocytes. Acetyldigitoxin  Chemical Structure
  34. GC30927 Acevaltrate Acevaltrate inhibits the Na+/K+-ATPase activity in the rat kidney and brain hemispheres with IC50s of 22.8 μM and 42.3 μM, respectively. Acevaltrate  Chemical Structure
  35. GC31100 ACT-709478 ACT-709478 is a potent, selective, orally active, and brain penetrating T-type calcium channel blocker. ACT-709478  Chemical Structure
  36. GC19729 Adenosine 5′-diphosphoribose sodium Adenosine 5′-diphosphoribose sodium (ADP ribose sodium) is a nicotinamide adenine nucleotide (NAD+) metabolite. Adenosine 5′-diphosphoribose sodium  Chemical Structure
  37. GC49231 Adenylosuccinic Acid (ammonium salt) A purine nucleotide and an intermediate in the purine nucleotide cycle Adenylosuccinic Acid (ammonium salt)  Chemical Structure
  38. GC13542 Adiphenine HCl Adiphenine HCl is a non-competitive inhibitor of nicotinic acetylcholine receptor (nAChR), with an IC50s of 1.9, 1.8, 3.7, and 6.3 μM for α1, α3β4, α4β2, and α4β4, respectively. Adiphenine HCl  Chemical Structure
  39. GC19021 Adjudin Adjudin is an extensively studied male contraceptive with a superior mitochondria-inhibitory effect. Adjudin  Chemical Structure
  40. GC11315 ADWX 1 Kv1.3 channel blocker,potent and selective ADWX 1  Chemical Structure
  41. GC32672 AE0047 Hydrochloride AE0047 Hydrochloride is a calcium blocker, used in the research of hypertensive disease. AE0047 Hydrochloride  Chemical Structure
  42. GC19022 AF-353 AF-353 is a novel, potent and orally bioavailable P2X3/P2X2/3 receptor antagonist, inhibits human and rat P2X3 (pIC50= 8.0). AF-353  Chemical Structure
  43. GC30844 Afloqualone An Analytical Reference Standard Afloqualone  Chemical Structure
  44. GC39248 Afoxolaner An isoxazoline insecticide and acaricide Afoxolaner  Chemical Structure
  45. GC14867 Agitoxin 2 Shaker K+ channel blocker, potent Agitoxin 2  Chemical Structure
  46. GC35273 Ajmaline Ajmaline  Chemical Structure
  47. GC45378 Alaproclate (hydrochloride)   Alaproclate (hydrochloride)  Chemical Structure
  48. GC30371 Alisol F Alisol F is a triterpene isolated from Alisma orientalis, has immunosuppressive and anti-virus functions. Alisol F  Chemical Structure
  49. GC40476 Allethrin Allethrin is a pyrethroid insecticide and modulator of voltage-gated sodium channels (NaV). Allethrin  Chemical Structure
  50. GC35293 Allocryptopine Allocryptopine, a derivative of tetrahydropalmatine, is extracted from Corydalis decumbens (Thunb. Allocryptopine  Chemical Structure
  51. GC46831 Alloisolithocholic Acid Alloisolithocholic Acid (3β-Hydroxy-5α-cholanic acid), a derivative of Lithocholic acid, is a T cell regulator. Alloisolithocholic Acid  Chemical Structure
  52. GC14192 Allopregnanolone

    Allopregnanolone, a 3alpha, 5alpha progesterone metabolite, acts as a potent allosteric modulator of the γ-aminobutyric acid type A (GABAA) receptor, exerts antidepressant and neuroprotective action.

    Allopregnanolone  Chemical Structure
  53. GC30891 Almitrine mesylate (Almitrine bismesylate) Almitrine mesylate (Almitrine bismesylate), a peripheral chemoreceptor agonist, inhibits selectively the Ca2+-dependent K+ channel. Almitrine mesylate (Almitrine bismesylate)  Chemical Structure
  54. GC32673 Almokalant (H 234/09) Almokalant (H 234/09) is a class III antiarrhythmic drug, acts as a potassium channel blocker, and inhibits a specific component (Ikr) of the time-dependent delayed rectifier K+ current. Almokalant (H 234/09)  Chemical Structure
  55. GC30983 alpha-Asarone (α-Asarone) alpha-Asarone (α-Asarone) (α-Asarone) is one of the main psychoactive compounds, and possesses an antidepressant-like activity in mice. alpha-Asarone (α-Asarone)  Chemical Structure
  56. GC13515 Alphaxalone activates and potentiates GABAA receptor-activated membrane current (IGABA) Alphaxalone  Chemical Structure
  57. GC15467 ALX 5407 hydrochloride GlyT1 inhibitor,selective non-transportable ALX 5407 hydrochloride  Chemical Structure
  58. GC12972 AM 1172 Inhibitor of anandamide uptake and FAAH,potent and selective AM 1172  Chemical Structure
  59. GC50475 AM 12 TRPC5 inhibitor AM 12  Chemical Structure
  60. GC12071 AM 404 Anandamide transport inhibitor AM 404  Chemical Structure
  61. GC10943 AM 92016 hydrochloride Potassium channel blocker AM 92016 hydrochloride  Chemical Structure
  62. GC19025 AM-0902 AM-0902 is a potent, selective transient receptor potential A1 (TRPA1) antagonist with IC50s of 71 and 131 nM for rTRPA1 and hTRPA1, respectively. AM-0902  Chemical Structure
  63. GC30917 AM-2099 AM-2099 is a potent and selective inhibitor of voltage-gated sodium channel Nav1.7 with an IC50 of 0.16 μM for human Nav1.7. AM-2099  Chemical Structure
  64. GC15458 Ambroxol HCl Ambroxol HCl (NA-872 hydrochloride), an active metabolite of the prodrug Bromhexine, has potent expectorant effects. Ambroxol HCl  Chemical Structure
  65. GC50058 AMG 21629 Potent and selective TRPV1 antagonist AMG 21629  Chemical Structure
  66. GC65611 AMG 333 AMG 333 is a potent and highly selective TRPM8 antagonist with an IC50 of 13 nM. AMG 333  Chemical Structure
  67. GC11926 AMG 9810 TRPV1 antagonist AMG 9810  Chemical Structure
  68. GC13003 AMG-517 TRPV1 antagonist,potent and highly selective AMG-517  Chemical Structure
  69. GC35316 AMG2850 AMG2850 is a potent, orally bioavailable and selective transient receptor potential melastatin 8 (TRPM8) antagonist. AMG2850  Chemical Structure
  70. GC31431 Amiloride (MK-870) Amiloride (MK-870) (MK-870) is an inhibitor of both epithelial sodium channel (ENaC[1]) and urokinase-type plasminogen activator receptor (uTPA[2]). Amiloride (MK-870)  Chemical Structure
  71. GC17853 Amiloride HCl Amiloride HCl (MK-870 hydrochloride) is an inhibitor of both epithelial sodium channel (ENaC[1]) and urokinase-type plasminogen activator receptor (uTPA[2]). Amiloride HCl  Chemical Structure
  72. GC12051 Amiloride HCl dihydrate Amiloride HCl dihydrate (MK-870 hydrochloride dihydrate) is an inhibitor of both epithelial sodium channel (ENaC[1]) and urokinase-type plasminogen activator receptor (uTPA[2]). Amiloride HCl dihydrate  Chemical Structure
  73. GC34064 Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) Aminooxyacetic acid (Carboxymethoxylamine) hemihydrochloride is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA degradating enzyme GABA-T. Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride)  Chemical Structure
  74. GC35322 Amiodarone Amiodarone is an antiarrhythmic drug for inhibition of ATP-sensitive potassium channel with an IC50 of 19.1 μM. Amiodarone  Chemical Structure
  75. GC11432 Amiodarone HCl Amiodarone HCl, a benzofuran-based Class III antiarrhythmic agent, inhibits WT outwardIhERG tails with an IC50 of ~45 nM. Amiodarone HCl  Chemical Structure
  76. GC18274 Amiprofos-methyl Amiprofos-methyl (APM) is a phosphoric amide herbicide. Amiprofos-methyl  Chemical Structure
  77. GC13723 Amitriptyline HCl Amitriptyline HCl is an inhibitor of serotonin reuptake transporter (SERT) and noradrenaline reuptake transporter (NET), with Kis of 3.45 nM and 13.3 nM for human SERT and NET, respectively. Amitriptyline HCl  Chemical Structure
  78. GC13523 Amlodipine Calcium channel blocker Amlodipine  Chemical Structure
  79. GC13146 Amlodipine Besylate Block of L-type calcium channel Amlodipine Besylate  Chemical Structure
  80. GC35325 Amlodipine maleate Amlodipine maleate is a dihydropyridine calcium channel blocker, acts as an orally active antianginal agent. Amlodipine maleate  Chemical Structure
  81. GC50334 AMP PNP AMP PNP (Adenylyl-imidodiphosphate tetralithium) is a non-hydrolysable analogue of ATP and inhibits KATP channels. AMP PNP  Chemical Structure
  82. GC62840 AMPA receptor modulator-2 AMPA receptor modulator-2 (Example 134) is a AMPA receptor modulator, with a pIC50 of 10.1 for TARPγ2 dependent AMPA receptor. AMPA receptor modulator-2  Chemical Structure
  83. GC68438 AMPA receptor modulator-3 AMPA receptor modulator-3  Chemical Structure
  84. GC13164 Ampalex An AMPA receptor modulator Ampalex  Chemical Structure
  85. GC14537 AMTB hydrochloride TRPM8 channel blocker AMTB hydrochloride  Chemical Structure
  86. GC30866 Anabasine ((S)-Anabasine) Anabasine ((S)-Anabasine) ((S)-Anabasine ((S)-Anabasine)) is an alkaloid that found as a minor component in tobacco (Nicotiana). Anabasine ((S)-Anabasine)  Chemical Structure
  87. GC39254 Anatabine dicitrate Anatabine dicitrate is a tobacco alkaloid that can cross the blood-brain barrier. Anatabine dicitrate  Chemical Structure
  88. GC46086 Ani 9 An inhibitor of ANO1 Ani 9  Chemical Structure
  89. GC32566 Anipamil Anipamil is a long-acting calcium channel blocker, used for the treatment of cardiovascular disease. Anipamil  Chemical Structure
  90. GC17695 Aniracetam Nootropic drug for senile dementia Aniracetam  Chemical Structure
  91. GC18203 Annonacin Annonacin is a potent and lipophilic acetogenin from A. Annonacin  Chemical Structure
  92. GC31141 Antihistamine-1 Antihistamine-1 is a H1-antihistamine (Ki=6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively. Antihistamine-1  Chemical Structure
  93. GC50471 AP 14145 hydrochloride KCa2 channel negative allosteric modulator AP 14145 hydrochloride  Chemical Structure
  94. GC18020 AP 18

    Reversible TRPA1 channel blocker

    AP 18  Chemical Structure
  95. GC42821 AP219 AP39 is a compound used to increase the levels of hydrogen sulfide (H2S) within mitochondria. AP219  Chemical Structure
  96. GC42823 AP39 AP39 is a compound used to increase the levels of hydrogen sulfide (H2S) within mitochondria. AP39  Chemical Structure
  97. GC14893 Apamin small-conductance Ca2+-activated K+-channel (KCa2, SK) inhibitor Apamin  Chemical Structure
  98. GC38557 Apamin TFA Apamin TFA (Apamine TFA) is an 18 amino acid peptide neurotoxin found in apitoxin (bee venom), is known as a specifically selective blocker of Ca2+-activated K+ (SK) channels and exhibits anti-inflammatory and anti-fibrotic activity. Apamin TFA  Chemical Structure
  99. GC17168 APETx2 acid-sensing ion channel 3 (ASIC3) channel blocker APETx2  Chemical Structure
  100. GC65272 APETx2 TFA APETx2 TFA, a sea anemone peptide from Anthopleura elegantissima, is a selective and reversible ASIC3 inhibitor, with an IC50 of 63 nM. APETx2 TFA  Chemical Structure
  101. GC30911 Apimostinel (NRX-1074) Apimostinel (NRX-1074) (NRX-1074; AGN-241660) is an orally active NMDA receptor partial agonist. Apimostinel (NRX-1074)  Chemical Structure

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