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Home >> Signaling Pathways >> Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Products for  Membrane Transporter/Ion Channel

  1. Cat.No. Product Name Information
  2. GC46841 Amiloride (hydrochloride) (hydrate)

    MK-870

     A neuropeptide with diverse biological activities Amiloride (hydrochloride) (hydrate) Chemical Structure
  3. GC31431 Amiloride (MK-870) Amiloride (MK-870) is a selective T-type calcium channel blocker and an inhibitor of epithelial sodium channels (ENaC) and urokinase-type plasminogen activator receptor (uTPA), Ki=7 µM. It is also polycystin-2 (PC2;TRPP2) channel blocker. Amiloride (MK-870) Chemical Structure
  4. GC17853 Amiloride HCl

    MK-870

     Amiloride HCl (MK-870 hydrochloride) is an inhibitor of both epithelial sodium channel (ENaC[1]) and urokinase-type plasminogen activator receptor (uTPA[2]). Amiloride HCl Chemical Structure
  5. GC12051 Amiloride HCl dihydrate Amiloride HCl dihydrate (MK-870 hydrochloride dihydrate) is an inhibitor of both epithelial sodium channel (ENaC[1]) and urokinase-type plasminogen activator receptor (uTPA[2]). Amiloride HCl dihydrate Chemical Structure
  6. GC34064 Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride)

    Aminooxyacetate

     Aminooxyacetic acid (Carboxymethoxylamine) hemihydrochloride is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA degradating enzyme GABA-T. Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) Chemical Structure
  7. GC35322 Amiodarone Amiodarone is an antiarrhythmic drug for inhibition of ATP-sensitive potassium channel with an IC50 of 19.1 μM. Amiodarone Chemical Structure
  8. GC11432 Amiodarone HCl Amiodarone HCl, a benzofuran-based Class III antiarrhythmic agent, inhibits WT outwardIhERG tails with an IC50 of ~45 nM. Amiodarone HCl Chemical Structure
  9. GC18274 Amiprofos-methyl

    APM, NSC 313446

     Amiprofos-methyl (APM) is a phosphoric amide herbicide. Amiprofos-methyl Chemical Structure
  10. GC13723 Amitriptyline HCl

    NIH 10794, Ro 4-1575

     Amitriptyline HCl is an inhibitor of serotonin reuptake transporter (SERT) and noradrenaline reuptake transporter (NET), with Kis of 3.45 nM and 13.3 nM for human SERT and NET, respectively. Amitriptyline HCl Chemical Structure
  11. GC13523 Amlodipine

    Intervask, Pelmec

     Calcium channel blocker Amlodipine Chemical Structure
  12. GC13146 Amlodipine Besylate Block of L-type calcium channel Amlodipine Besylate Chemical Structure
  13. GC35325 Amlodipine maleate Amlodipine maleate is a dihydropyridine calcium channel blocker, acts as an orally active antianginal agent. Amlodipine maleate Chemical Structure
  14. GC50334 AMP PNP AMP PNP (adenylyl-imidodiphosphate) is a non-hydrolyzable analog of ATP. AMP PNP Chemical Structure
  15. GC70946 AMPA receptor antagonist-3 AMPA receptor antagonist-3 is an AMPA receptor antagonist extracted from patent US20070027143A1. AMPA receptor antagonist-3 Chemical Structure
  16. GC70348 AMPA receptor modulator-1 AMPA receptor modulator-1 is a potent, orally active and selective AMPAR regulatory protein TARP γ-8 negative modulator with a pIC50 of 9.7, more selective over GluA1/γ-2 (pIC50=5). AMPA receptor modulator-1 Chemical Structure
  17. GC62840 AMPA receptor modulator-2 AMPA receptor modulator-2 (Example 134) is a AMPA receptor modulator, with a pIC50 of 10.1 for TARPγ2 dependent AMPA receptor. AMPA receptor modulator-2 Chemical Structure
  18. GC68438 AMPA receptor modulator-3 AMPA receptor modulator-3 Chemical Structure
  19. GC13164 Ampalex

    Ampalex, BDP-12, Benzoyl-Piperidine-12

     An AMPA receptor modulator Ampalex Chemical Structure
  20. GC14537 AMTB hydrochloride TRPM8 channel blocker AMTB hydrochloride Chemical Structure
  21. GC30866 Anabasine ((S)-Anabasine) Anabasine ((S)-Anabasine) ((S)-Anabasine ((S)-Anabasine)) is an alkaloid that found as a minor component in tobacco (Nicotiana). Anabasine ((S)-Anabasine) Chemical Structure
  22. GC39254 Anatabine dicitrate Anatabine dicitrate is a tobacco alkaloid that can cross the blood-brain barrier. Anatabine dicitrate Chemical Structure
  23. GC46086 Ani 9 An inhibitor of ANO1 Ani 9 Chemical Structure
  24. GC32566 Anipamil Anipamil is a long-acting calcium channel blocker, used for the treatment of cardiovascular disease. Anipamil Chemical Structure
  25. GC17695 Aniracetam

    Memodrin, Ro 13-5057, Sarpul

     Nootropic drug for senile dementia Aniracetam Chemical Structure
  26. GC68659 Anisatin

    Anisatin is a toxic substance isolated from the seeds of a Japanese plant (Illicium anisatum). It is a non-competitive b>GABA antagonist and belongs to the class of convulsant toxins. Anisatin inhibits GABA-induced currents in a concentration-dependent manner, with an EC50 of approximately 1.10 μM.

     Anisatin Chemical Structure
  27. GC18203 Annonacin Annonacin is a potent and lipophilic acetogenin from A. Annonacin Chemical Structure
  28. GC68663 ANO1-IN-1

    ANO1-IN-1 (Compound 9c) is a selective ANO1 channel blocker with IC50 values of 2.56 μM and 15.43 μM for ANO1 and ANO2, respectively. ANO1-IN-1 strongly inhibits the proliferation of glioma cells.

     ANO1-IN-1 Chemical Structure
  29. GC72240 Anthopleurin-A TFA Anthopleurin-A TFA is a soidum channel toxin. Anthopleurin-A TFA Chemical Structure
  30. GC31141 Antihistamine-1 Antihistamine-1 is a H1-antihistamine (Ki=6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively. Antihistamine-1 Chemical Structure
  31. GC50471 AP 14145 hydrochloride KCa2 channel negative allosteric modulator AP 14145 hydrochloride Chemical Structure
  32. GC18020 AP 18

    Reversible TRPA1 channel blocker

     AP 18 Chemical Structure
  33. GC42821 AP219 AP39 is a compound used to increase the levels of hydrogen sulfide (H2S) within mitochondria. AP219 Chemical Structure
  34. GC71431 AP30663 AP30663 is a KCa2 channel inhibitor that can be used for the study of atrial fibrillation. AP30663 Chemical Structure
  35. GC42823 AP39 AP39 is a compound used to increase the levels of hydrogen sulfide (H2S) within mitochondria. AP39 Chemical Structure
  36. GC14893 Apamin

    Ro 23-6721

     small-conductance Ca2+-activated K+-channel (KCa2, SK) inhibitor Apamin Chemical Structure
  37. GC38557 Apamin TFA

    Apamine TFA

     Apamin TFA (Apamine TFA) is an 18 amino acid peptide neurotoxin found in apitoxin (bee venom), is known as a specifically selective blocker of Ca2+-activated K+ (SK) channels and exhibits anti-inflammatory and anti-fibrotic activity. Apamin TFA Chemical Structure
  38. GC17168 APETx2 acid-sensing ion channel 3 (ASIC3) channel blocker APETx2 Chemical Structure
  39. GC65272 APETx2 TFA APETx2 TFA, a sea anemone peptide from Anthopleura elegantissima, is a selective and reversible ASIC3 inhibitor, with an IC50 of 63 nM. APETx2 TFA Chemical Structure
  40. GC30911 Apimostinel (NRX-1074)

    NRX-1074; AGN-241660

     Apimostinel (NRX-1074) (NRX-1074; AGN-241660) is an orally active NMDA receptor partial agonist. Apimostinel (NRX-1074) Chemical Structure
  41. GC42827 Apoptolidin

    Apoptolidin A

     Apoptolidin is an apoptosis inducer originally isolated from Nocardiopsis bacteria. Apoptolidin Chemical Structure
  42. GC71601 Aprindine hydrochloride Aprindine hydrochloride is a class I-b anti-arrhythmic agent and a hERG channel blocker with an IC50 of 0.23 μM. Aprindine hydrochloride Chemical Structure
  43. GC50226 AR-C 141990 hydrochloride MCT1 inhibitor AR-C 141990 hydrochloride Chemical Structure
  44. GC10680 AR-C155858 An inhibitor of MCT1 and 2 AR-C155858 Chemical Structure
  45. GC34049 Aranidipine (MPC1304) Aranidipine (MPC1304) (MPC1304) is a Ca2+ channel antagonist with potent and long-lasting antihypertensive effects. Aranidipine (MPC1304) Chemical Structure
  46. GC14470 Arcaine sulfate NMDA antagonist Arcaine sulfate Chemical Structure
  47. GC63879 Arecaidine hydrochloride Arecaidine hydrochloride, a pyridine alkaloid, is a potent GABA uptake inhibitor. Arecaidine hydrochloride Chemical Structure
  48. GC17225 ARL 67156 trisodium salt

    FPL 67156 trisodium

     ARL67156 (FPL 67156) trisodium is a selective ecto-ATPase inhibitor. ARL 67156 trisodium salt Chemical Structure
  49. GC74029 ASCT2-IN-1 ASCT2-IN-1 (compound 20k) is an ASCT2 inhibitor with IC50 values of 5.6 μM and 3.5 μM in cells A549 and HEK293, respectively. ASCT2-IN-1 Chemical Structure
  50. GC74030 ASCT2-IN-2 ASCT2-IN-2 (compound 25e) is an ASCT2 inhibitor with IC50 of 5.14 μM. ASCT2-IN-2 Chemical Structure
  51. GC35407 Asivatrep

    PAC-14028

     Asivatrep (PAC-14028) is a potent and selective transient receptor potential vanilloid type I (TRPV1) antagonist. Asivatrep Chemical Structure
  52. GC50115 ASP 7663 Selective TRPA1 activator ASP 7663 Chemical Structure
  53. GC38888 ASP2535 ASP2535 is a potent, orally bioavailable, selective, brain permeable and centrally-active glycine transporter-1 (GlyT1) inhibitor. ASP2535 Chemical Structure
  54. GC61960 ASP2905 ASP2905 is a potent and selective potassium channel Kv12.2 inhibitor encoded by the Kcnh3/BEC1 gene. ASP2905 Chemical Structure
  55. GC45387 Aspergillimide

    Asperparaline A, VM 55598

     Aspergillimide ((rel)-Aspergillimide), an anthelmintic metabolite, is isolated from okara that has been fermented with Aspergillus japonicas JV-23. Aspergillimide Chemical Structure
  56. GC16945 Astemizole

    NSC 329963

     anti-histamine compound, potent Astemizole Chemical Structure
  57. GC72112 Astressin 2B TFA Astressin 2B TFA is a potent and selective corticotropin-releasing factor receptor 2 (CRF2) antagonist, with the IC50 values of 1.3 nM and > 500 nM for CRF2 and CRF1, respectively. Astressin 2B TFA Chemical Structure
  58. GC12945 Atazanavir

    BMS 232632, CGP 73547

     An inhibitor of HIV-1 protease Atazanavir Chemical Structure
  59. GC10240 Atazanavir sulfate (BMS-232632-05) An inhibitor of HIV-1 protease Atazanavir sulfate (BMS-232632-05) Chemical Structure
  60. GC49421 Atorvastatin lactone-d5 An internal standard for the quantification of atorvastatin lactone Atorvastatin lactone-d5 Chemical Structure
  61. GC11109 ATP disodium salt

    5'-ATP, ATP, NSC 20268

     P2 purinoceptor agonist ATP disodium salt Chemical Structure
  62. GC35421 ATP synthase inhibitor 1 ATP synthase inhibitor 1 is a potent inhibitor of c subunit of the F1/FO-ATP synthase complex, inhibits mitochondrial permeability transition pore (mPTP) opening, does not affect ATP levels. ATP synthase inhibitor 1 Chemical Structure
  63. GC38497 ATPA ATPA Chemical Structure
  64. GC12721 ATPA GluR5 kainate receptor agonist ATPA Chemical Structure
  65. GC46891 ATPA (hydrate) An agonist of GluR5 ATPA (hydrate) Chemical Structure
  66. GC12574 ATPγS tetralithium salt

    ATPγS

     ATPγS (tetralithium salt) is a substrate for the nucleotide hydrolysis and RNA unwinding activities of eukaryotic translation initiation factor eIF4A. ATPγS tetralithium salt Chemical Structure
  67. GC15667 Atracurium Besylate

    BW 33A, Tracrium, Wellcome 33A74

     Neuromuscular blocking agent Atracurium Besylate Chemical Structure
  68. GC72125 ATX-II TFA ATX-II TFA is a specific Na+ channel Modulator toxin that can be isolated from the venom of sea anemone (Anemonia sulcata). ATX-II TFA Chemical Structure
  69. GC39699 Aurintricarboxylic acid Aurintricarboxylic acid is a nanomolar-potency, allosteric antagonist with selectivity towards αβ-methylene-ATP-sensitive P2X1Rs and P2X3Rs, with IC50s of 8.6 nM and 72.9 nM for rP2X1R and rP2X3R, respectively. Aurintricarboxylic acid Chemical Structure
  70. GC19480 AUT1

    Cell permeant modulator

     AUT1 Chemical Structure
  71. GC42876 Autocamtide 2 (trifluoroacetate salt) Autocamtide 2 is a peptide substrate for calcium/calmodulin-dependent protein kinase (CaMK) and CaMKII. Autocamtide 2 (trifluoroacetate salt) Chemical Structure
  72. GC15099 Autocamtide-2-related inhibitory peptide inhibitor of calmodulin-dependent protein kinase II (CaM-kinase II, CaMKII) Autocamtide-2-related inhibitory peptide Chemical Structure
  73. GC70456 AVE-0118 AVE-0118 is a nonselective Kv1.5 blocker with an IC50 of 1.1 μM. AVE-0118 Chemical Structure
  74. GC72973 AVE1231

    A293

     AVE1231 (A293) is a dual-pore potassium channel TASK-1 inhibitor with antiarrthmic activity. AVE1231 Chemical Structure
  75. GC10974 AWD 131-138

    ELB138, Imepitoin

     AWD 131-138 (AWD 131-138) is a new low-affinity partial benzodiazepine receptor agonist with potent anticonvulsant and anxiolytic properties in rodent models. AWD 131-138 Chemical Structure
  76. GC17375 AZ 10606120 dihydrochloride Potent P2X7 receptor antagonist AZ 10606120 dihydrochloride Chemical Structure
  77. GC18052 AZ 11645373 Human P2X7 antagonist,potent and selective AZ 11645373 Chemical Structure
  78. GC63799 AZ194 AZ194 is a first-in-class, orally active inhibitor of CRMP2-Ubc9 interaction and inhibitor of NaV1.7 (IC50=1.2 μM). AZ194 Chemical Structure
  79. GC11010 AZD 3965 Ki = 1.6 nM for MCT1

    AZD 3965 is a potent inhibitor of monocarboxylate transporter 1 (MCT1). AZD 3965 Chemical Structure

  80. GC64274 AZD-5672 AZD-5672 is an orally active, potent, and selective CCR5 antagonist (IC50=0.32 nM). AZD-5672 Chemical Structure
  81. GC31010 AZD-6280 AZD-6280 is a selective GABAA(α2/3) receptor modulator, used for treatment of generalized anxiety disorder. AZD-6280 Chemical Structure
  82. GC68713 AZD0095

    AZD0095 is a selective and orally active MCT4 inhibitor (IC50: 1.3 nM). When used in combination with Cediranib, AZD0095 effectively inhibits tumor growth of NCI-H358 xenografts.

     AZD0095 Chemical Structure
  83. GC31674 AZD9056 hydrochloride AZD9056 hydrochloride is a selective orally active inhibitor of P2X7 which plays a significant role in inflammation and pain-causing diseases. AZD9056 hydrochloride Chemical Structure
  84. GC15101 Azelnidipine

    CS 905, RS 9054

     L-type calcium channel blocker;antihypertensive Azelnidipine Chemical Structure
  85. GC35451 Azelnidipine D7 Azelnidipine D7 Chemical Structure
  86. GC14515 Azimilide class III anti-arrhythmic drug Azimilide Chemical Structure
  87. GC35453 Azimilide Dihydrochloride

    NE 10064

     A class III antiarrhythmic agent Azimilide Dihydrochloride Chemical Structure
  88. GC38738 Azosemide Azosemide, a sulfonamide loop diuretic, is a potent NKCC1 inhibitor with IC50s of 0.246??M and 0.197??M for hNKCC1A and NKCC1B, respectively. Azosemide Chemical Structure
  89. GC61493 Azumolene Azumolene (EU4093 free base), a Dantrolene analog, is a muscle relaxant. Azumolene Chemical Structure
  90. GC42893 Azumolene (sodium salt)

    EU4093

     Azumolene is a muscle relaxant that inhibits the release of calcium from skeletal muscle sarcoplasmic reticulum. Azumolene (sodium salt) Chemical Structure
  91. GC17597 Bafilomycin A1

    NSC 381866

    Bafilomycin A1, a macrolide antibiotic isolated from the Streptomyces species, is an inhibitor of vacuolar H ATPase (V-ATPase).

     Bafilomycin A1 Chemical Structure
  92. GC10934 Bafilomycin C1

    2-Demethyl-2-methoxy-24-methyl-hygrolidin,L-681,110A1

     vacuolar H+-ATPases (V-ATPases) inhibitor Bafilomycin C1 Chemical Structure
  93. GC12302 Bafilomycin D vacuolar H+ ATPases (V-ATPases) inhibitor Bafilomycin D Chemical Structure
  94. GC45820 Balsalazide-d4 A neuropeptide with diverse biological activities Balsalazide-d4 Chemical Structure
  95. GC31990 Bamaluzole Bamaluzole is a GABA receptor agonist extracted from patent WO 2012064642 A1. Bamaluzole Chemical Structure
  96. GC31426 Bamaquimast (F 10126)

    F 10126; L 0042

     Bamaquimast (F 10126) (F 10126; L 0042) is a potent antiasthmatic drug. Bamaquimast (F 10126) Chemical Structure
  97. GC68723 Bamocaftor

    VX-659

    Bamocaftor (VX-659) is a cystic fibrosis transmembrane conductance regulator (CFTR) corrector designed to restore the function of F508del-CFTR protein. Bamocaftor can be used in combination with Tezacaftor and Ivacaftor for research on cystic fibrosis.

     Bamocaftor Chemical Structure
  98. GC35469 Barnidipine Barnidipine (Mepirodipine) is an L-type calcium antagonist (CaA) with high affinity for [3H] initrendipine binding sites (Ki=0.21 nmol/l), has selective action against CaA receptors. Barnidipine Chemical Structure
  99. GC13289 Barnidipine (hydrochloride)

    YM 09730-5

     calcium-channel blocker Barnidipine (hydrochloride) Chemical Structure
  100. GC19057 Basmisanil

    RG-1662

     Basmisanil is a highly selective GABAAα5 negative allosteric modulator. Basmisanil Chemical Structure
  101. GC39344 BAY-1797 A P2X4receptor antagonist BAY-1797 Chemical Structure

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