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Home >> Signaling Pathways >> Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Products for  Membrane Transporter/Ion Channel

  1. Cat.No. Product Name Information
  2. GC68735 BAY-390

    BAY-390 is a selective, cross-species active, and brain-penetrant TRPA1 inhibitor. BAY-390 inhibits hTRPA1 FLIPR, hTRPA1 Ephys, rTRPA1 FLIPR and rDRG Ephys with IC50 values of 16, 82, 63 and 35 nM respectively. BAY-390 can be used for research on inflammation.

     BAY-390 Chemical Structure
  3. GC19000 BAY-588 BAY-588 is a glucose transporter inhibitor and derivative of BAY-876 . BAY-588 Chemical Structure
  4. GC19488 BAY-8002

    BAY-8002 is a potent, selective, orally active inhibitor of monocarboxylate transporter 1 (MCT1)

     BAY-8002 Chemical Structure
  5. GC72475 BBT BBT is an enhancer of impaired glucose-stimulated insulin secretion (GSIS). BBT Chemical Structure
  6. GC16516 BCH

    2-amino-2-Norbornanecarboxylic Acid

     BCH (BCH) is a selective and competitive inhibitor of large neutral amino acid transporter 1 (LAT1) significantly inhibit cellular uptake of amino acids and mTOR phosphorylation, which induces the suppression of cancer growth and apoptosis. BCH Chemical Structure
  7. GC14276 BCTC vanilloid receptor 1 (TRPV1 receptor) antagonist BCTC Chemical Structure
  8. GC13323 BDS I Kv3.4 potassium channel blocker, potent and reversible BDS I Chemical Structure
  9. GC33723 Becampanel (AMP 397)

    AMP 397

     Becampanel (AMP 397) (AMP397) is the first competitive AMPA antagonist and an antiepileptic agent. Becampanel (AMP 397) Chemical Structure
  10. GC50661 BeKm 1 BeKm 1 is a HERG (human ether-a-go-go-related gene) blocking compound. BeKm 1 Chemical Structure
  11. GC12414 Bemegride GABA receptor antagonist Bemegride Chemical Structure
  12. GC13888 Benidipine HCl

    (±)-Benidipine, KW-3049

     Benidipine HCl is a dihydropyridine calcium channel blocker for the treatment of high blood pressure (hypertension). Benidipine HCl Chemical Structure
  13. GC11693 Benzamil hydrochloride

    Na+/Ca2+ exhanger (NCX) inhibitor

     Benzamil hydrochloride Chemical Structure
  14. GC49403 Benzarone

    L 2197, NSC 82134

     An active metabolite of benzbromarone Benzarone Chemical Structure
  15. GC14339 Benzethonium Chloride Potent inhibitor of nAChRs Benzethonium Chloride Chemical Structure
  16. GC13125 Benzocaine

    Ethyl 4-Aminobenzoate, H-4-Abz-OEt, NSC 4688, NSC 41531

     Sodium channel inhibitor Benzocaine Chemical Structure
  17. GC25134 Benzocaine hydrochloride

    Ethyl 4-aminobenzoate hydrochloride, Benzocaine HCl, Ethyl p-aminobenzoate hydrochloride

     Benzocaine hydrochloride (Ethyl 4-aminobenzoate, Ethyl p-aminobenzoate) is a surface anesthetic that acts by preventing transmission of impulses along nerve fibers and at nerve endings. Benzocaine hydrochloride Chemical Structure
  18. GC68749 Benzocaine-(ethyl-d5)

    Benzocaine-(ethyl-d5) is the deuterated form of Benzocaine. Benzocaine acts as a co-receptor for voltage-gated Na+ channels, with an IC50 value of 0.8 mM measured at +30 mV.

     Benzocaine-(ethyl-d5) Chemical Structure
  19. GC42919 Benzonatate

    Benzonatate is a reversible voltage-gated sodium channel blocker.

     Benzonatate Chemical Structure
  20. GC15533 Bepridil hydrochloride Calcium channel blocker Bepridil hydrochloride Chemical Structure
  21. GC39743 Bepridil hydrochloride hydrate Bepridil hydrochloride hydrate ((±)-Bepridil hydrochloride hydrate) is a non-selective, long-acting Ca+ channel antagonist and Na+, K+ channel inhibitor, with antianginal and type I antiarrhythmic effects. Bepridil hydrochloride hydrate Chemical Structure
  22. GC35501 Beta-Eudesmol

    (+)-β-Eudesmol

     A sesquiterpene with diverse biological activities Beta-Eudesmol Chemical Structure
  23. GC39546 Bevantolol hydrochloride

    CI-755, DL-Bevantolol, NC-1400

     A β1-AR antagonist Bevantolol hydrochloride Chemical Structure
  24. GC14664 BHQ BHQ (DTBHQ), the indirect food additive, regulates the activity of 5-lipoxygenase as well as the activity of COX-2 (IC50=1.8 and 14.1 μM for 5-LO and COX-2, respectively) . BHQ Chemical Structure
  25. GC34486 BI 01383298 An NaCT inhibitor BI 01383298 Chemical Structure
  26. GC34489 BI-749327 BI-749327 is a potent, high selectivity and orally bioavailable TRPC6 antagonist, with IC50s of 13 nM, 19 nM and 15 nM for mouse, human and guinea pig TRPC6, respectively. BI-749327 Chemical Structure
  27. GC34492 BI-9627 An NHE1 inhibitor BI-9627 Chemical Structure
  28. GC34494 Bifenazate An acaricide Bifenazate Chemical Structure
  29. GC60642 Bifenthrin

    (±)-Bifenthrin

     A synthetic pyrethroid insecticide Bifenthrin Chemical Structure
  30. GC33338 Biricodar (VX-710)

    VX-710

     Biricodar (VX-710) (VX-710) is a modulator of P-glycoprotein and MRP-1; shows effective chemosensitizing activity in multidrug resistant cells. Biricodar (VX-710) Chemical Structure
  31. GC10206 Bitopertin

    RG-1678, RO-4917838

     An inhibitor of GlyT1 Bitopertin Chemical Structure
  32. GC35527 Bitopertin R enantiomer Bitopertin R enantiomer (RG1678 R enantiomer; RO4917838 R enantiomer) is the R-enantiomer of Bitopertin. Bitopertin R enantiomer Chemical Structure
  33. GC10094 BL 1249 K2P2.1 (TREK-1) channel opener BL 1249 Chemical Structure
  34. GC64658 Bliretrigine Bliretrigine is a sodium channel blocker. Bliretrigine Chemical Structure
  35. GC60090 BLU-5937 BLU-5937 Chemical Structure
  36. GC14239 BMS 191011

    BMS-A

     BKCa channel opener BMS 191011 Chemical Structure
  37. GC31405 BMS-191095 BMS-191095 is an activators of mitochondrial ATP-sensitive potassium (mitoKATP) channels. BMS-191095 Chemical Structure
  38. GC70402 BMS-192364 BMS-192364 is targeting the Gα-RGS interaction to produce an inactive Gα-RGS complex. BMS-192364 Chemical Structure
  39. GC35538 BNC375 BNC375 is a potent, selective, and orally available type I positive allosteric modulator of α7 nAChRs with an EC50 of 1.9 μM. BNC375 Chemical Structure
  40. GC71999 Boeravinone B Boeravinone B, a dual inhibitor of NorA bacterial efflux pump of Staphylococcus aureus and human P-Glycoprotein, reduces the biofilm formation and intracellular invasion of bacteria. Boeravinone B Chemical Structure
  41. GC42965 Bongkrekic Acid

    Bongkrek Acid

    An inhibitor of mitochondrial adenine nucleotide translocase

     Bongkrekic Acid Chemical Structure
  42. GC62874 BPAM344 BPAM344 is a kainate receptor (KAR) subunits GluK1b, GluK2a, and GluK3a positive allosteric modulator (PAM). BPAM344 Chemical Structure
  43. GC68798 BPDBA

    BPDBA is a selective and non-competitive inhibitor of betaine/GABA transporter (BGT-1), with IC50 values of 20 μM for human BGT-1 and 35 μM for mouse GAT2.

     BPDBA Chemical Structure
  44. GC73391 bPiDI bPiDI is a novel selective α6β2 nicotinic receptor antagonist. bPiDI inhibits nicotine-evoked striatal dopamine (DA) release through an interaction with α6β2-containing nAChRs. bPiDI Chemical Structure
  45. GC30537 BPO-27 racemate BPO-27 racemate is a potent CFTR inhibitor with an IC50 of 8 nM. BPO-27 racemate Chemical Structure
  46. GC68799 BPU-11

    BPU-11 is a ligand for the hyperpolarization-activated cyclic nucleotide-gated (HCN) C-linker pocket (CLP) of HCN4 CLP. It can be used in research on congenital immune diseases.

     BPU-11 Chemical Structure
  47. GC70230 Br-PBTC Br-PBTC is a potent, 2/4 subtype-selective positive allosteric modulator of nAChRs (nicotinic acetylcholine receptors) with α2β2，α2β4，α4β2，α4β4，(α4β2)2α4 and (α4β2)2β2 EC50 ranges from 0.1~0.6 μM. Br-PBTC Chemical Structure
  48. GC64064 Bradanicline

    TC-5619

     Bradanicline is a highly selective α7 nicotinic acetylcholine receptor (nAChR) agonist (humanα7 nAChR: EC50=17 nM; Ki= 1.4 nM). Bradanicline Chemical Structure
  49. GC17683 Brefeldin A

    Ascotoxin, BFA, Cyanein, Decumbin, Nectrolide, NSC 56310, NSC 89671, NSC 107456, NSC 244390, Synergisidin

     Brefeldin A (BFA) is a fungal macrocyclic lactone and a potent, reversible inhibitor of intracellular vesicle formation and protein trafficking between the endoplasmic reticulum (ER) and the Golgi apparatus. Brefeldin A Chemical Structure
  50. GC11565 Bretazenil

    Ro 16-6028

     GABAA benzodiazepine site partial agonist Bretazenil Chemical Structure
  51. GC49740 Brevetoxin 3

    PbTx-3, T-17 Toxin

     A neurotoxin Brevetoxin 3 Chemical Structure
  52. GC42976 Brevetoxin B

    Brevetoxin 2, BTX-B, GbTx-2, PbTx-2

    Brevetoxin B is a polyketide neurotoxin produced by Karenia species and other dinoflagellates.

     Brevetoxin B Chemical Structure
  53. GC12421 Brilliant blue G-250

    Acid Blue 90,CBBG,Coomassie Brilliant Blue G-250,NSC 328382

     Brilliant Blue G-250 is a dye commonly used for the visualization of proteins separated by SDS-PAGE, offering a simple staining procedure and high quantitation. Brilliant blue G-250 Chemical Structure
  54. GC30521 Broflanilide Broflanilide is a potential insecticide and metabolized to Desmethyl-Broflanilide, which is a potent antagonist at the insect resistant-to-dieldrin (RDL) GABA Receptor, and inhibits S. Broflanilide Chemical Structure
  55. GC25174 Brucine sulfate heptahydrate Brucine is an alkaloid that acts as an antagonist at glycine receptors and paralyzes inhibitory neurons. Brucine sulfate heptahydrate Chemical Structure
  56. GC16833 BTB06584

    BTB

     F1F0 ATP synthases BTB06584 Chemical Structure
  57. GC42984 BTC (potassium salt) BTC (potassium salt) is a low affinity calcium indicator (Kd approximately 7-26 μM) featuring many desirable properties for cellular calcium imaging, including long excitation wavelengths (400/485 nm), low sensitivity to Mg2+, and accuracy of ratiometric measurement. BTC (potassium salt) Chemical Structure
  58. GC42985 BTC AM BTC AM is a cell-permeable acetoxy-methyl ester of BTC. BTC AM Chemical Structure
  59. GC50617 BTD Selective TRPC5 activator BTD Chemical Structure
  60. GC68816 Budiodarone tartrate

    ATI-2042 tartrate

    Budiodarone (ATI-2042) tartrate is a chemical analogue of Amiodarone, with balanced inhibition activity on multiple cardiac ion channels including potassium, sodium and calcium channels. Budiodarone tartrate is an antiarrhythmic agent.

     Budiodarone tartrate Chemical Structure
  61. GN10365 Bufalin

    NSC 89595

     Bufalin Chemical Structure
  62. GC35567 Bullatine A Bullatine A, a diterpenoid alkaloid of the genus Aconitum, possesses anti-rheumatic, anti-inflammatory and anti-nociceptive effects. Bullatine A Chemical Structure
  63. GC35568 Bulleyaconitine A Bulleyaconitine A is an analgesic and antiinflammatory drug isolated from Aconitum plants; has several potential targets, including voltage-gated Na+ channels. Bulleyaconitine A Chemical Structure
  64. GC15524 Bumetanide

    PF-1593, Ro 10-6338

     NKCC cotransporter inhibitor Bumetanide Chemical Structure
  65. GC46957 Bumetanide-d5 An internal standard for the quantification of bumetanide Bumetanide-d5 Chemical Structure
  66. GC42990 Bupivacaine Bupivacaine is a sodium channel blocker and local anesthetic. Bupivacaine Chemical Structure
  67. GC12410 Bupivacaine HCl

    AH 2250, (±)-1-butyl-2′,6′-Pipecoloxylidide

     Bupivacaine HCl is a NMDA receptor inhibitor. Bupivacaine HCl Chemical Structure
  68. GC30914 Butamben (Butyl 4-aminobenzoate) Butamben (Butyl 4-aminobenzoate) (Butyl 4-aminobenzoate) results in long-lasting relief from pain, without impairing motor function or other sensory functions. Butamben (Butyl 4-aminobenzoate) Chemical Structure
  69. GC50200 BX 430

    Blocker of P2X4 Compound 3.0

     Selective P2X4 allosteric antagonist BX 430 Chemical Structure
  70. GC64574 BZAD-01 BZAD-01 is a potent, selective and orally active inhibitor of NMDA NR2B subunit, with a Ki of 72 nM. BZAD-01 Chemical Structure
  71. GC15898 BzATP triethylammonium salt P2X7 receptor agonist BzATP triethylammonium salt Chemical Structure
  72. GC30977 Ca2+ channel agonist 1 Ca2+ channel agonist 1 is an agonist of N-type Ca2+ channel and an inhibitor of Cdk2, with EC50s of 14.23 μM and 3.34 μM, respectively, and is used as a potential treatment for motor nerve terminal dysfunction. Ca2+ channel agonist 1 Chemical Structure
  73. GC14768 CaCCinh-A01

    TMEM16 Blocker I

     calcium-activated chloride channel (CaCC) inhibitor CaCCinh-A01 Chemical Structure
  74. GN10792 Caffeic acid

    3,4-Dihydroxycinnamic Acid

     Caffeic acid Chemical Structure
  75. GC43115 Cal Green™ 1 (potassium salt)

    Calcium Green-1

    Cal Green™ 1 is a cell-impermeant fluorescent calcium indicator that is characterized by high quantum yield and low phototoxicity.

     Cal Green™ 1 (potassium salt) Chemical Structure
  76. GC43116 Cal Green™ 1 AM

    Calcium Green-1 AM

     Cal Green™ 1 AM is a cell-permeant fluorescent calcium indicator (Excitation 506 nm; Emission 531 nm). Cal Green™ 1 AM Chemical Structure
  77. GC32616 Calcium channel-modulator-1 Calcium channel-modulator-1 is a calcium channel modulator; blocks aortic contraction with an IC50 of 0.8 μM. Calcium channel-modulator-1 Chemical Structure
  78. GC10949 Calcium Ionophore I

    CA 1001, ETH 1001

    Ca2+-selective ionophore

     Calcium Ionophore I Chemical Structure
  79. GC34041 Caldaret (MCC-135)

    MCC-135

     Caldaret (MCC-135) is an intracellular Ca2+ handling modulator that acts through reverse mode Na+/Ca2+ exchanger inhibition. Caldaret (MCC-135) Chemical Structure
  80. GC14326 Calmidazolium chloride

    R 24571

    Calmodulin antagonist

     Calmidazolium chloride Chemical Structure
  81. GC43128 Calmodulin-Dependent Protein Kinase II (290-309) (trifluoroacetate salt) Calmodulin-dependent protein kinase II (290-309) is a synthetic peptide derived from the rat brain protein sequence that contains the calmodulin binding domain. Calmodulin-Dependent Protein Kinase II (290-309) (trifluoroacetate salt) Chemical Structure
  82. GC47021 Caloxin 2A1 (trifluoroacetate salt)

    VSNSNWPSFPSSGGG-NH2

     A neuropeptide with diverse biological activities Caloxin 2A1 (trifluoroacetate salt) Chemical Structure
  83. GC62885 Caloxin 2A1 TFA Caloxin 2A1 TFA is an extracellular plasma membrane Ca2+-ATPase (PMCA) peptide inhibitor. Caloxin 2A1 TFA Chemical Structure
  84. GC12104 CALP1

    Calcium-like Peptide 1

    Cell-permeable calmodulin (CaM) agonist

     CALP1 Chemical Structure
  85. GC65081 CALP1 TFA CALP1 TFA is a calmodulin (CaM) agonist (Kd of 88 ?M) with binding to the CaM EF-hand/Ca2+-binding site. CALP1 TFA Chemical Structure
  86. GC14889 CALP2 Cell-permeable calmodulin (CaM) antagonist CALP2 Chemical Structure
  87. GC61508 CALP2 TFA CALP2 TFA is a calmodulin (CaM) antagonist (Kd of 7.9 ?M) with high affinity for binding to the CaM EF-hand/Ca2+-binding site. CALP2 TFA Chemical Structure
  88. GC17687 CALP3 Cell-permeable calmodulin (CaM) agonist CALP3 Chemical Structure
  89. GC68824 Camlipixant

    BLU-5937

    Camlipixant (BLU-5937) is an effective, selective, non-competitive and orally active P2X3 homotrimer receptor antagonist with an IC50 of 25 nM for hP2X3 homotrimer. Camlipixant exhibits strong antitussive effects without taste alteration. Camlipixant can be used in the research of unexplained and refractory chronic cough.

     Camlipixant Chemical Structure
  90. GC31953 Camphor ((±)-Camphor) Camphor ((±)-Camphor) ((±)-Camphor ((±)-Camphor)) is a topical anti-infective and anti-pruritic and internally as a stimulant and carminative. Camphor ((±)-Camphor) Chemical Structure
  91. GC15930 Camstatin analog of PEP-19 with antagonism of calmodulin Camstatin Chemical Structure
  92. GC14065 Capsaicin Capsaicin is a highly selective agonist for the transient receptor potential cation channel, subfamily V, member 1 (TRPV1), a ligand-gated, nonselective cation channel, preferentially expressed on small-diameter sensory neurons. Capsaicin Chemical Structure
  93. GC17918 Capsazepine Capsazepine is a specific antagonist of the transient receptor potential vanilloid 1 (TRPV1) receptor with an IC50 value of 562nM. Capsazepine Chemical Structure
  94. GC49433 Capsiate A capsaicin analog with diverse biological activities Capsiate Chemical Structure
  95. GC12636 Capsiconiate

    Coniferyl (E)-8-methyl-6-nonenoate

     TRPV1 agonist Capsiconiate Chemical Structure
  96. GC17340 Carbamazepine Inhibitor of neuronal voltage-gated Na+ channels Carbamazepine Chemical Structure
  97. GC16937 Carbamoylcholine chloride

    Carbachol

    Cholinergic receptor agonist

     Carbamoylcholine chloride Chemical Structure
  98. GC39646 Carboxyamidotriazole Orotate

    L-651582 Orotate; CAI Orotate

     Carboxyamidotriazole Orotate (L-651582 Orotate) is the orotate salt form of Carboxyamidotriazole (CAI), an orally bioavailable signal transduction inhibitor. Carboxyamidotriazole Orotate Chemical Structure
  99. GC31224 Carburazepam (RGH 3331) Carburazepam (RGH 3331) is a drug which derives from benzodiazepine. Carburazepam (RGH 3331) Chemical Structure
  100. GC18069 Cardamonin

    Alpinetin chalcone, Cardamomin

     Cardamonin ((E)-Cardamomin) is a novel antagonist of hTRPA1 cation channel with an IC50 of 454 nM. Cardamonin Chemical Structure
  101. GC17842 CARIPORIDE

    HOE 642

     Potent NHE inhibitor CARIPORIDE Chemical Structure

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