AMPAR
AMPAR is an glutamate ionotropic α-amino-3-hydroxy- 5-methylisoxazole-4-propionic acid receptor that mediates fast excitatory synaptic transmission in the central nervous system.
Products for AMPAR
- Cat.No. Product Name Information
-
GC11071
(R)-AMPA
inactive enantiomer of AMPA
-
GC13631
(RS)-AMPA
AMPA agonist
-
GC13032
(RS)-AMPA hydrobromide
AMPAR agonist
-
GC11889
(S)-(-)-5-Fluorowillardiine
AMPA receptor agonist
-
GC17213
(S)-AMPA
L-AMPA
AMPA agonist -
GC17313
(S)-CPW 399
AMPA agonist,subtype-selective,weakly desensitizing
-
GC12863
1-BCP
Piperonylic acid piperidide
potentiator of AMPA-mediated responses -
GC13164
Ampalex
Ampalex, BDP-12, Benzoyl-Piperidine-12
An AMPA receptor modulator -
GC17695
Aniracetam
Memodrin, Ro 13-5057, Sarpul
Nootropic drug for senile dementia -
GC18079
CFM-2
AMPA antagonist
-
GC15012
Cl-HIBO
desensitising AMPA receptor agonist
-
GC13290
CMPDA
positive allosteric modulator of AMPA receptors
-
GC11799
CNQX
6cyano7Nitroquinoxaline2,3dione, FG 9065
CNQX is an effective competitive antagonist of AMPA/kainate receptors, with IC50 values of 0.3µM and 1.5µM, respectively[1]. -
GC14480
CNQX disodium salt
FG9065 disodium
CNQX disodium salt (FG9065 disodium) is a potent and competitive AMPA/kainate receptor antagonist with IC50s of 0.3 μM and 1.5 μM, respectively. -
GC12589
CP 465022 hydrochloride
AMPA receptor antagonist, non-competitive and selective
-
GC12742
CP-465022 (maleate)
AMPA antagonist
-
GC14495
CX 546
AMPA receptor potentiator
-
GC50111
CX 614
Positive allosteric modulator of AMPA receptors
-
GC12207
Cyclothiazide
Doburil
positive allosteric modulator of AMPA receptors -
GC11598
Diazoxide
NSC 64198, NSC 76130, SRG 95213
positive allosteric modulator of the AMPA and kainate receptors
-
GC10275
DNQX disodium salt
6,7-Dinitroquinoxaline-2,3-dione
Selective non-NMDA receptor antagonist
-
GC11259
GYKI 47261 dihydrochloride
AMPA receptor antagonist, non-competitive and selective
-
GC11301
GYKI 52466 dihydrochloride
GYKI 52466 dihydrochloride is an orally active, highly selective and noncompetitive AMPA/kainate receptor antagonist with the IC50 values of 7.5 and 11μM, respectively.
-
GC14842
GYKI 53655 hydrochloride
LY300168 hydrochloride
AMPA and kainate receptor antagonist -
GC17928
IDRA 21
Inhibits AMPA receptor desensitization
-
GC14140
IEM 1460
AMPA receptors blocker
-
GC13235
IEM 1925 dihydrobromide
AMPA receptor antagonist
-
GC45989
JNJ-55511118
A negative modulator of AMPA receptors containing TARP-γ8
-
GC16011
L-Quisqualic acid
L-Quisqualic acid (L-L-Quisqualic acid), a natural analog of glutamate, is a potent and pan two subsets (iGluR and mGluR) of excitatory amino acid (EAA) agonist with an EC50 of 45 nM and a Ki of 10 nM for mGluR1R.
-
GC13010
LY451395
LY451395
LY451395 (LY451395) is a potent and highly selective potentiator of the AMPA receptors. -
GC13349
Naspm trihydrochloride
1-Naphthylacetyl spermine
Ca2+-permeable AMPA receptor antagonist -
GC14156
NBQX
NBQX is a highly selective and competitive AMPA receptor antagonist.
-
GC13482
NBQX disodium salt
NBQX disodium salt is a potent, highly selective and competitive antagonist of α-amino-3-hydroxy-5-methyl-4-isoxazolepropionate (AMPA) receptors (AMPARs).
-
GC10270
Noopept
GVS111, Noopept, SGS 111
An Analytical Reference Standard -
GC14579
NPEC-caged-(S)-AMPA
AMPA receptor agonist
-
GC12999
Pep1-AGL
Analog of Pep1-TGL
-
GC17103
Pep1-TGL
Peptide containing the 'TGL' motif that corresponds to the C-terminus of GluR1 subunit
-
GC11244
pep2-AVKI
Inhibitor peptide that selectively disrupts binding of the GluR2 subunit(at the C-terminal PDZ site) to PICK1
-
GC10669
pep2-EVKI
Inhibitor peptide that selectively disrupts binding of the GluR2 subunit(at the C-terminal PDZ site) to PICK1
-
GC16112
pep2-SVKE
Inactive control peptide analog of pep2-SVKI
-
GC10272
pep2-SVKI
Inhibitor peptide corresponding to last 10 amino acids of the C-terminus of the GluR2 subunit
-
GC17069
pep2m
Peptide inhibitor of the interaction between the C-terminus of the GluR2 subunit and N-ethylmaleimide-sensitive fusion protein
-
GC14372
Pep2m, myristoylated
Myr-Pep2m
inhibitor of the interaction between AMPA receptor and N-ethylmaleimide-sensitive fusion protein (NSF) -
GC10551
pep4c
Inactive control peptide analog of pep2m
-
GC13007
PEPA
Novel allosteric potentiator of AMPA receptor desensitization
-
GC14492
PF 4778574
positive allosteric modulator of AMPA receptors
-
GC12703
Philanthotoxin 74
PhTx74
Philanthotoxin 74 (PhTx 74) is an AMPAR antagonist; inhibits GluR3 and GluR1 with IC50s of 263 and 296 nM, respectively. -
GC13684
S 18986
positive allosteric modulator of AMPA receptors
-
GC13728
SYM 2206
AMPA receptor antagonist
-
GC50582
TAT-GluA2 3Y
Inhibitor of AMPA receptor endocytosis
-
GC10415
Tezampanel
LY 293558;LY293558;LY-293558
AMPA receptor antagonist -
GC11397
UBP 282
AMPA and kainate receptor antagonist
-
GC50428
UoS 12258
Positive allosteric modulator of AMPA receptors
-
GC16909
YM 90K hydrochloride
YM 90K hydrochloride is a potent and selective AMPA receptor antagonist with a Ki of 84 nM.
-
GC16300
ZK 200775
ZK200775; MPQX
ZK 200775 (ZK200775) is a highly selective AMPA/kainate antagonist with little activity against NMDA; have Ki values of 3.2 nM, 100 nM, and 8.5 μM against quisqualate, kainate, and NMDA, respectively.