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Calcium Channel

Calcium channel is an ion channel that selectively permeable to calcium ions. It serves vital functions in cellular signal transduction.

Products for  Calcium Channel

  1. Cat.No. Product Name Information
  2. GC31873 NecroX-5 A necrosis inhibitor NecroX-5  Chemical Structure
  3. GC36713 Ned 19 Ned 19 is a selective membrane-permeant non competitive NAADP antagonist and inhibits NAADP-mediated Ca2+ signaling, with an IC50 of 65 nM. Ned 19 strongly inhibits tumor growth and vascularization as well as lung metastases in mice. Ned 19  Chemical Structure
  4. GC50308 Ned K NAADP signaling inhibitor Ned K  Chemical Structure
  5. GC13352 Neomycin sulfate

    Aminoglycoside antibiotic

    Neomycin sulfate  Chemical Structure
  6. GC32563 Nexopamil racemate Nexopamil racemate is the racemate of Nexopamil. Nexopamil racemate  Chemical Structure
  7. GC30986 Nicardipine (YC-93) Nicardipine (YC-93) (YC-93 free base) is a calcium channel blocker with an IC50 of 1 μM for blocking cardiac calcium channels. Nicardipine (YC-93)  Chemical Structure
  8. GC10678 Nicardipine HCl Nicardipine HCl (YC-93) is a calcium channel blocker with an IC50 of 1 μM for blocking cardiac calcium channels. Nicardipine HCl  Chemical Structure
  9. GC64870 Nicardipine-d3 hydrochloride Nicardipine D3 hydrochloride (YC-93 D3) is the deuterium labeled Nicardipine hydrochloride. Nicardipine-d3 hydrochloride  Chemical Structure
  10. GC15024 Nifedipine L-type calcium channel blocker Nifedipine  Chemical Structure
  11. GC40207 Nifedipine-d6 Nifedipine-d6 is intended for use as an internal standard for the quantification of nifedipine by GC- or LC-MS. Nifedipine-d6  Chemical Structure
  12. GC13698 Nilvadipine

    Calcium channel inhibitor

    Nilvadipine  Chemical Structure
  13. GC16587 Nimodipine Calcium Channel inhibitor & Autophagy activator Nimodipine  Chemical Structure
  14. GC16889 Nisoldipine calcium channel blocker Nisoldipine  Chemical Structure
  15. GC62196 Nisoldipine-d7 Nisoldipine-d7  Chemical Structure
  16. GC16999 Nitrendipine Calcium channel blocker Nitrendipine  Chemical Structure
  17. GC69566 Nitrendipine-d5

    Nitrendipine-d5 is the deuterated form of Nitrendipine. Nitrendipine (BAY-E-5009) is a similar compound to Nifedipine. It is a dihydropyridine calcium channel blocker with vasodilatory properties and has antihypertensive effects.

    Nitrendipine-d5  Chemical Structure
  18. GC14417 NNC 55-0396 A selective T-type calcium channel inhibitor NNC 55-0396  Chemical Structure
  19. GC63118 Norverapamil D7 hydrochloride Norverapamil-d7 ((±)-Norverapamil-d7) hydrochloride is a deuterium labeled Norverapamil. Norverapamil D7 hydrochloride  Chemical Structure
  20. GC32518 Norverapamil hydrochloride ((±)-Norverapamil hydrochloride) Norverapamil hydrochloride ((±)-Norverapamil hydrochloride) ((±)-Norverapamil hydrochloride ((±)-Norverapamil hydrochloride)), an N-demethylated metabolite of Verapamil, is a L-type calcium channel blocker and a P-glycoprotein (P-gp) function inhibitor. Norverapamil hydrochloride ((±)-Norverapamil hydrochloride)  Chemical Structure
  21. GC61139 Nothofagin Nothofagin, a dihydrochalcone, is isolated from rooibos (Aspalathus linearis). Nothofagin  Chemical Structure
  22. GC36766 NP118809 NP118809 is a potent N-type calcium channel blocker, with an IC50 of 0.11 μM; also less potently inhibits L-type calcium channel with an IC50 of 12.2 μM. NP118809  Chemical Structure
  23. GC30997 NS-638 NS-638 is a small nonpeptide molecule with Ca2+-channel blocking properties. NS-638  Chemical Structure
  24. GC45536 Oleic Acid-13C   Oleic Acid-13C  Chemical Structure
  25. GC36843 Palonidipine Palonidipine is a calcium antagonist which is potential for the therapy of angina-pectoris and hypertension. Palonidipine  Chemical Structure
  26. GC11082 Paxilline High-conductance Ca2+-activated K+ (BKCa, KCa1.1) channels blocker Paxilline  Chemical Structure
  27. GC11678 PD 173212 N-type voltage-gated calcium channel blocker PD 173212  Chemical Structure
  28. GC32649 PD0176078 PD0176078 is a newly found N-type Calcium channel blocker. PD0176078  Chemical Structure
  29. GC10458 Penfluridol Dopamine receptor antagonist Penfluridol  Chemical Structure
  30. GC30055 Pinaverium bromide Pinaverium bromide is an L-type calcium channel blocker with selectivity for the gastrointestinal tract, effectively relieves pain, diarrhea and intestinal discomfort, provides good therapeutic efficacies without significant adverse effects on Irritable bowel syndrome (IBS) patients. Pinaverium bromide  Chemical Structure
  31. GC36955 Praeruptorin E Praeruptorin E is a main bioactive constituent of Peucedanum praeruptorum (also known as Bai-Hua Qian Hu). Praeruptorin E  Chemical Structure
  32. GC38230 Pranidipine Pranidipine (OPC-13340) is a potent, long acting 1,4-dihydropyridine calcium channel blocker with antihypertensive activity. Pranidipine  Chemical Structure
  33. GC61933 Propiverine hydrochloride Propiverine hydrochloride is a bladder spasmolytic with calcium antagonistic and anticholinergic properties. Propiverine hydrochloride  Chemical Structure
  34. GC10358 ProTx I CaV3.1 channel blocker ProTx I  Chemical Structure
  35. GC44796 Quin-2 (potassium salt) Quin-2 is a high-affinity fluorescent calcium indicator (Kd = 115 nM for calcium). Quin-2 (potassium salt)  Chemical Structure
  36. GC14487 Ranolazine Anti-ischemic Ranolazine  Chemical Structure
  37. GC13882 Ranolazine 2HCl Ranolazine 2HCl (CVT 303 dihydrochloride) is an anti-angina drug that achieves its effects by inhibiting the late phase of inward sodium current (INa and IKr with IC50 values of 6 μM and 12 μM, respectively) without affecting heart rate or blood pressure (BP). Ranolazine 2HCl  Chemical Structure
  38. GC44827 Rhod-2 (potassium salt) Rhod-2 (potassium salt) is a water-soluble, red fluorescent calcium indicator. Rhod-2 (potassium salt)  Chemical Structure
  39. GC44828 Rhod-2 (sodium salt)

    Rhod-2 (sodium salt) is a water-soluble, red fluorescent calcium indicator.

    Rhod-2 (sodium salt)  Chemical Structure
  40. GC44829 Rhod-5N (potassium salt) Rhod-5N is a low affinity fluorescent calcium probe (Kd = 320 μM). Rhod-5N (potassium salt)  Chemical Structure
  41. GC44830 Rhod-5N AM Rhod-5N AM is a cell-permeant acetoxymethyl ester of the fluorescent calcium indicator rhod-5N. Rhod-5N AM  Chemical Structure
  42. GC44834 Rhod-FF (potassium salt) Rhod-FF is a difluorinated analog of the cell-impermeant calcium indicator rhod-2. Rhod-FF (potassium salt)  Chemical Structure
  43. GC44835 Rhod-FF AM Rhod-FF AM is a cell-permeant acetoxymethyl ester of the fluorescent calcium indicator rhod-FF. Rhod-FF AM  Chemical Structure
  44. GC60330 Ru360 Ru360  Chemical Structure
  45. GC16766 Ruthenium Red

    Blocks Ca2+ uptake and release, and voltage-sensitive Ca2+ channels

    Ruthenium Red  Chemical Structure
  46. GC12607 Ryanodine Potent inhibitor of Ca2+ release from sarcoplasmic reticulum Ryanodine  Chemical Structure
  47. GC13016 Safinamide Safinamide  Chemical Structure
  48. GC50392 SAK 3 Potent CaV3.1 and 3.3 activator; orally bioavailable SAK 3  Chemical Structure
  49. GC32539 Semotiadil recemate fumarate Semotiadil recemate fumarate is the recemate of Semotiadil fumarate. Semotiadil recemate fumarate  Chemical Structure
  50. GC64311 SERCA2a activator 1 SERCA2a activator 1 (Compound A) is a sarco/endoplasmic reticulum Ca2+-dependent ATPase 2a (SERCA2a) activator. SERCA2a activator 1  Chemical Structure
  51. GC11041 Sipatrigine voltage-dependent sodium channels (NaV) blocker Sipatrigine  Chemical Structure
  52. GC32552 SM-6586 SM-6586 is a calcium channel antagonist and inhibitor of Na+/H+ and Na+/Ca2+ exchange transport, potentially for the treatment of cerebrovasular diseases and hypertension. SM-6586  Chemical Structure
  53. GC44905 SMI-481 SMI-481 is a selective inhibitor of the yeast phosphatidylinositol transfer protein (PITP) Sec14. SMI-481  Chemical Structure
  54. GC15237 SNX 482 voltage-dependent R-type CaV2.3 calcium channel blocker SNX 482  Chemical Structure
  55. GC69925 SOICR-IN-1

    SOICR-IN-1 (compound 32) is an inhibitor of store-overload induced calcium release (SOICR), with an IC50 value of 14.6 μM. SOICR-IN-1 can be used for research on cardiac arrhythmias.

    SOICR-IN-1  Chemical Structure
  56. GC32603 SQ-31765 (SQ31765) SQ-31765 (SQ31765) is a benzazepine calcium channel blocker. SQ-31765 (SQ31765)  Chemical Structure
  57. GC10351 SR 33805 oxalate Ca2+ channel antagonist SR 33805 oxalate  Chemical Structure
  58. GC61292 SR33805 SR33805 is a potent Ca2+ channel antagonist, with EC50s of 4.1 nM and 33 nM in depolarized and polarized conditions, respectively. SR33805  Chemical Structure
  59. GC15678 STO-609 acetate Ca2+-calmodulin-dependent protein kinase kinase inhibitor STO-609 acetate  Chemical Structure
  60. GC11819 Strontium Ranelate Calcium Channel activator Strontium Ranelate  Chemical Structure
  61. GC33732 Syntide 2 A protein kinase substrate Syntide 2  Chemical Structure
  62. GC37710 Syntide 2 (TFA) Syntide 2 (TFA)  Chemical Structure
  63. GC31038 TDN345 TDN345 is a Ca2+ antagonist, used for the treatment of vascular and senile dementia including Alzheimer's disease. TDN345  Chemical Structure
  64. GC33176 Teludipine hydrochloride (GR53992B) Teludipine is a lipophilic calcium channel blocker. Teludipine hydrochloride (GR53992B)  Chemical Structure
  65. GC39186 Terodiline hydrochloride Terodiline hydrochloride is an M1-selective muscarinic receptor (mAChR) antagonist with Kbs of 15, 160, 280, and 198 nM in rabbit vas deferens (M1), atria (M2), bladder (M3) and ileal muscle (M3), respectively. Terodiline hydrochloride  Chemical Structure
  66. GC12911 Tetracaine HCl Anaesthetic and allosteric inhibitor Tetracaine HCl  Chemical Structure
  67. GN10446 Tetrandrine Tetrandrine  Chemical Structure
  68. GC11482 Thapsigargin

    Thapsigargin?is an inhibitor of the sarcoplasmic/endoplasmic reticulum Ca2+ ATPase pump.

    Thapsigargin  Chemical Structure
  69. GC32549 Tiapamil hydrochloride (Ro 11-1781) Tiapamil hydrochloride (Ro 11-1781) is a calcium channel blocker. Tiapamil hydrochloride (Ro 11-1781)  Chemical Structure
  70. GC19438 TMB 8 (hydrochloride) TMB 8 is a non-competitive antagonist of nicotinic acetylcholine receptors (nAChRs) with IC50 values of 390 and 350 nM, respectively, for human muscle-type and α3β4 subunit-containing ganglionic nAChRs expressed in TE671/RD or SH-SY5Y cells. TMB 8 (hydrochloride)  Chemical Structure
  71. GC16149 Topiramate An anticonvulsant Topiramate  Chemical Structure
  72. GC50198 Topiramate - d12 Deuterated topiramate Topiramate - d12  Chemical Structure
  73. GC61342 TPC2-A1-N TPC2-A1-N is a powerful and Ca2+-permeable agonist of?two pore?channel?2?(TPC2), which plays its role by mimicking the physiological actions?of?NAADP. TPC2-A1-N  Chemical Structure
  74. GC15323 TRAM 39 Potent KCa3.1 blocker TRAM 39  Chemical Structure
  75. GC16322 trans-Ned 19 Nicotinic acid adenine dinucleotide phosphate (NAADP) antagonist trans-Ned 19  Chemical Structure
  76. GC49217 Trifluoperazine N-Glucuronide A metabolite of trifluoperazine Trifluoperazine N-Glucuronide  Chemical Structure
  77. GC48204 Trifluoperazine-d3 (hydrochloride) An internal standard for the quantification of trifluoperazine Trifluoperazine-d3 (hydrochloride)  Chemical Structure
  78. GC33458 Trimethadione (3,5,5,-Trimethyloxazolidine-2,4-dione) Trimethadione (3,5,5,-Trimethyloxazolidine-2,4-dione) (3,5,5,-Trimethyloxazolidine-2,4-dione) is an oxazolidinedione anticonvulsant agent widely used against absences seizures. Trimethadione (3,5,5,-Trimethyloxazolidine-2,4-dione)  Chemical Structure
  79. GC30950 TTA-Q6

    TTA-Q6 is a selective antagonist of T-type Ca2+ channel and can be used in neurological research.

    TTA-Q6  Chemical Structure
  80. GC50371 UK 59811 hydrochloride CaVAb blocker UK 59811 hydrochloride  Chemical Structure
  81. GC32571 UK51656 UK51656 is a calcium antagonist with IC50 of 4 nM. UK51656  Chemical Structure
  82. GC60377 Urolithin C Urolithin C, a gut-microbial metabolite of Ellagic acid, is a glucose-dependent activator of insulin secretion. Urolithin C  Chemical Structure
  83. GC61811 Verapamil Verapamil ((±)-Verapamil) is a calcium channel blocker and a potent and orally active first-generation P-glycoprotein (P-gp) inhibitor. Verapamil  Chemical Structure
  84. GC70115 Verapamil EP Impurity C hydrochloride

    NSC-609249 hydrochloride is an impurity of Verapamil. Verapamil is a calcium channel blocker and an effective oral first-generation P-glycoprotein (P-gp) inhibitor.

    Verapamil EP Impurity C hydrochloride  Chemical Structure
  85. GC17106 Verapamil HCl Verapamil HCl ((±)-Verapamil HCl) is a calcium channel blocker and a potent and orally active first-generation P-glycoprotein (P-gp) inhibitor. Verapamil HCl  Chemical Structure
  86. GC15583 W-13 hydrochloride

    calmodulin antagonist

    W-13 hydrochloride  Chemical Structure
  87. GC16962 W-5 hydrochloride calmodulin antagonist W-5 hydrochloride  Chemical Structure
  88. GC17496 W-7 hydrochloride calmodulin antagonist W-7 hydrochloride  Chemical Structure
  89. GC11260 W-9 hydrochloride calmodulin antagonist W-9 hydrochloride  Chemical Structure
  90. GC37950 Yangambin Yangambin, a furofuran lignan, is already isolated from plants such as member of the Annonaceae family, including species of the genus Rollinia: R. Yangambin  Chemical Structure
  91. GC14665 YM 58483 store-operated Ca2+ entry (SOCE) blocker YM 58483  Chemical Structure
  92. GC32648 YS-201 YS-201 is a dihydropyridine-type calcium channel antagonist. YS-201  Chemical Structure
  93. GC50432 Z 944 CaV3.x blocker Z 944  Chemical Structure
  94. GC63265 Ziconotide acetate Ziconotide acetate (SNX-111 acetate), a peptide, is a potent and selective block of N-type calcium channels antagonist. Ziconotide acetate  Chemical Structure
  95. GC11735 Zonisamide Antiepileptic with anticonvulsant and mechanistic effect Zonisamide  Chemical Structure
  96. GC17952 Zonisamide sodium Antiepileptic drug Zonisamide sodium  Chemical Structure
  97. GC30807 ZSET1446 (ST-101) ZSET1446 (ST-101) is a novel cognitive enhancer that significantly improves learning deficits in various types of Alzheimer disease (AD) models. ZSET1446 (ST-101)  Chemical Structure

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