GABA Receptor
GABA receptors are a class of receptors that respond to the GABA (neurotransmitter gamma-aminobutyric acid), the chief inhibitory neurotransmitter in the vertebrate central nervous system.
Products for GABA Receptor
- Cat.No. Product Name Information
- GC16353 N-ArachidonylGABA arachidonyl amino acid
- GC12169 NCS-382 γ-Hydroxybutyric acid antagonist
- GC11901 Nefiracetam GABA receptor activator
- GC31018 NEO 376 (SPI-376) NEO 376 (SPI-376) is a selective modulator of 5-HT1 receptor, GABA receptor and dopamine receptor, with anti-psychotic actively.
- GC16564 Niflumic acid Ca2+-activated Cl- channel blocker
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GC11821
NNC 05-2090 hydrochloride
GABA uptake inhibitor
- GC11748 NNC 711 NNC-711 (hydrochloride) is a potent and selective inhibitor of GAT-1 ( GABA transporter 1) with an IC50 of 40 nM for hGAT-1.
- GC11143 NS 11394 GABA(A) receptor-positive modulator
- GC16024 Ocinaplon GABAA receptors modulator
- GC19271 ONO-8590580 ONO-8590580 is a GABAA α5 negative allosteric modulator.
- GC14329 Org 20599 GABAA receptor agonist
- GC11963 Oxiracetam cyclic derivative of gamma-aminobutyric acid (GABA)
- GC31282 p-Hydroxybenzaldehyde p-Hydroxybenzaldehyde is a one of the major components in Dendrocalamus asper bamboo shoots, with antagonistic effect on GABAA receptor of the α1β2γ2S subtype at high concentrations.
- GC12357 Pentylenetetrazole CNS stimulant
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GC17691
Phaclofen
GABAB antagonist
- GC13557 PHP 501 trifluoroacetate GABAA antagonist
- GC30827 Pipequaline (PK-8165) Pipequaline (PK-8165) (PK 8165) is a partial benzodiazepine receptor agonist with anxiolytic activity.
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GC16569
PK 11195
peripheral benzodiazepine antagonist
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GC17399
Pregnanolone
GABAA receptor positive allosteric modulator
- GC15960 Primidone anticonvulsant of the pyrimidinedione class
- GC65057 Propofol-d18 Propofol-d18 is the deuterium labeled Propofol.
- GC16476 rac BHFF GABAB receptor positive allosteric modulator
- GC65513 Radequinil Radequinil (AC-3933) is a benzodiazepine receptor (BzR) partial inverse agonist.
- GC31257 Rilmazafone hydrochloride (450191S) Rilmazafone hydrochloride (450191S) (450191S) is a benzodiazepine (omega) ligand.
- GC13802 Riluzole Sodium channel protein inhibitor
- GC44841 Riluzole (hydrochloride) Riluzole is a benzothiazole derivative with anti-excitotoxic effects that acts by blocking the presynaptic release of glutamate, indirectly antagonizing glutamate receptors, and inactivating neuronal voltage-gated Na+ channels (ED50 = 2.3 μM).
- GC16780 Ro 15-4513 benzodiazepine ligand
- GC12377 Ro 19-4603 Benzodiazepine inverse agonist
- GC30433 Ru-32514 Ru-32514 is an agonist of benzodiazepine receptor.
- GC11612 RuBi GABA trimethylphosphine GABAB receptor agonist
- GC17321 RuBi-GABA Ruthenium-bipyridine-triphenylphosphine caged GABA
- GC13792 Rufinamide voltage-gated sodium channel blocker
- GC31049 RWJ-51204 RWJ-51204 is a partial agonist of GABA(A) receptor, with Ki of 0.2-2 nM to the benzodiazepine site on GABA(A) receptors.
- GC17257 Saclofen GABAB receptor antagonist
- GC16356 SB 205384 positive GABAA receptor modulator
- GC10888 SCH 50911 GABAB antagonist
- GC10844 SCS GABAA receptor antagonist
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GC69905
SJM-3
SJM-3 is a positive allosteric modulator of different subtypes of GABAA receptors. SJM-3 binds with high affinity to the α+/γ- subunit interface of the benzodiazepine binding site.
- GC15226 SKF 89976A hydrochloride GABA uptake inhibitor
- GC14942 SKF 97541 GABAB agonist
- GC10101 SR 95531 hydrobromide SR 95531 hydrobromide is a selective and competitive antagonist of GABAA receptor, with an IC50 of ~0.2 μM for GABA receptor.
- GC34362 SSD114 hydrochloride SSD114 hydrochloride is a novel GABAB receptor positive allosteric modulator.
- GC10967 TACA GABAA agonist
- GC17934 TB 21007 GABAA receptor inverse agonist
- GC15859 TCS 1105 GABAA benzodiazepine receptor (BZR) ligand
- GC10741 TCS 1205 TCS 1205 (compound 2b) is a potent and selective GABAA agonist.
- GC37784 THIP THIP (Gaboxadol) is a selective extrasynaptic GABAA receptors (eGABARs) agonist (with blood-brain barrier permeability), shows an EC50 value of 13 ?M for δ-GABAAR.
- GC10856 THIP hydrochloride THIP hydrochloride (Lu 02-030 hydrochloride) is a potent agonist of the GABAA receptor and an antagonist of GABAC receptors (IC50=25 μM).
- GC38215 Tiagabine
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GC17402
Tiagabine hydrochloride
GABA uptake inhibitor
- GC37788 Tiagabine hydrochloride hydrate Tiagabine hydrochloride hydrate is a potent and selective GABA uptake inhibitor, used as an anticonvulsant agent, with IC50s of 67, 446 and 182 nM for [3H]GABA uptake in Synaptosomes, Neurons and Glia, respectively.
- GC16360 TP 003 GABAA receptor (α3 subtype) partial agonist
- GC30865 TPA 023 TPA 023 is a GABAA α2/α3 subtype-selective agonist, with Ki of 0.19-0.41 nM.
- GC67996 TPA-023B
- GC10183 TPMPA GABAA-ρ antagonist
- GC10262 Tracazolate hydrochloride GABAA receptor modulator
- GC17381 trans-4-Hydroxycrotonic acid ligand of γ-hydroxybutyric acid (GHB) receptor
- GC14933 U 89843A Positive allosteric modulator of GABAA receptors
- GC13509 U 90042 GABAA receptor ligand
- GC11013 U 93631 GABAA receptor antagonist
- GC31013 U-101017 (PNU 101017) U-101017 (PNU 101017) is a partial agonist of benzodiazepine receptor and GABAA receptor, with anxiolytic effects.
- GC11600 Valerenic acid Positive allosteric modulator of GABAA receptor
- GC41613 Valnoctamide Valnoctamide is an isomer of the valproic acid amide, valpromide.
- GC37905 Vigabatrin Inhibitor of GABA transaminase
- GC13387 Vigabatrin Hydrochloride GABA transaminase inhibitor
- GC10313 ZAPA sulfate GABAA receptors agonist
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GC13922
ZK 93423 hydrochloride
GABAA receptor agonist
- GC16010 ZK 93426 hydrochloride benzodiazepine receptor antagonist,competitive