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GABA Receptor

GABA receptors are a class of receptors that respond to the GABA (neurotransmitter gamma-aminobutyric acid), the chief inhibitory neurotransmitter in the vertebrate central nervous system.

Products for  GABA Receptor

  1. Cat.No. Product Name Information
  2. GC16353 N-ArachidonylGABA arachidonyl amino acid N-ArachidonylGABA  Chemical Structure
  3. GC12169 NCS-382 γ-Hydroxybutyric acid antagonist NCS-382  Chemical Structure
  4. GC11901 Nefiracetam GABA receptor activator Nefiracetam  Chemical Structure
  5. GC31018 NEO 376 (SPI-376) NEO 376 (SPI-376) is a selective modulator of 5-HT1 receptor, GABA receptor and dopamine receptor, with anti-psychotic actively. NEO 376 (SPI-376)  Chemical Structure
  6. GC16564 Niflumic acid Ca2+-activated Cl- channel blocker Niflumic acid  Chemical Structure
  7. GC11821 NNC 05-2090 hydrochloride

    GABA uptake inhibitor

    NNC 05-2090 hydrochloride  Chemical Structure
  8. GC11748 NNC 711 NNC-711 (hydrochloride) is a potent and selective inhibitor of GAT-1 ( GABA transporter 1) with an IC50 of 40 nM for hGAT-1. NNC 711  Chemical Structure
  9. GC11143 NS 11394 GABA(A) receptor-positive modulator NS 11394  Chemical Structure
  10. GC16024 Ocinaplon GABAA receptors modulator Ocinaplon  Chemical Structure
  11. GC19271 ONO-8590580 ONO-8590580 is a GABAA α5 negative allosteric modulator. ONO-8590580  Chemical Structure
  12. GC14329 Org 20599 GABAA receptor agonist Org 20599  Chemical Structure
  13. GC11963 Oxiracetam cyclic derivative of gamma-aminobutyric acid (GABA) Oxiracetam  Chemical Structure
  14. GC31282 p-Hydroxybenzaldehyde p-Hydroxybenzaldehyde is a one of the major components in Dendrocalamus asper bamboo shoots, with antagonistic effect on GABAA receptor of the α1β2γ2S subtype at high concentrations. p-Hydroxybenzaldehyde  Chemical Structure
  15. GC12357 Pentylenetetrazole CNS stimulant Pentylenetetrazole  Chemical Structure
  16. GC17691 Phaclofen

    GABAB antagonist

    Phaclofen  Chemical Structure
  17. GC13557 PHP 501 trifluoroacetate GABAA antagonist PHP 501 trifluoroacetate  Chemical Structure
  18. GC30827 Pipequaline (PK-8165) Pipequaline (PK-8165) (PK 8165) is a partial benzodiazepine receptor agonist with anxiolytic activity. Pipequaline (PK-8165)  Chemical Structure
  19. GC16569 PK 11195

    peripheral benzodiazepine antagonist

    PK 11195  Chemical Structure
  20. GC17399 Pregnanolone

    GABAA receptor positive allosteric modulator

    Pregnanolone  Chemical Structure
  21. GC15960 Primidone anticonvulsant of the pyrimidinedione class Primidone  Chemical Structure
  22. GC65057 Propofol-d18 Propofol-d18 is the deuterium labeled Propofol. Propofol-d18  Chemical Structure
  23. GC16476 rac BHFF GABAB receptor positive allosteric modulator rac BHFF  Chemical Structure
  24. GC65513 Radequinil Radequinil (AC-3933) is a benzodiazepine receptor (BzR) partial inverse agonist. Radequinil  Chemical Structure
  25. GC31257 Rilmazafone hydrochloride (450191S) Rilmazafone hydrochloride (450191S) (450191S) is a benzodiazepine (omega) ligand. Rilmazafone hydrochloride (450191S)  Chemical Structure
  26. GC13802 Riluzole Sodium channel protein inhibitor Riluzole  Chemical Structure
  27. GC44841 Riluzole (hydrochloride) Riluzole is a benzothiazole derivative with anti-excitotoxic effects that acts by blocking the presynaptic release of glutamate, indirectly antagonizing glutamate receptors, and inactivating neuronal voltage-gated Na+ channels (ED50 = 2.3 μM). Riluzole (hydrochloride)  Chemical Structure
  28. GC16780 Ro 15-4513 benzodiazepine ligand Ro 15-4513  Chemical Structure
  29. GC12377 Ro 19-4603 Benzodiazepine inverse agonist Ro 19-4603  Chemical Structure
  30. GC30433 Ru-32514 Ru-32514 is an agonist of benzodiazepine receptor. Ru-32514  Chemical Structure
  31. GC11612 RuBi GABA trimethylphosphine GABAB receptor agonist RuBi GABA trimethylphosphine  Chemical Structure
  32. GC17321 RuBi-GABA Ruthenium-bipyridine-triphenylphosphine caged GABA RuBi-GABA  Chemical Structure
  33. GC13792 Rufinamide voltage-gated sodium channel blocker Rufinamide  Chemical Structure
  34. GC31049 RWJ-51204 RWJ-51204 is a partial agonist of GABA(A) receptor, with Ki of 0.2-2 nM to the benzodiazepine site on GABA(A) receptors. RWJ-51204  Chemical Structure
  35. GC17257 Saclofen GABAB receptor antagonist Saclofen  Chemical Structure
  36. GC16356 SB 205384 positive GABAA receptor modulator SB 205384  Chemical Structure
  37. GC10888 SCH 50911 GABAB antagonist SCH 50911  Chemical Structure
  38. GC10844 SCS GABAA receptor antagonist SCS  Chemical Structure
  39. GC69905 SJM-3

    SJM-3 is a positive allosteric modulator of different subtypes of GABAA receptors. SJM-3 binds with high affinity to the α+/γ- subunit interface of the benzodiazepine binding site.

    SJM-3  Chemical Structure
  40. GC15226 SKF 89976A hydrochloride GABA uptake inhibitor SKF 89976A hydrochloride  Chemical Structure
  41. GC14942 SKF 97541 GABAB agonist SKF 97541  Chemical Structure
  42. GC10101 SR 95531 hydrobromide SR 95531 hydrobromide is a selective and competitive antagonist of GABAA receptor, with an IC50 of ~0.2 μM for GABA receptor. SR 95531 hydrobromide  Chemical Structure
  43. GC34362 SSD114 hydrochloride SSD114 hydrochloride is a novel GABAB receptor positive allosteric modulator. SSD114 hydrochloride  Chemical Structure
  44. GC10967 TACA GABAA agonist TACA  Chemical Structure
  45. GC17934 TB 21007 GABAA receptor inverse agonist TB 21007  Chemical Structure
  46. GC15859 TCS 1105 GABAA benzodiazepine receptor (BZR) ligand TCS 1105  Chemical Structure
  47. GC10741 TCS 1205 TCS 1205 (compound 2b) is a potent and selective GABAA agonist. TCS 1205  Chemical Structure
  48. GC37784 THIP THIP (Gaboxadol) is a selective extrasynaptic GABAA receptors (eGABARs) agonist (with blood-brain barrier permeability), shows an EC50 value of 13 ?M for δ-GABAAR. THIP  Chemical Structure
  49. GC10856 THIP hydrochloride THIP hydrochloride (Lu 02-030 hydrochloride) is a potent agonist of the GABAA receptor and an antagonist of GABAC receptors (IC50=25 μM). THIP hydrochloride  Chemical Structure
  50. GC38215 Tiagabine Tiagabine  Chemical Structure
  51. GC17402 Tiagabine hydrochloride

    GABA uptake inhibitor

    Tiagabine hydrochloride  Chemical Structure
  52. GC37788 Tiagabine hydrochloride hydrate Tiagabine hydrochloride hydrate is a potent and selective GABA uptake inhibitor, used as an anticonvulsant agent, with IC50s of 67, 446 and 182 nM for [3H]GABA uptake in Synaptosomes, Neurons and Glia, respectively. Tiagabine hydrochloride hydrate  Chemical Structure
  53. GC16360 TP 003 GABAA receptor (α3 subtype) partial agonist TP 003  Chemical Structure
  54. GC30865 TPA 023 TPA 023 is a GABAA α2/α3 subtype-selective agonist, with Ki of 0.19-0.41 nM. TPA 023  Chemical Structure
  55. GC67996 TPA-023B TPA-023B  Chemical Structure
  56. GC10183 TPMPA GABAA-ρ antagonist TPMPA  Chemical Structure
  57. GC10262 Tracazolate hydrochloride GABAA receptor modulator Tracazolate hydrochloride  Chemical Structure
  58. GC17381 trans-4-Hydroxycrotonic acid ligand of γ-hydroxybutyric acid (GHB) receptor trans-4-Hydroxycrotonic acid  Chemical Structure
  59. GC14933 U 89843A Positive allosteric modulator of GABAA receptors U 89843A  Chemical Structure
  60. GC13509 U 90042 GABAA receptor ligand U 90042  Chemical Structure
  61. GC11013 U 93631 GABAA receptor antagonist U 93631  Chemical Structure
  62. GC31013 U-101017 (PNU 101017) U-101017 (PNU 101017) is a partial agonist of benzodiazepine receptor and GABAA receptor, with anxiolytic effects. U-101017 (PNU 101017)  Chemical Structure
  63. GC11600 Valerenic acid Positive allosteric modulator of GABAA receptor Valerenic acid  Chemical Structure
  64. GC41613 Valnoctamide Valnoctamide is an isomer of the valproic acid amide, valpromide. Valnoctamide  Chemical Structure
  65. GC37905 Vigabatrin Inhibitor of GABA transaminase Vigabatrin  Chemical Structure
  66. GC13387 Vigabatrin Hydrochloride GABA transaminase inhibitor Vigabatrin Hydrochloride  Chemical Structure
  67. GC10313 ZAPA sulfate GABAA receptors agonist ZAPA sulfate  Chemical Structure
  68. GC13922 ZK 93423 hydrochloride

    GABAA receptor agonist

    ZK 93423 hydrochloride  Chemical Structure
  69. GC16010 ZK 93426 hydrochloride benzodiazepine receptor antagonist,competitive ZK 93426 hydrochloride  Chemical Structure

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