Glucose Transporters
Products for Glucose Transporters
- Cat.No. Product Name Information
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GC64568
DRB18
DRB18 is a potent pan-class GLUT inhibitor. DRB18 alters energy-related metabolism in A549 cells by changing the abundance of metabolites in glucose-related pathways. DRB18 can eventually lead to G1/S phase arrest and increase oxidative stress and necrotic cell death. DRB18 has anti-tumor activity.
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GC43654
Fasentin
Fasentin is an inhibitor of glucose transport.
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GC64876
GLUT inhibitor-1
GLUT inhibitor-1 is a potent and orally active inhibitor of glucose transporters, targeting both GLUT1 and GLUT3, with IC50s of 242 nM and 179 nM, respectively.
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GC73808
Glutor
Glutor is a selective GLUT 1/2/3 inhibitor that can suppress glucose uptake.
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GC64014
KL-11743
KL-11743 is a potent, orally active, and glucose-competitive inhibitor of the class I glucose transporters, with IC50s of 115, 137, 90, and 68 nM for GLUT1, GLUT2, GLUT3, and GLUT4, respectively.
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GC70894
KPH2f
KPH2f is a safe, orally active, and effective dual URAT1/GLUT9 inhibitor with IC50s of 0.24 μM and 9.37 μM for URAT1 and GLUT9, respectively.
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GC45494
Lavendustin B
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GC69481
MMV009085
MMV009085 is an effective inhibitor of the Plasmodium falciparum hexose transporter PfHT1, making it a potential anti-malaria compound. It also inhibits human glucose transporters, with strong inhibitory effects on glucose uptake (IC50: 2.6 μM) and parasite growth (EC50: 1.23±0.04 μM; 3D7).
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GC72650
MSNBA
MSNBA is a specific inhibitor of GLUT5 fructose transport in proteoliposomes.
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GC71079
SLC26A3-IN-2
SLC26A3-IN-2 is an orally active inhibitor of anion exchanger protein SLC26A3 (IC50=360 nM).
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GC14803
STF 31
GLUT1 and NAMPT inhibitor
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GC66470
SW157765
SW157765 is a selective non-canonical glucose transporter GLUT8 (SLC2A8) inhibitor. KRAS/KEAP1 double mutant NSCLC cells are selectively sensitive to the SW157765, due to the convergent consequences of dual KRAS and NRF2 modulation of metabolic and xenobiotic gene regulatory programs.
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GC13381
WZB117
Glucose Transporter Inhibitor IV
Glucose transporter 1 (Glut1) inhibitor