Monoamine transporter
Monoamine transporters are a family of plasma membrane transporter that regulates the reuptake of neurotransmitters into nerve terminals. It divided into DAT (dopamine transporter), NET (norepinephrine transporter) and SERT (serotonin transporter).
Products for Monoamine transporter
- Cat.No. Product Name Information
- GC50649 FFN 200 dihydrochloride
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GC36705
NBI-98782
NBI-98782(alpha-dihydrotetrabenazine) is a vesicular monoamine transporter (VMAT2) inhibtior with an Ki value of 0.97 nM.
-
GC69565
Nisoxetine
Nisoxetine is an effective and selective norepinephrine transporter (NET) inhibitor with a Kd value of 0.76 nM. It is an antidepressant agent and local anesthetic that can block voltage-gated sodium channels.
- GC31060 Radafaxine hydrochloride (GW-353162A) Radafaxine hydrochloride (GW-353162A) (GW-353162A) is a DAT (dopamine transporter) and NET(norepinephrine transporter) transporters inhibitor, and nAChR family modulator.
- GN10779 Reserpine
- GC14792 Reserpine hydrochloride Blocker of VMAT
-
GC13672
Tetrabenazine
Tetrabenazine is the only US Food and Drug Administration-approved drug for Huntington's disease, indicated for treatment of chorea associated with Huntington's disease.
- GC37768 Tetrabenazine Racemate Tetrabenazine Racemate (Ro 1-9569 Racemate) is a selective and reversible inhibitor of vesicular monoamine transporter-2 (VMAT-2).
- GC40180 Tetrabenazine-d6 Tetrabenazine-d6 is intended for use as an internal standard for the quantification of tetrabenazine by GC- or LC-MS.
- GC37820 Trans (2,3)-Dihydrotetrabenazine Trans (2,3)-Dihydrotetrabenazine ((2R,3R,11bR)-rel-Dihydrotetrabenazine), a metabolite of Tetrabenazine, shows remarkable inhibition activity on vesicular monoamine transporter (VMAT2).
- GC19370 Valbenazine Valbenazine is a prodrug of the (+)-α isomer of tetrabenazine for tardive syndrome therapy, and inhibits VMAT2 function.
- GC26029 Valbenazine tosylate Valbenazine tosylate (NBI-98854) is the tosylate salt of valbenazine, a vesicular monoamine transporter 2 (VMAT2) inhibitor with a Ki value of 150 nM while displaying no significant binding to VAMT1(Ki<10 μM).
- GC30994 Vanilpyruvic acid (Vanylpyruvic acid) Vanilpyruvic acid (Vanylpyruvic acid) is a catecholamine metabolite and precursor to vanillactic acid.